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TargetMol | Compound Library

毒性化合物库现货

Toxic Compound Library

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产品编号 L5500

Targetmol 毒性化合物库包含 1520 个人工合成或天然存在的有机小分子,这些物质是能够改变细胞、代谢和膜功能的化合物,例如:DNA 合成干扰剂、酶抑制剂、受体阻断剂、膜活性化合物等细胞毒性化合物。这些化合物有些是没有继续研发的,有些是由于毒性或者其他原因停止了研究。也有些作为杀虫剂和除草剂使用。从 DNA 合成损害到细胞增殖毒性,从免疫抑制到内分泌干扰,Targetmol 毒性化合物库为您提供来源广泛、针对性强、研究明确的毒物小分子化合物,这些化合物的多样性可以增加科学家实验的视野,同时也可能揭示新的未知活性,是综合化筛选、针对性研究的有力工具。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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产品编号 L5500

毒性化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 1520个细胞毒性化合物的特有集合,可用于高通量、高内涵筛选。
  • 涵盖免疫、神经、呼吸、内分泌、心血管等各系统相关疾病。
  • 结构多样,药效显著,可渗透细胞。
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Apoptosis
Autophagy
Antibacterial
Antibiotic
5-HT Receptor
Adrenergic Receptor
Endogenous Metabolite
Dopamine Receptor
Parasite
DNA/RNA Synthesis
COX
Potassium Channel
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Histamine Receptor
HIV Protease
Sodium Channel
Calcium Channel
ROS
Cytochromes P450
SARS-CoV
NF-κB
Topoisomerase
Virus Protease
Ferroptosis
Antifungal
VEGFR
Mitophagy
Estrogen/progestogen Receptor
Serotonin Transporter
GABA Receptor
RAAS
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HCV Protease
c-Kit
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PDE
EGFR
PDGFR
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Influenza Virus
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Akt
Estrogen Receptor/ERR
iGluR
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HSV
Cholinesterase (ChE)
ribosome
Dehydrogenase
PPAR
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ERK
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c-Met/HGFR
PI3K
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MMP
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Src
JNK
MRP
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TLR
HDAC
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Proteasome
Prostaglandin Receptor
Nrf2
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ATPase
Progesterone Receptor
HBV
Antifolate
Bcl-2 Family
ALK
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PKC
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HSP
Phospholipase
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Thyroid hormone receptor(THR)
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P2Y Receptor
NADPH
ABC Transporter
glycosidase
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S1P Receptor
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IκB/IKK
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Aromatase
Melanocortin Receptor
MDM-2/p53
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PERK
GSK-3
Melatonin Receptor
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Na-K-Cl cotransporter
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CCR
DNA
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Ligands for Target Protein for PROTAC
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IRE1
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LDL
MT Receptor
Integrase
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ACK1
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Chk
Somatostatin
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cAMP
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TGF-beta/Smad
ATP Citrate Lyase
Wee1
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BCRP
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MAPK
Survivin
STING
GPCR19
Histone Acetyltransferase
transporter
CRFR
Casein Kinase
CRISPR/Cas9
PDK
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PLK
Platelet aggregation
NADPH-oxidase
NOD
S6 Kinase
NOD-like Receptor (NLR)
p53
PD-1/PD-L1
PGC-1α