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TargetMol | Compound Library

毒性化合物库现货

Toxic Compound Library
Rating icon 很棒
货号 L5500

Targetmol 毒性化合物库包含 1520 个人工合成或天然存在的有机小分子,这些物质是能够改变细胞、代谢和膜功能的化合物,例如:DNA 合成干扰剂、酶抑制剂、受体阻断剂、膜活性化合物等细胞毒性化合物。这些化合物有些是没有继续研发的,有些是由于毒性或者其他原因停止了研究。也有些作为杀虫剂和除草剂使用。从 DNA 合成损害到细胞增殖毒性,从免疫抑制到内分泌干扰,Targetmol 毒性化合物库为您提供来源广泛、针对性强、研究明确的毒物小分子化合物,这些化合物的多样性可以增加科学家实验的视野,同时也可能揭示新的未知活性,是综合化筛选、针对性研究的有力工具。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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毒性化合物库

货号:L5500

  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
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精选库规格 化合物库推荐

肝脏毒性化合物库
Drug-induced Liver Injury (DILI) Compound Library
L5510915 化合物
造血毒性小分子库
Hematopoietic Toxicity Compound Library
L3100125 化合物
心血管毒性化合物库
Cardiotoxicity Compound Library
L4900131 化合物
FDA 上市药物库
FDA-Approved Drug Library
L42002080 化合物

产品描述 产品描述

  • 1520个细胞毒性化合物的特有集合,可用于高通量、高内涵筛选。
  • 涵盖免疫、神经、呼吸、内分泌、心血管等各系统相关疾病。
  • 结构多样,药效显著,可渗透细胞。
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Apoptosis
Autophagy
Antibacterial
Antibiotic
5-HT Receptor
Adrenergic Receptor
Endogenous Metabolite
Parasite
Dopamine Receptor
Potassium Channel
DNA/RNA Synthesis
COX
Histamine Receptor
AChR
HIV Protease
Sodium Channel
Calcium Channel
ROS
Cytochromes P450
SARS-CoV
Topoisomerase
NF-κB
Virus Protease
Ferroptosis
Antifungal
VEGFR
Mitophagy
Estrogen/progestogen Receptor
RAAS
Serotonin Transporter
Reactive Oxygen Species
GABA Receptor
HCV Protease
Nucleoside Antimetabolite/Analog
PDE
EGFR
c-Kit
Influenza Virus
Microtubule Associated
PDGFR
Akt
Estrogen Receptor/ERR
Norepinephrine
Interleukin
Reverse Transcriptase
iGluR
Cholinesterase (ChE)
ribosome
Dehydrogenase
PPAR
Glucocorticoid Receptor
HSV
ERK
p38 MAPK
PI3K
c-Met/HGFR
MMP
FLT
Caspase
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FGFR
TNF
HMG-CoA Reductase
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Src
JNK
MRP
MAO
Bcr-Abl
HDAC
HIF/HIF Prolyl-Hydroxylase
DNA Alkylator/Crosslinker
TRP/TRPV Channel
Opioid Receptor
Prostaglandin Receptor
TLR
Nrf2
ATPase
Progesterone Receptor
HBV
Antifolate
Drug Metabolite
ALK
STAT
Anti-infection
Thrombin
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Transferase
Adenosine Receptor
PARP
Raf
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AMPK
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Androgen Receptor
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Endothelin Receptor
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Ras
DHFR
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ABC Transporter
GluR
SGLT
HSP
Phospholipase
ROS Kinase
Thyroid hormone receptor(THR)
LPL Receptor
P2Y Receptor
Reductase
GNRH Receptor
Leukotriene Receptor
PKC
glycosidase
CaMK
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TAM Receptor
S1P Receptor
ADC Cytotoxin
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Wnt/beta-catenin
ROCK
Mitochondrial Metabolism
Monoamine Transporter
Isocitrate Dehydrogenase (IDH)
DNA Alkylation
Telomerase
Antiviral
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HER
Kras
GPCR
Chloride channel
MTP
Serine Protease
Gamma-secretase
P2X Receptor
BTK
Glucosidase
Molecular Glues
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Xanthine Oxidase
Thrombopoietin Receptor
Lipoxygenase
OAT
Free radical scavengers
IκB/IKK
Retinoid Receptor
Melanocortin Receptor
MDM-2/p53
Integrin
Histone Demethylase
PERK
GSK-3
Melatonin Receptor
Na-K-Cl cotransporter
Guanylate cyclase
Ligands for E3 Ligase
Fatty Acid Synthase
CCR
DNA
FKBP
Aromatase
AhR
Vitamin
Proteasome
MALT
ASBT
ROR
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Ligands for Target Protein for PROTAC
Cell wall
Tie-2
Rho
Cysteine Protease
NR4A
Aryl Hydrocarbon Receptor
Immunology/Inflammation related
IRE1
Adenylate cyclase
UGT
LDL
MT Receptor
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Integrase
PAK
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Aurora Kinase
Epigenetic Reader Domain
IGF-1R
PANoptosis
Ephrin Receptor
Decarboxylase
GluCls
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FOXO
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CGRP Receptor
Cuproptosis
Complement System
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Sigma receptor
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Imidazoline Receptor
PKM
IKZF
PGC-1α
NPC1L1
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Hydrogenase
DNA-PK
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Na+/Ca2+ Exchanger
IFNAR
Necroptosis
TOPK
OCT
c-Myc
PKA
Photosensitizer
FXR
Glutaminase
LDLR
RANKL/RANK
CSF-1R
Myosin
RIP kinase
Adiponectin Receptor
GRK
GlyT
PROTAC Linker
HCN Channel
FAAH
ACK1
Bradykinin Receptor
CXCR
Somatostatin
Chk
Epoxide Hydrolase
cAMP
Mucin
DUB
TGF-beta/Smad
ATP Citrate Lyase
Wee1
BCRP
OXPHOS
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PGE Synthase
MAPK
Survivin
STING
GPCR19
Sirtuin
Histone Acetyltransferase
transporter
CRFR
Casein Kinase
CRISPR/Cas9
PDK
Aquaporin
PLK
NADPH-oxidase
S6 Kinase
NOD-like Receptor (NLR)
p53
PD-1/PD-L1