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毒性化合物库

毒性化合物库

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产品编号 L5500 Toxic Compound Library
  库化合物信息   Excel SDF

Targetmol 毒性化合物库包含 277 个人工合成或天然存在的有机小分子,这些物质是能够改变细胞、代谢和膜功能的化合物,例如:DNA 合成干扰剂、酶抑制剂、受体阻断剂、膜活性化合物等细胞毒性化合物。这些化合物有些是没有继续研发的,有些是由于毒性或者其他原因停止了研究。也有些作为杀虫剂和除草剂使用。从 DNA 合成损害到细胞增殖毒性,从免疫抑制到内分泌干扰,Targetmol 毒性化合物库为您提供来源广泛、针对性强、研究明确的毒物小分子化合物,这些化合物的多样性可以增加科学家实验的视野,同时也可能揭示新的未知活性,是综合化筛选、针对性研究的有力工具。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
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产品描述

  • 277个细胞毒性化合物的特有集合,可用于高通量、高内涵筛选。
  • 包括药物:222个;作用机制和毒理研究已有一定基础。
  • 包括天然产物:89个;活性明确,多为中药有效成分,是极具吸引力的毒理研究小分子。
  • 涉及的靶点超过150个;?涵盖免疫、神经、呼吸、内分泌、心血管等各系统相关疾病。
  • 结构多样,药效显著,可渗透细胞。
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L5500)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

DNA/RNA Synthesis (72)
Apoptosis (58)
Autophagy (57)
Antibacterial (49)
Antibiotic (46)
Endogenous Metabolite (32)
Parasite (21)
Nucleoside Antimetabolite/Analog (19)
DNA Alkylator/Crosslinker (13)
COX (13)
Potassium Channel (12)
Dehydrogenase (11)
Topoisomerase (11)
Antifungal (11)
Histamine Receptor (10)
Mitophagy (10)
HSV (9)
Reactive Oxygen Species (8)
Adrenergic Receptor (7)
HIV Protease (7)
SARS-CoV (7)
Ferroptosis (7)
AChR (7)
ribosome (7)
Dopamine Receptor (6)
Microtubule Associated (6)
PDE (5)
DNA Alkylation (5)
DNA (5)
5-HT Receptor (5)
PPAR (5)
Calcium Channel (5)
Influenza Virus (5)
Antifolate (5)
Sodium Channel (4)
HCV Protease (4)
NMDAR (4)
STAT (4)
Antifection (4)
P450 (4)
BCL (4)
ATPase (3)
MAO (3)
Antioxidant (3)
Chloride channel (3)
PKC (3)
EGFR (3)
HDAC (3)
HBV (3)
Virus Protease (3)
Phospholipase (3)
NF-κB (3)
mTOR (3)
Lipoxygenase (2)
iGluR (2)
Mitochondrial Metabolism (2)
PKA (2)
Monoamine Oxidase (2)
Norepinephrine (2)
Opioid Receptor (2)
Phosphatase (2)
ROS (2)
Sirtuin (2)
Thyroid hormone receptor(THR) (2)
TLR (2)
TNF (2)
Transferase (2)
Tyrosinase (2)
VEGFR (2)
AChE (2)
Wnt/beta-catenin (2)
HSP (2)
Akt (2)
DHFR (2)
DNA Methyltransferase (2)
Drug Metabolite (2)
CAT (2)
Casein Kinase (2)
Glucocorticoid Receptor (2)
Aromatase (2)
AMPK (2)
GABA Receptor (2)
Adenosine Receptor (2)
HIF/HIF Prolyl-Hydroxylase (2)
AhR (1)
CDK (1)
Proton pump (1)
Ras (1)
Adenosine deaminase (1)
CFTR (1)
Retinoid Receptor (1)
Reverse Transcriptase (1)
Rho (1)
Cell wall (1)
ROR (1)
RSV (1)
Amino Acids and Derivatives (1)
UGT (1)
Serotonin Transporter (1)
Sigma receptor (1)
Tyrosine Kinases (1)
Carbonic Anhydrase (1)
Prostaglandin Receptor (1)
CaMK (1)
Syk (1)
Adiponectin receptor (1)
TGF-beta/Smad (1)
TRP/TRPV Channel (1)
Trk receptor (1)
Proteasome (1)
CXCR (1)
c-Met/HGFR (1)
Gamma-secretase (1)
Histone Acetyltransferase (1)
IκB/IKK (1)
KLF (1)
HIF (1)
HER (1)
MEK (1)
Hedgehog/Smoothened (1)
GPR (1)
Glutathione Peroxidase (1)
MMP (1)
GluR (1)
MRP (1)
MTH1 (1)
NADPH (1)
NO Synthase (1)
Complement System (1)
PAD (1)
CRISPR/Cas9 (1)
HMG-CoA Reductase (1)
PI3K (1)
DNA gyrase (1)
P-gp (1)
PAK (1)
p53 (1)
FGFR (1)
DUB (1)
p38 MAPK (1)
Endothelin Receptor (1)
ERK (1)
Factor Xa (1)
Nrf2 (1)
IGF-1R (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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