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神经递质受体化合物库

神经递质受体化合物库

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产品编号 L2610 Neurotransmitter Receptor Compound Library
  库化合物信息   Excel SDF

神经递质是人类行为的化学基础。研究证实行为病理大都由一个或数个神经递质缺失或增多失平衡引起。躯体疾病也可由于特殊的神经径路障碍引起,例如帕金森病(PD)。脑内神经递质分为生物原胺类、氨基酸类、肽类、乙酰胆碱类等。生物原胺类神经递质包括:多巴胺(DA)、去甲肾上腺素(NE)、肾上腺素(E)、5-羟色胺(5-HT)也称(血清素)。氨基酸类神经递质包括:γ-氨基丁酸(GABA)、甘氨酸、谷氨酸、组胺。肽类神经递质分为:内源性阿片肽、P 物质、神经加压素、胆囊收缩素(CCK)、生长抑素、血管加压素和缩宫素、神经肽 Y。其它神经递质还有:核苷酸类、花生酸碱、阿南德酰胺、sigma 受体(σ受体)。在突触后膜或效应器细胞膜上有能与神经递质相结合的特殊蛋白质,称神经递质受体或突触后受体。许多精神药物作用于神经递质受体。

TargetMol 收集了 1513 种神经递质受体相关的化合物,可用于神经系统药物的开发。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
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产品描述

  • 1513种与神经递质受体相关的化合物,用于高通量、高内涵筛选;
  • 靶点包括5-HT receptor、AChR、GABA receptor、dopamine receptor、Opiod receptor等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L2610)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

5-HT Receptor (330)
AChR (287)
Dopamine Receptor (217)
Adrenergic Receptor (215)
Histamine Receptor (153)
GABA Receptor (130)
GluR (90)
Opioid Receptor (80)
Adenosine Receptor (72)
AChE (71)
iGluR (70)
NMDAR (65)
Autophagy (58)
Endogenous Metabolite (54)
Apoptosis (40)
Norepinephrine (33)
Serotonin Transporter (27)
Antibacterial (26)
Potassium Channel (24)
Calcium Channel (23)
Parasite (19)
Sodium Channel (19)
Neuropeptide Y Receptor (18)
Endothelin Receptor (17)
P450 (15)
PDE (13)
Influenza Virus (11)
cholecystokinin (9)
NF-κB (9)
Antibiotic (8)
Antifungal (7)
Mitophagy (7)
CaMK (7)
HIV Protease (7)
Sigma receptor (6)
Phospholipase (6)
HDAC (6)
Reactive Oxygen Species (6)
P-gp (5)
TRP/TRPV Channel (5)
Drug Metabolite (5)
TNF (5)
HCV Protease (5)
COX (5)
DNA/RNA Synthesis (4)
Adenosine deaminase (4)
Monoamine Transporter (4)
ERK (4)
NO Synthase (4)
Histone Methyltransferase (4)
Dehydrogenase (4)
Ferroptosis (4)
Caspase (3)
Virus Protease (3)
GPR (3)
Transferase (3)
AMPK (3)
Prostaglandin Receptor (3)
HSV (3)
Chloride channel (3)
PI3K (3)
VEGFR (3)
RAAS (3)
Tyrosinase (3)
BACE (3)
Cannabinoid Receptor (3)
Beta-Secretase (3)
Beta Amyloid (3)
ABC (3)
Glucocorticoid Receptor (3)
PPAR (2)
SARS-CoV (2)
Imidazoline Receptor (2)
RSV (2)
Aurora Kinase (2)
MAO (2)
cAMP (2)
Transaminase (2)
HER (2)
PARP (2)
mTOR (2)
NOS (2)
Adenylyl cyclase (2)
IL Receptor (2)
HBV (2)
Melatonin Receptor (2)
DYRK (2)
Gamma-secretase (2)
GSK-3 (2)
P2X Receptor (2)
PAFR (2)
MEK (2)
MRP (2)
ROS (2)
Antioxidant (2)
BCL (2)
PKA (2)
transporter (2)
Monoamine Oxidase (2)
STAT (1)
GST (1)
Reverse Transcriptase (1)
FLT (1)
CRISPR/Cas9 (1)
Hydroxylase (1)
FGFR (1)
Gap Junction Protein (1)
Platelet aggregation (1)
Syk (1)
Anti-infection (1)
NOD (1)
DNA Methyltransferase (1)
HMG-CoA Reductase (1)
Microtubule Associated (1)
HIF/HIF Prolyl-Hydroxylase (1)
FAK (1)
p53 (1)
GluCls (1)
Melanin-concentrating Hormone Receptor (MCHR) (1)
Nrf2 (1)
Progesterone Receptor (1)
Bcr-Abl (1)
Adiponectin receptor (1)
Annexin A (1)
IAP (1)
Immunology/Inflammation related (1)
Aryl Hydrocarbon Receptor (1)
Leukotriene Receptor (1)
FXR (1)
Antifolate (1)
Phosphatase (1)
Raf (1)
GTPase (1)
NADPH (1)
Na+/Ca2+ Exchanger (1)
Estrogen/progestogen Receptor (1)
p38 MAPK (1)
Amino Acids and Derivatives (1)
Integrin (1)
Carbonic Anhydrase (1)
CAT (1)
LDL (1)
GRK (1)
Aminopeptidase (1)
Lipoxygenase (1)
Trk receptor (1)
Acyltransferase (1)
MAPK (1)
Akt (1)
TGF-beta/Smad (1)
Interleukin (1)
Indoleamine 2,3-Dioxygenase (IDO) (1)
Androgen Receptor (1)
DNA (1)
Epigenetic Reader Domain (1)
MT Receptor (1)
ACK (1)
PAD (1)
MMP (1)
CCR (1)
Bombesin Receptor (1)
Fatty Acid Synthase (1)
Antifection (1)
Mitochondrial Metabolism (1)
Glucosidase (1)
GlyT (1)
Stearoyl-CoA Desaturase (SCD) (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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