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Endoplasmic Reticulum Stress Compound Library
内质网应激(Endoplasmic Reticulum stress)是细胞为应对内质网腔内错误折叠与未折叠蛋白聚集以及钙离子平衡紊乱等状况,而激活未折叠蛋白反应、内质网超负荷反应和 caspase-12 介导的凋亡通路等信号途径的反应过程。内质网应激既能诱导葡糖调节蛋白(glucose-regulated protein)GRP78、GRP94 等内质网分子伴侣表达而产生保护效应,亦能独立地诱导内源性细胞凋亡,并影响应激细胞的转归,如适应、损伤或凋亡。 内质网应激是一种重要的防御机制,参与多种疾病进程,是一种泛在的病因机制。近年来的研究表明,癌症、炎症性疾病、代谢性疾病、骨质疏松症及神经退行性疾病等有内质网应激信号传递参与。 TargetMol 内质网应激化合物库收录了 223 个内质网应激相关的化合物,靶向 PERK、IRE1、ATF6、GRP78等内质网应激信号通路相关靶点,是研究内质网应激及相关疾病的良好工具。
Empty | 99-66-1 | 98665-15-7 | 95975-55-6 | 951441-04-6 | 94805-82-0 | 940289-57-6 | 936498-64-5 | 934343-74-5 | 932986-18-0 | 929007-72-7 | Empty |
Valproic Acid | Ganoderic acid F | Guggulsterone | Icerguastat | Glycycoumarin | VER49009 | ICL-CCIC-0019 | NVP-HSP990 | Azoramide | DB07268 | ||
Empty | 919091-63-7 | 91-53-2 | 912999-49-6 | 908115-27-5 | 908112-43-6 | 90729-43-4 | 894804-07-0 | 892711-75-0 | 888216-25-9 | 88-58-4 | Empty |
RA-9 | Ethoxyquin | Onalespib | PF04929113 | SNX2112 | Ebastine | JNK Inhibitor VIII | CDN1163 | Ganetespib | 2,5-Di-tert-butylhydroquinone | ||
Empty | 88321-09-9 | 883065-90-5 | 88182-33-6 | 874101-00-5 | 867164-40-7 | 866405-64-3 | 865783-99-9 | 865273-97-8 | 864388-65-8 | 85650-56-2 | Empty |
Aloxistatin | BI-78D3 | Levistolide A | RO4987655 | TRC051384 | Dorsomorphin | Briciclib | ERAP1-IN-1 | MK-28 | Asenapine Maleate | ||
Empty | 851983-85-2 | 848695-25-0 | 848344-36-5 | 847559-80-2 | 84687-43-4 | 84057-84-1 | 834-28-6 | 819812-04-9 | 792-74-5 | 790186-68-4 | Empty |
Galeterone | BIIB021 | Bentamapimod | VER-82576 | Astragaloside IV | Lamotrigine | Phenformin hydrochloride | KW-2478 | Dimethyl biphenyl-4,4'-dicarboxylate | GW284543 | ||
Empty | 75747-14-7 | 74901-20-5 | 747413-08-7 | 747412-49-3 | 73-31-4 | 7085-55-4 | 6809-52-5 | 67920-52-9 | 67526-95-8 | 668467-91-2 | Empty |
Tanespimycin | MC2184 | VER-50589 | Luminespib | Melatonin | Troxerutin | Teprenone | Danshensu sodium salt | Thapsigargin | LDN-57444 | ||
Empty | 666859-49-0 | 6659-45-6 | 65914-17-2 | 64984-31-2 | 633-65-8 | 6100-05-6 | 608512-97-6 | 606-58-6 | 595-15-3 | 58-61-7 | Empty |
Antipsychotic agent 54 | Dihydrorotenone | (E/Z)-Polydatin | Pifithrin-μ | Berberine chloride | Hydroxycitric acid tripotassium hydrate | PKR-IN-C16 | Toyocamycin | Soyasapogenol B | Adenosine | ||
Empty | 57396-78-8 | 57-10-3 | 557795-19-4 | 548470-11-7 | 53452-16-7 | 529-44-2 | 52549-17-4 | 52286-59-6 | 511532-96-0 | 5104-49-4 | Empty |
Oroxin A | Palmitic acid | Sunitinib | ISRIB | Vaccarin | Myricetin | Pranoprofen | Ginsenoside Re | GP 1a | Flurbiprofen | ||
Empty | 50892-23-4 | 50773-41-6 | 501-36-0 | 500565-15-1 | 489-32-7 | 488832-69-5 | 475231-21-1 | 471-95-4 | 471-87-4 | 467214-21-7 | Empty |
Pirinixic Acid | Polyphyllin I | Resveratrol | HM03 | Icariin | Elesclomol | 3'-Hydroxypterostilbene | Bufotalin | Stachydrine | Alvespimycin hydrochloride |