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离子通道库

离子通道库

产品编号 L2300 Ion Channel Inhibitor Library
  库化合物信息   Excel SDF

离子跨膜通道的调节是治疗多种疾病的基础,离子通道是开发新的高效药物治疗的重要靶点,随着人类基因组计划的完成和转录机制研究的深入,离子通道分布的组织特异性逐渐得以阐明,这将使离子通道成为一类有选择性的组织特异性药物靶点。离子通道对于细胞间通讯至关重要,并调节多种重要的生理过程,这些过程功能障碍,可导致广泛的疾病和病理状况,如糖尿病、神经性疼痛、心血管疾病、大脑和外周血管疾病、哮喘、神经退行性疾病。

为满足客户离子通道相关研究的化合物需求,我们根据文献报道和其他公开资料精心整理 946 种与离子通道相关的生物活性小分子化合物,适用于离子通道相关的疾病和药物研究。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
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产品描述

  • 946种与离子通道相关的生物活性小分子化合物的特有集合,用于离子通道相关的疾病和药物研究,可用于高通量筛选和高内涵筛选;
  • 靶点含K+通道、Ca2+通道、Na+通道、质子泵等;
  • 通过前期临床研究和临床实验,生物活性和安全性已经得到验证;
  • 其中一些活性化合物已得到FDA批准上市;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR和HPLC检测技术保证产品高纯度和高质量;
  • 所有化合物现货供应。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L2300)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

Potassium Channel (169)
Calcium Channel (154)
Sodium Channel (126)
GABA Receptor (102)
TRP/TRPV Channel (99)
Autophagy (84)
iGluR (67)
ATPase (54)
Endogenous Metabolite (52)
AChR (48)
Apoptosis (38)
P-gp (35)
NMDAR (34)
Antibacterial (32)
Parasite (28)
P2X Receptor (26)
Proton pump (26)
Chloride channel (25)
P450 (20)
GluR (19)
Reactive Oxygen Species (17)
5-HT Receptor (17)
COX (16)
NF-κB (16)
CFTR (16)
Adrenergic Receptor (15)
Dopamine Receptor (15)
Antibiotic (13)
HIV Protease (13)
ABC (11)
PPAR (9)
Antifungal (9)
Monoamine Transporter (8)
CaMK (8)
GPR (8)
transporter (8)
HER (8)
Ferroptosis (8)
SGLT (8)
Monocarboxylate transporter (8)
Histamine Receptor (7)
BCRP (7)
OCT (7)
TNF (7)
Influenza Virus (7)
Carbonic Anhydrase (7)
SARS-CoV (6)
EGFR (6)
MRP (6)
AChE (6)
Na+/Ca2+ Exchanger (6)
OAT (6)
IL Receptor (6)
DNA/RNA Synthesis (6)
Phospholipase (5)
Mitochondrial Metabolism (5)
Drug Metabolite (5)
Topoisomerase (5)
PKC (5)
Virus Protease (5)
NPC1L1 (5)
CRM1 (5)
Antioxidant (5)
Mitophagy (5)
Cannabinoid Receptor (4)
Myosin (4)
PDE (4)
AMPK (4)
GluCls (3)
Hedgehog/Smoothened (3)
NO Synthase (3)
HSV (3)
STAT (3)
NADPH (3)
Lipoxygenase (3)
ERK (3)
PKA (3)
Caspase (3)
mTOR (3)
HDAC (3)
Serine/threonin kinase (3)
Norepinephrine (3)
VDAC (3)
CGRP Receptor (3)
TGF-beta/Smad (3)
MMP (2)
Prostaglandin Receptor (2)
Beta Amyloid (2)
Interleukin (2)
Lipid (2)
Akt (2)
Beta-Secretase (2)
GST (2)
IκB/IKK (2)
Fatty Acid Synthase (2)
RAAS (2)
Aquaporin (2)
HBV (2)
DNA Methyltransferase (2)
HMG-CoA Reductase (2)
Phosphatase (2)
TOPK (2)
Tyrosinase (2)
Anti-infection (2)
AhR (2)
NOD-like Receptor (NLR) (2)
p38 MAPK (2)
Integrin (2)
Src (2)
NOS (2)
Wnt/beta-catenin (2)
NOD (2)
Syk (2)
LDL (2)
Opioid Receptor (2)
ROS (2)
Na-K-Cl cotransporter (2)
GlyT (2)
FLT (2)
MEK (2)
Platelet aggregation (2)
Gamma-secretase (2)
ROCK (2)
VEGFR (2)
CRISPR/Cas9 (1)
S6 Kinase (1)
Sigma receptor (1)
FGFR (1)
Thrombin (1)
HIF/HIF Prolyl-Hydroxylase (1)
Gap Junction Protein (1)
HIF (1)
Reverse Transcriptase (1)
Hydroxylase (1)
PKM (1)
Proteasome (1)
HCN Channel (1)
RSV (1)
GSK-3 (1)
MAO (1)
Amylase (1)
FXR (1)
Cysteine Protease (1)
Serotonin Transporter (1)
PARP (1)
Estrogen Receptor/ERR (1)
N-Acetylglucosaminyltransferase (1)
CaSR (1)
JNK (1)
Glucocorticoid Receptor (1)
Reductase (1)
Adenosine Receptor (1)
LPL Receptor (1)
PI3K (1)
Dehydrogenase (1)
Estrogen/progestogen Receptor (1)
Piezo Channel (1)
Transaminase (1)
Transferase (1)
Taste receptor (1)
CSF-1R (1)
Adiponectin receptor (1)
Casein Kinase (1)
cAMP (1)
PAI-1 (1)
Nrf2 (1)
Trk receptor (1)
HSP (1)
MAPK (1)
Androgen Receptor (1)
DNA (1)
IGF-1R (1)
Epigenetic Reader Domain (1)
PAK (1)
UGT (1)
PDGFR (1)
BCL (1)
PROTAC Linker (1)
Anion Exchanger (1)
Antifection (1)
BTK (1)
DNA gyrase (1)
MT Receptor (1)
CDK (1)
PAFR (1)
S1P Receptor (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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