• TargetMol
    您的购物车当前为空
TargetMol | Compound Library

细胞凋亡化合物库现货

Apoptosis Compound Library

Rating icon 很棒
产品编号 L9000

细胞凋亡是一种发生在多细胞生物中的程序性细胞死亡。相对于细胞坏死,细胞凋亡是受基因调控的主动过程,细胞凋亡时会发生特征性的形态学变化,产生称为凋亡小体的细胞碎片被吞噬细胞吞噬。细胞凋亡受到促凋亡因子(Fas 受体和 caspases)和抑凋亡因子(Bcl-2蛋白和 IAP)的调控,异常凋亡过程牵涉到多种疾病中,细胞凋亡的抑制可导致癌症、自身免疫性疾病、炎性疾病和病毒感染。另一方面,过度的细胞凋亡可能导致神经退行性疾病、血液疾病和组织损伤。目前在细胞凋亡与癌症发生和自身免疫性疾病之间的关系有着很多研究,人们希望激发癌细胞的细胞凋亡,以达到治疗癌症的目的。“细胞凋亡在神经退化性疾病中所扮演的角色(如阿兹海默氏症、亨丁顿舞蹈症、帕金森病、肌肉萎缩性侧索硬化症),是目前热门的研究领域。” TargetMol 细胞凋亡化合物库精选 2394 种与凋亡相关的生物活性小分子化合物,适用于癌症和神经退行性疾病相关研究。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
资源下载
化合物库相关信息
Excel
SDF
联系我们获取更多批次信息

产品编号 L9000

细胞凋亡化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 2394种与凋亡相关的生物活性小分子化合物的特有集合,多用于研究肿瘤发生发展机制和抗癌药物筛选等。可用于高通量筛选和高内涵筛选;
  • 靶点含Bcl-2、Caspase、p53、TNF-α和survivin等;
  • 通过前期临床研究和临床实验,生物活性和安全性已经得到验证;
  • 其中一些活性化合物已得到FDA批准上市;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR和HPLC检测技术保证产品高纯度和高质量;
  • 所有化合物现货供应。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

使用TargetMol产品
发表顶级期刊文献

引用更多关于TargetMol产品的科学文献吧!

查看更多

Library Customization | TargetMol 化合物库定制

Compound Library | TargetMol
您可以通过点击按钮
定制您专属的化合物!
联系专属定制

Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
Endogenous Metabolite
EGFR
TNF
NF-κB
Antibacterial
Caspase
Ferroptosis
Bcl-2 Family
Reactive Oxygen Species
JAK
Akt
STAT
MDM-2/p53
CDK
p38 MAPK
PI3K
COX
ERK
Ras
DNA/RNA Synthesis
VEGFR
Parasite
p53
Antibiotic
Raf
IL Receptor
Antioxidant
Microtubule Associated
Antifungal
HDAC
Interleukin
FLT
JNK
Src
mTOR
RIP kinase
AMPK
c-RET
PARP
MEK
HIV Protease
PERK
Mitophagy
PDGFR
MAPK
FGFR
E1/E2/E3 Enzyme
c-Kit
Dehydrogenase
Nucleoside Antimetabolite/Analog
Tyrosine Kinases
Epigenetic Reader Domain
HSP
Nrf2
Aurora Kinase
Influenza Virus
Mdm2
PPAR
ROS
NO Synthase
Bcr-Abl
Cytochromes P450
Virus Protease
c-Met/HGFR
Topoisomerase
PKC
Mitochondrial Metabolism
Potassium Channel
Wnt/beta-catenin
GSK-3
PD-1/PD-L1
Phosphatase
Proteasome
Pim
MMP
IAP
Sirtuin
HER
Histone Methyltransferase
Calcium Channel
IκB/IKK
HSV
IGF-1R
Lipoxygenase
HIF/HIF Prolyl-Hydroxylase
FAK
SARS-CoV
PDE
Anti-infection
Estrogen Receptor/ERR
TGF-beta/Smad
Molecular Glues
Chk
DUB
Syk
ATPase
KRas
DNA-PK
RAAS
PKA
AChR
DNA Alkylator/Crosslinker
P-gp
Estrogen/progestogen Receptor
Beta Amyloid
S6 Kinase
PROTACs
Histone Demethylase
Cholinesterase (ChE)
Histone Acetyltransferase
TLR
Necroptosis
Gamma-secretase
Casein Kinase
Phospholipase
ALK
Prostaglandin Receptor
Drug Metabolite
HMG-CoA Reductase
Bcl-6
TRP/TRPV Channel
Adrenergic Receptor
Antiviral
PDK
5-HT Receptor
Trk receptor
c-Fms
Histamine Receptor
Ligand for E3 Ligase
HIF
Sodium Channel
OXPHOS
Pyroptosis
Retinoid Receptor
Tyrosinase
Dopamine Receptor
Serine Protease
S1P Receptor
ATM/ATR
TAM Receptor
GPCR
Rho
Reverse Transcriptase
GABA Receptor
Survivin
ASK
NADPH
CaMK
DNA Methyltransferase
NOD-like Receptor (NLR)
Monoamine Oxidase
PLK
HBV
Integrin
Reductase
DNA Alkylation
NOS
HCV Protease
Glutathione Peroxidase
PTEN
UGT
Kinesin
Telomerase
Immunology/Inflammation related
iGluR
GluR
Tie-2
c-Myc
MAO
Cysteine Protease
LPL Receptor
DAPK
Transferase
Angiotensin-converting Enzyme (ACE)
ROS Kinase
Opioid Receptor
MLK
MRP
Antifolate
Antifection
Fatty Acid Synthase
ADC Cytotoxin
Ligands for Target Protein for PROTAC
Cell Cycle Arrest
DPP-4
MNK
DNA
TOPK
CSF-1R
Glucosidase
IKZF
DYRK
Photosensitizer
PAK
PAI-1
GST
Proton pump
FXR
IRE1
GPX
Androgen Receptor
PGE Synthase
Cuproptosis
IFNAR
ROCK
transporter
SGK
MicroRNA
ROR
Amino Acids and Derivatives
Hexokinase
LTR
NR4A
p62
CRISPR/Cas9
Sigma receptor
DHFR
Cholecystokinin Receptor
Hedgehog/Smoothened
Beta-Secretase
FOXO
Adenosine Receptor
Liver X Receptor
BTK
NOD
Serine/threonin kinase
Leukotriene Receptor
Aryl Hydrocarbon Receptor
LDL
CXCR
Xanthine Oxidase
Free radical scavengers
FKBP
NADPH-oxidase
CRM1
PYK2
P2X Receptor
Indoleamine 2,3-Dioxygenase (IDO)
Wee1
YAP
BACE
IDO
SGLT
Lipid
FOXO3
Glucokinase
PAFR
NMDAR
GPCR19
PI4K
KLF
Carbonic Anhydrase
ATG
ABC Transporter
Hippo pathway
CFTR
FLAP
Smo
Endothelin Receptor
Acyltransferase
NAMPT
cAMP
AIM2
Aromatase
IRAK
Prolyl Endopeptidase (PREP)
KSP
STING
LRRK2
PAD
Aminopeptidase
p97
OCT
Hck
Glucocorticoid Receptor
Fas/FasL
Stearoyl-CoA Desaturase (SCD)
BMI-1
Apelin receptor
Dynamin
P2Y Receptor
Lipase
MTH1
Target Protein Ligand-Linker Conjugate
RSV
Protease
Hydrogenase
GDNF
NEDD8
VDA
VDAC
Monoamine Transporter
PROTAC Linker
FAAH
CCR
Transketolase
Hydroxylase
Imidazoline Receptor
Serotonin Transporter
LDLR
SIK
Myosin
Thioredoxin
Glutathione reductase
Neprilysin
Adenosine Deaminase
APC/C
Liposome
Y Box Binding Protein 1
Na+/Ca2+ Exchanger
gp120/CD4
GTPase
Progesterone Receptor
GNRH Receptor
ASCT
Ephrin Receptor
MELK
Melanocortin Receptor
Platelet aggregation
Lysosomal Autophagy
Chloride channel
RAR/RXR
MALT
Melatonin Receptor
Amylase
DNA gyrase
Guanylate cyclase
Cadherin
Norepinephrine
Cannabinoid Receptor
PKM
MIF
Glutaminase
Somatostatin
OX Receptor
Urea Transporter
Protease-activated Receptor
RANKL/RANK
Na-K-Cl cotransporter
ACK1
hCE
HuR
LPA Receptor
Thrombin
Vitamin
PGC-1α

Keywords