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血液病分子库

血液病分子库

产品编号 L8400 Hematonosis Compound Library
  库化合物信息   Excel SDF

血液病亦称为造血系统疾病,包括原发于造血系统疾病(如白血病原发于骨髓组织等)和主要累及造血系统疾病(如缺铁性贫血),例如白血病,血友病、再障、地中海贫血、骨髓增生异常综合症(MDS)、多发性骨髓瘤、淋巴瘤等。血液系统疾病多半是难治性疾病, 发病隐袭,病状隐匿。由于缺乏特效疗法,许多疾病曾被称为“不治之症”,近年来,随着医学研究的深入发展,血液病的治疗效果有了明显提高。现代医学对血液病的治疗多应用激素、化疗等方法,但副作用大,病人治愈率低、易复发。骨髓移植用于治疗白血病,治愈率有所提高,然而骨髓资源十分缺乏,即使移植成功,5年内复发率也高达70%。因此寻找新的治疗方法和治疗药物具有重要意义。

TargetMol 作为全球知名化合物库供应商,积极关注科研动态,为您提供大量造血系统疾病研究相关的优质产品,为您的新药筛选提供一站式服务平台。

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TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
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产品描述

  • 524种造血系统疾病相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 是研究造血系统功能及相关疾病的有效工具,例如白血病、血友病、β-地中海贫血等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

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包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
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化合物库组成

Apoptosis (156)
Autophagy (103)
PI3K (33)
DNA/RNA Synthesis (31)
Bcr-Abl (25)
Endogenous Metabolite (25)
FLT (24)
HDAC (24)
CDK (23)
Topoisomerase (21)
Histone Methyltransferase (18)
c-Kit (17)
Antibacterial (17)
ALK (16)
Dehydrogenase (16)
Src (16)
PDGFR (15)
mTOR (14)
JAK (14)
Nucleoside Antimetabolite/Analog (13)
VEGFR (12)
HIV Protease (11)
FGFR (10)
BCL (10)
TAM Receptor (10)
Antibiotic (10)
Epigenetic Reader Domain (10)
Microtubule Associated (9)
E1/E2/E3 Enzyme (9)
Proteasome (9)
PKC (9)
PLK (8)
Aurora Kinase (8)
AMPK (8)
Tyrosine Kinases (8)
Mitophagy (8)
Influenza Virus (8)
DNA Alkylator/Crosslinker (8)
c-Met/HGFR (8)
NF-κB (7)
BTK (7)
GSK-3 (7)
c-RET (7)
Trk receptor (7)
Reactive Oxygen Species (6)
STAT (6)
Antifolate (6)
Ligand for E3 Ligase (6)
COX (6)
HSP (6)
Caspase (5)
Akt (5)
c-Fms (5)
ROS (5)
TNF (5)
Retinoid Receptor (5)
Isocitrate Dehydrogenase (IDH) (5)
Antifungal (5)
Syk (5)
DNA Alkylation (4)
Histone Demethylase (4)
Ferroptosis (4)
ROS Kinase (4)
Virus Protease (4)
ERK (4)
Chk (4)
AChR (4)
MEK (4)
Raf (4)
IGF-1R (4)
DNA-PK (4)
Mdm2 (4)
Parasite (4)
Ras (4)
p53 (3)
Nrf2 (3)
IRAK (3)
Potassium Channel (3)
Rho (3)
Gamma-secretase (3)
Aminopeptidase (3)
CSF-1R (3)
Pim (3)
Transferase (3)
Ligands for Target Protein for PROTAC (3)
HIF/HIF Prolyl-Hydroxylase (3)
Smo (3)
IL Receptor (3)
Wnt/beta-catenin (3)
PROTACs (3)
Molecular Glues (3)
HBV (3)
Hedgehog/Smoothened (3)
Sirtuin (3)
DUB (3)
S6 Kinase (3)
DNA Methyltransferase (3)
IAP (3)
Adenosine Receptor (3)
Mitochondrial Metabolism (3)
P-gp (3)
ATM/ATR (3)
TOPK (2)
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transporter (2)
EGFR (2)
FAK (2)
BMI-1 (2)
Adenosine deaminase (2)
NAMPT (2)
MAPK (2)
Kinesin (2)
Sodium Channel (2)
HSV (2)
CaMK (2)
Phospholipase (2)
GABA Receptor (2)
Antiviral (2)
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Liver X Receptor (2)
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p38 MAPK (2)
IκB/IKK (2)
Phosphatase (2)
NEDD8 (2)
PKA (2)
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Histone Acetyltransferase (2)
IRE1 (2)
TGF-beta/Smad (1)
Methionine Adenosyltransferase (MAT) (1)
MNK (1)
GTPase (1)
PAK (1)
NO Synthase (1)
MLK (1)
JNK (1)
DNA (1)
ATPase (1)
ACK (1)
Hck (1)
Adrenergic Receptor (1)
Immunology/Inflammation related (1)
OXPHOS (1)
Serine/threonin kinase (1)
PD-1/PD-L1 (1)
HCV Protease (1)
Integrin (1)
Dopamine Receptor (1)
Histamine Receptor (1)
Glutaminase (1)
PPAR (1)
p97 (1)
Fatty Acid Synthase (1)
Chloride channel (1)
LTR (1)
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Amino Acids and Derivatives (1)
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Cysteine Protease (1)
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Haspin Kinase (1)
CXCR (1)
HIF (1)
BCRP (1)
Reverse Transcriptase (1)
CRM1 (1)
GluR (1)
Estrogen/progestogen Receptor (1)
TLR (1)
DNA gyrase (1)
NMDAR (1)
P450 (1)
Anti-infection (1)
Monocarboxylate transporter (1)
GPR (1)
MALT (1)
Antifection (1)
SGLT (1)
Tie-2 (1)
Lipoxygenase (1)
DYRK (1)
S1P Receptor (1)
VDAC (1)
Wee1 (1)
Aromatase (1)
Serine Protease (1)
Monoamine Transporter (1)
Drug Metabolite (1)
YAP (1)
PAD (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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