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TargetMol | Compound Library

抗肺癌化合物库现货

Anti-Lung Cancer Compound Library

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产品编号 L2190

根据《2018年全球癌症统计数据》报告,仅2018年,全球新增癌症病例1810万,死亡960万,其中亚洲占近70%,肺癌的发病率及死亡率居高不下(11.6%及18.4%)。肺癌的发病率和死亡率增长很快,对人群健康和生命威胁很大的恶性肿瘤之一。 由于缺乏有效的治疗手段,目前肺癌的治疗目标是延长生存期,尽可能长时间地实现和维持良好的生活质量。肺癌的治疗手段包括手术、放疗、化疗、免疫治疗或联合疗法。近年来,靶向治疗和肿瘤免疫疗法成为肺癌治疗的重要发展方向,并且取得了较好的治疗效果。但是靶向药物治疗易出现耐药性的问题,随着靶向药物的不断发展、全基因组测序的不断推进,开发新一代克服耐药的靶向治疗药物是肺癌药物开发的重中之重。 TargetMol 抗肺癌化合物库收集了2240 种与肺癌相关的化合物,包括已经报道有肺癌治疗作用的化合物,以及靶向肺癌相关靶点的化合物,是抗肺癌药物研发的良好工具。此外,我们还提供已知活性库、上市药物库、天然产物库以及一系列抗癌相关化合物库,可以用于抗癌药物的研发,如果您感兴趣,欢迎与我们联系~

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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产品编号 L2190

抗肺癌化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 2240种与肺癌相关的化合物,可以用于抗肺癌药物研发和药理研究;
  • 靶点包含EGFR, PI3K, FGFR, HER2, ALK, c-Met等;
  • 部分化合物已上市或进入临床期;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Apoptosis
Autophagy
NF-κB
PI3K
EGFR
VEGFR
Akt
mTOR
JAK
STAT
AMPK
PDGFR
FLT
FGFR
GSK-3
c-Met/HGFR
Wnt/beta-catenin
Endogenous Metabolite
Antibacterial
CDK
ALK
Ras
c-Kit
ERK
Src
ROS
TGF-beta/Smad
p53
Parasite
COX
Kras
DNA/RNA Synthesis
p38 MAPK
TNF
IGF-1R
MDM-2/p53
Tyrosine Kinases
Potassium Channel
DNA-PK
Bcr-Abl
S6 Kinase
Caspase
Raf
ATM/ATR
Antibiotic
Mitophagy
Reactive Oxygen Species
HIV Protease
c-RET
HER
Cytochromes P450
Bcl-2 Family
JNK
Interleukin
Pim
Aurora Kinase
Dehydrogenase
PARP
PKC
IL Receptor
MEK
Microtubule Associated
NO Synthase
HDAC
Ferroptosis
Topoisomerase
PDK
TAM Receptor
DNA Alkylator/Crosslinker
PPAR
FAK
Calcium Channel
MMP
Influenza Virus
c-Fms
Mdm2
MAPK
Trk receptor
IκB/IKK
PI4K
Phosphatase
PKA
DNA Alkylation
Nrf2
Casein Kinase
Lipoxygenase
SARS-CoV
Beta Amyloid
ROS Kinase
Antifungal
E1/E2/E3 Enzyme
PDE
HSV
HSP
TLR
5-HT Receptor
AChR
Drug Metabolite
Estrogen/progestogen Receptor
Antioxidant
Virus Protease
Chk
Epigenetic Reader Domain
Syk
HIF/HIF Prolyl-Hydroxylase
Histamine Receptor
ROCK
Adrenergic Receptor
Sodium Channel
NOS
PERK
Estrogen Receptor/ERR
Nucleoside Antimetabolite/Analog
PTEN
P-gp
Histone Methyltransferase
HCV Protease
Adenosine Receptor
CSF-1R
SIK
GABA Receptor
PLK
Tyrosinase
ADC Cytotoxin
Integrin
Reductase
DYRK
Tie-2
Glucocorticoid Receptor
Gamma-secretase
Mitochondrial Metabolism
Glucosidase
DUB
Prostaglandin Receptor
Sirtuin
Histone Acetyltransferase
ATPase
DHFR
Dopamine Receptor
Histone Demethylase
RAAS
Antifolate
IAP
RIP kinase
Antifection
Hedgehog/Smoothened
CaMK
MELK
NOD-like Receptor (NLR)
PD-1/PD-L1
BTK
PROTACs
MRP
Molecular Glues
Cholinesterase (ChE)
GluR
glycosidase
Antiviral
transporter
Retinoid Receptor
HIF
SGK
DNA Methyltransferase
NOD
MLK
Proteasome
Transferase
IFNAR
c-Myc
Rho
Serine Protease
PYK2
Aryl Hydrocarbon Receptor
iGluR
LDL
Opioid Receptor
CCR
Angiotensin-converting Enzyme (ACE)
DNA
PGE Synthase
Survivin
Porcupine
Ephrin Receptor
FKBP
Reverse Transcriptase
Cannabinoid Receptor
Discoidin Domain Receptor (DDR)
Anti-infection
Chloride channel
BACE
NADPH
Glutathione Peroxidase
Cholecystokinin Receptor
Leukotriene Receptor
TRP/TRPV Channel
NMDAR
ACK1
Lipid
STING
Hippo pathway
GST
Aromatase
IRAK
HMG-CoA Reductase
Kinesin
Monoamine Oxidase
GPCR
Proton pump
Carbonic Anhydrase
ROR
MyD88
Ligands for Target Protein for PROTAC
YAP
LTR
GTPase
Progesterone Receptor
HBV
Photosensitizer
Serotonin Transporter
Serine/threonin kinase
FXR
Glucokinase
RANKL/RANK
IDO
Immunology/Inflammation related
Prolyl Endopeptidase (PREP)
Myosin
IRE1
ABC Transporter
Monoamine Transporter
Smo
Fatty Acid Synthase
Bombesin Receptor
CXCR
cAMP
Indoleamine 2,3-Dioxygenase (IDO)
Androgen Receptor
ATP Citrate Lyase
BCRP
OXPHOS
Beta-Secretase
MNK
Acyltransferase
Pyroptosis
Ligand for E3 Ligase
ribosome
Phospholipase
GHSR
DAPK
S1P Receptor
IKZF
Melanin-concentrating Hormone Receptor (MCHR)
Adenylyl Cyclase
MicroRNA
NPC1L1
RAR/RXR
CD38
MALT
NEDD8
CRM1
Amino Acids and Derivatives
Y Box Binding Protein 1
P2Y Receptor
Na+/Ca2+ Exchanger
Lipase
gp120/CD4
TOPK
VDA
Melatonin Receptor
OCT
Galectin
Hck
ATG
Cell Cycle Arrest
Liver X Receptor
Neurotensin Receptor
LIM Kinase
Glutaminase
NR4A
MAO
UGT
PAFR
MTH1
FABP
Glucagon Receptor
P2X Receptor
Na-K-Cl cotransporter
Hexokinase
Guanylate cyclase
Neuropeptide Y Receptor
Thioredoxin
PAK
FAAH
Stearoyl-CoA Desaturase (SCD)
Xanthine Oxidase
KSP
Cadherin
Thrombopoietin Receptor
Wee1
LRRK2
Free radical scavengers
Aminopeptidase
AIM2
CD74
Decarboxylase
GluCls
hCE
PAI-1
RSV
Methionine Adenosyltransferase (MAT)
p62
CRISPR/Cas9
Adenosine Deaminase
Cuproptosis
Complement System
Gap Junction Protein
Neurokinin receptor
Platelet aggregation
NADPH-oxidase
Sigma receptor
CFTR
PKM
IGF-2R

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