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TargetMol | Compound Library

抗肺癌化合物库现货

Anti-Lung Cancer Compound Library
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货号 L2190

根据《2018年全球癌症统计数据》报告,仅2018年,全球新增癌症病例1810万,死亡960万,其中亚洲占近70%,肺癌的发病率及死亡率居高不下(11.6%及18.4%)。肺癌的发病率和死亡率增长很快,对人群健康和生命威胁很大的恶性肿瘤之一。 由于缺乏有效的治疗手段,目前肺癌的治疗目标是延长生存期,尽可能长时间地实现和维持良好的生活质量。肺癌的治疗手段包括手术、放疗、化疗、免疫治疗或联合疗法。近年来,靶向治疗和肿瘤免疫疗法成为肺癌治疗的重要发展方向,并且取得了较好的治疗效果。但是靶向药物治疗易出现耐药性的问题,随着靶向药物的不断发展、全基因组测序的不断推进,开发新一代克服耐药的靶向治疗药物是肺癌药物开发的重中之重。 TargetMol 抗肺癌化合物库收集了2240 种与肺癌相关的化合物,包括已经报道有肺癌治疗作用的化合物,以及靶向肺癌相关靶点的化合物,是抗肺癌药物研发的良好工具。此外,我们还提供已知活性库、上市药物库、天然产物库以及一系列抗癌相关化合物库,可以用于抗癌药物的研发,如果您感兴趣,欢迎与我们联系~

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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货号 L2190

抗肺癌化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 2240种与肺癌相关的化合物,可以用于抗肺癌药物研发和药理研究;
  • 靶点包含EGFR, PI3K, FGFR, HER2, ALK, c-Met等;
  • 部分化合物已上市或进入临床期;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
NF-κB
PI3K
EGFR
VEGFR
Akt
mTOR
JAK
STAT
PDGFR
AMPK
FLT
FGFR
GSK-3
c-Met/HGFR
Wnt/beta-catenin
Endogenous Metabolite
Antibacterial
CDK
ALK
Ras
c-Kit
ERK
Src
ROS
TGF-beta/Smad
p53
Kras
COX
Parasite
p38 MAPK
DNA/RNA Synthesis
TNF
IGF-1R
MDM-2/p53
Tyrosine Kinases
Potassium Channel
Bcr-Abl
DNA-PK
S6 Kinase
Caspase
Raf
Reactive Oxygen Species
ATM/ATR
Antibiotic
Mitophagy
HIV Protease
c-RET
HER
Cytochromes P450
Interleukin
Bcl-2 Family
JNK
Pim
Aurora Kinase
Microtubule Associated
Dehydrogenase
PARP
PKC
IL Receptor
MEK
NO Synthase
HDAC
Ferroptosis
Topoisomerase
PDK
TAM Receptor
DNA Alkylator/Crosslinker
PPAR
FAK
Calcium Channel
MMP
Influenza Virus
c-Fms
Mdm2
MAPK
Trk receptor
IκB/IKK
PI4K
Nrf2
Phosphatase
PKA
Casein Kinase
DNA Alkylation
Lipoxygenase
SARS-CoV
Beta Amyloid
ROS Kinase
PDE
E1/E2/E3 Enzyme
HSV
HSP
TLR
5-HT Receptor
AChR
Antifungal
Drug Metabolite
Estrogen/progestogen Receptor
Virus Protease
Chk
Epigenetic Reader Domain
Syk
HIF/HIF Prolyl-Hydroxylase
NOS
Histamine Receptor
Antioxidant
ROCK
Adrenergic Receptor
Sodium Channel
HCV Protease
Estrogen Receptor/ERR
Nucleoside Antimetabolite/Analog
P-gp
PTEN
Histone Methyltransferase
Adenosine Receptor
CSF-1R
SIK
GABA Receptor
PLK
Tyrosinase
ADC Cytotoxin
Reductase
DYRK
Tie-2
Integrin
PERK
IAP
Glucocorticoid Receptor
Mitochondrial Metabolism
Gamma-secretase
Glucosidase
DUB
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Histone Acetyltransferase
DHFR
RAAS
Dopamine Receptor
Histone Demethylase
Antifolate
RIP kinase
BTK
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MELK
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PROTACs
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GluR
glycosidase
Molecular Glues
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Survivin
Antiviral
SGK
MLK
Retinoid Receptor
HIF
DNA Methyltransferase
NOD
c-Myc
Proteasome
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IFNAR
Serine Protease
PYK2
iGluR
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Aryl Hydrocarbon Receptor
Opioid Receptor
Angiotensin-converting Enzyme (ACE)
DNA
PGE Synthase
transporter
CCR
Porcupine
Ephrin Receptor
FKBP
Reverse Transcriptase
Cannabinoid Receptor
Discoidin Domain Receptor (DDR)
Anti-infection
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BACE
NADPH
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LDL
NMDAR
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Leukotriene Receptor
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STING
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IRAK
HMG-CoA Reductase
Hippo pathway
Aromatase
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Monoamine Oxidase
GPCR
Carbonic Anhydrase
ROR
GTPase
Progesterone Receptor
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MyD88
Ligands for Target Protein for PROTAC
YAP
LTR
Photosensitizer
Serine/threonin kinase
Glucokinase
RANKL/RANK
IDO
Prolyl Endopeptidase (PREP)
IRE1
HBV
Hck
Serotonin Transporter
FXR
Immunology/Inflammation related
ABC Transporter
Monoamine Transporter
Smo
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CXCR
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ATP Citrate Lyase
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OXPHOS
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Ligands for E3 Ligase
Bombesin Receptor
Androgen Receptor
Indoleamine 2,3-Dioxygenase (IDO)
MNK
Pyroptosis
GST
ribosome
DAPK
Phospholipase
GHSR
S1P Receptor
IKZF
CD38
MALT
CRM1
P2Y Receptor
gp120/CD4
TOPK
Melatonin Receptor
Melanin-concentrating Hormone Receptor (MCHR)
MicroRNA
NPC1L1
RAR/RXR
NEDD8
Amino Acids and Derivatives
Y Box Binding Protein 1
Na+/Ca2+ Exchanger
Lipase
VDA
OCT
Galectin
MAO
Myosin
UGT
ATG
Cell Cycle Arrest
Liver X Receptor
LIM Kinase
Neurotensin Receptor
Glutaminase
NR4A
Adenylate cyclase
PAFR
MTH1
FABP
Glucagon Receptor
P2X Receptor
Na-K-Cl cotransporter
Hexokinase
Guanylate cyclase
Neuropeptide Y Receptor
Stearoyl-CoA Desaturase (SCD)
Xanthine Oxidase
KSP
Thrombopoietin Receptor
LRRK2
Free radical scavengers
AIM2
CD74
Decarboxylase
Thioredoxin
PAK
FAAH
Cadherin
Wee1
Aminopeptidase
GluCls
Methionine Adenosyltransferase (MAT)
p62
Cuproptosis
CFTR
PKM
hCE
PAI-1
RSV
Adenosine Deaminase
Complement System
Gap Junction Protein
Neurokinin receptor
Platelet aggregation
NADPH-oxidase
Sigma receptor
IGF-2R

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