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TargetMol | Compound Library

抗肺癌化合物库现货

Anti-Lung Cancer Compound Library

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产品编号 L2190

根据《2018年全球癌症统计数据》报告,仅2018年,全球新增癌症病例1810万,死亡960万,其中亚洲占近70%,肺癌的发病率及死亡率居高不下(11.6%及18.4%)。肺癌的发病率和死亡率增长很快,对人群健康和生命威胁很大的恶性肿瘤之一。 由于缺乏有效的治疗手段,目前肺癌的治疗目标是延长生存期,尽可能长时间地实现和维持良好的生活质量。肺癌的治疗手段包括手术、放疗、化疗、免疫治疗或联合疗法。近年来,靶向治疗和肿瘤免疫疗法成为肺癌治疗的重要发展方向,并且取得了较好的治疗效果。但是靶向药物治疗易出现耐药性的问题,随着靶向药物的不断发展、全基因组测序的不断推进,开发新一代克服耐药的靶向治疗药物是肺癌药物开发的重中之重。 TargetMol 抗肺癌化合物库收集了2240 种与肺癌相关的化合物,包括已经报道有肺癌治疗作用的化合物,以及靶向肺癌相关靶点的化合物,是抗肺癌药物研发的良好工具。此外,我们还提供已知活性库、上市药物库、天然产物库以及一系列抗癌相关化合物库,可以用于抗癌药物的研发,如果您感兴趣,欢迎与我们联系~

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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产品编号 L2190

抗肺癌化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 2240种与肺癌相关的化合物,可以用于抗肺癌药物研发和药理研究;
  • 靶点包含EGFR, PI3K, FGFR, HER2, ALK, c-Met等;
  • 部分化合物已上市或进入临床期;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Apoptosis
Autophagy
NF-κB
PI3K
EGFR
VEGFR
mTOR
Akt
JAK
STAT
PDGFR
AMPK
FLT
FGFR
GSK-3
c-Met/HGFR
Wnt/beta-catenin
Endogenous Metabolite
Antibacterial
CDK
ALK
Ras
c-Kit
ERK
Src
ROS
TGF-beta/Smad
p53
Parasite
COX
Kras
DNA/RNA Synthesis
p38 MAPK
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IGF-1R
MDM-2/p53
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S6 Kinase
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ATM/ATR
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c-RET
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Pim
JNK
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PARP
IL Receptor
Dehydrogenase
PKC
MEK
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NO Synthase
HDAC
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PDK
TAM Receptor
DNA Alkylator/Crosslinker
PPAR
FAK
Calcium Channel
MMP
c-Fms
Influenza Virus
Mdm2
MAPK
Trk receptor
PI4K
IκB/IKK
Casein Kinase
PKA
DNA Alkylation
Phosphatase
Nrf2
Lipoxygenase
ROS Kinase
Beta Amyloid
SARS-CoV
Antifungal
5-HT Receptor
E1/E2/E3 Enzyme
HSV
HSP
AChR
PDE
TLR
Drug Metabolite
Chk
Syk
HIF/HIF Prolyl-Hydroxylase
Antioxidant
Virus Protease
Epigenetic Reader Domain
Estrogen/progestogen Receptor
Sodium Channel
ROCK
Adrenergic Receptor
Histamine Receptor
PERK
Nucleoside Antimetabolite/Analog
Estrogen Receptor/ERR
NOS
PTEN
P-gp
Adenosine Receptor
GABA Receptor
PLK
CSF-1R
SIK
Histone Methyltransferase
HCV Protease
Tyrosinase
ADC Cytotoxin
DYRK
Histone Acetyltransferase
Gamma-secretase
Mitochondrial Metabolism
DUB
Glucocorticoid Receptor
Sirtuin
Integrin
Reductase
Tie-2
Glucosidase
Prostaglandin Receptor
MELK
PD-1/PD-L1
CaMK
NOD-like Receptor (NLR)
ATPase
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PROTACs
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glycosidase
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Transferase
IFNAR
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CCR
DNA
Porcupine
Proteasome
PYK2
PGE Synthase
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Aryl Hydrocarbon Receptor
LDL
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FKBP
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GST
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IRAK
NMDAR
BACE
NADPH
TRP/TRPV Channel
ACK1
Lipid
Monoamine Oxidase
Hippo pathway
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HMG-CoA Reductase
Kinesin
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Glutathione Peroxidase
Leukotriene Receptor
STING
GPCR
GTPase
Progesterone Receptor
Photosensitizer
cAMP
GHSR
ROR
Ligands for Target Protein for PROTAC
Glucokinase
Immunology/Inflammation related
MNK
S1P Receptor
YAP
Hck
RANKL/RANK
IDO
Bombesin Receptor
Carbonic Anhydrase
LTR
HBV
ABC Transporter
Monoamine Transporter
ATP Citrate Lyase
ribosome
Serotonin Transporter
Myosin
Smo
Beta-Secretase
Acyltransferase
Ligand for E3 Ligase
Phospholipase
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Indoleamine 2,3-Dioxygenase (IDO)
Androgen Receptor
BCRP
DAPK
Proton pump
MyD88
Serine/threonin kinase
FXR
Prolyl Endopeptidase (PREP)
IRE1
CXCR
OXPHOS
Pyroptosis
IKZF
Y Box Binding Protein 1
Na+/Ca2+ Exchanger
gp120/CD4
Liver X Receptor
MAO
PAK
AIM2
PAI-1
Gap Junction Protein
Platelet aggregation
MicroRNA
Amino Acids and Derivatives
P2Y Receptor
Lipase
Galectin
Cell Cycle Arrest
LIM Kinase
PAFR
MTH1
Glucagon Receptor
Hexokinase
RSV
Complement System
OCT
Na-K-Cl cotransporter
Neuropeptide Y Receptor
Stearoyl-CoA Desaturase (SCD)
hCE
CD38
NEDD8
VDA
ATG
NR4A
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CD74
p62
CRISPR/Cas9
Sigma receptor
CFTR
Melanin-concentrating Hormone Receptor (MCHR)
NPC1L1
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Thioredoxin
Decarboxylase
Adenosine Deaminase
Neurokinin receptor
Adenylyl Cyclase
CRM1
Neurotensin Receptor
Glutaminase
UGT
P2X Receptor
Thrombopoietin Receptor
Wee1
Aminopeptidase
Methionine Adenosyltransferase (MAT)
Cuproptosis
RAR/RXR
MALT
Melatonin Receptor
FABP
Guanylate cyclase
Xanthine Oxidase
KSP
Cadherin
LRRK2
Free radical scavengers
GluCls
NADPH-oxidase
PKM
IGF-2R

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