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Diflubenzuron

Name: Diflubenzuron
Brand: TargetMol
SKU: T7088
Price: 182 CNY
Availability: InStock
Rating: 5 (10 reviews)

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很棒

纯度: 99.96%

货号 T7088Cas号 35367-38-5

别名 氟脲杀, Larvakil, Dimilin, Difubenzuron, Difluron

Diflubenzuron (Larvakil) 是杀虫剂 Dimilin 的有效成分，具有杀幼虫和杀卵作用。

Diflubenzuron

一键复制产品信息

很棒

纯度: 99.96%

货号 T7088 别名 氟脲杀, Larvakil, Dimilin, Difubenzuron, DifluronCas号 35367-38-5

Diflubenzuron (Larvakil) 是杀虫剂 Dimilin 的有效成分，具有杀幼虫和杀卵作用。

规格	价格	库存
25 mg	¥ 208	现货
50 mg	¥ 293	现货
100 mg	¥ 397	现货
500 mg	¥ 938	现货
1 g	¥ 1,370	现货
1 mL x 10 mM (in DMSO)	¥ 182	现货

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纯度: 99.96%

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COA LCMS HNMR 产品操作手册

产品介绍

Diflubenzuron AI Summary

Diflubenzuron demonstrates a wide range of bioactivities, including significant antitumor, antiviral, insecticidal, and antifeedant properties. In vivo, it shows antitumor activity against 6C3HED lymphosarcoma with inhibition percentages of 6.0% and 33.0% at doses of 300 mg/kg and 1600 mg/kg respectively for 10 days. Additionally, it has an IC50 value of >20.0 ug/mL for inhibiting the growth of CCRF-CEM cells over 72 hours. The compound acts as an agonist for retinoid X receptor alpha, peroxisome proliferator-activated receptor gamma, Aryl hydrocarbon Receptor (AhR), and antioxidant response element (ARE) with Nrf2-dependent transcriptional activity. It also inhibits binding or entry into cells for Lassa Virus and Marburg Virus and exhibits antiviral activity against Foot and Mouth Disease Virus. In terms of insecticidal capabilities, Diflubenzuron exhibits potent activities against a variety of pests. It shows 100% mortality rates in Culex pipiens pallens mosquito larvae at 0.01 mg/L after 8 days and significant mortality in Mythimna separata (Oriental armyworm) larvae, with 100% mortality observed at 0.5 mg/L and 1 mg/L after 4 days. It is also effective against Chilo suppressalis larvae, inhibiting N-acetyl-[1-14C]glucosamine incorporation with an EC50 of 20.0 nM and inhibiting chitin synthesis with IC50 values of 19.05 nM and 20.42 nM. Moreover, Diflubenzuron effectively controls insect populations in agricultural settings, causing over 90% egg mortality in Spodoptera litura at 1 to 4 ppm and significant mortality in Plutella xylostella with an LC50 of 19.9 ug/mL in susceptible strains. However, it demonstrates reduced efficacy against fufenozide-resistant strains with a Resistance ratio of 17.2. Its toxicity is evident in Daphnia magna with an EC90 of 0.5 ppb. In summary, Diflubenzuron is highly effective as an antitumor agent, antiviral compound, and potent insecticide with varied applications across different pest species and settings..

Note: Summary generated by AI. Data source: ChEMBL

生物活性

产品描述	Diflubenzuron (Larvakil) is a benzoyl-urea insecticide, found to be a potent inhibitor of melanosome synthesis in mouse melanoma cells. Diflubenzuron has also been shown to inhibit TCDD-induced CYP1A1 expression in HepG2 cells.
别名	氟脲杀, Larvakil, Dimilin, Difubenzuron, Difluron

化学信息

分子量	310.68
分子式	C₁₄H₉ClF₂N₂O₂
CAS No.	35367-38-5
Smiles	Fc1cccc(F)c1C(=O)NC(=O)Nc1ccc(Cl)cc1
密度	1.4301 g/cm3 (Estimated)

储存&溶解度

存储

In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

溶解度信息

H2O: Insoluble

DMSO: 50 mg/mL (160.94 mM), Sonication is recommended.

溶液配制表

DMSO

	1mg	5mg	10mg	50mg
1 mM	3.2187 mL	16.0937 mL	32.1875 mL	160.9373 mL
5 mM	0.6437 mL	3.2187 mL	6.4375 mL	32.1875 mL
10 mM	0.3219 mL	1.6094 mL	3.2187 mL	16.0937 mL
20 mM	0.1609 mL	0.8047 mL	1.6094 mL	8.0469 mL
50 mM	0.0644 mL	0.3219 mL	0.6437 mL	3.2187 mL
100 mM	0.0322 mL	0.1609 mL	0.3219 mL	1.6094 mL

计算器

摩尔浓度计算器
稀释计算器
配液计算器
分子量计算器

体内实验配液计算器

请在以下方框中输入您的动物实验信息后点击计算，可以得到母液配置方法和体内配方的制备方法：

比如您的给药剂量是10 mg/kg，每只动物体重20 g，给药体积100 μL，一共给药动物10只，您使用的配方为 10% DMSO + 40% PEG300 + 5% Tween 80 + 45% Saline / PBS / ddH₂O，那么您的工作液浓度为2 mg/mL。

母液配置方法：2 mg 药物溶于 100 μL DMSO （母液浓度为 20 mg/mL ）, 如您需要配置的浓度超过该产品的溶解度，请先与我们联系。

体内配方的制备方法： 取 100 μL DMSO 母液，添加 400 μL PEG300 混匀澄清，再加 50 μL Tween 80, 混匀澄清, 再加 450 μL Saline / PBS / ddH₂O 混匀澄清

以上为“体内实验配液计算器”的使用方法举例，并不是具体某个化合物的推荐配制方式，请根据您的实验动物和给药方式选择适当的溶解方案。

方案所需的各类助溶剂如： DMSO， PEG300， PEG400， Tween 80， SBE-β-CD，玉米油等，均可在TargetMol网站点击购买。

剂量转换

对于不同动物的给药剂量换算，您也可以参考更多

关键词

synthesis ovicidal larvicida insecticide Inhibitor inhibit Diflubenzuron CYP1A1 chitin

Diflubenzuron

Diflubenzuron

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