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TargetMol | Compound Library

铁死亡化合物库现货

Ferroptosis Compound Library
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货号 L8700

铁死亡(ferroptosis)是近年来发现的一种由铁依赖的氧化损伤引起的细胞死亡模式,与凋亡、坏死、自噬不同,铁死亡的特征主要是细胞体积缩小和线粒体膜密度增加,没有典型的细胞凋亡和坏死表现。ferroptosis 与神经系统疾病、肿瘤(特别是乳腺癌、弥漫性大 B 细胞淋巴瘤)、缺血再灌注损伤、肾损伤、动脉粥样硬化、糖尿病、心脏病等疾病有关,进一步深入研究铁死亡的作用机理,研究其在不同疾病类型中的作用,对寻找相关疾病的治疗靶点、靶向药物的研发具有重要意义。

TargetMol 铁死亡化合物库,收集了 950 种与铁死亡通路相关的化合物,靶点包括 GPX4、ROS、p53、Nrf2等,另外还包含了铁螯合剂、抗氧化剂等多种类型小分子,助力您铁死亡通路相关的靶点鉴定和药物研发。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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货号 L8700

铁死亡化合物库

规格

  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 950种与铁死亡通路相关的化合物,可用于高通量和高内涵筛选;
  • 靶点含GPX4,ROS,p53,Nrf2等;
  • 部分化合物已被FDA批准上市;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

ROS
Apoptosis
Reactive Oxygen Species
Autophagy
Ferroptosis
Endogenous Metabolite
Nrf2
PPAR
NF-κB
Lipoxygenase
Antibacterial
Ras
p38 MAPK
p53
COX
MDM-2/p53
Antioxidant
Akt
Antifungal
Dehydrogenase
DNA/RNA Synthesis
Caspase
HMG-CoA Reductase
Parasite
FXR
Cytochromes P450
ERK
Interleukin
JNK
TNF
Bcl-2 Family
Antibiotic
Influenza Virus
HIV Protease
Raf
Glutathione Peroxidase
NADPH
PI3K
NO Synthase
Mdm2
HIF/HIF Prolyl-Hydroxylase
AMPK
PARP
Mitochondrial Metabolism
MMP
Mitophagy
Calcium Channel
TLR
CDK
STAT
NOD-like Receptor (NLR)
VEGFR
Potassium Channel
Virus Protease
Wnt/beta-catenin
TRP/TRPV Channel
Topoisomerase
NADPH-oxidase
Rho
SARS-CoV
5-HT Receptor
GPX
Kras
Beta Amyloid
Phosphatase
P-gp
IL Receptor
E1/E2/E3 Enzyme
Cholinesterase (ChE)
mTOR
Proteasome
TGF-beta/Smad
Estrogen/progestogen Receptor
Microtubule Associated
GSK-3
PKC
Pyroptosis
Tyrosinase
EGFR
GABA Receptor
HIF
JAK
HSP
AChR
Anti-infection
Monoamine Oxidase
Leukotriene Receptor
Opioid Receptor
Prostaglandin Receptor
MAO
Immunology/Inflammation related
MAPK
GPCR19
ATPase
Src
HBV
HSV
IGF-1R
Sirtuin
Reductase
Estrogen Receptor/ERR
IκB/IKK
HCV Protease
Xanthine Oxidase
Photosensitizer
NOD
Dopamine Receptor
Drug Metabolite
DPP-4
Angiotensin-converting Enzyme (ACE)
DUB
PERK
IAP
iGluR
Histamine Receptor
Adrenergic Receptor
IDO
Lipid
Antiviral
FLT
NOS
MyD88
Aryl Hydrocarbon Receptor
PDE
LDL
OXPHOS
Cannabinoid Receptor
Histone Acetyltransferase
Reverse Transcriptase
Aromatase
Sodium Channel
ROS Kinase
UGT
Antifection
Androgen Receptor
Indoleamine 2,3-Dioxygenase (IDO)
ROR
Amino Acids and Derivatives
Gamma-secretase
LTR
GluR
HDAC
Integrin
RAAS
PKA
Glucosidase
Epigenetic Reader Domain
Transferase
BACE
Necroptosis
CaMK
MEK
c-Kit
DNA Methyltransferase
AhR
DNA Alkylator/Crosslinker
Cysteine Protease
Free radical scavengers
Retinoid Receptor
PKM
Ferroportin
GTPase
c-Myc
Liver X Receptor
PAI-1
GST
Adenylate cyclase
Survivin
FGFR
FAK
Cell Cycle Arrest
Glucokinase
Syk
Carbonic Anhydrase
ABC Transporter
PDGFR
Hedgehog/Smoothened
Phospholipase
FOXO3
PGK1
YAP
IFNAR
ROCK
Glucocorticoid Receptor
Phosphorylase
SGLT
transporter
S6 Kinase
Thrombin
Chloride channel
Proton pump
Monocarboxylate transporter
RAR/RXR
Melatonin Receptor
Serine/threonin kinase
Prolyl Endopeptidase (PREP)
Bradykinin Receptor
PTEN
Epoxide Hydrolase
STING
LRRK2
Acetyl-CoA Carboxylase
MLK
GPCR
CAT
c-Met/HGFR
Adenosine Receptor
gp120/CD4
PAK
cAMP
AIM2
Gap Junction Protein
Platelet aggregation
IRAK
Lysosomal Autophagy
PD-1/PD-L1
RIP kinase
Bcr-Abl
Fatty Acid Synthase
Somatostatin
Aurora Kinase
PGE Synthase
Urea Transporter
ASK
Aquaporin
Cuproptosis
DAPK
Dynamin
Serine Protease
NMDAR
Trk receptor
RSV
c-Fms
Protease
PLK
Complement System
PROTACs
Hydrogenase
CD38
NR4A
glycosidase
DNA
Casein Kinase
p62
Hydroxylase
Sigma receptor
CFTR
HER
NPC1L1
DNA Alkylation
Beta-Secretase
Glutathione reductase
Acyltransferase
ATM/ATR
FOXO

Keywords