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别名 StemRegenin 1 盐酸盐, StemRegenin 1 (hydrochloride) (1227633-49-9 free base)
StemRegenin 1 Hydrochloride is an aryl hydrocarbon receptor (AhR) antagonist (IC₅₀ = 127 nM) that inhibits RANKL-induced osteoclast generation and differentiation while promoting the expansion of multipotent haematopoietic progenitor cells derived from human embryonic stem cells (hESCs).

StemRegenin 1 Hydrochloride is an aryl hydrocarbon receptor (AhR) antagonist (IC₅₀ = 127 nM) that inhibits RANKL-induced osteoclast generation and differentiation while promoting the expansion of multipotent haematopoietic progenitor cells derived from human embryonic stem cells (hESCs).
| 规格 | 价格 | 库存 | 数量 |
|---|---|---|---|
| 1 mg | ¥ 1,470 | In Stock | |
| 5 mg | ¥ 3,710 | In Stock | |
| 10 mg | ¥ 6,530 | In Stock | |
| 25 mg | ¥ 9,820 | In Stock | |
| 50 mg | ¥ 13,200 | In Stock | |
| 100 mg | ¥ 17,800 | In Stock |
StemRegenin 1 Hydrochloride 相关产品
| 产品描述 | StemRegenin 1 Hydrochloride是一种芳香烃受体(AhR)拮抗剂,IC50=127 nM,能够抑制RANKL诱导的破骨细胞生成和分化,还能够促进人胚胎干细胞(hESC)衍生的多能造血祖细胞的扩增。 |
| 靶点活性 | AhR:127 nM |
| 体外活性 | 将人外周血(mPB)CD34 + 细胞与细胞因子及 StemRegenin 1 Hydrochloride 共同培养 7 天,与对照细胞相比,CD34+、CD133 + 和 CD90 + 造血干祖细胞群体的数量分别增加了 2.6 倍、2.3 倍和 10 倍。在缺乏细胞因子的情况下,StemRegenin 1 Hydrochloride 无法诱导细胞增殖;且当 StemRegenin 1 Hydrochloride 浓度超过 1μM 时,其处理会产生抗增殖效应 [1]。 |
| 体内活性 | 方法:StemRegenin 1 Hydrochloride (30 μg/kg,每周 3 次,隔天 1 次,持续30天)通过腹腔注射给予接受全身照射(TBI)(照射剂量 6 Gy)4 小时后的小鼠,研究StemRegenin 1 Hydrochloride 对致死剂量照射小鼠的辐射缓解作用。 |
| 别名 | StemRegenin 1 盐酸盐, StemRegenin 1 (hydrochloride) (1227633-49-9 free base) |
| 分子量 | 466 |
| 分子式 | C24H24ClN5OS |
| CAS No. | 2319882-01-2 |
| 密度 | no data available |
| 颜色 | White |
| 物理性状 | Solid |
| 存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
| 溶解度信息 | DMSO: ≤ 2.5 mg/mL, Sonication is recommended. |
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