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TargetMol | Compound Library

神经信号分子库现货

Neuronal Signaling Compound Library

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产品编号 L2600

神经元之间和神经元内部的通信对于神经系统的所有功能至关重要,无论是从发育到衰老,还是从健康到疾病。在过去十年中,我们对神经系统内分子、细胞和系统信号通路的认识取得了巨大进步,在信号通路研究方面取得了重大突破,这些神经信号通路是神经发生、成瘾、自闭症以及情绪障碍的病理生理学和治疗基础。例如:G 蛋白偶联受体(GPCR),包括5-HT 受体、组胺受体、阿片受体等,是研究较多的神经元信号传导途径,GPCR 功能障碍会引起多种神经疾病;Notch 信号途径调节神经干细胞增殖、存活、自我更新和分化,Notch 信号传导异常参与中风、阿尔茨海默病和CNS 肿瘤等疾病中发生的病理过程。因此靶向神经元信号传导,可以用来治疗多种不同CNS 疾病。

TargetMol 神经信号分子库包含2771 种神经信号相关的小分子化合物,主要用于神经系统类疾病的药物研发,可用于高通量、高内涵筛选。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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产品编号 L2600

神经信号分子库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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产品描述 产品描述

  • 2771种CNS相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 靶点包括5-HT receptor、AChR、Histamine receptor、dopamine receptor、Opiod receptor等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

5-HT Receptor
AChR
Adrenergic Receptor
COX
Dopamine Receptor
Histamine Receptor
Calcium Channel
Apoptosis
GABA Receptor
GluR
Endogenous Metabolite
iGluR
Autophagy
TRP/TRPV Channel
Cholinesterase (ChE)
Adenosine Receptor
NMDAR
Opioid Receptor
MAO
Antibacterial
Beta Amyloid
Monoamine Oxidase
Potassium Channel
NF-κB
Parasite
Serotonin Transporter
P-gp
Gamma-secretase
Cannabinoid Receptor
Sodium Channel
P2X Receptor
Norepinephrine
CaMK
Reactive Oxygen Species
FAAH
Cytochromes P450
NO Synthase
TNF
Neurokinin receptor
ERK
Sigma receptor
Akt
GPCR
PDE
P2Y Receptor
BACE
Lipoxygenase
Antibiotic
PPAR
Caspase
OX Receptor
Interleukin
Influenza Virus
Neuropeptide Y Receptor
Beta-Secretase
HIV Protease
Antioxidant
Drug Metabolite
NOS
Prostaglandin Receptor
Ferroptosis
Virus Protease
IL Receptor
SARS-CoV
p38 MAPK
Antifungal
PI3K
Melatonin Receptor
PKC
ROS
Bcl-2 Family
VEGFR
DNA/RNA Synthesis
STAT
Phospholipase
Imidazoline Receptor
Mitophagy
EGFR
PGE Synthase
Adenylyl Cyclase
MT Receptor
GlyT
MMP
AMPK
Anti-infection
Dehydrogenase
PKA
Wnt/beta-catenin
IκB/IKK
Chloride channel
Carbonic Anhydrase
Transferase
HCV Protease
Estrogen/progestogen Receptor
Phosphatase
Glucocorticoid Receptor
Monoamine Transporter
HSV
Melanocortin Receptor
CGRP Receptor
HIF/HIF Prolyl-Hydroxylase
JNK
GSK-3
MRP
AAK1
Nucleoside Antimetabolite/Analog
Leukotriene Receptor
CDK
Mitochondrial Metabolism
mTOR
TLR
Hydroxylase
Tyrosinase
Histone Methyltransferase
Src
IFNAR
Histone Demethylase
Glutathione Peroxidase
Cholecystokinin Receptor
PARP
Serine/threonin kinase
Neuropeptide FF Receptor
PAFR
AAK1 (AP2 associated kinase 1)
ABC Transporter
Glucosidase
JAK
Epigenetic Reader Domain
TGF-beta/Smad
HDAC
MEK
Microtubule Associated
Melanin-concentrating Hormone Receptor (MCHR)
ATPase
Amino Acids and Derivatives
Reductase
Na+/Ca2+ Exchanger
NADPH
RAAS
Neurotensin Receptor
Immunology/Inflammation related
Topoisomerase
Antifection
CCR
Angiotensin-converting Enzyme (ACE)
Epoxide Hydrolase
cAMP
IGF-1R
Acyltransferase
transporter
Nrf2
Thyroid hormone receptor(THR)
Advanced Glycation End Products
Transaminase
Monocarboxylate transporter
Integrin
c-Met/HGFR
Arrestin
DYRK
Lipase
MIF
Progesterone Receptor
HBV
Estrogen Receptor/ERR
ROCK
IAP
UGT
Bcr-Abl
LDL
MAGL
Aurora Kinase
DNA
Androgen Receptor
BCRP
MAPK
Sirtuin
GluCls
RSV
ATM/ATR
GST
Oxytocin Receptor
FGFR
MDM-2/p53
Gap Junction Protein
Platelet aggregation
DNA Methyltransferase
NOD
S6 Kinase
ROS Kinase
NOD-like Receptor (NLR)
p53
FOXO3
Proteasome
MicroRNA
CAT
ROR
LPL Receptor
Glutaminyl Cyclase
LTR
Neuropeptide W
gp120/CD4
GTPase
OCT
Galectin
CaSR
N-Acetylglucosaminyltransferase
ASCT
Serine Protease
Antifolate
Cell Cycle Arrest
Cysteine Protease
FXR
LIM Kinase
Glutaminase
NR4A
Aryl Hydrocarbon Receptor
IDO
Prolyl Endopeptidase (PREP)
Myosin
Annexin A
FLAP
Adiponectin Receptor
Raf
Glucagon Receptor
Anion Exchanger
HCN Channel
Fatty Acid Synthase
Bombesin Receptor
PDGFR
PAK
Stearoyl-CoA Desaturase (SCD)
ACK1
CXCR
PTEN
Somatostatin
Indoleamine 2,3-Dioxygenase (IDO)
ATP Citrate Lyase
OXPHOS
Antiviral
HSP
STING
Trk receptor
Free radical scavengers
Aminopeptidase
GPCR19
Ephrin Receptor
Pyroptosis
Casein Kinase
Reverse Transcriptase
Retinoid Receptor
CRISPR/Cas9
FOXO
Adenosine Deaminase
FLT
Syk
NADPH-oxidase
HMG-CoA Reductase
Thrombin
Protease-activated Receptor
Lysosomal Autophagy
FAK
Liposome
AhR
CFTR
PD-1/PD-L1
S1P Receptor
NMU2R
NMUR