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TargetMol | Compound Library

神经信号分子库现货

Neuronal Signaling Compound Library
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货号 L2600

神经元之间和神经元内部的通信对于神经系统的所有功能至关重要,无论是从发育到衰老,还是从健康到疾病。在过去十年中,我们对神经系统内分子、细胞和系统信号通路的认识取得了巨大进步,在信号通路研究方面取得了重大突破,这些神经信号通路是神经发生、成瘾、自闭症以及情绪障碍的病理生理学和治疗基础。例如:G 蛋白偶联受体(GPCR),包括5-HT 受体、组胺受体、阿片受体等,是研究较多的神经元信号传导途径,GPCR 功能障碍会引起多种神经疾病;Notch 信号途径调节神经干细胞增殖、存活、自我更新和分化,Notch 信号传导异常参与中风、阿尔茨海默病和CNS 肿瘤等疾病中发生的病理过程。因此靶向神经元信号传导,可以用来治疗多种不同CNS 疾病。

TargetMol 神经信号分子库包含3500 种神经信号相关的小分子化合物,主要用于神经系统类疾病的药物研发,可用于高通量、高内涵筛选。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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货号 L2600

神经信号分子库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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产品描述 产品描述

  • 3500种CNS相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 靶点包括5-HT receptor、AChR、Histamine receptor、dopamine receptor、Opiod receptor等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

5-HT Receptor
AChR
COX
Adrenergic Receptor
Dopamine Receptor
Apoptosis
Histamine Receptor
GABA Receptor
Endogenous Metabolite
Calcium Channel
iGluR
Cholinesterase (ChE)
GluR
Autophagy
TRP/TRPV Channel
Adenosine Receptor
NF-κB
Beta Amyloid
Antibacterial
Opioid Receptor
NMDAR
Monoamine Oxidase
ROS
MAO
Parasite
Potassium Channel
P-gp
Serotonin Transporter
NO Synthase
Akt
TNF
Cytochromes P450
Interleukin
ERK
Gamma-secretase
CaMK
Neurokinin receptor
Sodium Channel
P2X Receptor
p38 MAPK
Reactive Oxygen Species
Cannabinoid Receptor
Norepinephrine
FAAH
Antibiotic
Caspase
Lipoxygenase
Sigma receptor
Drug Metabolite
Influenza Virus
PPAR
PI3K
PDE
P2Y Receptor
GPCR
Melanocortin Receptor
Antifungal
Ferroptosis
Antioxidant
OX Receptor
DNA/RNA Synthesis
HIV Protease
Bcl-2 Family
MMP
JNK
BACE
Neuropeptide Y Receptor
Beta-Secretase
Prostaglandin Receptor
IL Receptor
SARS-CoV
PKC
STAT
NOS
Virus Protease
mTOR
AMPK
Wnt/beta-catenin
Dehydrogenase
EGFR
Imidazoline Receptor
Mitochondrial Metabolism
MRP
PKA
Phospholipase
TLR
Nrf2
HIF/HIF Prolyl-Hydroxylase
GlyT
GSK-3
TGF-beta/Smad
Melatonin Receptor
HDAC
VEGFR
Immunology/Inflammation related
Microtubule Associated
Mitophagy
CDK
Epigenetic Reader Domain
IκB/IKK
Monoamine Transporter
Adenylyl Cyclase
PGE Synthase
Glucocorticoid Receptor
MT Receptor
Anti-infection
Chloride channel
Tyrosinase
PERK
Nucleoside Antimetabolite/Analog
HSV
Amino Acids and Derivatives
Histone Methyltransferase
Estrogen/progestogen Receptor
IFNAR
HCV Protease
Phosphatase
CGRP Receptor
Carbonic Anhydrase
Hydroxylase
PAFR
Transferase
transporter
AAK1
cAMP
Serine/threonin kinase
Leukotriene Receptor
ATPase
HBV
ABC Transporter
CCR
glycosidase
MEK
PARP
MDM-2/p53
Glutathione Peroxidase
Src
Histone Demethylase
MAPK
Antifection
NADPH
NOD-like Receptor (NLR)
Reductase
Glucosidase
Acyltransferase
HSP
FOXO
MAGL
LTR
IAP
Lipase
Angiotensin-converting Enzyme (ACE)
Trk receptor
Ras
Neurotensin Receptor
UGT
Aurora Kinase
AAK1 (AP2 associated kinase 1)
RAAS
Cholecystokinin Receptor
Neuropeptide FF Receptor
JAK
GST
Reverse Transcriptase
Platelet aggregation
ROS Kinase
Topoisomerase
Huntingtin
IGF-1R
RSV
Syk
Transaminase
LPL Receptor
Androgen Receptor
BCRP
Survivin
Aminopeptidase
FAK
S6 Kinase
Melanin-concentrating Hormone Receptor (MCHR)
Integrin
Estrogen Receptor/ERR
Na+/Ca2+ Exchanger
DYRK
Gap Junction Protein
NOD
Monocarboxylate transporter
CXCR
PTEN
Epoxide Hydrolase
GluCls
p53
Tyrosine Kinases
DNA
Sirtuin
ADC Linker
CFTR
Transmembrane Glycoprotein
OAT
Glutaminyl Cyclase
MIF
Bcr-Abl
Indoleamine 2,3-Dioxygenase (IDO)
FGFR
HMG-CoA Reductase
Advanced Glycation End Products
OCT
ROCK
IDO
GRK
Telomerase
Lipid
Antiviral
FLT
DNA Methyltransferase
AhR
Thyroid hormone receptor(THR)
Proteasome
ATM/ATR
CAT
c-Met/HGFR
Progesterone Receptor
Photosensitizer
PAK
PAI-1
Oxytocin Receptor
IRAK
Arrestin
Aryl Hydrocarbon Receptor
LDL
STING
Free radical scavengers
FOXO3
GDNF
N-Acetylglucosaminyltransferase
ATG
NR4A
Adiponectin Receptor
Anion Exchanger
PDGFR
ATP Citrate Lyase
CD74
Casein Kinase
p62
CRISPR/Cas9
MicroRNA
ROR
Galectin
Serine Protease
Cell Cycle Arrest
LIM Kinase
Glucagon Receptor
Orphan Receptor
GPCR19
Protease
Tight Junction Protein
S1P Receptor
Antifolate
Glutaminase
RIP kinase
Fatty Acid Synthase
Somatostatin
PAD
ASK
Protease-activated Receptor
Necroptosis
Annexin A
Raf
Phosphorylase
Na-K-Cl cotransporter
Molecular Glues
Bombesin Receptor
Stearoyl-CoA Desaturase (SCD)
ACK1
SGLT
BMI-1
Thrombin
Taste receptor
LDLR
Myosin
FLAP
Hedgehog/Smoothened
Ligand for E3 Ligase
Adenosine Deaminase
Liposome
Arginase
gp120/CD4
GTPase
c-Myc
CaSR
ASCT
Rho
Liver X Receptor
HCN Channel
Ephrin Receptor
Histone Acetyltransferase
ALK
Carboxypeptidase
Aromatase
HIF
Lysosomal Autophagy
PD-1/PD-L1
Proton pump
Neuropeptide W
Cysteine Protease
FXR
Amylase
Prolyl Endopeptidase (PREP)
Guanylate cyclase
OXPHOS
LRRK2
Pyroptosis
Retinoid Receptor
NADPH-oxidase
NMU2R
NMUR
BTK
PGC-1α