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TargetMol | Compound Library

神经信号分子库现货

Neuronal Signaling Compound Library

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产品编号 L2600

神经元之间和神经元内部的通信对于神经系统的所有功能至关重要,无论是从发育到衰老,还是从健康到疾病。在过去十年中,我们对神经系统内分子、细胞和系统信号通路的认识取得了巨大进步,在信号通路研究方面取得了重大突破,这些神经信号通路是神经发生、成瘾、自闭症以及情绪障碍的病理生理学和治疗基础。例如:G 蛋白偶联受体(GPCR),包括5-HT 受体、组胺受体、阿片受体等,是研究较多的神经元信号传导途径,GPCR 功能障碍会引起多种神经疾病;Notch 信号途径调节神经干细胞增殖、存活、自我更新和分化,Notch 信号传导异常参与中风、阿尔茨海默病和CNS 肿瘤等疾病中发生的病理过程。因此靶向神经元信号传导,可以用来治疗多种不同CNS 疾病。

TargetMol 神经信号分子库包含2771 种神经信号相关的小分子化合物,主要用于神经系统类疾病的药物研发,可用于高通量、高内涵筛选。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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产品编号 L2600

神经信号分子库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 2771种CNS相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 靶点包括5-HT receptor、AChR、Histamine receptor、dopamine receptor、Opiod receptor等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

Packaging And Storage | TargetMol 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

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Library Customization | TargetMol 化合物库组成

5-HT Receptor
AChR
COX
Adrenergic Receptor
Dopamine Receptor
Histamine Receptor
Calcium Channel
GABA Receptor
GluR
TRP/TRPV Channel
Cholinesterase (ChE)
Autophagy
Apoptosis
Adenosine Receptor
Endogenous Metabolite
NMDAR
iGluR
Opioid Receptor
MAO
Beta Amyloid
Antibacterial
NF-κB
Potassium Channel
P-gp
Gamma-secretase
Monoamine Oxidase
P2X Receptor
Cannabinoid Receptor
Serotonin Transporter
Norepinephrine
Parasite
Sodium Channel
CaMK
FAAH
Cytochromes P450
Neurokinin receptor
Reactive Oxygen Species
BACE
Neuropeptide Y Receptor
TNF
NO Synthase
P2Y Receptor
PDE
GPCR
Antibiotic
Sigma receptor
Lipoxygenase
OX Receptor
Influenza Virus
Antioxidant
HIV Protease
NOS
PPAR
Beta-Secretase
IL Receptor
Prostaglandin Receptor
Ferroptosis
Antifungal
ERK
ROS
Melatonin Receptor
Phospholipase
Imidazoline Receptor
Virus Protease
Caspase
MT Receptor
Akt
Adenylyl Cyclase
p38 MAPK
Mitophagy
Drug Metabolite
GlyT
EGFR
PGE Synthase
DNA/RNA Synthesis
Bcl-2 Family
STAT
Chloride channel
Carbonic Anhydrase
HCV Protease
Estrogen/progestogen Receptor
Transferase
Dehydrogenase
PKA
Wnt/beta-catenin
AAK1
Glucocorticoid Receptor
PKC
Interleukin
SARS-CoV
AMPK
Melanocortin Receptor
Phosphatase
GSK-3
MRP
Monoamine Transporter
HSV
MMP
IκB/IKK
CGRP Receptor
Histone Methyltransferase
Glutathione Peroxidase
ATPase
PI3K
Histone Demethylase
Serine/threonin kinase
Cholecystokinin Receptor
ABC Transporter
TGF-beta/Smad
TLR
Tyrosinase
Src
Reductase
NADPH
RAAS
JNK
Melanin-concentrating Hormone Receptor (MCHR)
Na+/Ca2+ Exchanger
PARP
VEGFR
Topoisomerase
Mitochondrial Metabolism
Neurotensin Receptor
Immunology/Inflammation related
PAFR
CDK
Antifection
cAMP
Acyltransferase
transporter
CCR
Epoxide Hydrolase
mTOR
MEK
HDAC
Anti-infection
HIF/HIF Prolyl-Hydroxylase
Transaminase
Arrestin
DYRK
Progesterone Receptor
Advanced Glycation End Products
Amino Acids and Derivatives
IFNAR
Lipase
Estrogen Receptor/ERR
ROCK
IAP
UGT
Bcr-Abl
LDL
HBV
Leukotriene Receptor
Glucosidase
Aurora Kinase
Epigenetic Reader Domain
DNA
BCRP
JAK
IGF-1R
Androgen Receptor
GluCls
ATM/ATR
GST
Nrf2
RSV
Hydroxylase
Gap Junction Protein
Platelet aggregation
DNA Methyltransferase
NOD
Microtubule Associated
p53
FOXO3
Monocarboxylate transporter
ROR
c-Met/HGFR
LPL Receptor
Glutaminyl Cyclase
Neuropeptide W
gp120/CD4
GTPase
Proteasome
MicroRNA
Integrin
LTR
Antifolate
Myosin
Annexin A
Adiponectin Receptor
Raf
Anion Exchanger
N-Acetylglucosaminyltransferase
Cell Cycle Arrest
Nucleoside Antimetabolite/Analog
Cysteine Protease
LIM Kinase
FXR
Aryl Hydrocarbon Receptor
FLAP
Glucagon Receptor
HCN Channel
Fatty Acid Synthase
Stearoyl-CoA Desaturase (SCD)
ACK1
Angiotensin-converting Enzyme (ACE)
Somatostatin
HSP
STING
Free radical scavengers
GPCR19
MAGL
Bombesin Receptor
PAK
Indoleamine 2,3-Dioxygenase (IDO)
MAPK
Antiviral
Aminopeptidase
FGFR
NMU2R
FLT
HMG-CoA Reductase
Protease-activated Receptor
AhR
CFTR
Casein Kinase
Reverse Transcriptase
Retinoid Receptor
CRISPR/Cas9
Adenosine Deaminase
Syk
NADPH-oxidase
Thrombin
Lysosomal Autophagy
FAK
ROS Kinase
NOD-like Receptor (NLR)
S1P Receptor