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TargetMol | Compound Library

神经信号分子库现货

Neuronal Signaling Compound Library
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货号 L2600

神经元之间和神经元内部的通信对于神经系统的所有功能至关重要,无论是从发育到衰老,还是从健康到疾病。在过去十年中,我们对神经系统内分子、细胞和系统信号通路的认识取得了巨大进步,在信号通路研究方面取得了重大突破,这些神经信号通路是神经发生、成瘾、自闭症以及情绪障碍的病理生理学和治疗基础。例如:G 蛋白偶联受体(GPCR),包括5-HT 受体、组胺受体、阿片受体等,是研究较多的神经元信号传导途径,GPCR 功能障碍会引起多种神经疾病;Notch 信号途径调节神经干细胞增殖、存活、自我更新和分化,Notch 信号传导异常参与中风、阿尔茨海默病和CNS 肿瘤等疾病中发生的病理过程。因此靶向神经元信号传导,可以用来治疗多种不同CNS 疾病。

TargetMol 神经信号分子库包含3500 种神经信号相关的小分子化合物,主要用于神经系统类疾病的药物研发,可用于高通量、高内涵筛选。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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货号 L2600

神经信号分子库

规格

  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 3500种CNS相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 靶点包括5-HT receptor、AChR、Histamine receptor、dopamine receptor、Opiod receptor等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

5-HT Receptor
AChR
Adrenergic Receptor
COX
Dopamine Receptor
Apoptosis
Histamine Receptor
GABA Receptor
Endogenous Metabolite
Calcium Channel
iGluR
Cholinesterase (ChE)
GluR
Autophagy
TRP/TRPV Channel
Adenosine Receptor
NF-κB
Beta Amyloid
Antibacterial
Opioid Receptor
NMDAR
Monoamine Oxidase
ROS
MAO
Parasite
Potassium Channel
P-gp
Serotonin Transporter
NO Synthase
Akt
TNF
Gamma-secretase
Cytochromes P450
ERK
Interleukin
CaMK
Sodium Channel
P2X Receptor
Neurokinin receptor
p38 MAPK
Reactive Oxygen Species
Cannabinoid Receptor
Norepinephrine
FAAH
Antibiotic
Caspase
Lipoxygenase
Sigma receptor
Drug Metabolite
PI3K
Influenza Virus
PPAR
PDE
Melanocortin Receptor
P2Y Receptor
GPCR
Ferroptosis
HIV Protease
DNA/RNA Synthesis
Bcl-2 Family
Antioxidant
Antifungal
OX Receptor
MMP
JNK
BACE
Neuropeptide Y Receptor
Prostaglandin Receptor
Beta-Secretase
IL Receptor
PKC
SARS-CoV
STAT
NOS
mTOR
Adenylate cyclase
Virus Protease
Wnt/beta-catenin
Dehydrogenase
EGFR
AMPK
Mitochondrial Metabolism
TLR
Nrf2
PKA
Phospholipase
Imidazoline Receptor
MRP
HIF/HIF Prolyl-Hydroxylase
Melatonin Receptor
Mitophagy
GSK-3
GlyT
VEGFR
Anti-infection
CDK
Epigenetic Reader Domain
TGF-beta/Smad
IκB/IKK
HDAC
Microtubule Associated
Immunology/Inflammation related
Glucocorticoid Receptor
MT Receptor
Chloride channel
Tyrosinase
PGE Synthase
Amino Acids and Derivatives
Transferase
IFNAR
HCV Protease
Phosphatase
CGRP Receptor
PERK
Nucleoside Antimetabolite/Analog
Monoamine Transporter
HSV
Histone Methyltransferase
Estrogen/progestogen Receptor
PAFR
cAMP
Leukotriene Receptor
Carbonic Anhydrase
ABC Transporter
Hydroxylase
transporter
MEK
PARP
MDM-2/p53
Glutathione Peroxidase
Serine/threonin kinase
Reductase
AAK1
ATPase
HBV
CCR
glycosidase
MAPK
NADPH
NOD-like Receptor (NLR)
MAGL
Glucosidase
Acyltransferase
HSP
Histone Demethylase
Antifection
FOXO
Lipase
Angiotensin-converting Enzyme (ACE)
Trk receptor
Ras
AAK1 (AP2 associated kinase 1)
GST
Reverse Transcriptase
Platelet aggregation
ROS Kinase
Topoisomerase
Huntingtin
Melanin-concentrating Hormone Receptor (MCHR)
RAAS
Cholecystokinin Receptor
Neuropeptide FF Receptor
JAK
Src
LTR
IAP
Neurotensin Receptor
UGT
Aurora Kinase
RSV
Syk
Na+/Ca2+ Exchanger
DYRK
Gap Junction Protein
NOD
Monocarboxylate transporter
CXCR
PTEN
Epoxide Hydrolase
GluCls
p53
Integrin
Estrogen Receptor/ERR
IGF-1R
CFTR
Transaminase
LPL Receptor
Androgen Receptor
BCRP
Survivin
Aminopeptidase
FAK
Transmembrane Glycoprotein
OAT
Advanced Glycation End Products
ROCK
IDO
GRK
Telomerase
Lipid
Antiviral
FLT
DNA Methyltransferase
S6 Kinase
AhR
CAT
c-Met/HGFR
Progesterone Receptor
Photosensitizer
PAK
PAI-1
IRAK
Arrestin
Aryl Hydrocarbon Receptor
LDL
STING
Free radical scavengers
Thyroid hormone receptor(THR)
Proteasome
ATM/ATR
Tyrosine Kinases
DNA
Sirtuin
ADC Linker
Glutaminyl Cyclase
MIF
Bcr-Abl
Indoleamine 2,3-Dioxygenase (IDO)
HMG-CoA Reductase
PGC-1α
MicroRNA
ROR
Galectin
Serine Protease
Cell Cycle Arrest
Glucagon Receptor
Orphan Receptor
GPCR19
Protease
Tight Junction Protein
S1P Receptor
Necroptosis
OCT
Annexin A
Raf
Phosphorylase
Na-K-Cl cotransporter
Molecular Glues
Bombesin Receptor
Stearoyl-CoA Desaturase (SCD)
ACK1
SGLT
FOXO3
BMI-1
Thrombin
Arginase
gp120/CD4
GTPase
c-Myc
CaSR
ASCT
Rho
Liver X Receptor
BTK
HCN Channel
Ephrin Receptor
Histone Acetyltransferase
ALK
Carboxypeptidase
Aromatase
Oxytocin Receptor
HIF
Lysosomal Autophagy
PD-1/PD-L1
Proton pump
Neuropeptide W
Cysteine Protease
FXR
Amylase
Prolyl Endopeptidase (PREP)
Guanylate cyclase
OXPHOS
LRRK2
Pyroptosis
Retinoid Receptor
NADPH-oxidase
Taste receptor
LDLR
Myosin
FLAP
Hedgehog/Smoothened
Adenosine Deaminase
Liposome
GDNF
N-Acetylglucosaminyltransferase
ATG
NR4A
Adiponectin Receptor
Anion Exchanger
PDGFR
ATP Citrate Lyase
CD74
Casein Kinase
p62
CRISPR/Cas9
Antifolate
Glutaminase
RIP kinase
Ligands for E3 Ligase
Fatty Acid Synthase
Somatostatin
PAD
ASK
FGFR
Protease-activated Receptor
NMU2R
NMUR