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TargetMol | Compound Library

神经信号分子库现货

Neuronal Signaling Compound Library
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货号 L2600

神经元之间和神经元内部的通信对于神经系统的所有功能至关重要,无论是从发育到衰老,还是从健康到疾病。在过去十年中,我们对神经系统内分子、细胞和系统信号通路的认识取得了巨大进步,在信号通路研究方面取得了重大突破,这些神经信号通路是神经发生、成瘾、自闭症以及情绪障碍的病理生理学和治疗基础。例如:G 蛋白偶联受体(GPCR),包括5-HT 受体、组胺受体、阿片受体等,是研究较多的神经元信号传导途径,GPCR 功能障碍会引起多种神经疾病;Notch 信号途径调节神经干细胞增殖、存活、自我更新和分化,Notch 信号传导异常参与中风、阿尔茨海默病和CNS 肿瘤等疾病中发生的病理过程。因此靶向神经元信号传导,可以用来治疗多种不同CNS 疾病。

TargetMol 神经信号分子库包含3500 种神经信号相关的小分子化合物,主要用于神经系统类疾病的药物研发,可用于高通量、高内涵筛选。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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货号 L2600

神经信号分子库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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产品描述 产品描述

  • 3500种CNS相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 靶点包括5-HT receptor、AChR、Histamine receptor、dopamine receptor、Opiod receptor等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

5-HT Receptor
AChR
COX
Adrenergic Receptor
Dopamine Receptor
Apoptosis
Histamine Receptor
GABA Receptor
Endogenous Metabolite
Calcium Channel
iGluR
Cholinesterase (ChE)
GluR
Autophagy
TRP/TRPV Channel
Adenosine Receptor
Beta Amyloid
NF-κB
Antibacterial
Opioid Receptor
NMDAR
Monoamine Oxidase
ROS
MAO
Parasite
Potassium Channel
P-gp
Serotonin Transporter
NO Synthase
Akt
TNF
ERK
Cytochromes P450
Interleukin
Gamma-secretase
CaMK
Neurokinin receptor
Sodium Channel
P2X Receptor
p38 MAPK
Reactive Oxygen Species
Cannabinoid Receptor
Norepinephrine
FAAH
Antibiotic
Caspase
Lipoxygenase
Sigma receptor
Drug Metabolite
Influenza Virus
PI3K
PPAR
PDE
GPCR
P2Y Receptor
Melanocortin Receptor
Ferroptosis
Antifungal
HIV Protease
Antioxidant
OX Receptor
DNA/RNA Synthesis
Bcl-2 Family
JNK
MMP
BACE
Neuropeptide Y Receptor
Beta-Secretase
Prostaglandin Receptor
IL Receptor
SARS-CoV
PKC
NOS
STAT
Virus Protease
mTOR
Dehydrogenase
Wnt/beta-catenin
AMPK
EGFR
MRP
PKA
Mitochondrial Metabolism
TLR
Nrf2
Phospholipase
Imidazoline Receptor
GSK-3
Melatonin Receptor
GlyT
TGF-beta/Smad
HIF/HIF Prolyl-Hydroxylase
Mitophagy
VEGFR
Immunology/Inflammation related
CDK
Epigenetic Reader Domain
IκB/IKK
HDAC
Microtubule Associated
Chloride channel
Adenylyl Cyclase
Glucocorticoid Receptor
MT Receptor
Monoamine Transporter
PGE Synthase
Anti-infection
Tyrosinase
Histone Methyltransferase
HCV Protease
Amino Acids and Derivatives
Estrogen/progestogen Receptor
IFNAR
PERK
Phosphatase
Nucleoside Antimetabolite/Analog
HSV
CGRP Receptor
Carbonic Anhydrase
Transferase
AAK1
Serine/threonin kinase
Leukotriene Receptor
PAFR
cAMP
Hydroxylase
ATPase
Glutathione Peroxidase
HBV
PARP
ABC Transporter
CCR
glycosidase
MAPK
transporter
MEK
MDM-2/p53
Src
Reductase
Histone Demethylase
NADPH
Glucosidase
Antifection
MAGL
Acyltransferase
HSP
FOXO
NOD-like Receptor (NLR)
LTR
RAAS
Lipase
Cholecystokinin Receptor
Neurotensin Receptor
IAP
Topoisomerase
Neuropeptide FF Receptor
UGT
AAK1 (AP2 associated kinase 1)
JAK
Angiotensin-converting Enzyme (ACE)
Aurora Kinase
Huntingtin
Trk receptor
GST
Reverse Transcriptase
Platelet aggregation
Ras
ROS Kinase
Melanin-concentrating Hormone Receptor (MCHR)
Transaminase
Monocarboxylate transporter
Integrin
LPL Receptor
Na+/Ca2+ Exchanger
DYRK
Estrogen Receptor/ERR
CXCR
PTEN
Epoxide Hydrolase
IGF-1R
Androgen Receptor
BCRP
Survivin
Aminopeptidase
GluCls
RSV
Gap Junction Protein
Syk
NOD
S6 Kinase
FAK
p53
Thyroid hormone receptor(THR)
Proteasome
Advanced Glycation End Products
CAT
c-Met/HGFR
Glutaminyl Cyclase
Arrestin
MIF
Progesterone Receptor
OCT
Tyrosine Kinases
Photosensitizer
ROCK
Aryl Hydrocarbon Receptor
IDO
Transmembrane Glycoprotein
Bcr-Abl
LDL
GRK
PAK
DNA
Indoleamine 2,3-Dioxygenase (IDO)
Telomerase
Lipid
OAT
Antiviral
STING
Free radical scavengers
Sirtuin
ADC Linker
PAI-1
ATM/ATR
Oxytocin Receptor
FGFR
FLT
DNA Methyltransferase
IRAK
HMG-CoA Reductase
AhR
CFTR
FOXO3
Proton pump
Taste receptor
MicroRNA
GDNF
ROR
Arginase
Neuropeptide W
Necroptosis
gp120/CD4
GTPase
Galectin
c-Myc
N-Acetylglucosaminyltransferase
CaSR
ASCT
Rho
ATG
Serine Protease
Antifolate
Cell Cycle Arrest
Cysteine Protease
Liver X Receptor
FXR
LIM Kinase
Glutaminase
NR4A
LDLR
Amylase
Prolyl Endopeptidase (PREP)
Myosin
Annexin A
FLAP
RIP kinase
Adiponectin Receptor
Raf
Glucagon Receptor
Phosphorylase
Na-K-Cl cotransporter
Anion Exchanger
Molecular Glues
Guanylate cyclase
HCN Channel
Fatty Acid Synthase
Hedgehog/Smoothened
Bombesin Receptor
PDGFR
Stearoyl-CoA Desaturase (SCD)
ACK1
Somatostatin
PAD
Orphan Receptor
SGLT
ATP Citrate Lyase
OXPHOS
LRRK2
GPCR19
Ephrin Receptor
Histone Acetyltransferase
CD74
ASK
Pyroptosis
ALK
Casein Kinase
p62
Carboxypeptidase
Retinoid Receptor
Ligand for E3 Ligase
Protease
Aromatase
CRISPR/Cas9
HIF
Adenosine Deaminase
NADPH-oxidase
BMI-1
Tight Junction Protein
Thrombin
Protease-activated Receptor
Lysosomal Autophagy
Liposome
PD-1/PD-L1
S1P Receptor
NMU2R
BTK
NMUR
PGC-1α