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糖代谢化合物库

糖代谢化合物库

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产品编号 L2520 Glycometabolism Compound Library
  库化合物信息   Excel SDF

糖类是血清代谢物质的一种,糖代谢对机体新陈代谢有重要意义,代谢异常时可引发机体各种疾病,如糖尿病及其并发症、蚕豆病、肝病等。

此外,糖代谢异常是肿瘤代谢突出的特征之一。糖酵解是生物体内普遍存在的能量代谢过程,指在氧气不充分的条件下,葡萄糖经一系列酶促反应生成丙酮酸,进而还原成乳酸的过程,也称无氧氧化。在有氧的情况下,机体细胞主要通过氧化磷酸化途径获得能量,糖酵解受到抑制。然而在恶性肿瘤中,即使氧供应充分,糖酵解也十分活跃。肿瘤细胞有氧糖酵解能力是正常细胞的20 ~ 30倍,为肿瘤代谢提供大量能量和中间产物,此即Warburg 效应。因此,靶向糖酵解等异常环节的代谢酶是抗肿瘤治疗的重点。一些研究显示,抑制肿瘤细胞糖酵解途径能够有效抑制肿瘤细胞的增殖甚至可以起到杀伤肿瘤细胞的作用。

研究糖代谢对某些相关疾病的治疗具有重要意义,TargetMol 糖代谢化合物库提供708 种糖代谢相关的化合物,作用靶点包含GLUTs、Hexokinase(HK)、Pyruvate Kinase(PK )、phosphofructokinase(PFK)、IDH1/2、LDH、AMPK 等糖代谢相关靶点,是研究糖代谢紊乱疾病、癌症等的有效工具。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
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产品描述

  • 708种糖代谢相关的化合物,可用于高通量和高内涵筛选;
  • 作用靶点包含GLUTs、Hexokinase(HK)、Pyruvate Kinase(PK)、phosphofructokinase(PFK)、IDH1/2、LDH、AMPK等糖代谢相关靶点;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • NMR和HPLC检测技术保证产品高纯度和高质量;
  • 所有化合物现货供应。

化合物库定制

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包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L2520)
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客户使用化合物库发表的文献

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化合物库组成

Apoptosis (117)
Autophagy (116)
PI3K (107)
Phosphatase (76)
PPAR (62)
mTOR (60)
AMPK (51)
Akt (44)
Glucokinase (40)
Endogenous Metabolite (36)
GSK-3 (35)
Dehydrogenase (32)
Antibacterial (30)
DNA-PK (25)
Carbonic Anhydrase (25)
p53 (23)
HIF/HIF Prolyl-Hydroxylase (21)
HIF (21)
NF-κB (19)
S6 Kinase (19)
Parasite (18)
ATM/ATR (18)
CDK (17)
IGF-1R (17)
PDK (16)
Antibiotic (16)
Mitochondrial Metabolism (16)
DPP-4 (15)
Glucocorticoid Receptor (14)
Ferroptosis (14)
Proteasome (14)
Reactive Oxygen Species (14)
COX (14)
SGLT (14)
transporter (14)
Reductase (11)
PKC (10)
Antifungal (10)
HIV Protease (9)
E1/E2/E3 Enzyme (9)
Isocitrate Dehydrogenase (IDH) (9)
Influenza Virus (9)
Wnt/beta-catenin (8)
P450 (8)
Mitophagy (8)
Tyrosinase (8)
Potassium Channel (8)
PKM (8)
Src (8)
VEGFR (7)
TNF (7)
PARP (7)
ERK (7)
PKA (7)
Virus Protease (7)
SGK (7)
NAMPT (6)
NADPH (6)
Calcium Channel (6)
MMP (6)
Mdm2 (6)
HSV (6)
ROCK (6)
PERK (5)
Chk (5)
MEK (5)
Lipoxygenase (5)
Histone Methyltransferase (5)
Casein Kinase (5)
STAT (5)
Interleukin (4)
FLT (4)
EGFR (4)
PDE (4)
PDGFR (4)
AChE (4)
FGFR (4)
ATPase (4)
JNK (4)
PI4K (4)
ALK (3)
Androgen Receptor (3)
p38 MAPK (3)
Sodium Channel (3)
NADPH-oxidase (3)
PTEN (3)
Chloride channel (3)
IL Receptor (3)
SIK (3)
Estrogen/progestogen Receptor (3)
c-Met/HGFR (3)
Adrenergic Receptor (3)
Aryl Hydrocarbon Receptor (3)
Hexokinase (3)
Sirtuin (3)
TRP/TRPV Channel (3)
Phosphorylase (3)
AhR (2)
Beta Amyloid (2)
AChR (2)
DNA/RNA Synthesis (2)
Epigenetic Reader Domain (2)
c-Fms (2)
Estrogen Receptor/ERR (2)
Anti-infection (2)
PAK (2)
BCL (2)
Antioxidant (2)
Integrin (2)
GluR (2)
Gamma-secretase (2)
Aurora Kinase (2)
Serine Protease (2)
HDAC (2)
GABA Receptor (2)
ATP Citrate Lyase (2)
Topoisomerase (2)
Microtubule Associated (2)
Tyrosine Kinases (2)
TGF-beta/Smad (2)
c-RET (2)
Raf (2)
MELK (2)
Bcr-Abl (2)
LRRK2 (2)
FAK (2)
Syk (2)
Trk receptor (1)
Proton pump (1)
Serine/threonin kinase (1)
Thrombin (1)
S1P Receptor (1)
Progesterone Receptor (1)
Prostaglandin Receptor (1)
Reverse Transcriptase (1)
PYK2 (1)
Retinoid Receptor (1)
ROS (1)
ABC (1)
PLK (1)
cell cycle arrest (1)
DNA Alkylator/Crosslinker (1)
DNA Alkylation (1)
DHFR (1)
Cysteine Protease (1)
CSF-1R (1)
Complement System (1)
c-Kit (1)
CaMK (1)
Fatty Acid Synthase (1)
Bombesin Receptor (1)
Beta-Secretase (1)
BACE (1)
Arginase (1)
Adenosine Receptor (1)
Adenosine deaminase (1)
ADC Cytotoxin (1)
Drug Metabolite (1)
Glucagon Receptor (1)
Phospholipase (1)
Immunology/Inflammation related (1)
NOS (1)
Myosin (1)
MRP (1)
MLK (1)
MAPK (1)
JAK (1)
IκB/IKK (1)
iGluR (1)
Glutaminase (1)
HSP (1)
Histone Demethylase (1)
Hedgehog/Smoothened (1)
HCV Protease (1)
Hck (1)
HBV (1)
Guanylate cyclase (1)
Glutathione Peroxidase (1)
YAP (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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