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Histone Modification Compound Library
组蛋白修饰(histone modification)是指组蛋白在相关酶作用下发生甲基化、乙酰化、磷酸化、腺苷酸化、泛素化、ADP 核糖基化等化学修饰的过程。组蛋白修饰可通过改变染色质结构或募集组蛋白修饰物来影响基因表达,因此组蛋白修饰在多种生物过程中起作用,例如转录激活与失活、染色体包装、DNA 损伤与修复等。定量检测各种组蛋白修饰将为更好地理解细胞代谢过程的表观遗传调节提供有用的信息,促进组蛋白修饰酶靶向药物的发展。 TargetMol 组蛋白修饰化合物库是由569 个组蛋白修饰研究相关的小分子的独特集合,用于组蛋白修饰相关的研究以及药物的筛选,可用于高通量、高内涵筛选。
Empty | 99873-43-5 | 99-66-1 | 96680-77-2 | 96017-59-3 | 955900-27-3 | 95480-80-1 | 950762-95-5 | 949912-58-7 | 946150-57-8 | 941521-45-5 | Empty |
Droxinostat | Valproic Acid | 2-methyl-2,3,4,5-tetrahydro-1,5-benzothiazepin-4-one | 2-hexyl-4-Pentynoic Acid | RK-9123016 | 5-Hydroxy-7-acetoxy-8-methoxyflavone | PCI-34051 | Remodelin | Remetinostat | BAZ1A-IN-1 | ||
Empty | 939228-52-1 | 937039-45-7 | 935881-37-1 | 935693-62-2 | 934828-12-3 | 932749-62-7 | 931596-95-1 | 930039-92-2 | 929016-96-6 | 92-78-4 | Empty |
CCI-007 | Pimelic diphenylamide 106 | AR42 | BIX-01294 | CXD101 | Histone Acetyltransferase Inhibitor II | P3FI-63 | BRD4 Inhibitor-27 | Pracinostat | Naphthol AS-E | ||
Empty | 926908-04-5 | 78574-94-4 | 780757-88-2 | 7761-45-7 | 76584-70-8 | 755038-02-9 | 74901-20-5 | 748777-47-1 | 743420-02-2 | 7389-87-9 | Empty |
HNHA | Cycloastragenol | ICG-001 | Metoprine | Divalproex Sodium | BI 2536 | MC2184 | CCT077791 | HDAC-IN-7 | Methyl L-histidinate dihydrochloride | ||
Empty | 732302-99-7 | 726169-73-9 | 709676-56-2 | 709002-46-0 | 6953-61-3 | 65604-80-0 | 652-37-9 | 6398-98-7 | 63512-50-5 | 604769-01-9 | Empty |
Givinostat hydrochloride monohydrate | Mocetinostat | TTK21 | SirReal2 | 1-Naphthohydroxamic acid | Ophiopogonin D' | Acefylline | Amodiaquine dihydrochloride dihydrate | L-2-Hydroxyglutaric acid disodium | R306465 | ||
Empty | 5967-84-0 | 593273-05-3 | 58944-73-3 | 58880-19-6 | 587850-67-7 | 926259-99-6 | 925434-55-5 | 925432-73-1 | 919973-83-4 | 916489-36-6 | Empty |
Theophylline monohydrate | DCH36_06 | Sinefungin | Trichostatin A | C-7280948 | BG45 | SRT 1720 | SRT 1460 | OF-1 | MS417 | ||
Empty | 914382-60-8 | 910462-43-0 | 907957-34-0 | 902279-44-1 | 901245-65-6 | 900305-37-5 | 89412-79-3 | 891002-11-2 | 890643-16-0 | 890190-22-4 | Empty |
Tefinostat | Domatinostat | NSC 694623 | CPUY074020 | GSK-5959 | PFI-4 | Raddeanin A | SIRT6-IN-5 | DC-05 | WDR5-0103 | ||
Empty | 887686-02-4 | 880813-42-3 | 875320-31-3 | 875320-29-9 | 866323-14-0 | 864814-88-0 | 86-42-0 | 86361-55-9 | 863589-52-0 | 852475-26-4 | Empty |
OSS_128167 | CMP-5 | Quisinostat dihydrochloride | Quisinostat | Belinostat | Resminostat | Amodiaquine | Gnetol | Benzamide, 3-methoxy-N-(3-thiazolo[5,4-b]pyridin-2-ylphenyl) | MC1568 | ||
Empty | 849234-64-6 | 848354-66-5 | 848193-69-1 | 848193-68-0 | 847591-62-2 | 847459-98-7 | 847249-57-4 | 824960-50-1 | 796-42-9 | 792946-69-1 | Empty |
BRD-6929 | PTACH | Selisistat R-enantiomer | Selisistat S-enantiomer | ICG001 | CRA-026440 hydrochloride | AES-350 | WDR5-0102 | AS8351 | DCLX069 |