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TargetMol | Compound Library

免疫/炎症分子化合物库现货

Immunology/Inflammation Compound Library

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产品编号 L4700

当某些触发因素引起免疫系统功能紊乱,使其不能区分正常组织和病原,开始攻击破坏自身正常组织时,就会发生自身免疫性疾病,受累部位包括血管、结缔组织、关节和皮肤等。随着19-20世纪的化学进展,开发了非甾体抗炎药(NSAIDs),尽管有效治疗炎性疾病,但NSAID 具有一些不良作用,例如溃疡,肾损伤和胃肠道出血。后来虽然被描述为抗肿瘤介质,但肿瘤坏死因子-α(TNF)通常被认为是主要的促炎细胞因子。它在炎性疾病的发病机制中起关键作用,因此,抗TNF 治疗已成为治疗自身免疫性疾病的主要方法。随着基础研究的快速进展,许多与自身免疫性疾病相关的信号传导途径及相关蛋白陆续被发现,这些蛋白是潜在治疗免疫性疾病的药物靶点,例如,很多小分子化合物或基于大环的药物具有抑制免疫蛋白酶体、抑制核输出蛋白、抑制 NF-kB 和肿瘤坏死因子-α(TNF)的活性,这些化合物有可能发展成用于治疗自身免疫疾病和慢性炎症疾病的药物。 TargetMol 免疫/炎症分子化合物库包含了5293 个抗炎活性化合物,用于抗免疫疾病药物高通量筛选,确认药物靶点以及其他医药研发和科研领域。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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产品编号 L4700

免疫/炎症分子化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 5293种具有抗炎症活性的化合物的特有集合,可用于高通量筛选和高内涵筛选;
  • 部分化合物已经得到FDA批准上市;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Apoptosis
Antibacterial
Autophagy
Antibiotic
Endogenous Metabolite
NF-κB
COX
Reactive Oxygen Species
PI3K
Histamine Receptor
EGFR
Ras
Parasite
HIV Protease
p38 MAPK
Antifungal
TNF
ERK
mTOR
Prostaglandin Receptor
NO Synthase
JAK
Akt
Antiviral
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STAT
DNA/RNA Synthesis
Interleukin
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Influenza Virus
5-HT Receptor
GSK-3
AMPK
TLR
ROS
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CDK
Raf
Cytochromes P450
Nrf2
Potassium Channel
AChR
Adrenergic Receptor
SARS-CoV
PDE
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MAPK
PPAR
NOS
JNK
VEGFR
Caspase
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HCV Protease
CCR
MMP
Ferroptosis
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Lipoxygenase
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Immunology/Inflammation related
Src
CXCR
MEK
FLT
NOD-like Receptor (NLR)
Kras
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Dopamine Receptor
PKC
HBV
Tyrosine Kinases
Wnt/beta-catenin
HSV
NOD
DNA-PK
Reverse Transcriptase
S6 Kinase
Topoisomerase
RIP kinase
Anti-infection
GPCR
Aryl Hydrocarbon Receptor
Antifection
Cholinesterase (ChE)
Mitophagy
Beta Amyloid
GABA Receptor
TRP/TRPV Channel
Phosphatase
ATM/ATR
TGF-beta/Smad
Sodium Channel
HER
Leukotriene Receptor
FGFR
Drug Metabolite
PDGFR
Epigenetic Reader Domain
Phospholipase
Estrogen/progestogen Receptor
Syk
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ribosome
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Pim
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IRAK
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STING
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MRP
PKA
PARP
HDAC
Microtubule Associated
ATPase
NADPH
Estrogen Receptor/ERR
S1P Receptor
RAAS
c-Kit
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Opioid Receptor
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P-gp
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IGF-1R
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ALK
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ROCK
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Sigma receptor
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P2Y Receptor
GluR
MNK
HIF
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FAK
p53
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PERK
IDO
FAAH
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Indoleamine 2,3-Dioxygenase (IDO)
transporter
MLK
Arginase
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Gamma-secretase
PTEN
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Necroptosis
Tie-2
FLAP
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NMDAR
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PAK
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cAMP
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CD73
AIM2
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SGK
Neurokinin receptor
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HMG-CoA Reductase
ADC Cytotoxin
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gp120/CD4
TOPK
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PYK2
PAFR
ABC Transporter
Smo
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Decarboxylase
PLK
RAR/RXR
EBI2/GPR183
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IAP
Myosin
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Somatostatin
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CRISPR/Cas9
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PKM
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Dynamin
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Melatonin Receptor
GNRH Receptor
Cell Cycle Arrest
Glucokinase
NR4A
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GlyT
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Integrase
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ACK1
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Y Box Binding Protein 1
Ligands for Target Protein for PROTAC
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VDA
OCT
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CaSR
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AAK1
ASCT
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PROTAC Linker
Neuropeptide Y Receptor
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Vasopressin Receptor
OX Receptor
Target Protein Ligand-Linker Conjugate
MRGPR
Urea Transporter
GluCls
hCE
CRFR
Methionine Adenosyltransferase (MAT)
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TMV
Protease
GHSR
FOXO
RXFP receptor
CGRP Receptor
BMI-1
TAM Receptor
CFTR
Kinesin