Powder: -20°C for 3 years | In solvent: -80°C for 1 year
hCAIX/XII-IN-1 是一种有效的CAIX/XII 抑制剂,KI 值分别为 0.48 μM 和 0.83 μM。hCAIX/XII-IN-1 显示出体外抗增殖活性。hCAIX/XII-IN-1 诱导 MCF-7 细胞凋亡apoptosis。
规格 | 价格/CNY | 货期 | 数量 | |
---|---|---|---|---|
25 mg | ¥ 10,600 | 10-14周 | ||
50 mg | ¥ 13,800 | 10-14周 | ||
100 mg | ¥ 17,500 | 10-14周 |
产品描述 | hCAIX/XII-IN-1, a potent inhibitor of both CAIX and CAXII, exhibits KI values of 0.48 μM for CAIX and 0.83 μM for CAXII, respectively. This compound demonstrates antiproliferative activity in vitro and induces apoptosis in MCF-7 cells [1]. |
体外活性 | hCAIX/XII-IN-1 (compound 11a) (3.125, 6.25, 12.5, 25, 50 μM, 48 h) shows antiproliferative activity with an IC 50 value of 0.48 μM in MCF-7 cells [1]. hCAIX/XII-IN-1 (0.48 μM; 24 h) increases the cell populations of Sub-G1 phase [1]. hCAIX/XII-IN-1 (0.48 μM) induces apoptosis in MCF-7 cells [1]. Cell Proliferation Assay [1] Cell Line: MCF-7 cells Concentration: 3.125, 6.25, 12.5, 25, 50 μM Incubation Time: 48 h Result: Showed antiproliferative activity with an IC 50 value of 0.48 μM in MCF-7 cells. Cell Cycle Analysis [1] Cell Line: MCF-7 cells Concentration: 0.48 μM Incubation Time: 24 h Result: Significantly increased the cell populations of Sub-G1 phase. Apoptosis Analysis [1] Cell Line: MCF-7 cells Concentration: 0.48 μM Incubation Time: Result: Induced apoptosis in MCF-7 cells. |
分子量 | 397.42 |
分子式 | C19H11NO5S2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
对于不同动物的给药剂量换算,您也可以参考 更多...
请在以下方框中输入您的动物实验信息后点击计算,可以得到母液配置方法和体内配方的制备方法: 比如您的给药剂量是10 mg/kg,每只动物体重20 g,给药体积100 μL,一共给药动物10 只,您使用的配方为5% DMSO+30% PEG300+5% Tween 80+60% ddH2O。那么您的工作液浓度为2 mg/mL。
母液配置方法:2 mg 药物溶于 50 μL DMSO (母液浓度为 40 mg/mL), 如您需要配置的浓度超过该产品的溶解度,请先与我们联系。
体内配方的制备方法:取 50 μL DMSO 主液,加入 300 μL PEG300, 混匀澄清,再加 50 μL Tween 80,混匀澄清,再加 600 μL ddH2O, 混匀澄清。
您可能有的问题的答案可以在抑制剂处理说明中找到,包括如何准备库存溶液,如何存储产品,以及基于细胞的分析和动物实验需要特别注意的问题。
hCAIX/XII-IN-1 Inhibitor inhibitor inhibit