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别名 阿伐斯汀, Semprex, BW825C, Acrivastin
Acrivastine (Acrivastin) 是一种短效组胺 1 受体拮抗剂,可用于研究过敏性鼻炎。


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Acrivastine (Acrivastin) 是一种短效组胺 1 受体拮抗剂,可用于研究过敏性鼻炎。
| 规格 | 价格 | 库存 | 数量 |
|---|---|---|---|
| 2 mg | ¥ 127 | In stock | |
| 5 mg | ¥ 189 | In stock | |
| 10 mg | ¥ 289 | In stock | |
| 25 mg | ¥ 579 | In stock | |
| 50 mg | ¥ 868 | In stock | |
| 100 mg | ¥ 1,280 | In stock | |
| 500 mg | ¥ 3,280 | In stock | |
| 1 mL x 10 mM (in DMSO) | ¥ 228 | In stock |
Acrivastine 相关产品
| 产品描述 | Acrivastine (Acrivastin) is a short-acting histamine 1 receptor antagonist. |
| 体内活性 | Acrivastine (usually 8mg three times daily) is an effective and well-tolerated antihistamine in the treatment of chronic urticaria and allergic rhinitis. Acrivastine causes less drowsiness than clemastine, the incidence of adverse effects being indistinguishable from that with placebo or terfenadine. In the treatment of dermatoses in which histamine has a pathogenetic role, the efficacy of acrivastine is superior to that of placebo and similar to that of usual dosages of clemastine, hydroxyzine, chlorpheniramine, cyproheptadine or terfenadine [1]. Both 4 mg and 8 mg acrivastine alleviate the symptoms of seasonal allergic rhinitis with significant improvements in the symptom scores for sneezing, running nose and the calculated overall score. In addition, 8 mg acrivastine reduces the symptom scores for watery eyes and itchy throat. Acrivastine is both well tolerated and effective in the treatment of seasonal allergic rhinitis [2]. |
| 别名 | 阿伐斯汀, Semprex, BW825C, Acrivastin |
| 分子量 | 348.44 |
| 分子式 | C22H24N2O2 |
| CAS No. | 87848-99-5 |
| Smiles | Cc1ccc(cc1)C(=C/CN1CCCC1)\c1cccc(\C=C\C(O)=O)n1 |
| 密度 | 1.170 g/cm3 (Predicted) |
| 存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. | ||||||||||||||||||||
| 溶解度信息 | DMSO: 5 mg/mL (14.35 mM), Sonication is recommended. | ||||||||||||||||||||
| 体内实验配方 | 10% DMSO+40% PEG300+5% Tween 80+45% Saline: 1 mg/mL (2.87 mM), Sonication is recommended. 请按顺序添加溶剂,在添加下一种溶剂之前,尽可能使溶液澄清。如有必要,可通过加热、超声、涡旋处理进行溶解。工作液建议现配现用。以上配方仅供参考,体内配方并不是绝对的,请根据不同情况进行调整。 | ||||||||||||||||||||
溶液配制表 | |||||||||||||||||||||
DMSO
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