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hMC1R agonist 1 是一种有效的选择性hMC1R 激动剂(EC50=3 nM),hMC1R agonist 1 对hMC1R 的选择性是hMC3R(b>EC50=902 nM),hMC4R(b>EC50=915 nM),和hMC5R(b>EC50=>1000 nM) 的 300 倍。hMC1R agonist 1 有研究和预防黑皮质素家族疾病的潜能。
hMC1R agonist 1 是一种有效的选择性hMC1R 激动剂(EC50=3 nM),hMC1R agonist 1 对hMC1R 的选择性是hMC3R(b>EC50=902 nM),hMC4R(b>EC50=915 nM),和hMC5R(b>EC50=>1000 nM) 的 300 倍。hMC1R agonist 1 有研究和预防黑皮质素家族疾病的潜能。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
5 mg | 待询 | 期货 | |
50 mg | 待询 | 期货 |
产品描述 | hMC1R agonist 1, with an EC 50 of 3 nM, exhibits at least 300-fold higher selectivity for hMC1R compared to hMC3R (EC 50 >902 nM), hMC4R (EC 50 >915 nM), and hMC5R (EC 50 >1000 nM). This compound demonstrates potential for therapeutic applications in targeting the melanocortin family [1]. |
分子量 | 1107.35 |
分子式 | C54H70N14O8S2 |
存储 | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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