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内分泌激素分子库

内分泌激素分子库

产品编号 L2400 Endocrinology-Hormone Compound Library
  库化合物信息   Excel SDF

内分泌腺是由一群合成并释放激素的细胞组成,激素随体液输送到靶细胞起作用,调节生长、发育、繁殖和代谢活动,维持内环境的稳态。常见的激素有甲状腺激素、肾上腺素、胰岛素、性激素等,根据化学结构不同,激素通常分为蛋白类、固醇类和氨基酸衍生物,不同激素的受体不同,作用方式不同。内分泌系统的疾病可由激素的过度分泌或分泌不足或目标器官或组织无法有效应对激素引起。

TargetMol 内分泌激素分子库包含784 个与内分泌系统及其信号通路相关的小分子化合物,用于人体内分泌系统的研究及相关疾病的药物筛选,可用于高通量、高内涵筛选。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
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产品描述

  • 784种与内分泌系统相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 是研究人体内分泌系统疾病和筛选相关药物的有效工具; 
  • 靶点含雌激素受体、甲状腺激素受体、去甲肾上腺素受体等等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L2400)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

Adrenergic Receptor (147)
Estrogen/progestogen Receptor (91)
Opioid Receptor (76)
Estrogen Receptor/ERR (76)
RAAS (75)
Dopamine Receptor (71)
GPR (71)
Autophagy (58)
Androgen Receptor (57)
Glucocorticoid Receptor (56)
Endogenous Metabolite (55)
Apoptosis (54)
5-HT Receptor (49)
Prostaglandin Receptor (30)
Reductase (25)
Thyroid hormone receptor(THR) (22)
AChR (21)
Progesterone Receptor (20)
Histamine Receptor (19)
Antibacterial (13)
Potassium Channel (11)
P450 (10)
Norepinephrine (10)
Calcium Channel (9)
COX (9)
Aromatase (9)
IGF-1R (8)
Influenza Virus (8)
Drug Metabolite (7)
PPAR (7)
NF-κB (7)
Cannabinoid Receptor (6)
Oxytocin Receptor (6)
Antibiotic (6)
Mitophagy (6)
Reactive Oxygen Species (6)
HSP (5)
ERK (5)
CaMK (5)
Endothelin Receptor (5)
Antifungal (5)
NO Synthase (5)
Virus Protease (4)
PDE (4)
Ferroptosis (4)
MRP (4)
OX Receptor (4)
Parasite (4)
Thrombin (4)
HIV Protease (4)
Annexin A (3)
Interleukin (3)
MMP (3)
TRP/TRPV Channel (3)
Vasopressin Receptor (3)
Arrestin (3)
Imidazoline Receptor (3)
Serotonin Transporter (3)
Sodium Channel (3)
ALK (3)
Kisspeptin (3)
Phosphatase (3)
TNF (3)
VEGFR (3)
Antioxidant (3)
Lipoxygenase (2)
AhR (2)
Tyrosinase (2)
Gap Junction Protein (2)
GluR (2)
AChE (2)
MEK (2)
GABA Receptor (2)
Phospholipase (2)
STAT (2)
mTOR (2)
Nrf2 (2)
SARS-CoV (2)
Akt (2)
P-gp (2)
Melanin-concentrating Hormone Receptor (MCHR) (2)
ROS (2)
Cysteine Protease (2)
Serine Protease (2)
Liver X Receptor (2)
PKC (2)
p38 MAPK (2)
GNRH Receptor (2)
iGluR (2)
Dehydrogenase (2)
PI3K (2)
ATPase (2)
Glucagon Receptor (2)
JNK (2)
Smo (2)
P2Y Receptor (1)
GHSR (1)
RAR/RXR  (1)
Ligands for Target Protein for PROTAC (1)
NADPH (1)
c-RET (1)
CGRP Receptor (1)
Integrin (1)
CRISPR/Cas9 (1)
HSV (1)
Src (1)
HCV Protease (1)
Glutathione Peroxidase (1)
Histone Methyltransferase (1)
ROR (1)
Platelet aggregation (1)
DNA Methyltransferase (1)
Transferase (1)
S6 Kinase (1)
Carbonic Anhydrase (1)
NOS (1)
Chloride channel (1)
FAK (1)
Apelin receptor (1)
advanced glycation end products (1)
Monoamine Oxidase (1)
LHRH (1)
Melatonin Receptor (1)
Ligand for E3 Ligase (1)
Caspase (1)
PROTAC Linker (1)
Monoamine Transporter (1)
Phosphorylase (1)
Thrombopoietin Receptor (1)
LDL (1)
Epigenetic Reader Domain (1)
Gamma-secretase (1)
Fas/FasL (1)
UGT (1)
Adiponectin receptor (1)
Immunology/Inflammation related (1)
MAO (1)
RANKL/RANK (1)
EGFR (1)
Antiviral (1)
HDAC (1)
Rho (1)
HBV (1)
Free radical scavengers (1)
Histone Acetyltransferase (1)
CaSR (1)
RSV (1)
ABC (1)
Neprilysin (1)
GST (1)
Acetyl-CoA Carboxylase (1)
Reverse Transcriptase (1)
IL Receptor (1)
Retinoid Receptor (1)
GSK-3 (1)
HER (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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