Name: D13-9001
Brand: TargetMol
SKU: T10944
Rating: 4.5 (1 reviews)

规格

价格

库存

数量

25 mg

¥ 22,200

3-6月

50 mg

¥ 27,800

3-6月

100 mg

¥ 34,500

3-6月

生物活性

产品描述	The KD values of D13-9001 in Escherichia coli and Pseudomonas aeruginosa were 1.15μM and 3.57μM, respectively. D13-9001 has antibiotic activity. It is an effective AcrB (AcrAB-TolC efflux pump subunit) and MexB (MexAB-OprM efflux pump subunit) inhibitor.
靶点活性	MexB:3.57 μM (kd), AcrB:(kd)1.15 μM
体外活性	D13-9001 has high solubility and good safety.
体内活性	Compared with AZT treated alone, D13-9001 (1.25-20 mg / kg; intravenous infusion; 2 hours) using aztreonam (AZT) can improve the survival rate of lethal pneumonia rats at the end of the seventh day .

化学信息

分子量	693.78
分子式	C₃₁H₃₉N₁₁O₆S
CAS No.	957471-96-4
Smiles	C(=C/C=1NN=NN1)\C2=C(N=C3N(C2=O)C=CC(C(NC4=NC(C(C)(C)C)=CS4)=O)=C3)N5C[C@H](OC(NCC[N+](CC([O-])=O)(C)C)=O)CCC5
密度	no data available

储存&溶解度

存储	Powder: -20°C for 3 years \| In solvent: -80°C for 1 year Shipping with blue ice/Shipping at ambient temperature. 实际储存温度请以COA为准

D13-9001