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Search Results for " inhibitor "

Targets Recommended: Carboxypeptidase

10000+

抑制剂 & 化合物

1000+

天然产物

17

化合物库

94

TargetMol 试剂盒

444

重组蛋白

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Cat. No.	Product Name
L2000	抑制剂库		8418 compounds
	8418 个小分子抑制剂的独特集合，主要用于细胞信号研究、新药筛选、高通量筛选和高内涵筛选；
L9100	磷酸酶抑制剂化合物库		80 compounds
	80 种已知活性的磷酸酶抑制剂的集合，可用于化合物筛选、化学基因组学、药理分析等方面；
L1600	激酶抑制剂库		2720 compounds
	2720 种激酶抑制剂/调节剂的独特集合，用于特定靶向激酶，可用于高通量筛选和高内涵筛选；
L7600	趋化因子抑制剂库		59 compounds
	59 种趋化因子或其受体抑制剂的独特集合，可用于高通量筛选和高内涵筛选；
L9400	PPI抑制剂库		490 compounds
	490 种已知活性的 PPI 相关的抑制剂，可用于高通量、高内涵筛选；
L1400	MAPK 抑制剂库		367 compounds
	367 种与MAPK 信号通路相关的生物活性小分子化合物的特有集合，可用于高通量筛选和高内涵筛选；
L1100	蛋白酶抑制剂库		344 compounds
	344 种已知的小分子蛋白酶抑制剂的特有集合，可用于高通量筛选和高内涵筛选；
L9410	共价抑制剂库		1949 compounds
	1949 种小分子的独特集合，包含已发现的共价抑制剂以及包含某些共价反应基团常见弹头的分子，如氯乙酰基，2-氯丙酰基，丙烯酰基，1-丙-2-炔基，1-丁-2-炔基，酮羰基，二硫键等，可以用于共价抑制剂药物研发；
L3600	细胞因子抑制剂库		613 compounds
	613 个与细胞因子紧密相关的化合物集合，是高通量、高内涵筛选的良好载体；
L2200	酪氨酸激酶分子库		1033 compounds
	1033 种酪氨酸激酶抑制剂的独特集合，可用于高通量筛选和高内涵筛选；
L2300	离子通道库		946 compounds
	946 种与离子通道相关的生物活性小分子化合物的特有集合，用于离子通道相关的疾病和药物研究，可用于高通量筛选和高内涵筛选；
L1610	FDA 上市激酶抑制剂库		266 compounds
	266种靶向激酶的上市药物集合，用于特定靶向激酶，可用于高通量筛选和高内涵筛选；
L2010	高选择性抑制剂库		580 compounds
	xunm种具有高选择性的抑制剂集合
L1510	核受体化合物库		546 compounds
	546 个核受体作用化合物的独特集合，可用于高通量筛选和高内涵筛选；
L8000	干细胞分化化合物库		1213 compounds
	1213 种干细胞分化信号通路相关的生物活性小分子化合物的特有集合，可用于高通量、高内涵筛选；
L7000	活性脂质化合物库		385 compounds
	385 种生物活性小分子化合物，用于高通量、高内涵筛选；
L7110	抗高血压化合物库		719 compounds
	719 种高血压相关的小分子，用于高通量和高内涵筛选；

化合物库

Cat.No: L2000

Compounds: 8418

磷酸酶抑制剂化合物库

Cat.No: L9100

Compounds: 80

激酶抑制剂库

Cat.No: L1600

Compounds: 2720

趋化因子抑制剂库

Cat.No: L7600

Compounds: 59

PPI抑制剂库

Cat.No: L9400

Compounds: 490

MAPK 抑制剂库

Cat.No: L1400

Compounds: 367

蛋白酶抑制剂库

Cat.No: L1100

Compounds: 344

共价抑制剂库

Cat.No: L9410

Compounds: 1949

细胞因子抑制剂库

Cat.No: L3600

Compounds: 613

酪氨酸激酶分子库

Cat.No: L2200

Compounds: 1033

离子通道库

Cat.No: L2300

Compounds: 946

FDA 上市激酶抑制剂库

Cat.No: L1610

Compounds: 266

高选择性抑制剂库

Cat.No: L2010

Compounds: 580

核受体化合物库

Cat.No: L1510

Compounds: 546

干细胞分化化合物库

Cat.No: L8000

Compounds: 1213

活性脂质化合物库

Cat.No: L7000

Compounds: 385

抗高血压化合物库

Cat.No: L7110

Compounds: 719

Cat. No.	Product Name	Form	Specificity Of Inhibition
C0002	Phosphatase Inhibitor Cocktail I (100× ddH2O) 磷酸酶抑制剂 Cocktail I (100× ddH2O)	Solution (100× in ddH2O)	Acid Phosphatase, Alkaline phosphatase, PTPs, ATPases
C0003	Phosphatase Inhibitor Cocktail II (100× DMSO) 磷酸酶抑制剂 Cocktail II (100× DMSO)	Solution (100× in DMSO)	Alkaline phosphatases, Ser/Thr phosphatases, Acid and PP1 and PP2A
C0004	Phosphatase Inhibitor Cocktail III (2 Tubes, 100x) 磷酸酶抑制剂 Cocktail III (2 Tubes, 100x)	2 Tube Solution (100×)	Each Tube has different specificity of inhibition
C0001	Protease Inhibitor Cocktail (EDTA-Free, 100× in DMSO) 蛋白酶抑制剂 Cocktail (EDTA-Free, 100× in DMSO)	Solution (EDTA-Free,100× in DMSO)	Serine proteases, Aminopeptidases, Cysteine proteases, Aspartic proteases
C0048	Deacetylase Inhibitor Cocktail (100× in 70% DMSO) 去乙酰化酶抑制剂 Cocktail（100× in 70% DMSO）	Solution (100× in 70% DMSO)	Class I/II/III HDAC
CL0064	PDE inhibitor kit PDE inhibitor kit
CL0140	BTK inhibitor kit BTK inhibitor kit
CL0128	HMGCR inhibitor kit HMGCR inhibitor kit
CL0131	SGLT inhibitor kit SGLT inhibitor kit
CL0142	MMP inhibitor kit MMP inhibitor kit
CL0121	ALK inhibitor kit ALK inhibitor kit
CL0052	HDAC inhibitor kit HDAC inhibitor kit
CL0062	Topoisomerase inhibitor kit Topoisomerase inhibitor kit
CL0081	Phosphatase inhibitor kit Phosphatase inhibitor kit
CL0100	Raf inhibitor kit Raf inhibitor kit
CL0072	BET inhibitor kit BET inhibitor kit
CL0127	NOS inhibitor kit NOS inhibitor kit
CL0085	HSP inhibitor kit HSP inhibitor kit
CL0132	DHFR inhibitor kit DHFR inhibitor kit
CL0133	CXCR inhibitor kit CXCR inhibitor kit
CL0087	mTOR inhibitor kit mTOR inhibitor kit
CL0045	COX inhibitor kit COX inhibitor kit
CL0116	MAO inhibitor kit MAO inhibitor kit
CL0056	CDK inhibitor kit CDK inhibitor kit
CL0114	ERK inhibitor kit ERK inhibitor kit
CL0109	Ras inhibitor kit Ras inhibitor kit
CL0084	FGFR inhibitor kit FGFR inhibitor kit
CL0139	ROS inhibitor kit ROS inhibitor kit
CL0069	JAK inhibitor kit JAK inhibitor kit
CL0091	MEK inhibitor kit MEK inhibitor kit
CL0071	PDGFR inhibitor kit PDGFR inhibitor kit
CL0130	DUB inhibitor kit DUB inhibitor kit
CL0083	Dehydrogenase inhibitor kit Dehydrogenase inhibitor kit
CL0101	STAT inhibitor kit STAT inhibitor kit
CL0125	AChE inhibitor kit AChE inhibitor kit
CL0146	JNK inhibitor kit JNK inhibitor kit
CL0068	VEGFR inhibitor kit VEGFR inhibitor kit
CL0058	EGFR inhibitor kit EGFR inhibitor kit
CL0112	PKC inhibitor kit PKC inhibitor kit
CL0122	ACE inhibitor kit ACE inhibitor kit
CL0093	PARP inhibitor kit PARP inhibitor kit
CL0135	ROCK inhibitor kit ROCK inhibitor kit
CL0098	HER2 inhibitor kit HER2 inhibitor kit
CL0077	Reverse Transcriptase inhibitor kit Reverse Transcriptase inhibitor kit
CL0102	Akt inhibitor/activator kit Akt inhibitor/activator kit
CL0129	Aurora Kinase inhibitor kit Aurora Kinase inhibitor kit
CL0076	PPAR inhibitor/activator kit PPAR inhibitor/activator kit
CL0138	Carbonic Anhydrase inhibitor kit Carbonic Anhydrase inhibitor kit
CL0066	P450 inhibitor kit P450 inhibitor kit
CL0094	FLT3 inhibitor kit FLT3 inhibitor kit
CL0115	Proton Pump inhibitor kit Proton Pump inhibitor kit
CL0107	Src inhibitor/activator kit Src inhibitor/activator kit
CL0082	TRP Channel inhibitor kit TRP Channel inhibitor kit
CL0074	Microtubule/Tubulin inhibitor kit Microtubule/Tubulin inhibitor kit
CL0059	Dopamine Receptor inhibitor kit Dopamine Receptor inhibitor kit
CL0063	Cytoskeleton pathway inhibitor kit Cytoskeleton pathway inhibitor kit
CL0105	Sirtuin inhibitor/activator kit Sirtuin inhibitor/activator kit
CL0118	p38 inhibitor kit p38 inhibitor kit
CL0117	DPP4 inhibitor kit DPP4 inhibitor kit
CL0057	PI3K inhibitor kit PI3K inhibitor kit
CL0092	GSK-3 inhibitor kit GSK-3 inhibitor kit
CL0075	c-Kit inhibitor kit c-Kit inhibitor kit
CL0145	Casein Kinase inhibitor kit Casein Kinase inhibitor kit
CL0136	ATM/ATR inhibitor kit ATM/ATR inhibitor kit
CL0055	Potassium Channel inhibitor kit Potassium Channel inhibitor kit
CL0088	Angiotensin Receptor inhibitor kit Angiotensin Receptor inhibitor kit
CL0067	Sodium Channel inhibitor kit Sodium Channel inhibitor kit
CL0119	Histone Demethylase inhibitor kit Histone Demethylase inhibitor kit
CL0079	Adenosine Receptor inhibitor kit Adenosine Receptor inhibitor kit
CL0070	GABA Receptor inhibitor kit GABA Receptor inhibitor kit
CL0060	Estrogen Receptor inhibitor kit Estrogen Receptor inhibitor kit
CL0061	Histone Methyltransferase inhibitor kit Histone Methyltransferase inhibitor kit
CL0141	Notch pathway inhibitor kit Notch pathway inhibitor kit
CL0123	AMPK inhibitor/activator kit AMPK inhibitor/activator kit
CL0149	β-/γ-secretase inhibitor kit β-/γ-secretase inhibitor kit
CL0147	c-FMS inhibitor kit c-FMS inhibitor kit
CL0134	p53 inhibitor/reactivator kit p53 inhibitor/reactivator kit
CL0150	DNA Methyltransferase/Demethylase inhibitor kit DNA Methyltransferase/Demethylase inhibitor kit
CL0090	RNA Synthesis inhibitor/activator kit RNA Synthesis inhibitor/activator kit
CL0073	DNA synthesis inhibitor/activator kit DNA synthesis inhibitor/activator kit
CL0143	PKA/cAMP inhibitor/activator kit PKA/cAMP inhibitor/activator kit
CL0078	Glucocorticoid Receptor inhibitor/activator kit Glucocorticoid Receptor inhibitor/activator kit
CL0089	c-Met/HGFR inhibitor kit c-Met/HGFR inhibitor kit
CL0053	NF-κB pathway inhibitor kit NF-κB pathway inhibitor kit
CL0080	TGFβ signaling pathway inhibitor/activator kit TGFβ signaling pathway inhibitor/activator kit
CL0120	Bcr-Abl inhibitor/degrader kit Bcr-Abl inhibitor/degrader kit
CL0095	Hedgehog signaling pathway inhibitor/activator kit Hedgehog signaling pathway inhibitor/activator kit
CL0113	ER stress pathway inhibitor/inducer kit ER stress pathway inhibitor/inducer kit
CL0106	HIF/HIF-PH inhibitor/activator kit HIF/HIF-PH inhibitor/activator kit
CL0096	Wnt/β-catenin/PORCN inhibitor/activator kit Wnt/β-catenin/PORCN inhibitor/activator kit
CL0137	E1/E2/E3 Enzyme inhibitor kit E1/E2/E3 Enzyme inhibitor kit
C0047	RIPA Lysis Buffer (Weak) RIPA裂解液(弱)	Solution in bottle
C0046	RIPA Lysis Buffer (Middle) RIPA裂解液(中)	Solution in bottle
C0045	RIPA Lysis Buffer (Strong) RIPA裂解液(强)	Solution in bottle

TargetMol 试剂盒

磷酸酶抑制剂 Cocktail I (100× ddH2O)

Cat.No: C0002

磷酸酶抑制剂 Cocktail II (100× DMSO)

Cat.No: C0003

磷酸酶抑制剂 Cocktail III (2 Tubes, 100x)

Cat.No: C0004

蛋白酶抑制剂 Cocktail (EDTA-Free, 100× in DMSO)

Cat.No: C0001

去乙酰化酶抑制剂 Cocktail（100× in 70% DMSO）

Cat.No: C0048

PDE inhibitor kit

Cat.No: CL0064

BTK inhibitor kit

Cat.No: CL0140

HMGCR inhibitor kit

Cat.No: CL0128

SGLT inhibitor kit

Cat.No: CL0131

MMP inhibitor kit

Cat.No: CL0142

ALK inhibitor kit

Cat.No: CL0121

HDAC inhibitor kit

Cat.No: CL0052

Topoisomerase inhibitor kit

Cat.No: CL0062

Phosphatase inhibitor kit

Cat.No: CL0081

Raf inhibitor kit

Cat.No: CL0100

BET inhibitor kit

Cat.No: CL0072

NOS inhibitor kit

Cat.No: CL0127

HSP inhibitor kit

Cat.No: CL0085

DHFR inhibitor kit

Cat.No: CL0132

CXCR inhibitor kit

Cat.No: CL0133

mTOR inhibitor kit

Cat.No: CL0087

COX inhibitor kit

Cat.No: CL0045

MAO inhibitor kit

Cat.No: CL0116

CDK inhibitor kit

Cat.No: CL0056

ERK inhibitor kit

Cat.No: CL0114

Ras inhibitor kit

Cat.No: CL0109

FGFR inhibitor kit

Cat.No: CL0084

ROS inhibitor kit

Cat.No: CL0139

JAK inhibitor kit

Cat.No: CL0069

MEK inhibitor kit

Cat.No: CL0091

PDGFR inhibitor kit

Cat.No: CL0071

DUB inhibitor kit

Cat.No: CL0130

Dehydrogenase inhibitor kit

Cat.No: CL0083

STAT inhibitor kit

Cat.No: CL0101

AChE inhibitor kit

Cat.No: CL0125

JNK inhibitor kit

Cat.No: CL0146

VEGFR inhibitor kit

Cat.No: CL0068

EGFR inhibitor kit

Cat.No: CL0058

PKC inhibitor kit

Cat.No: CL0112

ACE inhibitor kit

Cat.No: CL0122

PARP inhibitor kit

Cat.No: CL0093

ROCK inhibitor kit

Cat.No: CL0135

HER2 inhibitor kit

Cat.No: CL0098

Reverse Transcriptase inhibitor kit

Cat.No: CL0077

Akt inhibitor/activator kit

Cat.No: CL0102

Aurora Kinase inhibitor kit

Cat.No: CL0129

PPAR inhibitor/activator kit

Cat.No: CL0076

Carbonic Anhydrase inhibitor kit

Cat.No: CL0138

P450 inhibitor kit

Cat.No: CL0066

FLT3 inhibitor kit

Cat.No: CL0094

Proton Pump inhibitor kit

Cat.No: CL0115

Src inhibitor/activator kit

Cat.No: CL0107

TRP Channel inhibitor kit

Cat.No: CL0082

Microtubule/Tubulin inhibitor kit

Cat.No: CL0074

Dopamine Receptor inhibitor kit

Cat.No: CL0059

Cytoskeleton pathway inhibitor kit

Cat.No: CL0063

Sirtuin inhibitor/activator kit

Cat.No: CL0105

p38 inhibitor kit

Cat.No: CL0118

DPP4 inhibitor kit

Cat.No: CL0117

PI3K inhibitor kit

Cat.No: CL0057

GSK-3 inhibitor kit

Cat.No: CL0092

c-Kit inhibitor kit

Cat.No: CL0075

Casein Kinase inhibitor kit

Cat.No: CL0145

ATM/ATR inhibitor kit

Cat.No: CL0136

Potassium Channel inhibitor kit

Cat.No: CL0055

Angiotensin Receptor inhibitor kit

Cat.No: CL0088

Sodium Channel inhibitor kit

Cat.No: CL0067

Histone Demethylase inhibitor kit

Cat.No: CL0119

Adenosine Receptor inhibitor kit

Cat.No: CL0079

GABA Receptor inhibitor kit

Cat.No: CL0070

Estrogen Receptor inhibitor kit

Cat.No: CL0060

Histone Methyltransferase inhibitor kit

Cat.No: CL0061

Notch pathway inhibitor kit

Cat.No: CL0141

AMPK inhibitor/activator kit

Cat.No: CL0123

β-/γ-secretase inhibitor kit

Cat.No: CL0149

c-FMS inhibitor kit

Cat.No: CL0147

p53 inhibitor/reactivator kit

Cat.No: CL0134

DNA Methyltransferase/Demethylase inhibitor kit

Cat.No: CL0150

RNA Synthesis inhibitor/activator kit

Cat.No: CL0090

DNA synthesis inhibitor/activator kit

Cat.No: CL0073

PKA/cAMP inhibitor/activator kit

Cat.No: CL0143

Glucocorticoid Receptor inhibitor/activator kit

Cat.No: CL0078

c-Met/HGFR inhibitor kit

Cat.No: CL0089

NF-κB pathway inhibitor kit

Cat.No: CL0053

TGFβ signaling pathway inhibitor/activator kit

Cat.No: CL0080

Bcr-Abl inhibitor/degrader kit

Cat.No: CL0120

Hedgehog signaling pathway inhibitor/activator kit

Cat.No: CL0095

ER stress pathway inhibitor/inducer kit

Cat.No: CL0113

HIF/HIF-PH inhibitor/activator kit

Cat.No: CL0106

Wnt/β-catenin/PORCN inhibitor/activator kit

Cat.No: CL0096

E1/E2/E3 Enzyme inhibitor kit

Cat.No: CL0137

RIPA裂解液(弱)

Cat.No: C0047

RIPA裂解液(中)

Cat.No: C0046

RIPA裂解液(强)

Cat.No: C0045

Cat. No.	Product Name	Target	Signaling Pathways
T10876	CPA inhibitor Carboxypeptidase inhibitor	Carboxypeptidase	Proteases/Proteasome
	CPA inhibitor (Carboxypeptidase inhibitor) 是一种有效的羧肽酶 A (CPA) 抑制剂，Ki 值为 0.32 μM。
T5451	Eph inhibitor 2 Ehp-inhibitor-1	Ephrin Receptor	Tyrosine Kinase/Adaptors
	Eph inhibitor 2 是一种 Eph 家族酪氨酸激酶抑制剂。
T4338	USP7/USP47 inhibitor USP7/47 inhibitor-1	DUB	Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Ubiquitination
	USP7/USP47 inhibitor (USP7/47 inhibitor-1) 是一种选择性泛素特异性蛋白酶 7/47 抑制剂，EC50值分别为 0.42 μM 和 1.0 μM。
T1804	HPGDS inhibitor 1 HPGDS-inhibitor-1	PGE Synthase	Immunology/Inflammation
	HPGDS inhibitor 1 是口服具有活性的HPGDS 选择性抑制剂，在酶和细胞分析中的IC50值分别为 0.6 nM 和 32 nM，但对 L-PGDS、mPGES、COX-1、COX-2 、5-LOX 无抑制作用。
T8766	GOT1 inhibitor-1 GOT1 inhibitor 2c	Others	Others
	GOT1 inhibitor-1 (GOT1 inhibitor 2c) 是一种新型的、非共价的谷氨酸草酰乙酸转氨酶 1 (GOT1) 抑制剂(IC50:8.2 uM)，是一种戊酸衍生物。它可用于以及胰腺导管腺癌 (PDAC) 。
T38683	SCD1 inhibitor-3 SCD1-IN-3,SCD1 inhibitor-3,SCD1 inhibitor 17a	Dehydrogenase	Metabolism
	SCD1 inhibitor-3 (ML-270) 是一种高效、口服的化合物，可以抑制SCD1，且安全性极高。 SCD1 inhibitor-3 显示出在代谢疾病(包括肥胖、二型糖尿病和血脂异常，以及痤疮和癌症等各种皮肤病)方面的巨大研究潜力。
T5817	PKC-theta inhibitor hcl PKC-theta inhibitor	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKC-theta inhibitor hcl 是一种选择性 PKC-θ 抑制剂 (IC50:12 nM)。
T5524	Aurora kinase inhibitor-3 Aurora Kinase Inhibitor III	Aurora Kinase	Cell Cycle/Checkpoint; Chromatin/Epigenetic
	Aurora kinase inhibitor-3 (Aurora Kinase Inhibitor III) 是一种有效的，选择性 Aurora A 激酶抑制剂，IC50为 42 nM。
T2350	MALT1 inhibitor MI-2 MALT1 inhibitor,MI 2,MI 2 (MALT1 inhibitor)	MALT	Immunology/Inflammation
	MI 2 (MALT1 inhibitor) 是一种MALT1抑制剂 (IC50=5.84 μM)，对动物无毒性。它能够直接与 MALT1 结合，不可逆地抑制蛋白酶功能，并伴有 NF-κB 报告子活性抑制、c-REL 核定位抑制和 NF-κB 靶基因下调。
T2074	Raf inhibitor 1 B-Raf inhibitor 1	Raf	MAPK
	Raf inhibitor 1 (B-Raf inhibitor 1)是Raf 激酶抑制剂，对B-RafWT、B-RafV600E 和 C-Raf 的Ki 分别为 1、1 和 0.3 nM。
T3042	JAK2 Inhibitor V JAK2 Inhibitor V Z3,Z3	JAK	Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells
	JAK2 Inhibitor V (JAK2 Inhibitor V Z3) 是一种新型的 Jak2 特异性抑制剂，以剂量依赖性方式抑制 Jak2-V617F 和 Jak2-WT 自磷酸化。
T3593	Src Inhibitor 1 Src Kinase Inhibitor 1,Src-l1	Src	Angiogenesis; Tyrosine Kinase/Adaptors
	Src Inhibitor 1 (Src Kinase Inhibitor 1) 是一种选择性的、高效的、ATP-竞争性的双位点 Src 酪氨酸激酶抑制剂，能够抑制 Src (IC50:44 nM) 和 Lck (IC50:88 nM)。
T3189	B7/CD28 interaction inhibitor 1 CTLA-4 inhibitor	Others	Others
	B7/CD28 interaction inhibitor 1 (CTLA-4 inhibitor) 是B7.1-CD28相互作用抑制剂(IC50:50 nM)。
T4191	Multi-kinase inhibitor 1 Multi-kinase inhibitor I	Others; Bcr-Abl; PDGFR; c-Kit	Angiogenesis; Cytoskeletal Signaling; Others; Tyrosine Kinase/Adaptors
	Multi-kinase inhibitor 1 (Multi-kinase inhibitor I) 是多激酶抑制剂。它有用于导致与酪氨酸激酶活性异常或失控有关的疾病或失调的潜力，特别是与c-Kit，PDGF-R，Bcr-abl 活性相关的疾病。
T6335	Tie2 kinase inhibitor 1 Tie2 kinase inhibitor	Tie-2	Tyrosine Kinase/Adaptors
	Tie2 kinase inhibitor 1 (Tie2 kinase inhibitor) 是Tie2激酶选择性抑制剂9IC50:250 nM)，具有抗癌作用。
T4391	Syk Inhibitor II dihydrochloride Syk Inhibitor II (hydrochloride)	Others; Tyrosine Kinases; Syk; PKC; BTK	Angiogenesis; Chromatin/Epigenetic; Cytoskeletal Signaling; Others; Tyrosine Kinase/Adaptors
	Syk Inhibitor II (hydrochloride) 是一种非受体酪氨酸激酶，磷酸化后，它与 FcRγ 链的基于免疫受体酪氨酸的激活基序结合，并介导与血小板功能和炎症相关的下游信号传导。 Syk inhibitor II 是一种可渗透细胞的嘧啶-甲酰胺化合物，以 ATP 竞争性方式选择性和可逆地阻断 Syk (IC50 = 41 nM)。它对 PKCε、PKCβII、ZAP-70、Btk 和 Itk 的效力要低得多（IC50s 分别为5.1、11、11.2、15.5 和 22.6 μM）。
T10678	Carboxypeptidase G2 (CPG2) Inhibitor CPG2 Inhibitor,Carboxypeptidase G2 Inhibitor	Carboxypeptidase	Proteases/Proteasome
	Carboxypeptidase G2 (CPG2) Inhibitor (CPG2 Inhibitor) 是新型的羧肽酶 G2(CPG2)抑制剂，显示出抗癌活性。
T2457	IRAK-1-4 Inhibitor I IRAK-1/4 Inhibitor I,IRAK-1/4 Inhibitor	IRAK	Immunology/Inflammation; NF-κB
	IRAK-1-4 Inhibitor I 是一种IRAK1/4双重抑制剂，其IC50分别为 0.2 μM 和 0.3 μM。
T24141	HIV-1 Inhibitor 18A HIV-1 Inhibitor-18A	HIV Protease	Microbiology/Virology; Proteases/Proteasome
	HIV-1 Inhibitor 18A (HIV-1 Inhibitor-18A) 特异性抑制多种 HIV-1 分离株的进入。
T67767	HIF-1 inhibitor-4 HIF-1 inhibitor-4	HIF	Angiogenesis; Chromatin/Epigenetic
	HIF-1 inhibitor-4 (HIF-1 inhibitor-4) 是一种 HIF-1 抑制剂 (IC50: 560 nM)。HIF-1 inhibitor-4 减少 HIF-1α 蛋白水平，但不影响 mRNA 水平。
T4167	Raf inhibitor 1 dihydrochloride B-Raf inhibitor 1 dihydrochloride	Raf	MAPK
	Raf inhibitor 1 dihydrochloride (B-Raf inhibitor 1 dihydrochloride) 是 Raf 激酶抑制剂，对 B-RafWT、B-RafV600E 和 C-Raf 的Ki 分别为 1、1 和 0.3 nM。
T9040	Aurora kinase inhibitor-2 IUN-70219,Aurora Kinase Inhibitor II	Aurora Kinase	Cell Cycle/Checkpoint; Chromatin/Epigenetic
	Aurora kinase inhibitor-2 (IUN-70219) 是一种可渗透细胞的苯胺喹唑啉，可抑制极光激酶的活性，对Aurora A 和Aurora B 的IC50分别为 390 nM 和 240 nM。
T35827L	PKCε Inhibitor Peptide acetate PKCε Inhibitor Peptide acetate(182683-50-7 Free base)	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKCε Inhibitor Peptide acetate 是一种特异性 PKCε 抑制剂，含有其特定受体活化 C 激酶 (RACK) 的位点。 PKCε Inhibitor Peptide acetate 抑制 PKCε 的转运，但不抑制 αPKC，βPKC 和 δPKC 的转运。
T4491	LMPTP INHIBITOR 1 hydrochloride LMPTP INHIBITOR 1 hydrochloride (1908414-82-3(free base))	Phosphatase	Metabolism
	LMPTP INHIBITOR 1 hydrochloride 是一种高选择性的低分子量蛋白酪氨酸磷酸酶 (LMPTP) 抑制剂。LMPTP INHIBITOR 1 (hydrochloride) 能够抑制 LMPTP-A 的活性，IC50值为 0.8 μM。
T21954	EGFR/ErbB-2/ErbB-4 inhibitor-2 EGFR/ErbB2 Inhibitor	EGFR	Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
	EGFR/ErbB-2/ErbB-4 inhibitor-2 (EGFR/ErbB2 Inhibitor) 是EGFR 和ErbB 的抑制剂，对EGFR、ErbB2 和 ErbB4 的IC50分别为 0.017、0.08 和 1.91 μM。
TP2008L	Lyn peptide inhibitor acetate Lyn peptide inhibitor acetate(222018-18-0 free base)	IL Receptor	Immunology/Inflammation
	Lyn peptide inhibitor acetate(222018-18-0 free base) 是一种有效的细胞渗透性 Lyn 偶联 IL-5 受体信号通路抑制剂，同时保持其他信号完整。它阻断 Lyn 活化并抑制 Lyn 酪氨酸激酶与 IL-3/GM-CSF/IL-5 受体的 βc 亚基的结合。它可用于哮喘、过敏和其他嗜酸性粒细胞疾病的研究。
T17157	TRAF-STOP inhibitor 6877002 CD40-TRAF6 inhibitor	NF-κB	NF-κB
	TRAF-STOP inhibitor 6877002 (CD40-TRAF6 inhibitor)是一种 CD40-TRAF6 相互作用的选择性抑制剂，可以抑制 RAW 细胞中 NF-κB 活化。TRAF-STOP 6877002 可阻止小鼠动脉粥样硬化的恶化，减少白细胞募集和巨噬细胞的活化，减少动脉粥样硬化斑块中的巨噬细胞增殖。
T9178	(E/Z)-GSK-3β inhibitor 1 GSK-3β inhibitor 1	GSK-3	PI3K/Akt/mTOR signaling; Stem Cells
	(E/Z)-GSK-3β inhibitor 1 是 (E)-GSK-3β inhibitor 1 和 (Z)-GSK-3β inhibitor 1 的消旋体。它是一种糖原合成酶激酶 3β (GSK-3β)的抑制剂，可其对 GSK-3β 的 IC50=4.9 nM，用于糖尿病的研究。
T36933	Cdk2 Inhibitor II Cdk2 Inhibitor II,CDK2-IN-3	CDK	Cell Cycle/Checkpoint
	Cdk2 Inhibitor II 是一种具有选择性和有效性的 CDK2 抑制剂，50 为 60 nM。
T10927	Cyt-PTPε Inhibitor-1 Cyt-PTP\|A Inhibitor-1	Phosphatase; Src	Angiogenesis; Metabolism; Tyrosine Kinase/Adaptors
	Cyt-PTPε Inhibitor-1 (A Inhibitor-1) 是胞质蛋白酪氨酸磷酸酶 ε 的抑制剂。 Cyt-PTPε Inhibitor-1 阻断 c-Src 的去磷酸化并表现出抗破骨活性。
T36675	ERK Inhibitor
	ERK inhibitor is a cell-permeable inhibitor that binds ERK2 near its docking domain (KD = 5 μM). This prevents its interaction with protein substrates without inhibiting catalytic activity. ERK inhibitor blocks ERK-specific phosphorylation of ribosomal S6 kinase-1 and ternary complex factor Elk-1 but does not affect ERK1/2 phosphorylation by MEK1/2. Presumably through its effects on ERK, ERK inhibitor completely prevents proliferation of HeLa cells (IC50 = 15-20 μM), A549 lung carcinoma cells (I...
T10865L	Cot inhibitor-1 hydrochloride Cot inhibitor-1 hydrochloride(915365-57-0 Free base)	TNF; MAPK	Apoptosis; MAPK
	Cot inhibitor-1 hydrochloride 是肿瘤进展位点 2 激酶 (IC50 = 28 nM) 的抑制剂，可抑制人全血中 TNF-α 的产生 (IC50 = 5.7 nM)。
T22081	FBPase-1 inhibitor-1 Fructose 1,6-bisphosphatase-1 Inhibitor	Others	Others
	FBPase-1 inhibitor-1 (Fructose 1,6-bisphosphatase-1 Inhibitor) 是一种fructose-1,6-bisphosphatase (FBPase-1)的变构抑制剂。
T22136	PRL-3 Inhibitor I PRL-3 Inhibitor,BR-1	Phosphatase; Others	Metabolism; Others
	PRL-3 Inhibitor I (BR-1) 是 PRL-3 抑制剂，IC50=0.9 μM。它在细胞检测中显示降低侵袭性。
TP1523	PKG inhibitor peptide TFA (82801-73-8 free base) PKG inhibitor peptide TFA	PKA	Tyrosine Kinase/Adaptors
	PKG inhibitor peptide TFA (82801-73-8 free base) 是 ATP 竞争性 cGMP 依赖性蛋白激酶 (PKG) 的抑制剂。
T10599	BRAF inhibitor	Raf	MAPK
	BRAF inhibitor 是B-Raf 抑制剂。
T2649	Menin-MLL inhibitor MI-2 Menin-MLL Inhibitor,MI2,MI-2,Menin-MLL inhibitor 2,MI 2	Apoptosis; Epigenetic Reader Domain; Histone Methyltransferase	Apoptosis; Chromatin/Epigenetic
	Menin-MLL inhibitor MI-2 (MI2) 抑制Menin-MLL 相互作用，IC50为 446±28 nM。
T11184	EML4-ALK kinase inhibitor 1 EML4 ALK kinase inhibitor 1,EML4-ALK kinase inhibitor 1	ALK	Angiogenesis; Tyrosine Kinase/Adaptors
	EML4-ALK kinase inhibitor 1 (EML4 ALK kinase inhibitor 1) 是有效的、具有口服活性的类棘皮细胞微管相关蛋白4-间变性淋巴瘤激酶 (EML4-ALK) 的抑制剂，其 IC50 值为 1 nM。
TP1890L1	MLCK inhibitor peptide 18 acetate MLCK inhibitor peptide 18 acetate(224579-74-2 free base)	Serine/threonin kinase	Cell Cycle/Checkpoint; Metabolism
	MLCK inhibitor peptide 18 acetate(224579-74-2 free base) 是肌球蛋白轻链激酶的选择性竞争性抑制剂 (IC50 = 50 nM)。显示出比 CaM 激酶 II 高 4000 倍的选择性，并且不抑制 PKA。细胞可渗透。
T7541	PTP inhibitor 1 PTP Inhibitor II,alpha-溴-4-甲氧基苯乙酮	Phosphatase	Metabolism
	PTP inhibitor 1 是蛋白酪氨酸磷酸酶 (PTP) 抑制剂，具有抗血管生成作用。
TP1015	NFAT Inhibitor VIVIT peptide	Others	Others
	NFAT Inhibitor (VIVIT peptide) 是NFAT 的细胞渗透性肽抑制剂，能够选择性抑制钙调磷酸酶介导的NFAT 脱磷酸作用。
T2159	CaMKP Inhibitor	CaMK	Neuroscience
	CaMKP Inhibitor 可以抑制 CaMKP。
T60108	PDGFR Tyrosine Kinase Inhibitor III PDGF Receptor Tyrosine Kinase Inhibitor III	PDGFR	Angiogenesis; Tyrosine Kinase/Adaptors
	PDGFR Tyrosine Kinase Inhibitor III (PDGF Receptor Tyrosine Kinase Inhibitor III) (PDGF Receptor Tyrosine Kinase Inhibitor III)是一种多激酶抑制剂，可抑制 PDGFR、EGFR、FGFR、PKA 和 PKC 等。PDGFR Tyrosine Kinase Inhibitor III 可用于肌萎缩侧索硬化症的研究。
T12502	PLpro inhibitor 5-(乙酰氨基)-2-甲基-N-[(1R)-1-(1-萘基)乙基]苯甲酰胺	SARS-CoV	Microbiology/Virology
	PLpro inhibitor 是一种木瓜蛋白酶抑制剂，IC50为 2.6 µM，能抑制 SARS-CoV-2 PLpro。
T60119	SOD1-Derlin-1 inhibitor-1 SOD1-Derlin-1 Inhibitor 56-20	Others	Others
	SOD1-Derlin-1 inhibitor-1 (SOD1-Derlin-1 Inhibitor 56-20) (compound 56-20) 是 SOD1-Derlin-1相互作用的抑制剂。SOD1-Derlin-1 inhibitor-1 抑制 SOD1G93A-Derlin-1 复合物，IC50值为 7.11 μM。SOD1-Derlin-1 inhibitor-1 可用于肌萎缩性侧索硬化症的研究。
T10276L	AKT Kinase Inhibitor HCl AKT Kinase Inhibitor HCl(842148-40-7 Free base)	Akt	Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
	AKT Kinase Inhibitor HCl 是一种 Akt 抑制剂，具有抗肿瘤活性。
T69757	PDDC inhibitor
	PDDC is the first nSMase2 inhibitor that possesses both favorable pharmacodynamics and pharmacokinetic (PK) parameters, including substantial oral bioavailability, brain penetration, and significant inhibition of exosome release from the brain in vivo.
T5452	Ehp-inhibitor-2	Ephrin Receptor	Tyrosine Kinase/Adaptors
	Ehp-inhibitor-2 是一种靶向 Eph 受体的 Eph 家族酪氨酸激酶抑制剂。
T36802L	Bisubstrate Inhibitor 78 HCl Bisubstrate Inhibitor 78 HCl(2368247-39-4 Free base)	Others	Others
	Bisubstrate Inhibitor 78 HCl 是一种 NNMT 抑制剂（IC50 = 1.41 μM），具有潜在的抗癌活性，在 100μM 时抑制HSC-2口腔癌细胞增殖。
T69730	F092 inhibitor
	F092 inhibitor, also called Prostaglandin D synthase (hematopoietic-type) inhibitor F092, is an inhibitor of hematopoietic-type prostaglandin D synthase (H-PGDS).

化合物

CPA inhibitor

Cat.No: T10876

Synonym: Carboxypeptidase inhibitor

Target: Carboxypeptidase

Eph inhibitor 2

Cat.No: T5451

Synonym: Ehp-inhibitor-1

Target: Ephrin Receptor

USP7/USP47 inhibitor

Cat.No: T4338

Synonym: USP7/47 inhibitor-1

Target: DUB

HPGDS inhibitor 1

Cat.No: T1804

Synonym: HPGDS-inhibitor-1

Target: PGE Synthase

GOT1 inhibitor-1

Cat.No: T8766

Synonym: GOT1 inhibitor 2c

Target: Others

SCD1 inhibitor-3

Cat.No: T38683

Synonym: SCD1-IN-3,SCD1 inhibitor-3,SCD1 inhibitor 17a

Target: Dehydrogenase

PKC-theta inhibitor hcl

Cat.No: T5817

Synonym: PKC-theta inhibitor

Target: PKC

Aurora kinase inhibitor-3

Cat.No: T5524

Synonym: Aurora Kinase Inhibitor III

Target: Aurora Kinase

MALT1 inhibitor MI-2

Cat.No: T2350

Synonym: MALT1 inhibitor,MI 2,MI 2 (MALT1 inhibitor)

Target: MALT

Raf inhibitor 1

Cat.No: T2074

Synonym: B-Raf inhibitor 1

Target: Raf

JAK2 Inhibitor V

Cat.No: T3042

Synonym: JAK2 Inhibitor V Z3,Z3

Target: JAK

Src Inhibitor 1

Cat.No: T3593

Synonym: Src Kinase Inhibitor 1,Src-l1

Target: Src

B7/CD28 interaction inhibitor 1

Cat.No: T3189

Synonym: CTLA-4 inhibitor

Target: Others

Multi-kinase inhibitor 1

Cat.No: T4191

Synonym: Multi-kinase inhibitor I

Target: Others, Bcr-Abl, PDGFR, c-Kit

Tie2 kinase inhibitor 1

Cat.No: T6335

Synonym: Tie2 kinase inhibitor

Target: Tie-2

Syk Inhibitor II dihydrochloride

Cat.No: T4391

Synonym: Syk Inhibitor II (hydrochloride)

Target: Others, Tyrosine Kinases, Syk, PKC, BTK

Carboxypeptidase G2 (CPG2) Inhibitor

Cat.No: T10678

Synonym: CPG2 Inhibitor,Carboxypeptidase G2 Inhibitor

Target: Carboxypeptidase

IRAK-1-4 Inhibitor I

Cat.No: T2457

Synonym: IRAK-1/4 Inhibitor I,IRAK-1/4 Inhibitor

Target: IRAK

HIV-1 Inhibitor 18A

Cat.No: T24141

Synonym: HIV-1 Inhibitor-18A

Target: HIV Protease

HIF-1 inhibitor-4

Cat.No: T67767

Synonym: HIF-1 inhibitor-4

Target: HIF

Raf inhibitor 1 dihydrochloride

Cat.No: T4167

Synonym: B-Raf inhibitor 1 dihydrochloride

Target: Raf

Aurora kinase inhibitor-2

Cat.No: T9040

Synonym: IUN-70219,Aurora Kinase Inhibitor II

Target: Aurora Kinase

PKCε Inhibitor Peptide acetate

Cat.No: T35827L

Synonym: PKCε Inhibitor Peptide acetate(182683-50-7 Free base)

Target: PKC

LMPTP INHIBITOR 1 hydrochloride

Cat.No: T4491

Synonym: LMPTP INHIBITOR 1 hydrochloride (1908414-82-3(free base))

Target: Phosphatase

EGFR/ErbB-2/ErbB-4 inhibitor-2

Cat.No: T21954

Synonym: EGFR/ErbB2 Inhibitor

Target: EGFR

Lyn peptide inhibitor acetate

Cat.No: TP2008L

Synonym: Lyn peptide inhibitor acetate(222018-18-0 free base)

Target: IL Receptor

TRAF-STOP inhibitor 6877002

Cat.No: T17157

Synonym: CD40-TRAF6 inhibitor

Target: NF-κB

(E/Z)-GSK-3β inhibitor 1

Cat.No: T9178

Synonym: GSK-3β inhibitor 1

Target: GSK-3

Cdk2 Inhibitor II

Cat.No: T36933

Synonym: Cdk2 Inhibitor II,CDK2-IN-3

Target: CDK

Cyt-PTPε Inhibitor-1

Cat.No: T10927

Synonym: Cyt-PTP|A Inhibitor-1

Target: Phosphatase, Src

ERK Inhibitor

Cat.No: T36675

Cot inhibitor-1 hydrochloride

Cat.No: T10865L

Synonym: Cot inhibitor-1 hydrochloride(915365-57-0 Free base)

Target: TNF, MAPK

FBPase-1 inhibitor-1

Cat.No: T22081

Synonym: Fructose 1,6-bisphosphatase-1 Inhibitor

Target: Others

PRL-3 Inhibitor I

Cat.No: T22136

Synonym: PRL-3 Inhibitor,BR-1

Target: Phosphatase, Others

PKG inhibitor peptide TFA (82801-73-8 free base)

Cat.No: TP1523

Synonym: PKG inhibitor peptide TFA

Target: PKA

BRAF inhibitor

Cat.No: T10599

Target: Raf

Menin-MLL inhibitor MI-2

Cat.No: T2649

Synonym: Menin-MLL Inhibitor,MI2,MI-2,Menin-MLL inhibitor 2,MI 2

Target: Apoptosis, Epigenetic Reader Domain, Histone Methyltransferase

EML4-ALK kinase inhibitor 1

Cat.No: T11184

Synonym: EML4 ALK kinase inhibitor 1,EML4-ALK kinase inhibitor 1

Target: ALK

MLCK inhibitor peptide 18 acetate

Cat.No: TP1890L1

Synonym: MLCK inhibitor peptide 18 acetate(224579-74-2 free base)

Target: Serine/threonin kinase

PTP inhibitor 1

Cat.No: T7541

Synonym: PTP Inhibitor II,alpha-溴-4-甲氧基苯乙酮

Target: Phosphatase

NFAT Inhibitor

Cat.No: TP1015

Synonym: VIVIT peptide

Target: Others

CaMKP Inhibitor

Cat.No: T2159

Target: CaMK

PDGFR Tyrosine Kinase Inhibitor III

Cat.No: T60108

Synonym: PDGF Receptor Tyrosine Kinase Inhibitor III

Target: PDGFR

PLpro inhibitor

Cat.No: T12502

Synonym: 5-(乙酰氨基)-2-甲基-N-[(1R)-1-(1-萘基)乙基]苯甲酰胺

Target: SARS-CoV

SOD1-Derlin-1 inhibitor-1

Cat.No: T60119

Synonym: SOD1-Derlin-1 Inhibitor 56-20

Target: Others

AKT Kinase Inhibitor HCl

Cat.No: T10276L

Synonym: AKT Kinase Inhibitor HCl(842148-40-7 Free base)

Target: Akt

PDDC inhibitor

Cat.No: T69757

Ehp-inhibitor-2

Cat.No: T5452

Target: Ephrin Receptor

Bisubstrate Inhibitor 78 HCl

Cat.No: T36802L

Synonym: Bisubstrate Inhibitor 78 HCl(2368247-39-4 Free base)

Target: Others

F092 inhibitor

Cat.No: T69730

Cat. No.	Product Name	Target	Signaling Pathways
T3384	Wedelolactone 蟛蜞菊内酯,IKK Inhibitor II	Apoptosis; NF-κB; Lipoxygenase; Caspase	Apoptosis; Metabolism; NF-κB; Proteases/Proteasome
	Wedelolactone (IKK Inhibitor II) 是来自旱莲草的一种天然产物，通过阻断 IκBα 的磷酸化和降解来抑制细胞中 NF-κB 介导的基因转录，具有抗癌，抗炎和抗氧化活性。
T14961	Chrysene 䓛,屈	Others	Others
	Chrysene 是高分子量 (HMW) 多环芳烃，有极强的顽固性和致癌性。
T5813	BYAKANGELICIN	Reductase	Endocrinology/Hormones; Metabolism
	Byakangelicin 是发现于当归根中的一种活性化合物，可作为调节剂，改善各种活性化合物 (Umb，Cur 和 Dox) 的脑积累，增强研究效果。它提高所有PXR 靶基因 (如MDR1) 的表达，并广泛的诱导药物-药物相互作用。它可抑制性激素的作用，可能会增加内源激素的分解代谢。
T3817	Darutigenol	Others	Others
	Darutigenol 是一种戊二萜，从Siegesbecikia orientalis L.中分离得到。
T4953	Neotuberostemonine	NOS	Immunology/Inflammation
	Neotuberostemonine 是一种结核分枝杆菌根中主要的止咳生物碱，能够阻碍巨噬细胞的募集和活化，从而减轻博来霉素 (Bleomycin) 诱导的肺纤维化。
T3928	Neoliquiritin	Others	Others
	Neoliquiritin 是从甘草 Glycyrrhiza uralensis 分离得到，具有抗炎作用。它可能具有细胞毒性和肿瘤特异性。
TN2058	Persicogenin	Anti-infection	Microbiology/Virology
	Persicogenin 是分离自 Rhus retinorrhoea 中，具有抗癌作用。
T6S1049	Wilforine	ATPase	Membrane transporter/Ion channel
	Wilforine 是一倍半萜吡啶化合物，T. wilfordii 植物中的重要生物活性化合物，可有效治疗特发性肺纤维化。它具有抗炎和杀虫活性。
T3S2027	Rubusoside	Others	Others
	Rubusoside 是天然的增溶剂及甜味剂，具有良好的抗血管新生和抗过敏药的特性。
TN1816	Kadsurin	Antioxidant	oxidation-reduction
	Kadsurin 是一种提取自异形南五味子茎中的天然产物，能够显著降低小鼠肝脏中CCL4诱导的脂质过氧化产物（例如TBA-RS、共轭二烯和荧光产物）。
T13693	Fibrin	Others	Others
	Fibrin, the primary constituent of blood clots, is an insoluble protein essential for coagulation. Isolated from bovine blood, this protein is notably synthesized in response to bleeding.
T19231	Cellulase	Others	Others
	Cellulase 是一种能够催化纤维素和其他碳水化合物水解的酶。
T5S0661	Koumine	Others	Others
	Koumine 是一种从钩吻中得到的生物碱，具有高效抗肿瘤活性，在肿瘤细胞中能够提高 Bax/Bcl-2 的蛋白比例和 caspase-3 的表达。在类风湿性关节炎动物模型中，它能够预防关节炎的发展。它具有抗焦虑、抗应激、抗银屑病作用，也可用于缓解疼痛的研究。
T8161	Vicine	Others	Others
	Vicine 是一种主要存在于蚕豆中的生物碱糖苷，对人体有毒，可引起溶血性贫血。
TN1640	Fabiatrin	Others	Others
	Fabiatrin 是从 Przewalskia tangutica 的正丁醇提取物中分离和鉴定的天然产物。
T6S1657	Paeonolide	Others	Others
	Paeonolide 是一种广泛存在于 Paeonia 属植物根中的植物糖苷，含有一个非还原性末端 α-1-阿拉伯吡喃糖苷。
T6S0234	Toosendanin	Others	Others
	Toosendanin 是一种从杜鹃花果实皮中提取的三萜，具有杀虫和抗炎活性，可用于研究缓解疼痛。
T7033	Rosmanol	Antioxidant; COX	Immunology/Inflammation; Neuroscience; oxidation-reduction
	Rosmanol 能够显著抑制脂多糖诱导的 INOS、COX-2 的表达，抑制低密度脂蛋白的氧化，并具有抗炎作用。
T3A2414	Manninotriose	Others	Others
	Manninotriose 是小野芝麻（芝麻属，唇形科）主要的碳水化合物，参与RFO代谢并可能发挥重要作用
TN1081	Hirsuteine	Dopamine Receptor	GPCR/G Protein; Neuroscience
	Hirsuteine 是提取自钩藤属植物中的吲哚生物碱。它可阻断离子渗透通过烟碱受体通道复合物，非竞争性地拮抗烟碱介导的多巴胺释放。
TJS0851	Plantagoside	Others	Others
	Plantagoside 是α-mannosidase 的非竞争性特异性抑制剂(IC50:5 μM)，分离自Plantago asiatica 种子中。
TWS1563	Incensole	Others	Others
	Incensole 是一种 14-membered 二萜类化合物，分离自烯属植物的香精油和乳香树脂中。它能够激活脑中离子通道，并可以缓解焦虑或抑郁，从而显示出抗炎和抗抑郁的特性。
T6S1676	Cimigenoside	Others	Others
	Cimigenoside 是升麻属中的一种成分。
T5777	Phaseoloidin	Others	Others
	Phaseoloidin 是来自烟草细毛虫的高纯酸苷，有助于植物抵抗鳞翅目草食动物。它能够抑制Manduca sexta 和Spodoptera littoralis 的幼虫生长。它具有抗补体特性。
T8208	androsin	Others	Others
	Androsin 分离于印度胡黄连中，具有抗哮喘作用。
TN1982	Neoglycyrol	Others	Others
	Neoglycyrol 是分离自甘草的根中的化合物。它是由传统专利药通脉养心丸中筛选得到，具有潜在心肌保护作用。
TN1453	Bruceantinol	Anti-infection	Microbiology/Virology
	Bruceantinol 是一种quassinol 化合物，分离自Brucea javanica 的 CH3OH 提取物。它能够将系统性寄主植物中灭活。有效的抑制浓度为 10 μM。
T3931	Isobavachin	Others	Others
	Isobavachin 是一种分离自Psoralea morisiana 中的抗氧化剂，在A 环的8号位置有一个prenyl 基团，具有潜在的促进神经元的分化和其蛋白异戊烯化作用。
T19431	Moluccanin	Others	Others
	Moluccanin 是来自 Aleurites moluccana 的香豆素类。
T3873	griffonilide	Others	Others
	Griffonilide 是一种提取自Semiaquilegia adoxoides 根中的丁烯内酯类化合物，常与紫草甙一起出现。它是一种传统抗癌药草。
T14291	Anisindione	Others	Others
	Anisindione 是合成的抗凝血剂，对活性促凝因子II，VII，IX 和X 的形成具有抑制作用。
T8077	Dihydrojasmone	Others	Others
	Dihydrojasmone 是一种重要的香料成分，是佛手柑油的成分。
T5S1331	Herbacetin	c-Met/HGFR; Akt	Cytoskeletal Signaling; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors
	Herbacetin 是一种亚麻籽中的天然类黄酮，具有多种药理活性，如抗氧化、抗炎、抗癌作用。它是鸟氨酸脱羧酶Ornithine decarboxylase (ODC)变构抑制剂，能够直接与 ODC 上的 Asp44，Asp243 和 Glu384 结合。其中鸟氨酸脱羧酶是多胺生物合成中的限速酶。
TN6723	Lactiflorin	Others	Others
	Lactiflorin 是一种具有肾脏保护作用的单萜苷。
TN1983	Neoisoastilbin	IL Receptor; TNF; NO Synthase	Apoptosis; Immunology/Inflammation
	Neoisoastilbin 具有抗炎、抗氧化、抗尿酸过多等生物特性。
T2O2770	Agarotetrol	Others	Others
	Agarotetrol 是一种色酮衍生物，从沉香中分离得到。
TN1984	Neoisoliquiritin	Others	Others
	Neoisoliquiritin 是一种提取自甘草中的活性物质。
T6S0525	Farrerol	ERK; p38 MAPK; Akt	Cytoskeletal Signaling; MAPK; PI3K/Akt/mTOR signaling
	Farrerol 是一种杜鹃花的生物活性成分，具有抗氧化、抗肿瘤、抗炎、神经保护和肝保护等多种功能。
TN1075	Adynerin	Others	Others
	Adynerin 是一种发现于夹竹桃中的天然类固醇。
TN1800	Isosakuranin	Others	Others
	Isosakuranin 是一种提取自Paliurus ramosissimus 果实中的天然产物。
TN1626	Eugenin	Others	Others
	Eugenin 是一种色酮，分离自滨海前胡，能够抗血小板聚集。
TN1137	Isobutylshikonin	Others	Others
	Isobutylshikonin 是分离自Lithospermum canescens 毛状根培养的一种紫草素色素。
T5733	Xylotetraose	Others	Others
	Xylotetraose 是木聚糖的水解产物，可用于酶生化分析。Xylan 是由木糖单元组成的多糖，主要包含由纤维素连接的 β-D- 木糖单位。
TN1923	Mesaconine	IL Receptor; NF-κB	Immunology/Inflammation; NF-κB
	Mesaconine 是来自 Aconitum carmichaelii Debx 的一种成分。Mesaconine 具有心脏作用和抗 NF-κB 活性。 Mesaconine 可能是麻黄附子细辛汤抗炎和免疫抑制的部分物质基础。
TN4818	Poriol	Others	Others
	Poriol 是一种黄酮类化合物，分离自Pseudotsuga sinensis。
TN1829	Kakkalide	Dehydrogenase	Metabolism
	Kakkalide 是提取自葛根花中的一种异黄酮。它可以抑制活性氧相关炎症，并改善内皮细胞胰岛素抵抗作用。
T3S0693	Blinin	Others	Others
	Blinin 是一种二萜，分离自植物 Conyza blinii 中。
T8195	Lotusine	Others	Others
	Lotusine 是一种提取自Nelumbo nucifera Gaertn 的绿色种胚中的纯生物碱。它能够作用于心肌中动作电位及心脏浦肯野纤维缓慢内向电流。
TN1028	Militarine	Others	Others
	Militarine 是一种糖苷化合物，分离自 Bletilla striata，能够抑制植物生长。
T39049	Yubeinine	Others	Others
	Yubeinine 是一种生物碱类天然产物，可以起到气管松弛作用。
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天然产物

Cat.No: T3384

Synonym: 蟛蜞菊内酯,IKK Inhibitor II

Target: Apoptosis, NF-κB, Lipoxygenase, Caspase

Cat.No: T14961

Synonym: 䓛,屈

Target: Others

Cat.No: T5813

Target: Reductase

Cat.No: T3817

Target: Others

Neotuberostemonine

Cat.No: T4953

Target: NOS

Cat.No: T3928

Target: Others

Cat.No: TN2058

Target: Anti-infection

Cat.No: T6S1049

Target: ATPase

Cat.No: T3S2027

Target: Others

Cat.No: TN1816

Target: Antioxidant

Cat.No: T13693

Target: Others

Cat.No: T19231

Target: Others

Cat.No: T5S0661

Target: Others

Cat.No: T8161

Target: Others

Cat.No: TN1640

Target: Others

Cat.No: T6S1657

Target: Others

Cat.No: T6S0234

Target: Others

Cat.No: T7033

Target: Antioxidant, COX

Cat.No: T3A2414

Target: Others

Cat.No: TN1081

Target: Dopamine Receptor

Cat.No: TJS0851

Target: Others

Cat.No: TWS1563

Target: Others

Cat.No: T6S1676

Target: Others

Cat.No: T5777

Target: Others

Cat.No: T8208

Target: Others

Cat.No: TN1982

Target: Others

Cat.No: TN1453

Target: Anti-infection

Cat.No: T3931

Target: Others

Cat.No: T19431

Target: Others

Cat.No: T3873

Target: Others

Cat.No: T14291

Target: Others

Cat.No: T8077

Target: Others

Cat.No: T5S1331

Target: c-Met/HGFR, Akt

Cat.No: TN6723

Target: Others

Cat.No: TN1983

Target: IL Receptor, TNF, NO Synthase

Cat.No: T2O2770

Target: Others

Neoisoliquiritin

Cat.No: TN1984

Target: Others

Cat.No: T6S0525

Target: ERK, p38 MAPK, Akt

Cat.No: TN1075

Target: Others

Cat.No: TN1800

Target: Others

Cat.No: TN1626

Target: Others

Isobutylshikonin

Cat.No: TN1137

Target: Others

Cat.No: T5733

Target: Others

Cat.No: TN1923

Target: IL Receptor, NF-κB

Cat.No: TN4818

Target: Others

Cat.No: TN1829

Target: Dehydrogenase

Cat.No: T3S0693

Target: Others

Cat.No: T8195

Target: Others

Cat.No: TN1028

Target: Others

Cat.No: T39049

Target: Others

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Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPY-04815	C1 inhibitor Protein, Rat, Recombinant (His) serpin peptidase inhibitor, clade G (C1 inhibit...	Rat	HEK293
	Plasma protease C1 inhibitor, also known as C1-inhibiting factor, C1-INH, C1 esterase inhibitor, SERPING1 and C1IN, is a serine proteinase inhibitor (serpin) that regulates activation of both the complement and contact systems. By its C-terminal part (serpin domain), characterized by three beta-sheets and an exposed mobile reactive loop, C1-INH binds, and blocks the activity of its target proteases. The N-terminal end (nonserpin domain) confers to C1-INH the capacity to bind lipopolysaccharides ...
TMPY-01183	C1 inhibitor Protein, Human, Recombinant (His) serpin peptidase inhibitor, clade G (C1 inhibit...	Human	HEK293
	Plasma protease C1 inhibitor, also known as C1-inhibiting factor, C1-INH, C1 esterase inhibitor, SERPING1 and C1IN, is a serine proteinase inhibitor (serpin) that regulates activation of both the complement and contact systems. By its C-terminal part (serpin domain), characterized by three beta-sheets and an exposed mobile reactive loop, C1-INH binds, and blocks the activity of its target proteases. The N-terminal end (nonserpin domain) confers to C1-INH the capacity to bind lipopolysaccharides ...
TMPY-01030	TFPI Protein, Human, Recombinant (His) TFPI1,tissue factor pathway inhibitor (lipoprotein-...	Human	HEK293
	Tissue factor pathway inhibitor (TFPI) is the natural inhibitor of TF coagulant and signaling activities. It is a Kunitz-type serine proteinase inhibitor that down-regulates tissue factor-initiated blood coagulation. With its Kunitz domains, TFPI exhibits significant homology with human inter-alpha-trypson inhibitor and bovin basic pancreatic trypsin inhibitor. TFPI is the natural inhibitor of TF coagulant and signaling activities. The importance of TFPI in the regulation of blood coagulation is...
TMPY-01174	DKK1 Protein, Rhesus, Recombinant (N256Q, His) dickkopf WNT signaling pathway inhibitor 1	Rhesus	HEK293
	Dickkopf (DKK) family proteins, consisting of DKK-1, DKK-2, DKK-3 and DKK-4, function as secreted Wnt antagonists by inhibiting Wnt coreceptors LRP5/6. DKK-1, DKK-2, and DKK-4 also bind cell surface Kremen-1 or Kremen-2 and promote the internalization of LRP5/6. Dickkopf related protein 1 (DKK-1) was initially identified as an inducer of head formation in Xenopus embryos. DKK-1 protein modulates Wnt signaling pathway during embryonic development. Increased levels of DKK-1 are found in the majori...
TMPY-04811	DKK1 Protein, Mouse, Recombinant (His) dickkopf WNT signaling pathway inhibitor 1,mdkk-1	Mouse	HEK293
	Dickkopf (DKK) family proteins, consisting of DKK-1, DKK-2, DKK-3 and DKK-4, function as secreted Wnt antagonists by inhibiting Wnt coreceptors LRP5/6. DKK-1, DKK-2, and DKK-4 also bind cell surface Kremen-1 or Kremen-2 and promote the internalization of LRP5/6. Dickkopf related protein 1 (DKK-1) was initially identified as an inducer of head formation in Xenopus embryos. DKK-1 protein modulates Wnt signaling pathway during embryonic development. Increased levels of DKK-1 are found in the majori...
TMPY-01121	DKK3 Protein, Mouse, Recombinant (His) dickkopf WNT signaling pathway inhibitor 3,C87148,A...	Mouse	HEK293
	DKK3 (dickkopf related protein 3) is a member of the dickkopf-related family consisting of DKK1, DKK2, DKK3 and DKK4. It is a secreted protein, and also known as REIC (Reduced Expansion in Immortalized Cells). The DKK3 protein is proposed to function as a secreted tumor suppressor since it is downregulated in a number of cancer cells and prostate cancer tissue and may be a promising candidate molecule for therapeutic interference. DKK3 protein is also a negative regulator of beta-catenin and its...
TMPY-00775	DKK1 Protein, Human, Recombinant (His) dickkopf WNT signaling pathway inhibitor 1,SK,DKK-1	Human	HEK293
	Dickkopf (DKK) family proteins, consisting of DKK-1, DKK-2, DKK-3 and DKK-4, function as secreted Wnt antagonists by inhibiting Wnt coreceptors LRP5/6. DKK-1, DKK-2, and DKK-4 also bind cell surface Kremen-1 or Kremen-2 and promote the internalization of LRP5/6. Dickkopf related protein 1 (DKK-1) was initially identified as an inducer of head formation in Xenopus embryos. DKK-1 protein modulates Wnt signaling pathway during embryonic development. Increased levels of DKK-1 are found in the majori...
TMPY-02731	SPINK4 Protein, Mouse, Recombinant (hFc) MPGC60,serine peptidase inhibitor, Kazal type 4,RP2...	Mouse	HEK293
	Serine protease inhibitor Kazal-type 4, also known as Peptide PEC-6 homolog and SPINK4, is a secreted protein that contains one Kazal-like domain. SPINK4 is a member of the SPINK protein family. The gene family of serine protease inhibitors of the Kazal type (SPINK) are functional and positional candidate genes for celiac disease (CD). SPINK1 plays an important role in protecting the pancreas against excessive trypsinogen activation. It is a potent natural inhibitor of pancreatic trypsin activit...
TMPY-06074	B7-H4 Protein, Cynomolgus, Rhesus, Recombinant (His) V-set domain containing T cell activation inhibitor...	Cynomolgus,Rhesus	HEK293
	V-set domain-containing T-cell activation inhibitor 1, also known as B7X, B7H4, B7S1, and VTCN1, is a single-pass type-III membrane protein belonging to the B7 family of costimulatory proteins. These proteins are expressed on the surface of antigen-presenting cells and interact with ligands on T lymphocytes. They provide costimulatory signals that regulate T cell responses. A soluble form of B7H4 has also been detected. B7X / VTCN1 / B7H4 negatively regulates T-cell-mediated immune response by i...
TMPY-01474	PAI-1 Protein, Human, Recombinant (His) PAI,SERPINE1,PAI-1,serpin peptidase inhibitor, clad...	Human	HEK293
	Plasminogen activator inhibitor 1, also known as PAI-1, Endothelial plasminogen activator inhibitor, SerpinE1 and PLANH1, is a secreted glycoprotein that belongs to the serpin family. SerpinE1 is the primary physiological inhibitor of the two plasminogen activators urokinase (uPA) and tissue plasminogen activator (tPA). Its rapid interaction with TPA may function as a major control point in the regulation of fibrinolysis. Defects in SerpinE1 are the cause of plasminogen activator inhibitor-1 def...
TMPY-05322	B7-H4 Protein, Mouse, Recombinant (His) BC032925,B7h4,B7x,V-set domain containing T cell activation ...	Mouse	HEK293
	V-set domain-containing T-cell activation inhibitor 1, also known as B7X, B7H4, B7S1, and VTCN1, is a single-pass type-III membrane protein belonging to the B7 family of costimulatory proteins. These proteins are expressed on the surface of antigen-presenting cells and interact with ligands on T lymphocytes. They provide costimulatory signals that regulate T cell responses. A soluble form of B7H4 has also been detected. B7X / VTCN1 / B7H4 negatively regulates T-cell-mediated immune response by i...
TMPY-00915	Serpin A1 Protein, Human, Recombinant (His) PRO2275,SerpinA1,serpin peptidase inhibitor, clade ...	Human	HEK293
	SerpinA1, also known as Alpha-1 antitrypsin (AAT), is a prototype member of the Serpin superfamily of the serine protease inhibitors. This serine protease inhibitor blocks the protease, neutrophil elastase. Alpha-1 antitrypsin is mainly produced in the liver and acts as an antiprotease. Its principal function is to inactivate neutrophil elastase, preventing tissue damage. SerpinA1 (alpha1-antitrypsin), an acute phase protein and the classical neutrophil elastase inhibitor, is localized within li...
TMPY-00916	Antithrombin III Protein, Human, Recombinant (His) AT3D,THPH7,ATIII,AT3,Serpin C1,MGC22579,serpin peptidase	Human	HEK293
	SerpinC1, also known as antithrombin III (AT III), is a member of the serpin superfamily of serine protease inhibitors, and has been found to be a marker for disseminated intravascular coagulation (DIC) and to be of prognostic significance in septic patients. SerpinC1 synthesized in the liver is the principal plasma serpin of blood coagulation proteases and inhibits thrombin and other factors such as Xa by the formation of covalently linked complexes. Thus it is one of the most important coagula...
TMPJ-00603	TL1A Protein, Mouse, Recombinant TNFSF15,Tumor Necrosis Factor Ligand Superfamily Member 15,V...	Mouse	E. coli
	Tumor Necrosis Factor Ligand Superfamily Member 15 (TNFSF15) is a new member of the tumor necrosis factor family. TNFSF15 is predominantly an endothelial cell-specific gene, and recombinant TNFSF15 is a potent inhibitor of endothelial cell proliferation, angiogenesis and tumor growth. TNFSF15 exerts two activities on endothelial cells: early G1 arrest of G0/G1-cells responding to growth stimuli and programmed cell death of proliferating cells. These activities are highly specific to endothelial ...
TMPJ-00916	TIMP-2 Protein, Mouse, Recombinant (His) metalloproteinase inhibitor 2,Tissue inhibitor<...	Mouse	Human Cells
	Mouse Metalloproteinase inhibitor 2(TIMP-2), belongs to a family of proteins that regulate the activation and proteolytic activity of matrix metalloproteinases (MMPs). There are four mammalian members of the family; TIMP‑1, TIMP‑2, TIMP‑3, and TIMP‑4. The TIMP-2 is detected in testis, retina, hippocampus and cerebral cortex. The function of TIMP 2 protein is to inhibit MMPs non covalently by the formation of binary complexes. Complexes with metalloproteinases (such as collagenases) and irreversi...
TMPY-03524	B7-H4 Protein, Human, Recombinant (His) PRO1291,B7X,B7H4,B7-H4,VCTN1,B7S1,B7h.5,V-set domain contain...	Human	HEK293
	V-set domain-containing T-cell activation inhibitor 1, also known as B7X, B7H4, B7S1, and VTCN1, is a single-pass type-III membrane protein belonging to the B7 family of costimulatory proteins. These proteins are expressed on the surface of antigen-presenting cells and interact with ligands on T lymphocytes. They provide costimulatory signals that regulate T cell responses. A soluble form of B7H4 has also been detected. B7X / VTCN1 / B7H4 negatively regulates T-cell-mediated immune response by i...
TMPH-00554	Trypsin inhibitor DE-3 Protein, Erythrina caffra, Recombinant (His)	Erythrina caffra	Yeast
	Inhibition of trypsin.
TMPH-00155	Barstar Protein, Bacillus amyloliquefaciens, Recombinant (His & Myc) Barstar,Ribonuclease inhibitor	Bacillus amyloliquefaciens	E. coli
	Barstar Protein, Bacillus amyloliquefaciens, Recombinant (His & Myc) is expressed in E. coli.
TMPJ-00490	Serpin A5 Protein, Human, Recombinant (His) Plasminogen Activator Inhibitor 3,Acrosomal Serine ...	Human	Human Cells
	Serpin A5 is a member of the human Serpin superfamily consists of at least 35 members. It is synthesized in the liver and has been detected in saliva, cerebral spinal fluid, amniotic fluid, tears and semen. As a potent inhibitor of the protein C anticoagulant pathway at the levels of both zymogen activation and enzyme inhibition, Serpin A5 additionally inhibits a variety of serine protease including thrombin, factor Xa, several kallekreins and acrosin. It plays a critical role in the processes o...
TMPJ-01289	TIMP-4 Protein, Human, Recombinant (His) TIMP4,TIMP-4,Metalloproteinase inhibitor 4,Tissue <...	Human	Human Cells
	Metalloproteinase inhibitor 4 is an enzyme that in humans is encoded by the TIMP4 gene, belongs to the protease inhibitor I35 (TIMP) family. The protein complexes with metalloproteinases (such as collagenases) and irreversibly inactivates them by binding to their catalytic zinc cofactor. Known to act on MMP-1, MMP-2, MMP-3, MMP-7 and MMP-9.
TMPY-02912	TIMP-1 Protein, Rat, Recombinant TIMP metallopeptidase inhibitor 1	Rat	HEK293
	TIMP metallopeptidase inhibitor 1, also known as TIMP-1/TIMP1, Collagenase inhibitor 16C8 fibroblast Erythroid-potentiating activity, TPA-S1TPA-induced proteinTissue inhibitor of metalloproteinases 1, is a natural inhibitors of the matrix metalloproteinases (MMPs), a group of peptidases involved in degradation of the extracellular matrix. TIMP-1/TIMP1 is found in fetal and adult tissues. Highest levels are found in bone, lung, ovary and uterus. Complexes with metalloproteinases and irreversibly ...
TMPY-03876	PTGFRN Protein, Cynomolgus, Recombinant (His) prostaglandin F2 receptor inhibitor	Cynomolgus	HEK293
	EWI-F, also known as PTGFRN, is inversely related to the loss of CD9. Its expression correlates with the metastatic status of hLT. EWI-F inhibits the binding of prostaglandin F2-alpha (PGF2-alpha) to its specific FP receptor, by decreasing the receptor number rather than the affinity constant. EWI-F expression positively correlates with the metastatic status of hLT, and that the upregulation of EWI-F expression could be one of the mechanisms underlying the loss of CD9 in solid tumours.
TMPJ-00733	SPINK1 Protein, Human, Recombinant (His) PSTI,Pancreatic Secretory Trypsin Inhibitor,TATI,Se...	Human	Human Cells
	Serine Protease Inhibitor Kazal-Type 1 (SPINK1) is a trypsin inhibitor that prevent the trypsin-catalyzed premature activation of zymogens within the pancreas. Defects in SPINK1 are a cause of pancreatitis (PCTT). A disease characterized by the presence of calculi in pancreatic ducts. It causes severe abdominal pain attacks. Defects in SPINK1 are the cause of susceptibility to tropical calcific pancreatitis (TCP). Recombinant SPINK1 protein (rSPINK1) stimulated cell proliferation in benign RWPE ...
TMPY-05179	TFPI Protein, Human, Recombinant (His), Biotinylated TFI,TFPI1,EPI,LACI,tissue factor pathway inhibitor ...	Human	HEK293
	Tissue factor pathway inhibitor (TFPI) is the natural inhibitor of TF coagulant and signaling activities. It is a Kunitz-type serine proteinase inhibitor that down-regulates tissue factor-initiated blood coagulation. With its Kunitz domains, TFPI exhibits significant homology with human inter-alpha-trypson inhibitor and bovin basic pancreatic trypsin inhibitor. TFPI is the natural inhibitor of TF coagulant and signaling activities. The importance of TFPI in the regulation of blood coagulation is...
TMPH-00478	DIT33 Protein, Dirofilaria immitis, Recombinant (His & Myc) Pepsin inhibitor Dit33,DIT33	Dirofilaria immitis	E. coli
	DIT33 Protein, Dirofilaria immitis, Recombinant (His & Myc) is expressed in E. coli.
TMPY-05800	IKB beta/NFKBIB Protein, Human, Recombinant (GST) NFKB inhibitor β,NFKB inhibitor beta,TRIP9...	Human	E. coli
	NFKBIB (NFKB Inhibitor Beta) is a Protein Coding gene. The protein encoded by this gene belongs to the NF-kappa-B inhibitor family, which inhibits NF-kappa-B by complexing with and trapping it in the cytoplasm. Phosphorylation of serine residues on these proteins by kinases marks them for destruction via the ubiquitination pathway, thereby allowing activation of the NF-kappa-B, which translocates to the nucleus to function as a transcription factor. NF-kappaB regulation involves the inhibitor pr...
TMPJ-00625	Serpin E1 Protein, Mouse, Recombinant (His) Pai1,Planh1,Plasminogen activator inhibitor 1,Serpi...	Mouse	Human Cells
	Plasminogen activator inhibitor-1 (serpin E1) is a serine protease inhibitor which belongs to the serpin family. Serpin E1 acts as 'bait' for tissue plasminogen activator, urokinase, protein C and matriptase-3/TMPRSS7. Its rapid interaction with PLAT may function as a major control point in the regulation of fibrinolysis.
TMPJ-00101	TIMP-2 Protein, Human, Recombinant (His) Tissue Inhibitor of Metalloproteinases 2,TIMP2,CSC-...	Human	Human Cells
	Tissue inhibitors of metalloproteinases or TIMPs are a family of proteins that regulate the activation and proteolytic activity of the zinc enzymes known as matrix metalloproteinases (MMPs). There are four members of the family, TIMP-1, TIMP-2, TIMP-3, and TIMP-4. Tissue Inhibitor of Metalloproteinases 2 (TIMP-2) is a non N-glycosylated protein with a molecular mass of 22 kDa. It produced by a wide range of cell types, which inhibits MMPs non-covalently by the formation of binary complexes and i...
TMPJ-00972	CDKN1B Protein, Human, Recombinant (His) KIP1,CDKN1B,Cyclin-Dependent Kinase Inhibitor p27,C...	Human	E. coli
	Cyclin-Dependent Kinase Inhibitor 1B (CDKN1B) is a Kinesin-related motor protein necessary for mitotic spindle assembly and chromosome segregation. CDKN1B is expressed in all tissues with highest levels observed in skeletal muscle. CDKN1B is a potent inhibitor of Cyclin E- and Cyclin A-CDK2 complexes. CDKN1B forms a complex with Cyclin Type D-CDK4 complexes and is involved in the assembly, stability, and modulation of CCND1-CDK4 complex activation. In addition, CDKN1B acts as an inhibitor or an ...
TMPY-00163	SPINK2 Protein, Human, Recombinant (hFc) serine peptidase inhibitor, Kazal type 2 (acrosin-t...	Human	HEK293
	Human serine proteinase inhibitor Kazal-type 2 (SPINK2) functions as a trypsin/acrosin inhibitor and is synthesized mainly in the testis and seminal vesicle where its activity is engaged in fertility. The SPINK2 protein contains a typical Kazal domain composed by six cysteine residues forming three disulfide bridges. The expression of SPINK2 is closely related to cancer such as lymphomas, in that a high transcript level of SPINK2 in patients with primary cutaneous follicle center cell lymphomas ...
TMPY-00928	TFPI Protein, Mouse, Recombinant (His) AW552122,A630013F22Rik,tissue factor pathway inhibitor	Mouse	HEK293
	Tissue factor pathway inhibitor (TFPI) is the natural inhibitor of TF coagulant and signaling activities. It is a Kunitz-type serine proteinase inhibitor that down-regulates tissue factor-initiated blood coagulation. With its Kunitz domains, TFPI exhibits significant homology with human inter-alpha-trypson inhibitor and bovin basic pancreatic trypsin inhibitor. TFPI is the natural inhibitor of TF coagulant and signaling activities. The importance of TFPI in the regulation of blood coagulation is...
TMPJ-01383	Serpin A10 Protein, Human, Recombinant (His) PZI,Protein Z-Dependent Protease Inhibitor,Serpin A...	Human	Human Cells
	Serpin A10 is a secreted protein that belongs to the serpin family. It is predominantly expressed in the liver and secreted in the plasma. Its phosphorylation sites are present in the extracelllular medium. It inhibits factors Xa and XIa of the coagulation cascade in the presence of protein Z, calcium, and phospholipid. Mutations in SERPINA10 are associated with venous thrombosis.
TMPJ-00931	Serpin A4 Protein, Human, Recombinant (His) Kallistatin,Peptidase Inhibitor 4,KST,Kallikrein	Human	Human Cells
	Serpin Peptidase Inhibitor, Clade A (α-1 Antiproteinase, Antitrypsin), Member 4 (Serpin A4) is a member of the Serpin family. Serpin A4 exists as a monomer and some homodimers. Serpin A4 is expressed by the liver and secreted in plasma. Serpin A4 is a regulator of vascular homeostasis capable of controlling a wide spectrum of biological actions in the cardiovascular and renal systems. It can inhibit intracellular reactive oxygen species formation in cultured cardiac and renal cells. In addition,...
TMPY-05797	DKK1 Protein, Rat, Recombinant (His) dickkopf WNT signaling pathway inhibitor 1	Rat	HEK293
	Dickkopf (DKK) family proteins, consisting of DKK-1, DKK-2, DKK-3 and DKK-4, function as secreted Wnt antagonists by inhibiting Wnt coreceptors LRP5/6. DKK-1, DKK-2, and DKK-4 also bind cell surface Kremen-1 or Kremen-2 and promote the internalization of LRP5/6. Dickkopf related protein 1 (DKK-1) was initially identified as an inducer of head formation in Xenopus embryos. DKK-1 protein modulates Wnt signaling pathway during embryonic development. Increased levels of DKK-1 are found in the majori...
TMPY-01175	DKK1 Protein, Rhesus, Recombinant (N256Q, mFc) dickkopf WNT signaling pathway inhibitor 1	Rhesus	HEK293
	Dickkopf (DKK) family proteins, consisting of DKK-1, DKK-2, DKK-3 and DKK-4, function as secreted Wnt antagonists by inhibiting Wnt coreceptors LRP5/6. DKK-1, DKK-2, and DKK-4 also bind cell surface Kremen-1 or Kremen-2 and promote the internalization of LRP5/6. Dickkopf related protein 1 (DKK-1) was initially identified as an inducer of head formation in Xenopus embryos. DKK-1 protein modulates Wnt signaling pathway during embryonic development. Increased levels of DKK-1 are found in the majori...
TMPJ-01064	Serpin G1 Protein, Mouse, Recombinant (His) Serping1,Plasma protease C1 inhibitor,C1 Inh,C1 est...	Mouse	Human Cells
	SERPIN G1 is a member of the serpin family, The C-terminal serpin domain is similar to other serpins, and this part of C1-INH provides the inhibitory activity. SERPIN G1 is involved in the inhibition of the complement system to prevent spontaneous activation. SERPIN G1 may play a potentially crucial role in regulating important physiological pathways including complement activation, blood coagulation, fibrinolysis and the generation of kinins. SERPIN G1 prevents the proteolytic cleavage of later...
TMPH-02532	BIRC5 Protein, Mouse, Recombinant (E. coli, His) Apoptosis inhibitor 4,Apoptosis inhibitor ...	Mouse	E. coli
	Multitasking protein that has dual roles in promoting cell proliferation and preventing apoptosis. Component of a chromosome passage protein complex (CPC) which is essential for chromosome alignment and segregation during mitosis and cytokinesis. Acts as an important regulator of the localization of this complex; directs CPC movement to different locations from the inner centromere during prometaphase to midbody during cytokinesis and participates in the organization of the center spindle by ass...
TMPJ-01069	Serpin A1e Protein, Mouse, Recombinant (His) Dom5,α-1-antitrypsin 1-5,Serpina1e,Spi1-5,Serine protease	Mouse	Human Cells
	Alpha-1-antitrypsin 1-5(SERPIN A1) is a secreted protein and belongs to the serpin family. Serpins bind the protease active site resulting in a major conformational rearrangement that traps the enzyme in a covalent acyl-enzyme intermediate. Mouse SERPIN A1 is a serine protease inhibitor whose targets include elastase,plasmin, thrombin, trypsin, chymotrypsin, and plasminogen activator. Defects in this gene can cause emphysema orliver disease. Several transcript variants encoding the same protein ...
TMPY-02981	ING5 Protein, Human, Recombinant (GST) p28ING5,inhibitor of growth family, member 5	Human	E. coli
	ING5 belongs to the ING family. It contains 1 PHD-type zinc finger and is a component of the HBO1 complex. HBO1 complex has a histone H4-specific acetyltransferase activity, a reduced activity toward histone H3 and is responsible for the bulk of histone H4 acetylation in vivo. HBO1 complex composed at least of ING4 or ING5, KAT7/HBO1, MEAF6, and one of PHF15, PHF16, and PHF17. ING5 also is a component of the MOZ/MORF complex which is composed at least of ING5, KAT6A, KAT6B, MEAF6, and one of BRP...
TMPY-03127	BAMBI Protein, Mouse, Recombinant (hFc) 2610003H06Rik,BMP and activin membrane-bound inhibitor	Mouse	HEK293
	BMP and activin membrane-bound inhibitor (BAMBI) is a transmembrane glycoprotein that is a pseudoreceptor of type 1 receptors. BAMBI structurally lacks intracellular serine/ threonine kinase domain but with an extracellular domain and a short cytoplasmic region that share sequence similarities with type 1 receptors, whose members have functions in signal transduction in various developing and pathological processes. BAMBI competes with the type 1 receptor, a receptor of the transforming growth f...
TMPY-02187	SEMA5A Protein, Human, Recombinant (hFc) SEMAF,serpin peptidase inhibitor, clade F,semF	Human	HEK293
	Semaphorins are secreted, transmembrane, and GPI-linked proteins, defined by cysteine-rich semaphorin protein domains, that have important roles in a variety of tissues. Humans have 2 semaphorins, Drosophila has five, and two are known from DNA viruses. Semaphorins are found in nematodes and crustaceans but not in non-animals. They are grouped into eight classes on the basis of phylogenetic tree analyses and the presence of additional protein motifs. Semaphorins have been implicated in diverse d...
TMPH-00992	BIRC5 Protein, Human, Recombinant (His & SUMO) API4,Apoptosis inhibitor survivin,BIRC5,IAP4,Baculo...	Human	E. coli
	BIRC5 Protein, Human, Recombinant (His & SUMO) is expressed in E. coli.
TMPH-02533	BIRC5 Protein, Mouse, Recombinant (His) BIRC5,Baculoviral IAP repeat-containing protein 5,API4,Apopt...	Mouse	Yeast
	Multitasking protein that has dual roles in promoting cell proliferation and preventing apoptosis. Component of a chromosome passage protein complex (CPC) which is essential for chromosome alignment and segregation during mitosis and cytokinesis. Acts as an important regulator of the localization of this complex; directs CPC movement to different locations from the inner centromere during prometaphase to midbody during cytokinesis and participates in the organization of the center spindle by ass...
TMPY-02559	PAI-1 Protein, Rat, Recombinant (His) serpin peptidase inhibitor, clade E (nexin, plasmin...	Rat	HEK293
	Plasminogen activator inhibitor 1, also known as PAI-1, Endothelial plasminogen activator inhibitor, SerpinE1 and PLANH1, is a secreted glycoprotein that belongs to the serpin family. SerpinE1 is the primary physiological inhibitor of the two plasminogen activators urokinase (uPA) and tissue plasminogen activator (tPA). Its rapid interaction with TPA may function as a major control point in the regulation of fibrinolysis. Defects in SerpinE1 are the cause of plasminogen activator inhibitor-1 def...
TMPH-00520	Host-nuclease inhibitor protein gam Protein, Enterobacteria phage lambda, Recombinant (His & Myc)	Escherichia phage lambda	E. coli
	Binds to host RecBCD nuclease and inhibits it thereby protecting the viral DNA against recBCD mediated degradation.
TMPJ-00452	Serpin A1a Protein, Mouse, Recombinant (His) Alpha-1-antitrypsin 1-1, Alpha-1 protease inhibitor...	Mouse	Human Cells
	Serpin A1a is also known as alpha-1-antitrypsin, is a member of the serpin superfamily of serine proteinase inhibitors that are involved in the regulation of a number of proteolytic processes. Its primary target is elastase, but it also has a moderate affinity for plasmin and thrombin.
TMPJ-00243	Serpin B6 Protein, Human, Recombinant (E. coli, His) CAP,PI6,SERPINB6,Placental Thrombin Inhibitor,Cytop...	Human	E. coli
	Serpin B6 belongs to the serpin family. Serpin B6 localizes to the cytoplasm. Serpin B6 is expressed in many tissues, abundantly by mast cells in different tissues and mastocytoma lesions. Serpin B6 may be involved in the regulation of serine proteinases present in the brain or extravasated from the blood. In addition, Serpin B6 may play an important role in the inner ear in the protection against leakage of lysosomal content during stress and loss of this protection results in cell death and se...
TMPY-00266	PEDF Protein, Rat, Recombinant (His) serpin peptidase inhibitor, clade F，member 1	Rat	HEK293
	Pigment epithelium-derived factor, also known as PEDF, Serpin F1, and SERPINF1, is a multiple functional protein that has both anti-angiogenic activity and neurotrophic activity at the same time. PEDF is a secreted glycoprotein that belongs to the noninhibitory serpin. It has an alpha/beta core serine-protease inhibitor domain, three major beta-sheets, and ten alpha-helices. PEDF does not inhibit either serine or cysteine proteinases. PEDF exerts diverse physiological activities including anti-a...
TMPY-04334	BAMBI Protein, Mouse, Recombinant (His) BMP and activin membrane-bound inhibitor,2610003H06...	Mouse	HEK293
	BMP and activin membrane-bound inhibitor (BAMBI) is a transmembrane glycoprotein that is a pseudoreceptor of type 1 receptors. BAMBI structurally lacks intracellular serine/ threonine kinase domain but with an extracellular domain and a short cytoplasmic region that share sequence similarities with type 1 receptors, whose members have functions in signal transduction in various developing and pathological processes. BAMBI competes with the type 1 receptor, a receptor of the transforming growth f...
TMPY-01456	BAMBI Protein, Human, Recombinant (His) BMP and activin membrane-bound inhibitor,NMA	Human	HEK293
	BMP and activin membrane-bound inhibitor (BAMBI) is a transmembrane glycoprotein that is a pseudoreceptor of type 1 receptors. BAMBI structurally lacks intracellular serine/ threonine kinase domain but with an extracellular domain and a short cytoplasmic region that share sequence similarities with type 1 receptors, whose members have functions in signal transduction in various developing and pathological processes. BAMBI competes with the type 1 receptor, a receptor of the transforming growth f...
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重组蛋白

C1 inhibitor Protein, Rat, Recombinant (His)

Cat.No: TMPY-04815

Species: Rat

Expression System: HEK293

C1 inhibitor Protein, Human, Recombinant (His)

Cat.No: TMPY-01183

Species: Human

Expression System: HEK293

TFPI Protein, Human, Recombinant (His)

Cat.No: TMPY-01030

Species: Human

Expression System: HEK293

DKK1 Protein, Rhesus, Recombinant (N256Q, His)

Cat.No: TMPY-01174

Species: Rhesus

Expression System: HEK293

DKK1 Protein, Mouse, Recombinant (His)

Cat.No: TMPY-04811

Species: Mouse

Expression System: HEK293

DKK3 Protein, Mouse, Recombinant (His)

Cat.No: TMPY-01121

Species: Mouse

Expression System: HEK293

DKK1 Protein, Human, Recombinant (His)

Cat.No: TMPY-00775

Species: Human

Expression System: HEK293

SPINK4 Protein, Mouse, Recombinant (hFc)

Cat.No: TMPY-02731

Species: Mouse

Expression System: HEK293

B7-H4 Protein, Cynomolgus, Rhesus, Recombinant (His)

Cat.No: TMPY-06074

Species: Cynomolgus,Rhesus

Expression System: HEK293

PAI-1 Protein, Human, Recombinant (His)

Cat.No: TMPY-01474

Species: Human

Expression System: HEK293

B7-H4 Protein, Mouse, Recombinant (His)

Cat.No: TMPY-05322

Species: Mouse

Expression System: HEK293

Serpin A1 Protein, Human, Recombinant (His)

Cat.No: TMPY-00915

Species: Human

Expression System: HEK293

Antithrombin III Protein, Human, Recombinant (His)

Cat.No: TMPY-00916

Species: Human

Expression System: HEK293

TL1A Protein, Mouse, Recombinant

Cat.No: TMPJ-00603

Species: Mouse

Expression System: E. coli

TIMP-2 Protein, Mouse, Recombinant (His)

Cat.No: TMPJ-00916

Species: Mouse

Expression System: Human Cells

B7-H4 Protein, Human, Recombinant (His)

Cat.No: TMPY-03524

Species: Human

Expression System: HEK293

Trypsin inhibitor DE-3 Protein, Erythrina caffra, Recombinant (His)

Cat.No: TMPH-00554

Species: Erythrina caffra

Expression System: Yeast

Barstar Protein, Bacillus amyloliquefaciens, Recombinant (His & Myc)

Cat.No: TMPH-00155

Species: Bacillus amyloliquefaciens

Expression System: E. coli

Serpin A5 Protein, Human, Recombinant (His)

Cat.No: TMPJ-00490

Species: Human

Expression System: Human Cells

TIMP-4 Protein, Human, Recombinant (His)

Cat.No: TMPJ-01289

Species: Human

Expression System: Human Cells

TIMP-1 Protein, Rat, Recombinant

Cat.No: TMPY-02912

Species: Rat

Expression System: HEK293

PTGFRN Protein, Cynomolgus, Recombinant (His)

Cat.No: TMPY-03876

Species: Cynomolgus

Expression System: HEK293

SPINK1 Protein, Human, Recombinant (His)

Cat.No: TMPJ-00733

Species: Human

Expression System: Human Cells

TFPI Protein, Human, Recombinant (His), Biotinylated

Cat.No: TMPY-05179

Species: Human

Expression System: HEK293

DIT33 Protein, Dirofilaria immitis, Recombinant (His & Myc)

Cat.No: TMPH-00478

Species: Dirofilaria immitis

Expression System: E. coli

IKB beta/NFKBIB Protein, Human, Recombinant (GST)

Cat.No: TMPY-05800

Species: Human

Expression System: E. coli

Serpin E1 Protein, Mouse, Recombinant (His)

Cat.No: TMPJ-00625

Species: Mouse

Expression System: Human Cells

TIMP-2 Protein, Human, Recombinant (His)

Cat.No: TMPJ-00101

Species: Human

Expression System: Human Cells

CDKN1B Protein, Human, Recombinant (His)

Cat.No: TMPJ-00972

Species: Human

Expression System: E. coli

SPINK2 Protein, Human, Recombinant (hFc)

Cat.No: TMPY-00163

Species: Human

Expression System: HEK293

TFPI Protein, Mouse, Recombinant (His)

Cat.No: TMPY-00928

Species: Mouse

Expression System: HEK293

Serpin A10 Protein, Human, Recombinant (His)

Cat.No: TMPJ-01383

Species: Human

Expression System: Human Cells

Serpin A4 Protein, Human, Recombinant (His)

Cat.No: TMPJ-00931

Species: Human

Expression System: Human Cells

DKK1 Protein, Rat, Recombinant (His)

Cat.No: TMPY-05797

Species: Rat

Expression System: HEK293

DKK1 Protein, Rhesus, Recombinant (N256Q, mFc)

Cat.No: TMPY-01175

Species: Rhesus

Expression System: HEK293

Serpin G1 Protein, Mouse, Recombinant (His)

Cat.No: TMPJ-01064

Species: Mouse

Expression System: Human Cells

BIRC5 Protein, Mouse, Recombinant (E. coli, His)

Cat.No: TMPH-02532

Species: Mouse

Expression System: E. coli

Serpin A1e Protein, Mouse, Recombinant (His)

Cat.No: TMPJ-01069

Species: Mouse

Expression System: Human Cells

ING5 Protein, Human, Recombinant (GST)

Cat.No: TMPY-02981

Species: Human

Expression System: E. coli

BAMBI Protein, Mouse, Recombinant (hFc)

Cat.No: TMPY-03127

Species: Mouse

Expression System: HEK293

SEMA5A Protein, Human, Recombinant (hFc)

Cat.No: TMPY-02187

Species: Human

Expression System: HEK293

BIRC5 Protein, Human, Recombinant (His & SUMO)

Cat.No: TMPH-00992

Species: Human

Expression System: E. coli

BIRC5 Protein, Mouse, Recombinant (His)

Cat.No: TMPH-02533

Species: Mouse

Expression System: Yeast

PAI-1 Protein, Rat, Recombinant (His)

Cat.No: TMPY-02559

Species: Rat

Expression System: HEK293

Host-nuclease inhibitor protein gam Protein, Enterobacteria phage lambda, Recombinant (His & Myc)

Cat.No: TMPH-00520

Species: Escherichia phage lambda

Expression System: E. coli

Serpin A1a Protein, Mouse, Recombinant (His)

Cat.No: TMPJ-00452

Species: Mouse

Expression System: Human Cells

Serpin B6 Protein, Human, Recombinant (E. coli, His)

Cat.No: TMPJ-00243

Species: Human

Expression System: E. coli

PEDF Protein, Rat, Recombinant (His)

Cat.No: TMPY-00266

Species: Rat

Expression System: HEK293

BAMBI Protein, Mouse, Recombinant (His)

Cat.No: TMPY-04334

Species: Mouse

Expression System: HEK293

BAMBI Protein, Human, Recombinant (His)

Cat.No: TMPY-01456

Species: Human

Expression System: HEK293

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