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Bifenazate
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很棒纯度: 99.62%
货号 T14571Cas号 149877-41-8
Bifenazate 是 GABA 受体的正向变构调节剂。 Bifenazate 是一种杀螨剂，可在 25 ppm 的浓度下控制 100% 的螨虫。
Bifenazate
一键复制产品信息 很棒纯度: 99.62%
货号 T14571Cas号 149877-41-8
Bifenazate 是 GABA 受体的正向变构调节剂。 Bifenazate 是一种杀螨剂，可在 25 ppm 的浓度下控制 100% 的螨虫。
| 规格 | 价格 | 库存 | 数量 |
|---|---|---|---|
| 25 mg | ¥ 148 | 现货 | |
| 1 mL x 10 mM (in DMSO) | ¥ 113 | 现货 |
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产品介绍
Bifenazate AI Summary
Bifenazate shows high bioactivity against various strains of Tetranychus urticae (two-spotted spider mite), including those resistant to bifenazate and METI, exhibiting resistance ratios exceeding 2780.0 in most cases. It also displays high toxicity towards adult spider mites, with low LC50 values. The compound demonstrates insecticidal activity against Panonychus ulmi strains, with LC50 values of 1.3 ug/mL for PSR-TK and 1.42 ug/mL for HS, and a resistance ratio of 1.0. Additionally, it is active against both spirodiclofen-resistant and spirodiclofen-susceptible Tetranychus urticae, with respective LC50 values of 2.4 ug/mL and 1.2 ug/mL, and a resistance ratio of 2.0.
In various signaling pathways, Bifenazate acts as both agonist and antagonist:
- Agonist in the retinoid X receptor alpha pathway (35481.3 nM potency).
- Antagonist in the thyroid hormone receptor beta pathway (50118.7 nM potency) and estrogen receptor alpha pathway (50118.7 nM potency).
- Agonist in the Aryl hydrocarbon Receptor (AhR) pathway (44668.4 nM potency).
- Agonist in the antioxidant response element (ARE) pathway (54482.7 nM potency).
The compound exhibits contact toxicity against Apis mellifera (honey bee) with an LD50 of less than 1.0 ug, but lower toxicity against Bombus terrestris (bumblebee) with an LD50 greater than 100.0 ug. For bumblebees, it has a NOAEL of 0.096 mgAi/L and an LC50 of 9.6 mgAi/L when administered through sugar water over 11 weeks, inducing 95.0% mortality at a concentration of 96 mg a.i./L, while topically applying less than 25.0% mortality on the dorsal thorax..
Note: Summary generated by AI. Data source: ChEMBL 
生物活性
化学信息
储存&溶解度
| 产品描述 | Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm. |
| 分子量 | 300.35 |
| 分子式 | C17H20N2O3 |
| CAS No. | 149877-41-8 |
| Smiles | COc1ccc(cc1NNC(=O)OC(C)C)-c1ccccc1 |
| 密度 | 1.19. Temperature:25 °C. |
| 存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. | |||||||||||||||||||||||||||||||||||
| 溶解度信息 | H2O: < 0.1 mg/mL (insoluble) DMSO: 250 mg/mL (832.36 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
| 体内实验配方 | 10% DMSO+40% PEG300+5% Tween 80+45% Saline: 5 mg/mL (16.65 mM), Sonication is recommended. 请按顺序添加溶剂，在添加下一种溶剂之前，尽可能使溶液澄清。如有必要，可通过加热、超声、涡旋处理进行溶解。工作液建议现配现用。以上配方仅供参考，体内配方并不是绝对的，请根据不同情况进行调整。 | |||||||||||||||||||||||||||||||||||
溶液配制表 | ||||||||||||||||||||||||||||||||||||
DMSO
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计算器
体内实验配液计算器
请在以下方框中输入您的动物实验信息后点击计算，可以得到母液配置方法和体内配方的制备方法：
比如您的给药剂量是10 mg/kg，每只动物体重20 g，给药体积100 μL， 一共给药动物10只，您使用的配方为 10% DMSO + 40% PEG300 + 5% Tween 80 + 45% Saline / PBS / ddH2O， 那么您的工作液浓度为2 mg/mL。
母液配置方法：2 mg 药物溶于 100 μL DMSO （ 母液浓度为 20 mg/mL ）, 如您需要配置的浓度超过该产品的溶解度，请先与我们联系。
体内配方的制备方法： 取 100 μL DMSO 母液， 添加 400 μL PEG300 混匀澄清， 再加 50 μL Tween 80, 混匀澄清, 再加 450 μL Saline / PBS / ddH2O 混匀澄清
以上为“体内实验配液计算器”的使用方法举例，并不是具体某个化合物的推荐配制方式，请根据您的实验动物和给药方式选择适当的溶解方案。
剂量转换
对于不同动物的给药剂量换算，您也可以参考 更多
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