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NPPB 是外向整流氯化物通道阻断剂,IC50 为 80 nM。
NPPB 是外向整流氯化物通道阻断剂,IC50 为 80 nM。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
5 mg | ¥ 281 | In stock | |
10 mg | ¥ 460 | In stock | |
25 mg | ¥ 837 | In stock | |
50 mg | ¥ 1,474 | In stock | |
100 mg | ¥ 2,615 | In stock | |
1 mL x 10 mM (in DMSO) | ¥ 401 | In stock |
NPPB 相关产品
产品描述 | NPPB is a chloride channel blocker with IC50 of 80 nM . |
靶点活性 | Cl- channel:80 nM |
体外活性 | NPPB has been shown to activate the GPR35-Gαi/o and GPR35-Gα16 pathways in HEK293 cells, inducing intracellular calcium mobilization[1]. |
别名 | 5-硝基-2-(3-苯丙胺)苯甲酸 |
分子量 | 300.31 |
分子式 | C16H16N2O4 |
CAS No. | 107254-86-4 |
Smiles | OC(=O)c1cc(ccc1NCCCc1ccccc1)[N+]([O-])=O |
密度 | 1.323 g/cm3 (Predicted) |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. | |||||||||||||||||||||||||||||||||||
溶解度信息 | DMSO: 150 mg/mL (499.48 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
溶液配制表 | ||||||||||||||||||||||||||||||||||||
DMSO
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以上为“体内实验配液计算器”的使用方法举例,并不是具体某个化合物的推荐配制方式,请根据您的实验动物和给药方式选择适当的溶解方案。
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