规格

价格

库存

数量

1 mg

¥ 593

现货

5 mg

¥ 1,490

现货

10 mg

¥ 2,480

现货

25 mg

¥ 3,970

现货

50 mg

¥ 5,860

现货

100 mg

¥ 7,890

现货

200 mg

¥ 10,600

现货

生物活性

产品描述	RSM-932A (TCD-717) is a specific ChoKα inhibitor with IC50s of 1 and 33 μM against human recombinant ChoKα and ChoKβ enzymes, respectively. RSM-932A possesses potent ex vivo antitumor activity and low toxicity.
体外活性	RSM-932A exhibits effective anti proliferative activity against most tumor derived cell lines tested, including those from breast, lung, colon, bladder, liver, ovary, bone, cervix, kidney, pancreas, melanoma, and brain tumors, with an IC50 of 1.3-7.1 μM at 72 hours [1]
体内活性	RSM-932A exhibits strong in vivo anticancer activity and is not toxic at effective doses [1].
别名	TCD-717

化学信息

分子量	877.54
分子式	C₄₆H₃₈Cl₂N₄Br₂
CAS No.	850807-63-5
Smiles	[Br-].[Br-].CN(c1ccc(Cl)cc1)c1cc[n+](Cc2ccc(cc2)-c2ccc(C[n+]3ccc(N(C)c4ccc(Cl)cc4)c4ccccc34)cc2)c2ccccc12
密度	1.31g/cm3

储存&溶解度

存储

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

溶解度信息

DMSO: 55 mg/mL (62.68 mM), Sonication is recommended.

体内实验配方

10% DMSO+90% Saline: 1.67 mg/mL (1.9 mM), Sonication is recommeded.

请按顺序添加溶剂，在添加下一种溶剂之前，尽可能使溶液澄清。如有必要，可通过加热、超声、涡旋处理进行溶解。工作液建议现配现用。以上配方仅供参考，体内配方并不是绝对的，请根据不同情况进行调整。

溶液配制表

DMSO

RSM-932A