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Targets Recommended: Carboxypeptidase

10000+

抑制剂 & 化合物

1000+

天然产物

21

化合物库

8

TargetMol 试剂盒

343

重组蛋白

277

同位素标记化合物

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Cat. No.	Product Name
L9410	共价抑制剂库		1920 compounds
	1920 种小分子的独特集合，包含已发现的共价抑制剂以及包含某些共价反应基团常见弹头的分子，如氯乙酰基，2-氯丙酰基，丙烯酰基，1-丙-2-炔基，1-丁-2-炔基，酮羰基，二硫键等，可以用于共价抑制剂药物研发；
LF9000	半胱氨酸靶向共价抑制剂库		3400 compounds
	It contains over 3,400 potential covalent modifiers.
L2000	抑制剂库		8328 compounds
	8328 个小分子抑制剂的独特集合，主要用于细胞信号研究、新药筛选、高通量筛选和高内涵筛选；
L9100	磷酸酶抑制剂化合物库		79 compounds
	79 种已知活性的磷酸酶抑制剂的集合，可用于化合物筛选、化学基因组学、药理分析等方面；
L1600	激酶抑制剂库		2720 compounds
	2720 种激酶抑制剂/调节剂的独特集合，用于特定靶向激酶，可用于高通量筛选和高内涵筛选；
L7600	趋化因子抑制剂库		59 compounds
	59 种趋化因子或其受体抑制剂的独特集合，可用于高通量筛选和高内涵筛选；
L3600	细胞因子抑制剂库		604 compounds
	604 个与细胞因子紧密相关的化合物集合，是高通量、高内涵筛选的良好载体；
L9400	PPI抑制剂库		485 compounds
	485 种已知活性的 PPI 相关的抑制剂，可用于高通量、高内涵筛选；
L1400	MAPK 抑制剂库		365 compounds
	365 种与MAPK 信号通路相关的生物活性小分子化合物的特有集合，可用于高通量筛选和高内涵筛选；
L1100	蛋白酶抑制剂库		343 compounds
	343 种已知的小分子蛋白酶抑制剂的特有集合，可用于高通量筛选和高内涵筛选；
L2300	离子通道库		1147 compounds
	1147 种与离子通道相关的生物活性小分子化合物的特有集合，用于离子通道相关的疾病和药物研究，可用于高通量筛选和高内涵筛选；
L2200	酪氨酸激酶分子库		1016 compounds
	1016 种酪氨酸激酶抑制剂的独特集合，可用于高通量筛选和高内涵筛选；
L1610	FDA 上市激酶抑制剂库		263 compounds
	263种靶向激酶的上市药物集合，用于特定靶向激酶，可用于高通量筛选和高内涵筛选；
L2010	高选择性抑制剂库		575 compounds
	575种具有高选择性的抑制剂集合
LF9100	丝氨酸靶向共价抑制剂库		2700 compounds
	Over 2,700 small-molecule screening compounds in the library.
L1510	核受体化合物库		531 compounds
	531 个核受体作用化合物的独特集合，可用于高通量筛选和高内涵筛选；
DO2200	共价抑制剂库CD		12000 compounds
	数量多：超过12000种共价结合化合物，并且数量在持续增加；
DF4100	Smart共价抑制剂库		1787 compounds
	ChemDiv’s Smart Library of Covalent Inhibitors contains 1152 compounds
L8000	干细胞分化化合物库		1197 compounds
	1197 种干细胞分化信号通路相关的生物活性小分子化合物的特有集合，可用于高通量、高内涵筛选；
L7000	活性脂质化合物库		385 compounds
	385 种生物活性小分子化合物，用于高通量、高内涵筛选；
L7110	抗高血压化合物库		678 compounds
	678 种高血压相关的小分子，用于高通量和高内涵筛选；

化合物库

共价抑制剂库

Cat.No: L9410

Compounds: 1920

半胱氨酸靶向共价抑制剂库

Cat.No: LF9000

Compounds: 3400

Cat.No: L2000

Compounds: 8328

磷酸酶抑制剂化合物库

Cat.No: L9100

Compounds: 79

激酶抑制剂库

Cat.No: L1600

Compounds: 2720

趋化因子抑制剂库

Cat.No: L7600

Compounds: 59

细胞因子抑制剂库

Cat.No: L3600

Compounds: 604

PPI抑制剂库

Cat.No: L9400

Compounds: 485

MAPK 抑制剂库

Cat.No: L1400

Compounds: 365

蛋白酶抑制剂库

Cat.No: L1100

Compounds: 343

离子通道库

Cat.No: L2300

Compounds: 1147

酪氨酸激酶分子库

Cat.No: L2200

Compounds: 1016

FDA 上市激酶抑制剂库

Cat.No: L1610

Compounds: 263

高选择性抑制剂库

Cat.No: L2010

Compounds: 575

丝氨酸靶向共价抑制剂库

Cat.No: LF9100

Compounds: 2700

核受体化合物库

Cat.No: L1510

Compounds: 531

共价抑制剂库CD

Cat.No: DO2200

Compounds: 12000

Smart共价抑制剂库

Cat.No: DF4100

Compounds: 1787

干细胞分化化合物库

Cat.No: L8000

Compounds: 1197

活性脂质化合物库

Cat.No: L7000

Compounds: 385

抗高血压化合物库

Cat.No: L7110

Compounds: 678

Cat. No.	Product Name	Form	Specificity Of Inhibition
C0002	Phosphatase Inhibitor Cocktail I (100× ddH2O) 磷酸酶抑制剂 Cocktail I (100× ddH2O)	Solution (100× in ddH2O)	Acid Phosphatase, Alkaline phosphatase, PTPs, ATPases
C0001	Protease Inhibitor Cocktail (EDTA-Free, 100× in DMSO) 蛋白酶抑制剂 Cocktail (EDTA-Free, 100× in DMSO)	Solution (EDTA-Free,100× in DMSO)	Serine proteases, Aminopeptidases, Cysteine proteases, Aspartic proteases
C0048	Deacetylase Inhibitor Cocktail (100× in 70% DMSO) 去乙酰化酶抑制剂 Cocktail（100× in 70% DMSO）	Solution (100× in 70% DMSO)	Class I/II/III HDAC
C0003	Phosphatase Inhibitor Cocktail II (100× DMSO) 磷酸酶抑制剂 Cocktail II (100× DMSO)	Solution (100× in DMSO)	Alkaline phosphatases, Ser/Thr phosphatases, Acid and PP1 and PP2A
C0004	Phosphatase Inhibitor Cocktail III (2 Tubes, 100x) 磷酸酶抑制剂 Cocktail III (2 Tubes, 100x)	2 Tube Solution (100×)	Each Tube has different specificity of inhibition
C0047	RIPA Lysis Buffer (Weak) RIPA裂解液(弱)	Solution in bottle
C0046	RIPA Lysis Buffer (Medium) RIPA裂解液(中)	Solution in bottle
C0045	RIPA Lysis Buffer (Strong) RIPA裂解液(强)	Solution in bottle

TargetMol 试剂盒

磷酸酶抑制剂 Cocktail I (100× ddH2O)

Cat.No: C0002

蛋白酶抑制剂 Cocktail (EDTA-Free, 100× in DMSO)

Cat.No: C0001

去乙酰化酶抑制剂 Cocktail（100× in 70% DMSO）

Cat.No: C0048

磷酸酶抑制剂 Cocktail II (100× DMSO)

Cat.No: C0003

磷酸酶抑制剂 Cocktail III (2 Tubes, 100x)

Cat.No: C0004

RIPA裂解液(弱)

Cat.No: C0047

RIPA裂解液(中)

Cat.No: C0046

RIPA裂解液(强)

Cat.No: C0045

Cat. No.	Product Name	Target	Signaling Pathways
T10876	CPA inhibitor Carboxypeptidase inhibitor	Carboxypeptidase	Proteases/Proteasome
	CPA inhibitor (Carboxypeptidase inhibitor) 是一种有效的羧肽酶 A (CPA) 抑制剂，Ki 值为 0.32 μM。
T5451	Eph inhibitor 2 Ehp-inhibitor-1	Ephrin Receptor	Tyrosine Kinase/Adaptors
	Eph inhibitor 2 是一种 Eph 家族酪氨酸激酶抑制剂。
T1804	HPGDS inhibitor 1 HPGDS-inhibitor-1	PGE Synthase	Immunology/Inflammation
	HPGDS inhibitor 1 是口服具有活性的HPGDS 选择性抑制剂，在酶和细胞分析中的IC50值分别为 0.6 nM 和 32 nM，但对 L-PGDS、mPGES、COX-1、COX-2 、5-LOX 无抑制作用。
TP2325L	Endotoxin Inhibitor acetate Endotoxin Inhibitor acetate(147396-10-9 free base)	Others	Others
	Endotoxin Inhibitor acetate(147396-10-9 free base) 对细菌生理活性有很强的阻断作用，从而产生具有二硫键和大量赖氨酸的抗菌毒素抑制剂序列。内毒素抑制剂醋酸盐在酸性条件下更可能发挥生理活性
T4338	USP7/USP47 inhibitor USP7/47 inhibitor-1	DUB	Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Ubiquitination
	USP7/USP47 inhibitor (USP7/47 inhibitor-1) 是一种选择性泛素特异性蛋白酶 7/47 抑制剂，EC50值分别为 0.42 μM 和 1.0 μM。
T38683	SCD1 inhibitor-3 SCD1-IN-3,SCD1 inhibitor-3,SCD1 inhibitor 17a	Dehydrogenase	Metabolism
	SCD1 inhibitor-3 (ML-270) 是一种高效、口服的化合物，可以抑制SCD1，且安全性极高。 SCD1 inhibitor-3 显示出在代谢疾病(包括肥胖、二型糖尿病和血脂异常，以及痤疮和癌症等各种皮肤病)方面的巨大研究潜力。
T8766	GOT1 inhibitor-1 GOT1 inhibitor 2c	Others	Others
	GOT1 inhibitor-1 (GOT1 inhibitor 2c) 是一种新型的、非共价的谷氨酸草酰乙酸转氨酶 1 (GOT1) 抑制剂(IC50:8.2 uM)，是一种戊酸衍生物。它可用于以及胰腺导管腺癌 (PDAC) 。
T2074	Raf inhibitor 1 B-Raf inhibitor 1	Raf	MAPK
	Raf inhibitor 1 (B-Raf inhibitor 1)是Raf 激酶抑制剂，对B-RafWT、B-RafV600E 和 C-Raf 的Ki 分别为 1、1 和 0.3 nM。
T3593	Src Inhibitor 1 Src Kinase Inhibitor 1,Src-l1	Src	Angiogenesis; Tyrosine Kinase/Adaptors
	Src Inhibitor 1 (Src Kinase Inhibitor 1) 是一种选择性的、高效的、ATP-竞争性的双位点 Src 酪氨酸激酶抑制剂，能够抑制 Src (IC50:44 nM) 和 Lck (IC50:88 nM)。
T5524	Aurora kinase inhibitor-3 Aurora Kinase Inhibitor III	Aurora Kinase	Cell Cycle/Checkpoint; Chromatin/Epigenetic
	Aurora kinase inhibitor-3 (Aurora Kinase Inhibitor III) 是一种有效的，选择性 Aurora A 激酶抑制剂，IC50为 42 nM。
T5817	PKC-theta inhibitor hcl PKC-theta inhibitor	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKC-theta inhibitor hcl 是一种选择性 PKC-θ 抑制剂 (IC50:12 nM)。
T2350	MALT1 inhibitor MI-2 MALT1 inhibitor,MI 2,MI 2 (MALT1 inhibitor)	MALT	Immunology/Inflammation
	MI 2 (MALT1 inhibitor) 是一种MALT1抑制剂 (IC50=5.84 μM)，对动物无毒性。它能够直接与 MALT1 结合，不可逆地抑制蛋白酶功能，并伴有 NF-κB 报告子活性抑制、c-REL 核定位抑制和 NF-κB 靶基因下调。
T3189	B7/CD28 interaction inhibitor 1 CTLA-4 inhibitor	Others	Others
	B7/CD28 interaction inhibitor 1 (CTLA-4 inhibitor) 是B7.1-CD28相互作用抑制剂(IC50:50 nM)。
T3042	JAK2 Inhibitor V JAK2 Inhibitor V Z3,Z3,NSC42834	JAK	Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells
	JAK2 Inhibitor V (JAK2 Inhibitor V Z3) 是一种新型的 Jak2 特异性抑制剂，以剂量依赖性方式抑制 Jak2-V617F 和 Jak2-WT 自磷酸化。
T6335	Tie2 kinase inhibitor 1 Tie2 kinase inhibitor	Tie-2	Tyrosine Kinase/Adaptors
	Tie2 kinase inhibitor 1 (Tie2 kinase inhibitor) 是Tie2激酶选择性抑制剂9IC50:250 nM)，具有抗癌作用。
T4391	Syk Inhibitor II dihydrochloride Syk Inhibitor II (hydrochloride)	Others; Tyrosine Kinases; Syk; PKC; BTK	Angiogenesis; Chromatin/Epigenetic; Cytoskeletal Signaling; Others; Tyrosine Kinase/Adaptors
	Syk Inhibitor II (hydrochloride) 是一种非受体酪氨酸激酶，磷酸化后，它与 FcRγ 链的基于免疫受体酪氨酸的激活基序结合，并介导与血小板功能和炎症相关的下游信号传导。 Syk inhibitor II 是一种可渗透细胞的嘧啶-甲酰胺化合物，以 ATP 竞争性方式选择性和可逆地阻断 Syk (IC50 = 41 nM)。它对 PKCε、PKCβII、ZAP-70、Btk 和 Itk 的效力要低得多（IC50s 分别为5.1、11、11.2、15.5 和 22.6 μM）。
T4191	Multi-kinase inhibitor 1 Multi-kinase inhibitor I	Others; Bcr-Abl; PDGFR; c-Kit	Angiogenesis; Cytoskeletal Signaling; Others; Tyrosine Kinase/Adaptors
	Multi-kinase inhibitor 1 (Multi-kinase inhibitor I) 是多激酶抑制剂。它有用于导致与酪氨酸激酶活性异常或失控有关的疾病或失调的潜力，特别是与c-Kit，PDGF-R，Bcr-abl 活性相关的疾病。
T10678	Carboxypeptidase G2 (CPG2) Inhibitor CPG2 Inhibitor,Carboxypeptidase G2 Inhibitor	Carboxypeptidase	Proteases/Proteasome
	Carboxypeptidase G2 (CPG2) Inhibitor (CPG2 Inhibitor) 是新型的羧肽酶 G2(CPG2)抑制剂，显示出抗癌活性。
T2457	IRAK-1-4 Inhibitor I IRAK-1/4 Inhibitor I,IRAK-1/4 Inhibitor	IRAK	Immunology/Inflammation; NF-κB
	IRAK-1-4 Inhibitor I 是一种IRAK1/4双重抑制剂，其IC50分别为 0.2 μM 和 0.3 μM。
T24141	HIV-1 Inhibitor 18A HIV-1 Inhibitor-18A	HIV Protease	Microbiology/Virology; Proteases/Proteasome
	HIV-1 Inhibitor 18A (HIV-1 Inhibitor-18A) 特异性抑制多种 HIV-1 分离株的进入。
T67767	HIF-1 inhibitor-4 HIF-1 inhibitor-4	HIF	Angiogenesis; Chromatin/Epigenetic
	HIF-1 inhibitor-4 (HIF-1 inhibitor-4) 是一种 HIF-1 抑制剂 (IC50: 560 nM)。HIF-1 inhibitor-4 减少 HIF-1α 蛋白水平，但不影响 mRNA 水平。
T9040	Aurora kinase inhibitor-2 IUN-70219,Aurora Kinase Inhibitor II	Aurora Kinase	Cell Cycle/Checkpoint; Chromatin/Epigenetic
	Aurora kinase inhibitor-2 (IUN-70219) 是一种可渗透细胞的苯胺喹唑啉，可抑制极光激酶的活性，对Aurora A 和Aurora B 的IC50分别为 390 nM 和 240 nM。
T4167	Raf inhibitor 1 dihydrochloride B-Raf inhibitor 1 dihydrochloride	Raf	MAPK
	Raf inhibitor 1 dihydrochloride (B-Raf inhibitor 1 dihydrochloride) 是 Raf 激酶抑制剂，对 B-RafWT、B-RafV600E 和 C-Raf 的Ki 分别为 1、1 和 0.3 nM。
T35827L	PKCε Inhibitor Peptide acetate PKCε Inhibitor Peptide acetate(182683-50-7 Free base)	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKCε Inhibitor Peptide acetate 是一种特异性 PKCε 抑制剂，含有其特定受体活化 C 激酶 (RACK) 的位点。 PKCε Inhibitor Peptide acetate 抑制 PKCε 的转运，但不抑制 αPKC，βPKC 和 δPKC 的转运。
T4491	LMPTP INHIBITOR 1 hydrochloride LMPTP INHIBITOR 1 hydrochloride (1908414-82-3(free base))	Phosphatase	Metabolism
	LMPTP INHIBITOR 1 hydrochloride 是一种高选择性的低分子量蛋白酪氨酸磷酸酶 (LMPTP) 抑制剂。LMPTP INHIBITOR 1 (hydrochloride) 能够抑制 LMPTP-A 的活性，IC50值为 0.8 μM。
T21954	EGFR/ErbB-2/ErbB-4 inhibitor-2 EGFR/ErbB2 Inhibitor	EGFR	Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
	EGFR/ErbB-2/ErbB-4 inhibitor-2 (EGFR/ErbB2 Inhibitor) 是EGFR 和ErbB 的抑制剂，对EGFR、ErbB2 和 ErbB4 的IC50分别为 0.017、0.08 和 1.91 μM。
T9178	(E/Z)-GSK-3β inhibitor 1 GSK-3β inhibitor 1	GSK-3	PI3K/Akt/mTOR signaling; Stem Cells
	(E/Z)-GSK-3β inhibitor 1 是 (E)-GSK-3β inhibitor 1 和 (Z)-GSK-3β inhibitor 1 的消旋体。它是一种糖原合成酶激酶 3β (GSK-3β)的抑制剂，可其对 GSK-3β 的 IC50=4.9 nM，用于糖尿病的研究。
TP2008L	Lyn peptide inhibitor acetate Lyn peptide inhibitor acetate(222018-18-0 free base)	IL Receptor	Immunology/Inflammation
	Lyn peptide inhibitor acetate(222018-18-0 free base) 是一种有效的细胞渗透性 Lyn 偶联 IL-5 受体信号通路抑制剂，同时保持其他信号完整。它阻断 Lyn 活化并抑制 Lyn 酪氨酸激酶与 IL-3/GM-CSF/IL-5 受体的 βc 亚基的结合。它可用于哮喘、过敏和其他嗜酸性粒细胞疾病的研究。
T17157	TRAF-STOP inhibitor 6877002 CD40-TRAF6 inhibitor	NF-κB	NF-κB
	TRAF-STOP inhibitor 6877002 (CD40-TRAF6 inhibitor)是一种 CD40-TRAF6 相互作用的选择性抑制剂，可以抑制 RAW 细胞中 NF-κB 活化。TRAF-STOP 6877002 可阻止小鼠动脉粥样硬化的恶化，减少白细胞募集和巨噬细胞的活化，减少动脉粥样硬化斑块中的巨噬细胞增殖。
TP1015L	NFAT Inhibitor acetate VIVIT peptide acetate,NFAT Inhibitor acetate（249537-73-3 free base）
	NFAT Inhibitor acetate (VIVIT peptide acetate) 是一种具有细胞渗透性和选择性的 NFAT 多肽抑制，对钙调磷酸酶介导的 NFAT 脱磷酸作用有抑制作用。
T36933	Cdk2 Inhibitor II Cdk2 Inhibitor II,CDK2-IN-3	CDK	Cell Cycle/Checkpoint
	Cdk2 Inhibitor II 是一种具有选择性和有效性的 CDK2 抑制剂，50 为 60 nM。
T10927	Cyt-PTPε Inhibitor-1 Cyt-PTP\|A Inhibitor-1	Phosphatase; Src	Angiogenesis; Metabolism; Tyrosine Kinase/Adaptors
	Cyt-PTPε Inhibitor-1 (A Inhibitor-1) 是胞质蛋白酪氨酸磷酸酶 ε 的抑制剂。 Cyt-PTPε Inhibitor-1 阻断 c-Src 的去磷酸化并表现出抗破骨活性。
T22081	FBPase-1 inhibitor-1 Fructose 1,6-bisphosphatase-1 Inhibitor	Others	Others
	FBPase-1 inhibitor-1 (Fructose 1,6-bisphosphatase-1 Inhibitor) 是一种fructose-1,6-bisphosphatase (FBPase-1)的变构抑制剂。
T22136	PRL-3 Inhibitor I PRL-3 Inhibitor,BR-1	Phosphatase; Others	Metabolism; Others
	PRL-3 Inhibitor I (BR-1) 是 PRL-3 抑制剂，IC50=0.9 μM。它在细胞检测中显示降低侵袭性。
TP1523	PKG inhibitor peptide TFA (82801-73-8 free base) PKG inhibitor peptide TFA	PKA	Tyrosine Kinase/Adaptors
	PKG inhibitor peptide TFA (82801-73-8 free base) 是 ATP 竞争性 cGMP 依赖性蛋白激酶 (PKG) 的抑制剂。
T10865L	Cot inhibitor-1 hydrochloride Cot inhibitor-1 hydrochloride(915365-57-0 Free base)	TNF; MAPK	Apoptosis; MAPK
	Cot inhibitor-1 hydrochloride 是肿瘤进展位点 2 激酶 (IC50 = 28 nM) 的抑制剂，可抑制人全血中 TNF-α 的产生 (IC50 = 5.7 nM)。
T7676	LSKL, Inhibitor of Thrombospondin TSP-1 2TFA LSKL, Inhibitor of Thrombospondin TSP-1	TGF-beta/Smad	Stem Cells
	LSKL, Inhibitor of Thrombospondin TSP-1 2TFA 是 TGF-β 的激活剂。
T10599	BRAF inhibitor	Raf	MAPK
	BRAF inhibitor 是B-Raf 抑制剂。
TP1890L1	MLCK inhibitor peptide 18 acetate MLCK inhibitor peptide 18 acetate(224579-74-2 free base)	Serine/threonin kinase	Cell Cycle/Checkpoint; Metabolism
	MLCK inhibitor peptide 18 acetate(224579-74-2 free base) 是肌球蛋白轻链激酶的选择性竞争性抑制剂 (IC50 = 50 nM)。显示出比 CaM 激酶 II 高 4000 倍的选择性，并且不抑制 PKA。细胞可渗透。
T7541	PTP inhibitor 1 PTP Inhibitor II,alpha-溴-4-甲氧基苯乙酮	Phosphatase	Metabolism
	PTP inhibitor 1 是蛋白酪氨酸磷酸酶 (PTP) 抑制剂，具有抗血管生成作用。
T11184	EML4-ALK kinase inhibitor 1 EML4 ALK kinase inhibitor 1,EML4-ALK kinase inhibitor 1	ALK	Angiogenesis; Tyrosine Kinase/Adaptors
	EML4-ALK kinase inhibitor 1 (EML4 ALK kinase inhibitor 1) 是有效的、具有口服活性的类棘皮细胞微管相关蛋白4-间变性淋巴瘤激酶 (EML4-ALK) 的抑制剂，其 IC50 值为 1 nM。
T2649	Menin-MLL inhibitor MI-2 Menin-MLL Inhibitor,MI2,MI-2,Menin-MLL inhibitor 2,MI 2	Apoptosis; Epigenetic Reader Domain; Histone Methyltransferase	Apoptosis; Chromatin/Epigenetic
	Menin-MLL inhibitor MI-2 (MI2) 抑制Menin-MLL 相互作用，IC50为 446±28 nM。
TP1015	NFAT Inhibitor VIVIT peptide	Others	Others
	NFAT Inhibitor (VIVIT peptide) 是NFAT 的细胞渗透性肽抑制剂，能够选择性抑制钙调磷酸酶介导的NFAT 脱磷酸作用。
T2159	CaMKP Inhibitor	CaMK	Neuroscience
	CaMKP Inhibitor 可以抑制 CaMKP。
T12502	PLpro inhibitor 5-(乙酰氨基)-2-甲基-N-[(1R)-1-(1-萘基)乙基]苯甲酰胺	SARS-CoV	Microbiology/Virology
	PLpro inhibitor 是一种木瓜蛋白酶抑制剂，IC50为 2.6 µM，能抑制 SARS-CoV-2 PLpro。
T60108	PDGFR Tyrosine Kinase Inhibitor III PDGF Receptor Tyrosine Kinase Inhibitor III	PDGFR	Angiogenesis; Tyrosine Kinase/Adaptors
	PDGFR Tyrosine Kinase Inhibitor III (PDGF Receptor Tyrosine Kinase Inhibitor III) (PDGF Receptor Tyrosine Kinase Inhibitor III)是一种多激酶抑制剂，可抑制 PDGFR、EGFR、FGFR、PKA 和 PKC 等。PDGFR Tyrosine Kinase Inhibitor III 可用于肌萎缩侧索硬化症的研究。
T60119	SOD1-Derlin-1 inhibitor-1 SOD1-Derlin-1 Inhibitor 56-20	Others	Others
	SOD1-Derlin-1 inhibitor-1 (SOD1-Derlin-1 Inhibitor 56-20) (compound 56-20) 是 SOD1-Derlin-1相互作用的抑制剂。SOD1-Derlin-1 inhibitor-1 抑制 SOD1G93A-Derlin-1 复合物，IC50值为 7.11 μM。SOD1-Derlin-1 inhibitor-1 可用于肌萎缩性侧索硬化症的研究。
T10276L	AKT Kinase Inhibitor HCl AKT Kinase Inhibitor HCl(842148-40-7 Free base)	Akt	Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
	AKT Kinase Inhibitor HCl 是一种 Akt 抑制剂，具有抗肿瘤活性。
T36802L	Bisubstrate Inhibitor 78 HCl Bisubstrate Inhibitor 78 HCl(2368247-39-4 Free base)	Others	Others
	Bisubstrate Inhibitor 78 HCl 是一种 NNMT 抑制剂（IC50 = 1.41 μM），具有潜在的抗癌活性，在 100μM 时抑制HSC-2口腔癌细胞增殖。
T5452	Ehp-inhibitor-2	Ephrin Receptor	Tyrosine Kinase/Adaptors
	Ehp-inhibitor-2 是一种靶向 Eph 受体的 Eph 家族酪氨酸激酶抑制剂。

化合物

CPA inhibitor

Cat.No: T10876

Synonym: Carboxypeptidase inhibitor

Target: Carboxypeptidase

Eph inhibitor 2

Cat.No: T5451

Synonym: Ehp-inhibitor-1

Target: Ephrin Receptor

HPGDS inhibitor 1

Cat.No: T1804

Synonym: HPGDS-inhibitor-1

Target: PGE Synthase

Endotoxin Inhibitor acetate

Cat.No: TP2325L

Synonym: Endotoxin Inhibitor acetate(147396-10-9 free base)

Target: Others

USP7/USP47 inhibitor

Cat.No: T4338

Synonym: USP7/47 inhibitor-1

Target: DUB

SCD1 inhibitor-3

Cat.No: T38683

Synonym: SCD1-IN-3,SCD1 inhibitor-3,SCD1 inhibitor 17a

Target: Dehydrogenase

GOT1 inhibitor-1

Cat.No: T8766

Synonym: GOT1 inhibitor 2c

Target: Others

Raf inhibitor 1

Cat.No: T2074

Synonym: B-Raf inhibitor 1

Target: Raf

Src Inhibitor 1

Cat.No: T3593

Synonym: Src Kinase Inhibitor 1,Src-l1

Target: Src

Aurora kinase inhibitor-3

Cat.No: T5524

Synonym: Aurora Kinase Inhibitor III

Target: Aurora Kinase

PKC-theta inhibitor hcl

Cat.No: T5817

Synonym: PKC-theta inhibitor

Target: PKC

MALT1 inhibitor MI-2

Cat.No: T2350

Synonym: MALT1 inhibitor,MI 2,MI 2 (MALT1 inhibitor)

Target: MALT

B7/CD28 interaction inhibitor 1

Cat.No: T3189

Synonym: CTLA-4 inhibitor

Target: Others

JAK2 Inhibitor V

Cat.No: T3042

Synonym: JAK2 Inhibitor V Z3,Z3,NSC42834

Target: JAK

Tie2 kinase inhibitor 1

Cat.No: T6335

Synonym: Tie2 kinase inhibitor

Target: Tie-2

Syk Inhibitor II dihydrochloride

Cat.No: T4391

Synonym: Syk Inhibitor II (hydrochloride)

Target: Others, Tyrosine Kinases, Syk, PKC, BTK

Multi-kinase inhibitor 1

Cat.No: T4191

Synonym: Multi-kinase inhibitor I

Target: Others, Bcr-Abl, PDGFR, c-Kit

Carboxypeptidase G2 (CPG2) Inhibitor

Cat.No: T10678

Synonym: CPG2 Inhibitor,Carboxypeptidase G2 Inhibitor

Target: Carboxypeptidase

IRAK-1-4 Inhibitor I

Cat.No: T2457

Synonym: IRAK-1/4 Inhibitor I,IRAK-1/4 Inhibitor

Target: IRAK

HIV-1 Inhibitor 18A

Cat.No: T24141

Synonym: HIV-1 Inhibitor-18A

Target: HIV Protease

HIF-1 inhibitor-4

Cat.No: T67767

Synonym: HIF-1 inhibitor-4

Target: HIF

Aurora kinase inhibitor-2

Cat.No: T9040

Synonym: IUN-70219,Aurora Kinase Inhibitor II

Target: Aurora Kinase

Raf inhibitor 1 dihydrochloride

Cat.No: T4167

Synonym: B-Raf inhibitor 1 dihydrochloride

Target: Raf

PKCε Inhibitor Peptide acetate

Cat.No: T35827L

Synonym: PKCε Inhibitor Peptide acetate(182683-50-7 Free base)

Target: PKC

LMPTP INHIBITOR 1 hydrochloride

Cat.No: T4491

Synonym: LMPTP INHIBITOR 1 hydrochloride (1908414-82-3(free base))

Target: Phosphatase

EGFR/ErbB-2/ErbB-4 inhibitor-2

Cat.No: T21954

Synonym: EGFR/ErbB2 Inhibitor

Target: EGFR

(E/Z)-GSK-3β inhibitor 1

Cat.No: T9178

Synonym: GSK-3β inhibitor 1

Target: GSK-3

Lyn peptide inhibitor acetate

Cat.No: TP2008L

Synonym: Lyn peptide inhibitor acetate(222018-18-0 free base)

Target: IL Receptor

TRAF-STOP inhibitor 6877002

Cat.No: T17157

Synonym: CD40-TRAF6 inhibitor

Target: NF-κB

NFAT Inhibitor acetate

Cat.No: TP1015L

Synonym: VIVIT peptide acetate,NFAT Inhibitor acetate（249537-73-3 free base）

Cdk2 Inhibitor II

Cat.No: T36933

Synonym: Cdk2 Inhibitor II,CDK2-IN-3

Target: CDK

Cyt-PTPε Inhibitor-1

Cat.No: T10927

Synonym: Cyt-PTP|A Inhibitor-1

Target: Phosphatase, Src

FBPase-1 inhibitor-1

Cat.No: T22081

Synonym: Fructose 1,6-bisphosphatase-1 Inhibitor

Target: Others

PRL-3 Inhibitor I

Cat.No: T22136

Synonym: PRL-3 Inhibitor,BR-1

Target: Phosphatase, Others

PKG inhibitor peptide TFA (82801-73-8 free base)

Cat.No: TP1523

Synonym: PKG inhibitor peptide TFA

Target: PKA

Cot inhibitor-1 hydrochloride

Cat.No: T10865L

Synonym: Cot inhibitor-1 hydrochloride(915365-57-0 Free base)

Target: TNF, MAPK

LSKL, Inhibitor of Thrombospondin TSP-1 2TFA

Cat.No: T7676

Synonym: LSKL, Inhibitor of Thrombospondin TSP-1

Target: TGF-beta/Smad

BRAF inhibitor

Cat.No: T10599

Target: Raf

MLCK inhibitor peptide 18 acetate

Cat.No: TP1890L1

Synonym: MLCK inhibitor peptide 18 acetate(224579-74-2 free base)

Target: Serine/threonin kinase

PTP inhibitor 1

Cat.No: T7541

Synonym: PTP Inhibitor II,alpha-溴-4-甲氧基苯乙酮

Target: Phosphatase

EML4-ALK kinase inhibitor 1

Cat.No: T11184

Synonym: EML4 ALK kinase inhibitor 1,EML4-ALK kinase inhibitor 1

Target: ALK

Menin-MLL inhibitor MI-2

Cat.No: T2649

Synonym: Menin-MLL Inhibitor,MI2,MI-2,Menin-MLL inhibitor 2,MI 2

Target: Apoptosis, Epigenetic Reader Domain, Histone Methyltransferase

NFAT Inhibitor

Cat.No: TP1015

Synonym: VIVIT peptide

Target: Others

CaMKP Inhibitor

Cat.No: T2159

Target: CaMK

PLpro inhibitor

Cat.No: T12502

Synonym: 5-(乙酰氨基)-2-甲基-N-[(1R)-1-(1-萘基)乙基]苯甲酰胺

Target: SARS-CoV

PDGFR Tyrosine Kinase Inhibitor III

Cat.No: T60108

Synonym: PDGF Receptor Tyrosine Kinase Inhibitor III

Target: PDGFR

SOD1-Derlin-1 inhibitor-1

Cat.No: T60119

Synonym: SOD1-Derlin-1 Inhibitor 56-20

Target: Others

AKT Kinase Inhibitor HCl

Cat.No: T10276L

Synonym: AKT Kinase Inhibitor HCl(842148-40-7 Free base)

Target: Akt

Bisubstrate Inhibitor 78 HCl

Cat.No: T36802L

Synonym: Bisubstrate Inhibitor 78 HCl(2368247-39-4 Free base)

Target: Others

Ehp-inhibitor-2

Cat.No: T5452

Target: Ephrin Receptor

Cat. No.	Product Name	Target	Signaling Pathways
T3384	Wedelolactone 蟛蜞菊内酯,IKK Inhibitor II	Apoptosis; NF-κB; Lipoxygenase; Caspase	Apoptosis; Metabolism; NF-κB; Proteases/Proteasome
	Wedelolactone (IKK Inhibitor II) 是来自旱莲草的一种天然产物，通过阻断 IκBα 的磷酸化和降解来抑制细胞中 NF-κB 介导的基因转录，具有抗癌，抗炎和抗氧化活性。
T14961	Chrysene 䓛,屈	Others	Others
	Chrysene 是高分子量 (HMW) 多环芳烃，有极强的顽固性和致癌性。
TJS0851	Plantagoside	Others	Others
	Plantagoside 是α-mannosidase 的非竞争性特异性抑制剂(IC50:5 μM)，分离自Plantago asiatica 种子中。
T39049	Yubeinine	Others	Others
	Yubeinine 是一种生物碱类天然产物，可以起到气管松弛作用。
TN1455	Bryodulcosigenin	Immunology/Inflammation related	Immunology/Inflammation
	Bryodulcosigenin 是一种 Bryoniadioica 根的提取物，具有抗炎活性。
T8194	Isoflavone	Antioxidant	oxidation-reduction
	Isoflavone 是大豆植物雌激素和生物活性成分，存在于大豆、青豆、花生、鹰嘴豆和苜蓿等几种重要的豆类作物中。
T3S0693	Blinin	Others	Others
	Blinin 是一种二萜，分离自植物 Conyza blinii 中。
T8195	Lotusine	Others	Others
	Lotusine 是一种提取自Nelumbo nucifera Gaertn 的绿色种胚中的纯生物碱。它能够作用于心肌中动作电位及心脏浦肯野纤维缓慢内向电流。
TN1028	Militarine	Others	Others
	Militarine 是一种糖苷化合物，分离自 Bletilla striata，能够抑制植物生长。
TN3548	Bulleyanin	Others	Others
	Bulleyanin 是从 isodon species (Labiatae) 中分离出来的一种物质。
T5747	ISOBERGAPTEN	Others	Others
	Isobergapten 是一种化感抑制剂，分离自Hevacleum laciniatum 种子。
TN1785	Isomagnolone	Others	Others
	Isomagnolone 是一种分离自八角茴香中的天然产物，具有抗炎作用。
TN1829	Kakkalide	Dehydrogenase	Metabolism
	Kakkalide 是提取自葛根花中的一种异黄酮。它可以抑制活性氧相关炎症，并改善内皮细胞胰岛素抵抗作用。
T8203	Gentianose	Others	Others
	Gentianose 是一种碳水化合储备物，来源于多年生黄龙胆贮藏根中。
T3S1729	Dihydrolycorine	Others	Others
	Dihydrolycorine 是分离自Lycoris radiate 草药中，是一种真核细胞中蛋白质合成的抑制剂。
Fr13711	Tropinone	Others	Others
	Tropinone 是一种可用作合成 Atropine 中间体的生物碱。
TN6712	yibeissine	Others	Others
	Yibeissine 是一种甾体生物碱，分离自贝母球茎中。
TQ0096	Scabertopin	Others	Others
	Scabertopin 是一种从地胆草中分离得到倍半萜内酯，具有抗癌和抑菌活性。
T8212	Dichotomitin	Others	Others
	Dichotomitin 是一种提取自Belamcanda chinensis 根茎中的异黄酮。
T3S1850	Bayogenin	Others	Others
	Bayogenin 是紫花苜蓿皂苷，一定程度上能够抑制糖原磷酸化酶的活性。
T3S2019	Lathyrol	Others	Others
	Lathyrol 是一种具有抗癌功能的天然产物。
T16943	Stigmastanol	Endogenous Metabolite	Metabolism
	Stigmastanol 是分离自Hypericum riparium 的 6-氨基衍生物。Hypericum riparium 是属于杜仲科的药用植物。
T13350	Wushanicaritin	Others	Others
	Wushanicaritin 在 DPPH 自由基清除活性测试中显示出显著的抗氧化活性，其IC50值为35.3 μM，具有抗肿瘤作用和抗炎活性。
T5789	XYLOTRIOSE	Others	Others
	Xylotriose 是双歧杆菌促生因子，是天然的低聚木糖。
T7032	Eupatorin	Others; P450	Metabolism; Others
	Eupatorin 是天然存在的黄酮，可捕获 G2-M 细胞周期，激活多个 caspase、细胞色素 C 的释放、多聚 (ADP-核糖) 聚合酶的裂解，促使凋亡细胞死亡。
TN1002	Blumeatin	ROS	Immunology/Inflammation
	Blumeatin 是从Blumea balsamiferaDC 中分离得到，对 CCl4 和硫代乙酰胺 (TAA) 所致的肝损伤表现出保护活性。
TN1833	Karacoline	NF-κB	NF-κB
	Karacoline 是发现于植物Aconitum kusnezoffii 中的一种二萜生物碱，通过 NF-κB 信号通路，抑制椎间盘退变中细胞外基质的降解。
TN1111	Arnidiol	Immunology/Inflammation related	Immunology/Inflammation
	Arnidiol 是一种五环三萜烯，从Barleria Longiflora LinnF. 中提取得到。
T8169	Decursinol	Others	Others
	Decursinol 是一种分离自Angelica gigas 的根中的、口服具有活性的抗伤害药物。它具有抗肿瘤和抗转移作用。
TN2197	Secoisolariciresinol	TNF	Apoptosis
	Secoisolariciresinol 是一种属于苯丙素类的木脂素。
T6S2252	Sweroside	Others	Others
	Sweroside 是分离自Lonicera japonica 中，具有细胞保护、抗骨质疏松和保护肝脏活性。
TN1800	Isosakuranin	Others	Others
	Isosakuranin 是一种提取自Paliurus ramosissimus果实中的天然产物,具有抗糖尿病作用。
T6S1676	Cimigenoside	Others; Gamma-secretase	Neuroscience; Others; Proteases/Proteasome; Stem Cells
	Cimigenoside 是升麻属中的一种成分,是一种 γ-分泌酶抑制剂，通过 γ-分泌酶/Notch 轴抑制人类乳腺癌细胞的增殖或转移。
TN1982	Neoglycyrol	Others	Others
	Neoglycyrol 是分离自甘草的根中的化合物。它是由传统专利药通脉养心丸中筛选得到，具有潜在心肌保护作用。
T6S0525	Farrerol	ERK; p38 MAPK; Akt	Cytoskeletal Signaling; MAPK; PI3K/Akt/mTOR signaling
	Farrerol 是一种杜鹃花的生物活性成分，具有抗氧化、抗肿瘤、抗炎、神经保护和肝保护等多种功能。
TN1075	Adynerin	Others	Others
	Adynerin 是一种发现于夹竹桃中的天然类固醇。
T5733	Xylotetraose	Others	Others
	Xylotetraose 是木聚糖的水解产物，可用于酶生化分析。Xylan 是由木糖单元组成的多糖，主要包含由纤维素连接的 β-D- 木糖单位。
TN1626	Eugenin	Others	Others
	Eugenin 是一种色酮，分离自滨海前胡，能够抗血小板聚集。
TN1137	Isobutylshikonin	Others	Others
	Isobutylshikonin 是分离自Lithospermum canescens 毛状根培养的一种紫草素色素。
TN4818	Poriol	Others	Others
	Poriol 是一种黄酮类化合物，分离自Pseudotsuga sinensis。
TN1984	Neoisoliquiritin	Others	Others
	Neoisoliquiritin 是一种提取自甘草中的活性物质。
T2O2770	Agarotetrol	Others	Others
	Agarotetrol 是一种色酮衍生物，从沉香中分离得到。
TN1983	Neoisoastilbin	IL Receptor; TNF; NO Synthase	Apoptosis; Immunology/Inflammation
	Neoisoastilbin 具有抗炎、抗氧化、抗尿酸过多等生物特性。
TN1923	Mesaconine	IL Receptor; NF-κB	Immunology/Inflammation; NF-κB
	Mesaconine 是来自 Aconitum carmichaelii Debx 的一种成分。Mesaconine 具有心脏作用和抗 NF-κB 活性。 Mesaconine 可能是麻黄附子细辛汤抗炎和免疫抑制的部分物质基础。
T5813	BYAKANGELICIN	Reductase	Endocrinology/Hormones; Metabolism
	Byakangelicin 是发现于当归根中的一种活性化合物，可作为调节剂，改善各种活性化合物 (Umb，Cur 和 Dox) 的脑积累，增强研究效果。它提高所有PXR 靶基因 (如MDR1) 的表达，并广泛的诱导药物-药物相互作用。它可抑制性激素的作用，可能会增加内源激素的分解代谢。
T3873	griffonilide	Others	Others
	Griffonilide 是一种提取自Semiaquilegia adoxoides 根中的丁烯内酯类化合物，常与紫草甙一起出现。它是一种传统抗癌药草。
T3931	Isobavachin	Others	Others
	Isobavachin 是一种分离自Psoralea morisiana 中的抗氧化剂，在A 环的8号位置有一个prenyl 基团，具有潜在的促进神经元的分化和其蛋白异戊烯化作用。
T8208	androsin	Others	Others
	Androsin 分离于印度胡黄连中，具有抗哮喘作用。
T19431	Moluccanin	Others	Others
	Moluccanin 是来自 Aleurites moluccana 的香豆素类。
TN6723	Lactiflorin	Others	Others
	Lactiflorin 是一种具有肾脏保护作用的单萜苷。
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天然产物

Cat.No: T3384

Synonym: 蟛蜞菊内酯,IKK Inhibitor II

Target: Apoptosis, NF-κB, Lipoxygenase, Caspase

Cat.No: T14961

Synonym: 䓛,屈

Target: Others

Cat.No: TJS0851

Target: Others

Cat.No: T39049

Target: Others

Bryodulcosigenin

Cat.No: TN1455

Target: Immunology/Inflammation related

Cat.No: T8194

Target: Antioxidant

Cat.No: T3S0693

Target: Others

Cat.No: T8195

Target: Others

Cat.No: TN1028

Target: Others

Cat.No: TN3548

Target: Others

Cat.No: T5747

Target: Others

Cat.No: TN1785

Target: Others

Cat.No: TN1829

Target: Dehydrogenase

Cat.No: T8203

Target: Others

Dihydrolycorine

Cat.No: T3S1729

Target: Others

Cat.No: Fr13711

Target: Others

Cat.No: TN6712

Target: Others

Cat.No: TQ0096

Target: Others

Cat.No: T8212

Target: Others

Cat.No: T3S1850

Target: Others

Cat.No: T3S2019

Target: Others

Cat.No: T16943

Target: Endogenous Metabolite

Cat.No: T13350

Target: Others

Cat.No: T5789

Target: Others

Cat.No: T7032

Target: Others, P450

Cat.No: TN1002

Target: ROS

Cat.No: TN1833

Target: NF-κB

Cat.No: TN1111

Target: Immunology/Inflammation related

Cat.No: T8169

Target: Others

Secoisolariciresinol

Cat.No: TN2197

Target: TNF

Cat.No: T6S2252

Target: Others

Cat.No: TN1800

Target: Others

Cat.No: T6S1676

Target: Others, Gamma-secretase

Cat.No: TN1982

Target: Others

Cat.No: T6S0525

Target: ERK, p38 MAPK, Akt

Cat.No: TN1075

Target: Others

Cat.No: T5733

Target: Others

Cat.No: TN1626

Target: Others

Isobutylshikonin

Cat.No: TN1137

Target: Others

Cat.No: TN4818

Target: Others

Neoisoliquiritin

Cat.No: TN1984

Target: Others

Cat.No: T2O2770

Target: Others

Cat.No: TN1983

Target: IL Receptor, TNF, NO Synthase

Cat.No: TN1923

Target: IL Receptor, NF-κB

Cat.No: T5813

Target: Reductase

Cat.No: T3873

Target: Others

Cat.No: T3931

Target: Others

Cat.No: T8208

Target: Others

Cat.No: T19431

Target: Others

Cat.No: TN6723

Target: Others

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Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPY-04815	C1 inhibitor Protein, Rat, Recombinant (His) serpin peptidase inhibitor, clade G (C1 inhibit...	Rat	HEK293 Cells
	C1 inhibitor Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 54.7 kDa and the accession number is A6HMR4.
TMPY-01183	C1 inhibitor Protein, Human, Recombinant (His) serpin peptidase inhibitor, clade G (C1 inhibit...	Human	HEK293 Cells
	C1 inhibitor Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 54.3 kDa and the accession number is E9KL26.
TMPH-00554	Trypsin inhibitor DE-3 Protein, Erythrina caffra, Recombinant (His) Trypsin inhibitor DE-3	Erythrina caffra	P. pastoris (Yeast)
	Inhibition of trypsin.
TMPY-01030	TFPI Protein, Human, Recombinant (His) TFPI1,tissue factor pathway inhibitor (lipoprotein-...	Human	HEK293 Cells
	TFPI Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 30.6 kDa and the accession number is P10646-1.
TMPY-01174	DKK1 Protein, Rhesus, Recombinant (N256Q, His) dickkopf WNT signaling pathway inhibitor 1	Rhesus	HEK293 Cells
	DKK1 Protein, Rhesus, Recombinant (N256Q, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 27.2 kDa and the accession number is XP_001098844.1.
TMPH-00520	Host-nuclease inhibitor protein gam Protein, Enterobacteria phage lambda, Recombinant (His & Myc) Host-nuclease inhibitor protein gam,gam	Escherichia phage lambda	E. coli
	Binds to host RecBCD nuclease and inhibits it thereby protecting the viral DNA against recBCD mediated degradation.
TMPY-04811	DKK1 Protein, Mouse, Recombinant (His) dickkopf WNT signaling pathway inhibitor 1,mdkk-1	Mouse	HEK293 Cells
	DKK1 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 27.6 kDa and the accession number is O54908.
TMPY-01121	DKK3 Protein, Mouse, Recombinant (His) dickkopf WNT signaling pathway inhibitor 3,C87148,A...	Mouse	HEK293 Cells
	DKK3 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 38 kDa and the accession number is Q9QUN9.
TMPY-00775	DKK1 Protein, Human, Recombinant (His) dickkopf WNT signaling pathway inhibitor 1,SK,DKK-1	Human	HEK293 Cells
	DKK1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 27.22 kDa and the accession number is I1W660.
TMPY-02731	SPINK4 Protein, Mouse, Recombinant (hFc) MPGC60,serine peptidase inhibitor, Kazal type 4,RP2...	Mouse	HEK293 Cells
	SPINK4 Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 34.5 kDa and the accession number is O35679.
TMPH-02895	Serpin A3K Protein, Mouse, Recombinant (His) Contrapsin,SPI-2,Serpina3k,Serine protease inhibitor	Mouse	P. pastoris (Yeast)
	Contrapsin inhibits trypsin-like proteases. Serpin A3K Protein, Mouse, Recombinant (His) is expressed in yeast with C-6xHis tag. The predicted molecular weight is 45.7 kDa and the accession number is P07759.
TMPY-06074	B7-H4 Protein, Cynomolgus, Rhesus, Recombinant (His) V-set domain containing T cell activation inhibitor...	Cynomolgus,Rhesus	HEK293 Cells
	B7-H4 Protein, Cynomolgus, Rhesus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.8 kDa and the accession number is A0A2K5U6P5-1.
TMPY-01474	PAI-1 Protein, Human, Recombinant (His) PAI,SERPINE1,PAI-1,serpin peptidase inhibitor, clad...	Human	HEK293 Cells
	PAI-1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 44.2 kDa and the accession number is A0A024QYT5.
TMPY-01107	TIMP-1 Protein, Human, Recombinant EPO,TIMP metallopeptidase inhibitor 1,TIMP-1,HCI,CL...	Human	HEK293 Cells
	TIMP-1 Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 21 kDa and the accession number is P01033.
TMPY-05322	B7-H4 Protein, Mouse, Recombinant (His) BC032925,B7h4,B7x,V-set domain containing T cell activation ...	Mouse	HEK293 Cells
	B7-H4 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.6 kDa and the accession number is Q7TSP5.
TMPY-01256	TBG Protein, Human, Recombinant (His) Serpin A7,serpin peptidase inhibitor, clade A (α-1 ...	Human	HEK293 Cells
	TBG Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 45.5 kDa and the accession number is P05543.
TMPY-00915	Serpin A1 Protein, Human, Recombinant (His) PRO2275,SerpinA1,serpin peptidase inhibitor, clade ...	Human	HEK293 Cells
	Serpin A1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 45.7 kDa and the accession number is P01009-1.
TMPH-02048	RNH1 Protein, Human, Recombinant (His & Myc) RNH1,Ribonuclease/angiogenin inhibitor 1,Placental ...	Human	E. coli
	RNH1 Protein, Human, Recombinant (His & Myc) is expressed in E. coli.
TMPY-00916	Antithrombin III Protein, Human, Recombinant (His) AT3D,THPH7,ATIII,AT3,Serpin C1,MGC22579,serpin peptidase	Human	HEK293 Cells
	Antithrombin III Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 50.5 kDa and the accession number is A0A024R944.
TMPH-03211	TFPI Protein, Rabbit, Recombinant (His) TFPI,Lipoprotein-associated coagulation inhibitor,E...	Rabbit	HEK293 Cells
	Inhibits factor X (X(a)) directly and, in a Xa-dependent way, inhibits VIIa/tissue factor activity, presumably by forming a quaternary Xa/LACI/VIIa/TF complex. It possesses an antithrombotic action and also the ability to associate with lipoproteins in plasma. TFPI Protein, Rabbit, Recombinant (His) is expressed in HEK293 mammalian cells with N-10xHis tag. The predicted molecular weight is 35.4 kDa and the accession number is P19761.
TMPJ-00603	TL1A/TNFSF15 Protein, Mouse, Recombinant TNFSF15,Tumor Necrosis Factor Ligand Superfamily Member 15,V...	Mouse	E. coli
	Tumor Necrosis Factor Ligand Superfamily Member 15 (TNFSF15) is a new member of the tumor necrosis factor family. TNFSF15 is predominantly an endothelial cell-specific gene, and recombinant TNFSF15 is a potent inhibitor of endothelial cell proliferation, angiogenesis and tumor growth. TNFSF15 exerts two activities on endothelial cells: early G1 arrest of G0/G1-cells responding to growth stimuli and programmed cell death of proliferating cells. These activities are highly specific to endothelial ...
TMPH-03210	TFPI Protein, Rabbit, Recombinant (E. coli, His) Lipoprotein-associated coagulation inhibitor,Extrin...	Rabbit	E. coli
	Inhibits factor X (X(a)) directly and, in a Xa-dependent way, inhibits VIIa/tissue factor activity, presumably by forming a quaternary Xa/LACI/VIIa/TF complex. It possesses an antithrombotic action and also the ability to associate with lipoproteins in plasma. TFPI Protein, Rabbit, Recombinant (E. coli, His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 35.8 kDa and the accession number is P19761.
TMPJ-00916	TIMP-2 Protein, Mouse, Recombinant (His) metalloproteinase inhibitor 2,Tissue inhibitor<...	Mouse	HEK293 Cells
	Mouse Metalloproteinase inhibitor 2(TIMP-2), belongs to a family of proteins that regulate the activation and proteolytic activity of matrix metalloproteinases (MMPs). There are four mammalian members of the family; TIMP‑1, TIMP‑2, TIMP‑3, and TIMP‑4. The TIMP-2 is detected in testis, retina, hippocampus and cerebral cortex. The function of TIMP 2 protein is to inhibit MMPs non covalently by the formation of binary complexes. Complexes with metalloproteinases (such as collagenases) and irreversi...
TMPY-03524	B7-H4 Protein, Human, Recombinant (His) PRO1291,B7X,B7H4,B7-H4,VCTN1,B7S1,B7h.5,V-set domain contain...	Human	HEK293 Cells
	B7-H4 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.8 kDa and the accession number is Q7Z7D3-1.
TMPH-02832	Serpin A5 Protein, Mouse, Recombinant (His) Protein C inhibitor,Plasminogen activator inhib...	Mouse	Baculovirus Insect Cells
	Heparin-dependent serine protease inhibitor acting in body fluids and secretions. Inactivates serine proteases by binding irreversibly to their serine activation site. Involved in the regulation of intravascular and extravascular proteolytic activities. Plays hemostatic roles in the blood plasma. Acts as a procoagulant and proinflammatory factor by inhibiting the anticoagulant activated protein C factor as well as the generation of activated protein C factor by the thrombin/thrombomodulin comple...
TMPH-00155	Barstar Protein, Bacillus amyloliquefaciens, Recombinant (His & Myc) Barstar,Ribonuclease inhibitor	Bacillus amyloliquefaciens	E. coli
	Inhibitor of the ribonuclease barnase. Forms a one-to-one non-covalent complex. Barstar Protein, Bacillus amyloliquefaciens, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 17.7 kDa and the accession number is P11540.
TMPH-02782	TIMP4 Protein, Mouse, Recombinant (His & SUMO) Timp4,Metalloproteinase inhibitor 4,Tissue inhi...	Mouse	E. coli
	TIMP4 Protein, Mouse, Recombinant (His & SUMO) is expressed in E. coli.
TMPH-02408	SPI Protein, Lentinula edodes, Recombinant (His) Serine protease inhibitor	Lentinula edodes	E. coli
	Serine protease inhibitor. Active against beta-trypsin and alpha-chymotrypsin with dissociation constants of 0.35 nM and 40 nM respectively. Inhibits factor XIa, but not other enzymes involved in coagulation and fibrinolysis. Does not inhibit subtilisin, lysyl endopeptidase, arginyl endopeptidase or papain.
TMPJ-00490	Serpin A5 Protein, Human, Recombinant (His) Plasminogen Activator Inhibitor 3,Acrosomal Serine ...	Human	HEK293 Cells
	Serpin A5 is a member of the human Serpin superfamily consists of at least 35 members. It is synthesized in the liver and has been detected in saliva, cerebral spinal fluid, amniotic fluid, tears and semen. As a potent inhibitor of the protein C anticoagulant pathway at the levels of both zymogen activation and enzyme inhibition, Serpin A5 additionally inhibits a variety of serine protease including thrombin, factor Xa, several kallekreins and acrosin. It plays a critical role in the processes o...
TMPJ-01289	TIMP-4 Protein, Human, Recombinant (His) TIMP4,TIMP-4,Metalloproteinase inhibitor 4,Tissue <...	Human	HEK293 Cells
	Metalloproteinase inhibitor 4 is an enzyme that in humans is encoded by the TIMP4 gene, belongs to the protease inhibitor I35 (TIMP) family. The protein complexes with metalloproteinases (such as collagenases) and irreversibly inactivates them by binding to their catalytic zinc cofactor. Known to act on MMP-1, MMP-2, MMP-3, MMP-7 and MMP-9.
TMPH-01869	PAI-2 Protein, Human, Recombinant (His) SERPINB2,Urokinase inhibitor,Placental plasminogen ...	Human	HEK293 Cells
	Inhibits urokinase-type plasminogen activator. The monocyte derived PAI-2 is distinct from the endothelial cell-derived PAI-1. PAI-2 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with N-10xHis tag. The predicted molecular weight is 50.1 kDa and the accession number is P05120.
TMPY-03876	PTGFRN Protein, Cynomolgus, Recombinant (His) prostaglandin F2 receptor inhibitor	Cynomolgus	HEK293 Cells
	EWI-F, also known as PTGFRN, is inversely related to the loss of CD9. Its expression correlates with the metastatic status of hLT. EWI-F inhibits the binding of prostaglandin F2-alpha (PGF2-alpha) to its specific FP receptor, by decreasing the receptor number rather than the affinity constant. EWI-F expression positively correlates with the metastatic status of hLT, and that the upregulation of EWI-F expression could be one of the mechanisms underlying the loss of CD9 in solid tumours.
TMPY-02912	TIMP-1 Protein, Rat, Recombinant TIMP metallopeptidase inhibitor 1	Rat	HEK293 Cells
	TIMP-1 Protein, Rat, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 21.5 kDa and the accession number is P01860.
TMPH-03119	SERPINB1 Protein, Pig, Recombinant (His & Myc) Leukocyte elastase inhibitor,Serpin B1,Leukocyte ne...	Sus scrofa (Pig)	E. coli
	SERPINB1 Protein, Pig, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 50.0 kDa and the accession number is P80229.
TMPJ-00733	SPINK1 Protein, Human, Recombinant (His) PSTI,Pancreatic Secretory Trypsin Inhibitor,TATI,Se...	Human	HEK293 Cells
	Serine Protease Inhibitor Kazal-Type 1 (SPINK1) is a trypsin inhibitor that prevent the trypsin-catalyzed premature activation of zymogens within the pancreas. Defects in SPINK1 are a cause of pancreatitis (PCTT). A disease characterized by the presence of calculi in pancreatic ducts. It causes severe abdominal pain attacks. Defects in SPINK1 are the cause of susceptibility to tropical calcific pancreatitis (TCP). Recombinant SPINK1 protein (rSPINK1) stimulated cell proliferation in benign RWPE ...
TMPY-05179	TFPI Protein, Human, Recombinant (His), Biotinylated TFI,TFPI1,EPI,LACI,tissue factor pathway inhibitor ...	Human	HEK293 Cells
	TFPI Protein, Human, Recombinant (His), Biotinylated is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 30.6 kDa and the accession number is P10646-1.
TMPH-02834	PAI-1 Protein, Mouse, Recombinant (His & SUMO) Endothelial plasminogen activator inhibitor,Serpine...	Mouse	E. coli
	Serine protease inhibitor. Inhibits TMPRSS7. Is a primary inhibitor of tissue-type plasminogen activator (PLAT) and urokinase-type plasminogen activator (PLAU). As PLAT inhibitor, it is required for fibrinolysis down-regulation and is responsible for the controlled degradation of blood clots. As PLAU inhibitor, it is involved in the regulation of cell adhesion and spreading. Acts as a regulator of cell migration, independently of its role as protease inhibitor. It is required for stimulation of ...
TMPH-01994	GDI2 Protein, Human, Recombinant (His) Rab GDP dissociation inhibitor beta,Guanosine dipho...	Human	P. pastoris (Yeast)
	Regulates the GDP/GTP exchange reaction of most Rab proteins by inhibiting the dissociation of GDP from them, and the subsequent binding of GTP to them. GDI2 Protein, Human, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 52.7 kDa and the accession number is P50395.
TMPH-02833	PAI-1 Protein, Mouse, Recombinant (His) Endothelial plasminogen activator inhibitor,Plasmin...	Mouse	P. pastoris (Yeast)
	PAI-1 Protein, Mouse, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 44.9 kDa and the accession number is P22777.
TMPY-05800	IKB beta/NFKBIB Protein, Human, Recombinant (GST) NFKB inhibitor β,NFKB inhibitor beta,TRIP9...	Human	E. coli
	NFKBIB (NFKB Inhibitor Beta) is a Protein Coding gene. The protein encoded by this gene belongs to the NF-kappa-B inhibitor family, which inhibits NF-kappa-B by complexing with and trapping it in the cytoplasm. Phosphorylation of serine residues on these proteins by kinases marks them for destruction via the ubiquitination pathway, thereby allowing activation of the NF-kappa-B, which translocates to the nucleus to function as a transcription factor. NF-kappaB regulation involves the inhibitor pr...
TMPH-00478	DIT33 Protein, Dirofilaria immitis, Recombinant (His & Myc) Pepsin inhibitor Dit33,DIT33	Dirofilaria immitis	E. coli
	Aspartyl protease inhibitor. DIT33 Protein, Dirofilaria immitis, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 32.0 kDa and the accession number is Q27384.
TMPY-00163	SPINK2 Protein, Human, Recombinant (hFc) serine peptidase inhibitor, Kazal type 2 (acrosin-t...	Human	HEK293 Cells
	Human serine proteinase inhibitor Kazal-type 2 (SPINK2) functions as a trypsin/acrosin inhibitor and is synthesized mainly in the testis and seminal vesicle where its activity is engaged in fertility. The SPINK2 protein contains a typical Kazal domain composed by six cysteine residues forming three disulfide bridges. The expression of SPINK2 is closely related to cancer such as lymphomas, in that a high transcript level of SPINK2 in patients with primary cutaneous follicle center cell lymphomas ...
TMPH-00832	PAI-1 Protein, Horse, Recombinant (E. coli) Endothelial plasminogen activator inhibitor,PAI-1,P...	Horse	E. coli
	PAI-1 Protein, Horse, Recombinant (E. coli) is expressed in E. coli expression system. The predicted molecular weight is 32.1 kDa and the accession number is Q8MI31.
TMPH-00356	PAI-1 Protein, Feline, Recombinant PAI-1,Endothelial plasminogen activator inhibitor,S...	Feline	E. coli
	PAI-1 Protein, Feline, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 29.7 kDa and the accession number is A9NJ78.
TMPJ-00101	TIMP-2 Protein, Human, Recombinant (His) Tissue Inhibitor of Metalloproteinases 2,TIMP2,CSC-...	Human	HEK293 Cells
	Tissue inhibitors of metalloproteinases or TIMPs are a family of proteins that regulate the activation and proteolytic activity of the zinc enzymes known as matrix metalloproteinases (MMPs). There are four members of the family, TIMP-1, TIMP-2, TIMP-3, and TIMP-4. Tissue Inhibitor of Metalloproteinases 2 (TIMP-2) is a non N-glycosylated protein with a molecular mass of 22 kDa. It produced by a wide range of cell types, which inhibits MMPs non-covalently by the formation of binary complexes and i...
TMPH-01665	TIMP3 Protein, Human, Recombinant (His) Tissue inhibitor of metalloproteinases 3,TIMP3,Prot...	Human	E. coli
	Complexes with metalloproteinases (such as collagenases) and irreversibly inactivates them by binding to their catalytic zinc cofactor. May form part of a tissue-specific acute response to remodeling stimuli. Known to act on MMP-1, MMP-2, MMP-3, MMP-7, MMP-9, MMP-13, MMP-14 and MMP-15.
TMPJ-00625	Serpin E1 Protein, Mouse, Recombinant (His) Pai1,Planh1,Plasminogen activator inhibitor 1,Serpi...	Mouse	HEK293 Cells
	Plasminogen activator inhibitor-1 (serpin E1) is a serine protease inhibitor which belongs to the serpin family. Serpin E1 acts as 'bait' for tissue plasminogen activator, urokinase, protein C and matriptase-3/TMPRSS7. Its rapid interaction with PLAT may function as a major control point in the regulation of fibrinolysis.
TMPY-00928	TFPI Protein, Mouse, Recombinant (His) AW552122,A630013F22Rik,tissue factor pathway inhibitor	Mouse	HEK293 Cells
	TFPI Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 31 kDa and the accession number is O54819-1.
TMPJ-00972	CDKN1B Protein, Human, Recombinant (His) KIP1,CDKN1B,Cyclin-Dependent Kinase Inhibitor p27,C...	Human	E. coli
	Cyclin-Dependent Kinase Inhibitor 1B (CDKN1B) is a Kinesin-related motor protein necessary for mitotic spindle assembly and chromosome segregation. CDKN1B is expressed in all tissues with highest levels observed in skeletal muscle. CDKN1B is a potent inhibitor of Cyclin E- and Cyclin A-CDK2 complexes. CDKN1B forms a complex with Cyclin Type D-CDK4 complexes and is involved in the assembly, stability, and modulation of CCND1-CDK4 complex activation. In addition, CDKN1B acts as an inhibitor or an ...
TMPH-03578	SCIN Protein, S. aureus, Recombinant (His & Myc) scn,Staphylococcal complement inhibitor	Staphylococcus aureus	E. coli
	Involved in countering the first line of host defense mechanisms. Efficiently inhibits opsonization, phagocytosis and killing of S.aureus by human neutrophils. Acts by binding and stabilizing human C3 convertases (C4b2a and C3bBb), leading to their inactivation. The convertases are no longer able to cleave complement C3, therefore preventing further C3b deposition on the bacterial surface and phagocytosis of the bacterium. Also prevents C5a-induced neutrophil responses. SCIN Protein, S. aureus, ...
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重组蛋白

C1 inhibitor Protein, Rat, Recombinant (His)

Cat.No: TMPY-04815

Species: Rat

Expression System: HEK293 Cells

C1 inhibitor Protein, Human, Recombinant (His)

Cat.No: TMPY-01183

Species: Human

Expression System: HEK293 Cells

Trypsin inhibitor DE-3 Protein, Erythrina caffra, Recombinant (His)

Cat.No: TMPH-00554

Species: Erythrina caffra

Expression System: P. pastoris (Yeast)

TFPI Protein, Human, Recombinant (His)

Cat.No: TMPY-01030

Species: Human

Expression System: HEK293 Cells

DKK1 Protein, Rhesus, Recombinant (N256Q, His)

Cat.No: TMPY-01174

Species: Rhesus

Expression System: HEK293 Cells

Host-nuclease inhibitor protein gam Protein, Enterobacteria phage lambda, Recombinant (His & Myc)

Cat.No: TMPH-00520

Species: Escherichia phage lambda

Expression System: E. coli

DKK1 Protein, Mouse, Recombinant (His)

Cat.No: TMPY-04811

Species: Mouse

Expression System: HEK293 Cells

DKK3 Protein, Mouse, Recombinant (His)

Cat.No: TMPY-01121

Species: Mouse

Expression System: HEK293 Cells

DKK1 Protein, Human, Recombinant (His)

Cat.No: TMPY-00775

Species: Human

Expression System: HEK293 Cells

SPINK4 Protein, Mouse, Recombinant (hFc)

Cat.No: TMPY-02731

Species: Mouse

Expression System: HEK293 Cells

Serpin A3K Protein, Mouse, Recombinant (His)

Cat.No: TMPH-02895

Species: Mouse

Expression System: P. pastoris (Yeast)

B7-H4 Protein, Cynomolgus, Rhesus, Recombinant (His)

Cat.No: TMPY-06074

Species: Cynomolgus,Rhesus

Expression System: HEK293 Cells

PAI-1 Protein, Human, Recombinant (His)

Cat.No: TMPY-01474

Species: Human

Expression System: HEK293 Cells

TIMP-1 Protein, Human, Recombinant

Cat.No: TMPY-01107

Species: Human

Expression System: HEK293 Cells

B7-H4 Protein, Mouse, Recombinant (His)

Cat.No: TMPY-05322

Species: Mouse

Expression System: HEK293 Cells

TBG Protein, Human, Recombinant (His)

Cat.No: TMPY-01256

Species: Human

Expression System: HEK293 Cells

Serpin A1 Protein, Human, Recombinant (His)

Cat.No: TMPY-00915

Species: Human

Expression System: HEK293 Cells

RNH1 Protein, Human, Recombinant (His & Myc)

Cat.No: TMPH-02048

Species: Human

Expression System: E. coli

Antithrombin III Protein, Human, Recombinant (His)

Cat.No: TMPY-00916

Species: Human

Expression System: HEK293 Cells

TFPI Protein, Rabbit, Recombinant (His)

Cat.No: TMPH-03211

Species: Rabbit

Expression System: HEK293 Cells

TL1A/TNFSF15 Protein, Mouse, Recombinant

Cat.No: TMPJ-00603

Species: Mouse

Expression System: E. coli

TFPI Protein, Rabbit, Recombinant (E. coli, His)

Cat.No: TMPH-03210

Species: Rabbit

Expression System: E. coli

TIMP-2 Protein, Mouse, Recombinant (His)

Cat.No: TMPJ-00916

Species: Mouse

Expression System: HEK293 Cells

B7-H4 Protein, Human, Recombinant (His)

Cat.No: TMPY-03524

Species: Human

Expression System: HEK293 Cells

Serpin A5 Protein, Mouse, Recombinant (His)

Cat.No: TMPH-02832

Species: Mouse

Expression System: Baculovirus Insect Cells

Barstar Protein, Bacillus amyloliquefaciens, Recombinant (His & Myc)

Cat.No: TMPH-00155

Species: Bacillus amyloliquefaciens

Expression System: E. coli

TIMP4 Protein, Mouse, Recombinant (His & SUMO)

Cat.No: TMPH-02782

Species: Mouse

Expression System: E. coli

SPI Protein, Lentinula edodes, Recombinant (His)

Cat.No: TMPH-02408

Species: Lentinula edodes

Expression System: E. coli

Serpin A5 Protein, Human, Recombinant (His)

Cat.No: TMPJ-00490

Species: Human

Expression System: HEK293 Cells

TIMP-4 Protein, Human, Recombinant (His)

Cat.No: TMPJ-01289

Species: Human

Expression System: HEK293 Cells

PAI-2 Protein, Human, Recombinant (His)

Cat.No: TMPH-01869

Species: Human

Expression System: HEK293 Cells

PTGFRN Protein, Cynomolgus, Recombinant (His)

Cat.No: TMPY-03876

Species: Cynomolgus

Expression System: HEK293 Cells

TIMP-1 Protein, Rat, Recombinant

Cat.No: TMPY-02912

Species: Rat

Expression System: HEK293 Cells

SERPINB1 Protein, Pig, Recombinant (His & Myc)

Cat.No: TMPH-03119

Species: Sus scrofa (Pig)

Expression System: E. coli

SPINK1 Protein, Human, Recombinant (His)

Cat.No: TMPJ-00733

Species: Human

Expression System: HEK293 Cells

TFPI Protein, Human, Recombinant (His), Biotinylated

Cat.No: TMPY-05179

Species: Human

Expression System: HEK293 Cells

PAI-1 Protein, Mouse, Recombinant (His & SUMO)

Cat.No: TMPH-02834

Species: Mouse

Expression System: E. coli

GDI2 Protein, Human, Recombinant (His)

Cat.No: TMPH-01994

Species: Human

Expression System: P. pastoris (Yeast)

PAI-1 Protein, Mouse, Recombinant (His)

Cat.No: TMPH-02833

Species: Mouse

Expression System: P. pastoris (Yeast)

IKB beta/NFKBIB Protein, Human, Recombinant (GST)

Cat.No: TMPY-05800

Species: Human

Expression System: E. coli

DIT33 Protein, Dirofilaria immitis, Recombinant (His & Myc)

Cat.No: TMPH-00478

Species: Dirofilaria immitis

Expression System: E. coli

SPINK2 Protein, Human, Recombinant (hFc)

Cat.No: TMPY-00163

Species: Human

Expression System: HEK293 Cells

PAI-1 Protein, Horse, Recombinant (E. coli)

Cat.No: TMPH-00832

Species: Horse

Expression System: E. coli

PAI-1 Protein, Feline, Recombinant

Cat.No: TMPH-00356

Species: Feline

Expression System: E. coli

TIMP-2 Protein, Human, Recombinant (His)

Cat.No: TMPJ-00101

Species: Human

Expression System: HEK293 Cells

TIMP3 Protein, Human, Recombinant (His)

Cat.No: TMPH-01665

Species: Human

Expression System: E. coli

Serpin E1 Protein, Mouse, Recombinant (His)

Cat.No: TMPJ-00625

Species: Mouse

Expression System: HEK293 Cells

TFPI Protein, Mouse, Recombinant (His)

Cat.No: TMPY-00928

Species: Mouse

Expression System: HEK293 Cells

CDKN1B Protein, Human, Recombinant (His)

Cat.No: TMPJ-00972

Species: Human

Expression System: E. coli

SCIN Protein, S. aureus, Recombinant (His & Myc)

Cat.No: TMPH-03578

Species: Staphylococcus aureus

Expression System: E. coli

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Cat. No.	Product Name	Target	Signaling Pathways
T24046	WNK-IN-11-d3 WNK inhibitor-12,WNKIN12,WNK IN 12,WNK inhibitor 12,WNK-IN-12
	WNK-IN-12 is an effective, selective, and orally active WNK1 kinase inhibitor.
T14687	Deucravacitinib BMS-986165	Tyrosine Kinases; JAK; IFNAR; Interleukin	Angiogenesis; Chromatin/Epigenetic; Immunology/Inflammation; JAK/STAT signaling; Stem Cells; Tyrosine Kinase/Adaptors
	Deucravacitinib (BMS-986165) 是一种高选择性、口服生物可利用的变构 TYK2 抑制剂，用于治疗自身免疫性疾病。它通过稳定调节 JH2 结构域来阻断受体介导的 Tyk2 激活，可抑制IL-12/23和 I 型IFN 途径。它选择性结合 TYK2 假激酶 (JH2) 结构域，IC50为1.0 nM。
T22301	L-838417 D9 CTP354,CTP354 (C-21191),C-21191	GABA Receptor	Membrane transporter/Ion channel; Neuroscience
	L-838417 D9 (C-21191) 是 L-838417 的氘代物。其中L-838417 是亚型选择性GABAA 正变构调节剂，在 α2, α3 和 α5 亚型中作为部分激动剂。
T9087	Creatine-d3 hydrate CREATINE-(METHYL-D3) MONOHYDRATE,肌氨酸酐-甲基-D3 一水合物	Endogenous Metabolite	Metabolism
	Creatine-d3 hydrate (CREATINE-(METHYL-D3) MONOHYDRATE) 是一种氘标记的肌酸水合物。其中肌酸水合物在肌肉和脑细胞的能量代谢中起着关键作用。
T40376	L-Phenylalanine-15N L-苯丙氨酸 15N,(S)-2-Amino-3-phenylpropionic acid-15N,L-Phenylalanine-15N	Calcium Channel	Membrane transporter/Ion channel; Metabolism
	L-Phenylalanine-15N ((S)-2-Amino-3-phenylpropionic acid-15N) 是 15N 标记的 L-Phenylalanine。L-Phenylalanine 是从大肠杆菌中分离出来的一种必需氨基酸。 L-Phenylalanine 广泛用于食品香精和药物的生产。
T13446	(S)-Rivastigmine D6 tartrate 酒石酸卡巴拉汀 D6,(R)-卡巴拉汀酒石盐酸-D6,(R)-Rivastigmine D6 tartrate	AChE	Neuroscience
	(S)-Rivastigmine D6 tartrate 是一种 (S)-Rivastigmine 氘代化合物。
T16909	Donafenib Sorafenib (D3),Bay 43-9006 (D3),Sorafenib-d3	Raf; VEGFR	Angiogenesis; MAPK; Tyrosine Kinase/Adaptors
	Donafenib (Bay 43-9006 (D3)) 是一种氘标记的 Sorafenib，Sorafenib 是一种多激酶抑制剂(对 Raf-1、B-Raf 和 VEGFR-3 的 IC50 分别为 6 nM、20 nM 和 22 nM)。
T11067	VX-984 M9831	DNA-PK	DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
	VX-984 (M9831) 是一种可口服的、具有选择性的的、可透过血脑屏障的 DNA-PK 抑制剂。VX-984 对非同源性末端 NHEJ 的接合具有抑制作用，可作用于 DSBs 使 DNA 双链断裂。VX-984常见于对胶质母细胞瘤 (GBM) 和非小细胞肺癌 (NSC-LC) 的研究。
T10948	MMAE-d8 D8-MMAE,D8-Monomethyl auristatin E	ADC Cytotoxin	Antibody-drug Conjugate/ADC Related
	D8-MMAE (D8-Monomethyl auristatin E) is an effective mitotic inhibitor and tubulin inhibitor, deuterated MMAE.
T69462	Deulinoleic acid
	Deulinoleic acid is a lipid peroxidation inhibitor and antioxidant.
T27097	CTP518 CTP 518,Deuterated Atazanivir-D3-1,CTP-518
	CTP518, a deuterated Atazanivir derivative, is a HIV protease inhibitor.
T26871	BMT-052 BMT052
	BMT-052 is a potent and selective Pan-genotypic HCV NS5B Polymerase Inhibitor (EC50 = 7 nM).
T11192	Enalapril D5 maleate MK-421 D5 maleate,马来酸依那普利D5	Others	Others
	Enalapril D5 maleate is deuterium labeled Enalapril, which is an angiotensin converting enzyme (ACE) inhibitor.
T11194	Enalaprilat D5 MK-422 D5,依那普利拉 D5	Others	Others
	Enalaprilat D5 is the deuterium labeled Enalaprilat, which is an angiotensin-converting enzyme (ACE) inhibitor.
T12571	PSI-6206 13C,d3 Sofosbuvir metabolite GS-331007 13CD3,RO-2433 13CD3,PSI-6206 13CD3,GS-331007 13CD3	Others	Others
	PSI-6206 13CD3 is the deuterium labeled PSI-6206. PSI-6206 is a potent and selective HCV NS5B polymerase inhibitor.
T13181	Tolcapone D7 Ro 40-7592 D7	Transferase	Metabolism
	Tolcapone D7 is a deuterium-labeled Tolcapone. Tolcapone is a selective and orally active inhibitor of COMT.
T11193	Enalaprilat-d5 sodium MK-422 D5 Sodium Salt,依那普利拉钠 D5,Enalaprilat D5 Sodium Salt	Others	Others
	Enalaprilat D5 Sodium Salt is the deuterium labeled Enalaprilat, which is an angiotensin-converting enzyme (ACE) inhibitor.
TMIH-0297	Ledipasvir-d6
	Ledipasvir-d6 是 Ledipasvir 的氘代化合物。Ledipasvir 的 CAS 号为 1256388-51-8。Ledipasvir 是一种丙型肝炎病毒 NS5A 抑制剂。它也是 P-糖蛋白抑制剂和乳腺癌抗性蛋白抑制剂。
T11814	Lamivudine 13C,15N2	Others	Others
	Lamivudine 13C,15N2, an impurity of Lamivudine (BCH-189), functions as an inhibitor of both HIV-1/2 reverse transcriptase and hepatitis B virus reverse transcriptase, classifying it as a nucleoside reverse transcriptase inhibitor (NRTIs).
T13235	Tyk2-IN-7	Others	Others
	Tyk2-IN-7 is an inhibitor of TYK2 JH2, binds to the TYK2 JH2 domain (IC50: 0.00053 μM; Ki.app: 0.00007 μM).
TMIJ-0326	Cyclosporin A-d4 (Major)
	Cyclosporin A-d4 (Major) 是 Cyclosporin A 的氘代化合物。Cyclosporin A 的 CAS 号为 59865-13-3。Cyclosporine A 是一种能与亲环素结合的抑制剂。根据它的作用机制可作为钙调神经磷酸酶抑制剂、细胞色素 P450 3A4 抑制剂和 P-糖蛋白抑制剂。
T12046	Mirtazapine D3 Org3770 D3,6-Azamianserin D3,米氮平 D3	5-HT Receptor	GPCR/G Protein; Neuroscience
	Mirtazapine D3 is a deuterium labeled Mirtazapine. Mirtazapine is an inhibitor of 5-HT receptor .
T11270	Febuxostat D9 非布司他D9	Others	Others
	Febuxostat D9 is deuterium labeled Febuxostat, which is a selective xanthine oxidase inhibitor with Ki of 0.6 nM.
T11610	Idelalisib D5 CAL-101 D5,GS-1101 D5	PI3K	PI3K/Akt/mTOR signaling
	Idelalisib D5 is a deuterium-labeled Idelalisib. Idelalisib is a highly selective and orally bioavailable p110δ inhibitor.
T11229	Erlotinib-d6 OSI-774 D6,NSC 718781 D6,CP-358774 D6	Others	Others
	Erlotinib is a directly acting inhibitor EGFR tyrosine kinase inhibitor with an IC50 of 2 nM for human EGFR. Erlotinib D6 is a deuterium labeled Erlotinib .
T10256	Afatinib D6 BIBW 2992 D6	EGFR	Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
	Afatinib D6 (BIBW 2992 D6) is a deuterium-labeled Afatinib. Afatinib is an irreversible EGFR family inhibitor.
T10915	Cycloguanil D6 Nitrate Chlorguanide triazine D6 Nitrate	Others	Others
	Cycloguanil D6 Nitrate is a dihydrofolate reductase inhibitor, deuterium-labeled Cycloguanil.
T12587	Pyridostigmine-d6 bromide Pyridostigmine D6 bromide,溴化吡啶斯的明 D6	Others	Others
	Pyridostigmine D6 bromide is the deuterium labeled Pyridostigmine, which is a parasympathomimetic and a reversible inhibitor of cholinesterase.
T12308	Omeprazole-d3 奥美拉挫 D3,H 16868 D3	Others	Others
	Omeprazole D3 is deuterium labeled Omeprazole. Omeprazole is a proton pump inhibitor (PPI)
T11816	Lansoprazole-d4 AG-1749 D4,Lansoprazole D4	Proton pump	Membrane transporter/Ion channel
	Lansoprazole D4 (AG-1749 D4) is a deuterium labeled Lansoprazole. Lansoprazole is an inhibitor of proton pump which prevents the stomach from producing acid.
T10669	Canagliflozin-d4 Canagliflozin D4	Others	Others
	Canagliflozin D4 is a deuterium-labeled Canagliflozin. Canagliflozin is an SGLT2 inhibitor.
TMIH-0187	Dexlansoprazole-d4 (R)-Lansoprazole-d4
	Dexlansoprazole-d4 是 Dexlansoprazole 的氘代化合物。Dexlansoprazole 的 CAS 号为 138530-94-6。(R)-Lansoprazole 是Lansoprazole 的R型异构体。Lansoprazole 是口服有效的质子泵抑制剂，能抑制胃酸生成。Lansoprazole 是中性鞘磷脂酶(N-SMase)的抑制剂(外泌体抑制剂)，能透过血脑屏障。
T10916	Cycloguanil D6 Chlorguanide triazine D6	Others	Others
	Cycloguanil D6 is a dihydrofolate reductase inhibitor, deuterium-labeled Cycloguanil.
T10284	ALK-IN-6	Others	Others
	ALK-IN-6 is an orally bioavailable inhibitor of anaplastic lymphoma kinase (ALK, IC50s: 71 nM, 18.72 nM, and 36.81 nM for ALK wild, ALK F1196M and ALK F1174L).
T10231	Acetazolamide-d3 醋氮酰胺 D3	Others	Others
	Acetazolamide D3 is a deuterium-labeled Acetazolamide. Acetazolamide is a potent carbonic anhydrase inhibitor.
T10958	Dapagliflozin-d5 BMS-512148 D5	Others	Others
	Dapagliflozin D5 (BMS-512148 D5) is deuterated Dapagliflozin. Dapagliflozin is a competitive SGLT2 inhibitor.
T12355	Palbociclib-d8 PD 0332991 D8,Palbociclib D8	CDK	Cell Cycle/Checkpoint
	Palbociclib D8 is a deuterium labeled Palbociclib. Palbociclib is a selective and orally active inhibitor of CDK4 and CDK6 (IC50s of 11 and 16 nM, respectively).
T12208	Nepafenac-d5 奈帕芬胺 D5,AHR-9434 D5,AL-6515 D5	Others	Others
	Nepafenac D5 is the deuterium labeled Nepafenac, which is a selective inhibitor of COX-2 .
T13137	TGFβRI-IN-1	TGF-beta/Smad	Stem Cells
	TGFβRI-IN-1 is an oral active and selective inhibitor of TGFβ receptor type I (TGFβRI) kinase(IC50 values of 2 nM and 7.6 μM for TGFβRI and TGFβRII, respectively ).
TMID-0196	Allopurinol-d2
	Allopurinol-d2 是 Allopurinol 的氘代化合物。Allopurinol 的 CAS 号为 315-30-0。Allopurinol 是一种黄嘌呤氧化酶（XO）抑制剂，IC50=7.82±0.12 μM。
TMIJ-0110	Clarithromycin-13C-d3
	Clarithromycin-13C-d3 是 Clarithromycin 的 13C 和氘代化合物。Clarithromycin 的 CAS 号为 81103-11-9。Clarithromycin 具有广谱的抗菌活性。它抑制CYP3A4催化的三唑仑 α-羟基化，IC50(Ki) 值为 56 (43) μM。它抑制 HERG 钾电流。它可削弱连接 hERG1 和 PI3K 的信号通路影响自噬流。
T70214	BMS-986202
	BMS-986202 is a novel Tyk2 inhibitor, binding to Tyk2 JH2, showing efficacies for IL-23-driven acanthosis, anti-CD40-induced colitis, and spontaneous lupus.
T11601	Ibrutinib-d5 PCI-32765 D5,Ibrutinib D5	Others	Others
	Ibrutinib D5 is a deuterium-labeled Ibrutinib. Ibrutinib is an irreversible Btk inhibitor.
T10288	Alogliptin (13CD3) SYR-322 (13CD3)	Others	Others
	Alogliptin (SYR-322) 13CD3 is the deuterium-labeled Alogliptin. Alogliptin is a selective inhibitor of DPP-4.
T12701	(rel)-Tranylcypromine D5 hydrochloride 2-Phenylcyclopropylamine D5 hydrochloride	Histone Demethylase	Chromatin/Epigenetic
	(rel)-Tranylcypromine D5 hydrochloride is a deuterium labeled (rel)-Tranylcypromine hydrochloride. (rel)-Tranylcypromine hydrochloride is an irreversible, nonselective inhibitor of monoamine oxidase (MAO) used in the treatment of depression.
T12292	Olaparib-d5 KU0059436 D5,AZD2281 D5,Olaparib D5	Others	Others
	Olaparib D5 is a deuterium labeled Olaparib. Olaparib is a potent and oral inhibitor of PARP.
TMIJ-0133	Empagliflozin-d4
	Empagliflozin-d4 是 Empagliflozin 的氘代化合物。Empagliflozin 的 CAS 号为 864070-44-0。Empagliflozin 是有效的、选择性的钠葡萄糖协同转运蛋白-2 (SGLT-2) 抑制剂，对人 SGLT-2 的IC50为 3.1 nM。
T11250	Ezetimibe-d4 SCH 58235 D4	Others	Others
	Ezetimibe D4, a deuterium-labeled variant of Ezetimibe, functions as an inhibitor of Niemann-Pick C1-like1 (NPC1L1) and is recognized for its potent activation of Nrf2.
T10962	Dasatinib-d8 BMS-354825 D8	Others	Others
	Dasatinib D8 is deuterium-labeled dasatinib. Dasatinib is a dual Bcr-Abl and Src family tyrosine kinase inhibitor.
TMIH-0294	Lapatinib-d4
	Lapatinib-d4 是 Lapatinib 的氘代化合物。Lapatinib 的 CAS 号为 231277-92-2。Lapatinib 是一种ErbB2和EGFR酪氨酸激酶结构域的抑制剂，对纯化的ErbB2和EGFR的IC50值分别为 9.2 和 10.8 nM。Lapatinib
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同位素标记化合物

Cat.No: T24046

Synonym: WNK inhibitor-12,WNKIN12,WNK IN 12,WNK inhibitor 12,WNK-IN-12

Deucravacitinib

Cat.No: T14687

Synonym: BMS-986165

Target: Tyrosine Kinases, JAK, IFNAR, Interleukin

Cat.No: T22301

Synonym: CTP354,CTP354 (C-21191),C-21191

Target: GABA Receptor

Creatine-d3 hydrate

Cat.No: T9087

Synonym: CREATINE-(METHYL-D3) MONOHYDRATE,肌氨酸酐-甲基-D3 一水合物

Target: Endogenous Metabolite

L-Phenylalanine-15N

Cat.No: T40376

Synonym: L-苯丙氨酸 15N,(S)-2-Amino-3-phenylpropionic acid-15N,L-Phenylalanine-15N

Target: Calcium Channel

(S)-Rivastigmine D6 tartrate

Cat.No: T13446

Synonym: 酒石酸卡巴拉汀 D6,(R)-卡巴拉汀酒石盐酸-D6,(R)-Rivastigmine D6 tartrate

Target: AChE

Cat.No: T16909

Synonym: Sorafenib (D3),Bay 43-9006 (D3),Sorafenib-d3

Target: Raf, VEGFR

Cat.No: T11067

Synonym: M9831

Target: DNA-PK

Cat.No: T10948

Synonym: D8-MMAE,D8-Monomethyl auristatin E

Target: ADC Cytotoxin

Deulinoleic acid

Cat.No: T69462

Cat.No: T27097

Synonym: CTP 518,Deuterated Atazanivir-D3-1,CTP-518

Cat.No: T26871

Synonym: BMT052

Enalapril D5 maleate

Cat.No: T11192

Synonym: MK-421 D5 maleate,马来酸依那普利D5

Target: Others

Cat.No: T11194

Synonym: MK-422 D5,依那普利拉 D5

Target: Others

PSI-6206 13C,d3

Cat.No: T12571

Synonym: Sofosbuvir metabolite GS-331007 13CD3,RO-2433 13CD3,PSI-6206 13CD3,GS-331007 13CD3

Target: Others

Cat.No: T13181

Synonym: Ro 40-7592 D7

Target: Transferase

Enalaprilat-d5 sodium

Cat.No: T11193

Synonym: MK-422 D5 Sodium Salt,依那普利拉钠 D5,Enalaprilat D5 Sodium Salt

Target: Others

Cat.No: TMIH-0297

Lamivudine 13C,15N2

Cat.No: T11814

Target: Others

Cat.No: T13235

Target: Others

Cyclosporin A-d4 (Major)

Cat.No: TMIJ-0326

Cat.No: T12046

Synonym: Org3770 D3,6-Azamianserin D3,米氮平 D3

Target: 5-HT Receptor

Cat.No: T11270

Synonym: 非布司他D9

Target: Others

Cat.No: T11610

Synonym: CAL-101 D5,GS-1101 D5

Target: PI3K

Cat.No: T11229

Synonym: OSI-774 D6,NSC 718781 D6,CP-358774 D6

Target: Others

Cat.No: T10256

Synonym: BIBW 2992 D6

Target: EGFR

Cycloguanil D6 Nitrate

Cat.No: T10915

Synonym: Chlorguanide triazine D6 Nitrate

Target: Others

Pyridostigmine-d6 bromide

Cat.No: T12587

Synonym: Pyridostigmine D6 bromide,溴化吡啶斯的明 D6

Target: Others

Cat.No: T12308

Synonym: 奥美拉挫 D3,H 16868 D3

Target: Others

Lansoprazole-d4

Cat.No: T11816

Synonym: AG-1749 D4,Lansoprazole D4

Target: Proton pump

Canagliflozin-d4

Cat.No: T10669

Synonym: Canagliflozin D4

Target: Others

Dexlansoprazole-d4

Cat.No: TMIH-0187

Synonym: (R)-Lansoprazole-d4

Cat.No: T10916

Synonym: Chlorguanide triazine D6

Target: Others

Cat.No: T10284

Target: Others

Acetazolamide-d3

Cat.No: T10231

Synonym: 醋氮酰胺 D3

Target: Others

Dapagliflozin-d5

Cat.No: T10958

Synonym: BMS-512148 D5

Target: Others

Cat.No: T12355

Synonym: PD 0332991 D8,Palbociclib D8

Target: CDK

Cat.No: T12208

Synonym: 奈帕芬胺 D5,AHR-9434 D5,AL-6515 D5

Target: Others

Cat.No: T13137

Target: TGF-beta/Smad

Cat.No: TMID-0196

Clarithromycin-13C-d3

Cat.No: TMIJ-0110

Cat.No: T70214

Cat.No: T11601

Synonym: PCI-32765 D5,Ibrutinib D5

Target: Others

Alogliptin (13CD3)

Cat.No: T10288

Synonym: SYR-322 (13CD3)

Target: Others

(rel)-Tranylcypromine D5 hydrochloride

Cat.No: T12701

Synonym: 2-Phenylcyclopropylamine D5 hydrochloride

Target: Histone Demethylase

Cat.No: T12292

Synonym: KU0059436 D5,AZD2281 D5,Olaparib D5

Target: Others

Empagliflozin-d4

Cat.No: TMIJ-0133

Cat.No: T11250

Synonym: SCH 58235 D4

Target: Others

Cat.No: T10962

Synonym: BMS-354825 D8

Target: Others

Cat.No: TMIH-0294

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