gr

NXT629 是一种具有选择性和高效性的 PPAR-α 拮抗剂，具有抗癌活性，抑制 PPARδ，PPARγ，Erβ，GR 和 TRβ，可用于研究卵巢癌和黑色素瘤。

OP-3633 is an effective and selective steroidal glucocorticoid receptor (GR) antagonist (IC50: 29 nM). OP-3633 shows low progesterone receptor (PR) agonism and androgen receptor (AR) antagonism. It also has an inhibition of GR transcriptional activity.

Exicorilant is a selective and oral active glucocorticoid receptor (GR) antagonist (Ki: 7 nM) and it also has the potential to overcome adiposity, glucose intolerance, and dyslipidemia.

GR-95168 ((+)-C-BVDU) 是一种抗病毒化合物，可用于研究1型和2型单纯疱疹病毒感染。

Potent and selective tachykinin NK2 receptor agonist (EC50 = 3.7 nM in rat colon). Displays > 1000- and > 300-fold selectivity over NK1 and NK3 receptors respectively. Active in vivo.

GR 175737 is a bioactive chemical.

Potent neuropeptide Y (NPY) Y1 receptor antagonist (pA2 = 10 and 10.5 at rY1 and hY1, receptors respectively). Also a potent and selective NPY Y4 receptor agonist (pEC50 values are 6.0, 8.6 and 6.1 for rY2, hY4 and rY5 receptors respectively). Suppresses

platelet fibrinogen receptor glycoprotein IIb IIIa (GpIIb IIIa) antagonist

GR 196429, a melatonin receptor agonist, exhibits selectivity for the MT1 subtype. This compound not only promotes sleep and alters circadian rhythms but also stimulates melatonin release in mice.

GR 125487 sulfamate is a 5-HT4 receptor antagonist.

GR-92549 is an HMG-CoA reductase inhibitor.

GR 128107 is an antagonist of melatonin receptor.

GR203040 inhibits cyclophosphamide-induced damage in the rat and ferret bladder. GR-203040 is a selective NK1 receptor antagonist.

GR148672X 是三酰甘油水解酶抑制剂(IC50:4 nM)。

GR 63799 is a bioactive chemical.

GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.

GR 94800 TFA 是有效的、选择性的神经激肽 2(NK2)受体的肽类拮抗剂，其对 NK2、NK1和 NK3受体的 pKB 值分别为 9.6、6.4 和 6.0。

GR-36246 is a Thromboxane A2-receptor blocker.

GR-112000 is a peptide-based tachykinin NK2 receptor antagonist.

5-HT1B 1D receptor antagonist

GR 89696 fumarate 是一种高效选择性的κ2 opioid receptor 受体激动剂(IC50 = 0.04 nM)，具有预防瘙痒、体内抗伤害和神经保护作用。

Tachykinin NK1 receptor antagonist.

GR 94800 acetate 是一种有效的选择性神经激肽 2(NK-2) 拮抗剂。

GR-127935 is a potent and selective 5-HT1B 1D receptor antagonist.