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抗结直肠癌化合物库

抗结直肠癌化合物库

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产品编号 L2194 Anti-Colorectal Cancer Compound Library
  库化合物信息   Excel SDF

结直肠癌(Colorectal Cancer,CRC),又称大肠癌,包括结肠癌和直肠癌,是全球范围内致命的恶性肿瘤之一,严重威胁人类健康,近年来其发病率和死亡率均呈上升趋势,并且发病率随着年龄的增加而增加,人口老龄化和不良生活习惯是主要诱因,缺乏运动、肥胖、抽烟也使得患结直肠癌的风险显著增加。结直肠癌的治疗手段包括手术、放疗、化疗和靶向治疗。早期癌症可以通过手术治愈,晚期转移性癌通常选择化疗联合靶向治疗,研究表明,多个信号通路和靶点的失调与结直肠癌有关,如: VEGFREGFR、Wnt/β-catenin、p53、TGF-β等 TargetMol 抗结直肠癌化合物库收集了1565 种与结直肠癌相关的化合物,包括已经报道具有结直肠癌治疗作用的化合物,以及靶向结直肠癌相关靶点的化合物,是抗结直肠癌药物研发的良好工具。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
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产品描述

  • 1565种与结直肠癌相关的化合物,可以用于高通量和高内涵筛选;
  • 部分化合物已上市或已进入临床期;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L2194)
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客户使用化合物库发表的文献

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化合物库组成

Apoptosis (280)
Autophagy (211)
PI3K (163)
EGFR (150)
VEGFR (144)
COX (117)
Akt (88)
mTOR (88)
ERK (84)
p38 MAPK (83)
Wnt/beta-catenin (79)
Raf (69)
c-Met/HGFR (66)
NF-κB (64)
PDGFR (63)
AMPK (62)
Ras (58)
CDK (56)
GSK-3 (55)
STAT (54)
TGF-beta/Smad (52)
JNK (48)
c-Kit (45)
MAPK (43)
Src (43)
Antibacterial (43)
MEK (43)
Endogenous Metabolite (42)
FLT (40)
FGFR (40)
DNA-PK (37)
p53 (36)
S6 Kinase (32)
DNA/RNA Synthesis (29)
HER (29)
ALK (25)
Parasite (24)
ATM/ATR (22)
Reactive Oxygen Species (21)
PKC (20)
c-RET (20)
PDK (19)
Bcr-Abl (18)
E1/E2/E3 Enzyme (18)
Antibiotic (18)
Mdm2 (18)
Gamma-secretase (18)
Ferroptosis (17)
JAK (17)
Caspase (16)
Mitophagy (16)
Aurora Kinase (16)
TNF (15)
Antifungal (15)
PARP (14)
TAM Receptor (14)
PI4K (14)
Casein Kinase (13)
IGF-1R (13)
PKA (13)
Rho (12)
Influenza Virus (12)
Dehydrogenase (12)
P450 (11)
Potassium Channel (11)
PPAR (11)
c-Fms (11)
Trk receptor (11)
BCL (11)
Tyrosine Kinases (10)
IL Receptor (10)
FAK (10)
HIV Protease (10)
Sirtuin (10)
Topoisomerase (9)
Lipoxygenase (9)
MMP (9)
Chk (9)
Phosphatase (8)
PTEN (8)
Nucleoside Antimetabolite/Analog (8)
HDAC (8)
NOS (8)
Sodium Channel (8)
Calcium Channel (8)
ROCK (8)
Beta Amyloid (8)
Prostaglandin Receptor (7)
HSV (7)
HCV Protease (7)
ROS (7)
PDE (7)
Epigenetic Reader Domain (6)
Tyrosinase (6)
Microtubule Associated (5)
Antiviral (5)
Virus Protease (5)
Carbonic Anhydrase (5)
Estrogen/progestogen Receptor (5)
Tie-2 (5)
Interleukin (5)
Antioxidant (5)
BTK (5)
IκB/IKK (5)
MELK (5)
TLR (5)
MNK (5)
TOPK (5)
HSP (5)
Aryl Hydrocarbon Receptor (5)
MLK (5)
ASK (5)
Phospholipase (5)
Ephrin Receptor (5)
SIK (5)
SGK (5)
Porcupine (5)
Glucosidase (4)
PLK (4)
ATPase (4)
Estrogen Receptor/ERR (4)
ROS Kinase (4)
Drug Metabolite (4)
PGE Synthase (4)
AChR (4)
Adrenergic Receptor (4)
Serine Protease (4)
Integrin (4)
NO Synthase (4)
IAP (4)
Hydroxylase (4)
GABA Receptor (3)
MRP (3)
Nrf2 (3)
Mitochondrial Metabolism (3)
Proton pump (3)
Syk (3)
DNA Alkylation (3)
Glutathione Peroxidase (3)
Adenosine Receptor (3)
DNA Alkylator/Crosslinker (3)
Antifection (3)
GTPase (3)
KLF (3)
P-gp (3)
HIF (3)
CSF-1R (3)
AChE (3)
Antifolate (3)
Transferase (2)
TRP/TRPV Channel (2)
transporter (2)
S1P Receptor (2)
SARS-CoV (2)
Pim (2)
RIP kinase (2)
5-HT Receptor (2)
HIF/HIF Prolyl-Hydroxylase (2)
CCR (2)
CaMK (2)
BMI-1 (2)
HBV (2)
Beta-Secretase (2)
Hck (2)
Gap Junction Protein (2)
Histamine Receptor (2)
Histone Acetyltransferase (2)
Histone Methyltransferase (2)
IRAK (2)
IRE1 (2)
Kinesin (2)
BACE (2)
APC (2)
LRRK2 (2)
Androgen Receptor (2)
Fatty Acid Synthase (2)
NADPH (2)
FAAH (2)
DYRK (2)
Discoidin Domain Receptor (DDR) (2)
Chloride channel (2)
c-Myc (1)
CRISPR/Cas9 (1)
DAPK (1)
Serine/threonin kinase (1)
cholecystokinin (1)
DHFR (1)
Somatostatin (1)
NPC1L1 (1)
CD73 (1)
Cannabinoid Receptor (1)
cAMP (1)
DNA Methyltransferase (1)
BCRP (1)
ATP Citrate Lyase (1)
Aromatase (1)
Arginase (1)
Apelin receptor (1)
UGT (1)
Amino Acids and Derivatives (1)
AhR (1)
Wee1 (1)
ACK (1)
DNA (1)
Reverse Transcriptase (1)
RSV (1)
hCE (1)
OCT (1)
Opioid Receptor (1)
Neurotensin Receptor (1)
NADPH-oxidase (1)
Myosin (1)
PAI-1 (1)
MTH1 (1)
PD-1/PD-L1 (1)
Leukotriene Receptor (1)
LDL (1)
KSP (1)
PERK (1)
Immunology/Inflammation related (1)
GPX (1)
Dopamine Receptor (1)
GPR (1)
Progesterone Receptor (1)
GluR (1)
Glucokinase (1)
Glucocorticoid Receptor (1)
PYK2 (1)
RAAS (1)
FXR (1)
FLAP (1)
Reductase (1)
Retinoid Receptor (1)
NMDAR (1)
ROR (1)
DUB (1)
YAP (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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