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抗前列腺癌化合物库

抗前列腺癌化合物库

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产品编号 L2195 Anti-Prostate Cancer Compound Library
  库化合物信息   Excel SDF

前列腺癌是指发生在前列腺的上皮性恶性肿瘤,是男性生殖系统中常见的恶性肿瘤,具有复杂的疾病发病机制。Androgen Receptor、Hedgehog、TGF-β、Wnt、PI3K-AKT-mTOR 等多个信号通路和靶点参与前列腺癌的进展。 TargetMol 抗前列腺癌化合物库收集了2096 种与前列腺癌相关的化合物,包括已经报道具有前列腺癌治疗作用的化合物,以及靶向前列腺癌相关靶点的化合物,是抗前列腺癌药物研发的良好工具。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
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产品描述

  • 2096种与前列腺癌相关的化合物,可以用于高通量和高内涵筛选;
  • 部分化合物已上市或已进入临床期;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L2195)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

Apoptosis (374)
Autophagy (269)
NF-κB (208)
PI3K (163)
Reactive Oxygen Species (163)
EGFR (151)
VEGFR (143)
COX (130)
Endogenous Metabolite (101)
JAK (89)
mTOR (88)
Akt (87)
ERK (84)
CDK (84)
p38 MAPK (82)
STAT (81)
Wnt/beta-catenin (79)
FGFR (73)
Raf (69)
PARP (69)
Antibacterial (68)
PDGFR (68)
Androgen Receptor (64)
AMPK (62)
Ras (58)
GSK-3 (55)
c-Kit (51)
Src (49)
FLT (49)
JNK (48)
MEK (43)
MAPK (43)
HER (41)
IκB/IKK (38)
DNA-PK (37)
TNF (35)
S6 Kinase (32)
Parasite (31)
Ferroptosis (29)
Tyrosine Kinases (29)
Hedgehog/Smoothened (29)
Antifungal (28)
IL Receptor (27)
Bcr-Abl (27)
P450 (26)
Caspase (26)
c-Met/HGFR (26)
Antibiotic (24)
NOD (23)
Mitophagy (22)
RIP kinase (22)
PKC (22)
Potassium Channel (22)
Influenza Virus (22)
ATM/ATR (22)
Aurora Kinase (21)
PPAR (21)
HIV Protease (21)
Antioxidant (20)
c-RET (20)
PDK (19)
Gamma-secretase (18)
Pim (18)
IRAK (17)
NO Synthase (16)
MMP (16)
Casein Kinase (16)
ROS (15)
Lipoxygenase (15)
IGF-1R (14)
PI4K (14)
DNA/RNA Synthesis (14)
NOD-like Receptor (NLR) (14)
BCL (14)
Calcium Channel (14)
PKA (14)
Estrogen/progestogen Receptor (13)
Rho (13)
Mitochondrial Metabolism (12)
Epigenetic Reader Domain (12)
c-Fms (12)
Smo (12)
NOS (12)
Interleukin (11)
Virus Protease (11)
Estrogen Receptor/ERR (10)
Nrf2 (10)
p53 (10)
Topoisomerase (10)
Microtubule Associated (10)
Beta Amyloid (10)
Sodium Channel (9)
Chk (9)
TGF-beta/Smad (9)
Dehydrogenase (9)
Prostaglandin Receptor (9)
GABA Receptor (9)
Trk receptor (9)
ROCK (9)
AChR (8)
HSP (8)
PLK (8)
HIF/HIF Prolyl-Hydroxylase (8)
TAM Receptor (8)
FAK (8)
PTEN (8)
Drug Metabolite (8)
Tyrosinase (8)
HDAC (7)
HCV Protease (7)
E1/E2/E3 Enzyme (7)
GNRH Receptor (7)
Syk (7)
Phosphatase (7)
TLR (7)
PDE (7)
5-HT Receptor (6)
HSV (6)
Antiviral (6)
Ephrin Receptor (6)
P-gp (6)
BTK (6)
NADPH (6)
PGE Synthase (6)
CSF-1R (6)
Proteasome (6)
RAAS (5)
MELK (5)
MLK (5)
AChE (5)
MNK (5)
Adrenergic Receptor (5)
SARS-CoV (5)
ASK (5)
SGK (5)
Tie-2 (5)
Histone Methyltransferase (5)
TOPK (5)
Transferase (5)
SIK (5)
Carbonic Anhydrase (5)
Glucocorticoid Receptor (5)
Porcupine (4)
Free radical scavengers (4)
Anti-infection (4)
Glucosidase (4)
Glutathione Peroxidase (4)
Retinoid Receptor (4)
CXCR (4)
HBV (4)
ALK (4)
HIF (4)
ATPase (4)
Histamine Receptor (4)
Histone Acetyltransferase (4)
Progesterone Receptor (4)
Serine Protease (4)
TRP/TRPV Channel (4)
Integrin (4)
IFNAR (4)
CaMK (4)
Antifection (4)
IAP (4)
Aryl Hydrocarbon Receptor (4)
Opioid Receptor (3)
BACE (3)
Adenosine Receptor (3)
c-Myc (3)
cholecystokinin (3)
Chloride channel (3)
Cannabinoid Receptor (3)
Fatty Acid Synthase (3)
Hippo pathway (3)
S1P Receptor (3)
IRE1 (3)
KLF (3)
Leukotriene Receptor (3)
LRRK2 (3)
GTPase (3)
Sirtuin (3)
RANKL/RANK (2)
GST (2)
Phospholipase (2)
Hck (2)
CCR (2)
Mdm2 (2)
GPR (2)
transporter (2)
MAO (2)
Beta-Secretase (2)
Proton pump (2)
NADPH-oxidase (2)
Gap Junction Protein (2)
PERK (2)
FAAH (2)
Reverse Transcriptase (2)
ROR (2)
AhR (2)
Glutathione reductase (2)
MRP (2)
DYRK (2)
STING (2)
Dopamine Receptor (2)
Reductase (2)
DNA Alkylation (2)
Discoidin Domain Receptor (DDR) (2)
PD-1/PD-L1 (2)
Sigma receptor (1)
Somatostatin (1)
Serine/threonin kinase (1)
SGLT (1)
Wee1 (1)
VDA (1)
Survivin (1)
RSV (1)
UGT (1)
RAR/RXR  (1)
Immunology/Inflammation related (1)
Platelet aggregation (1)
CD73 (1)
DUB (1)
DPP-4 (1)
DNA (1)
DHFR (1)
DAPK (1)
Cysteine Protease (1)
CRISPR/Cas9 (1)
cGAS (1)
CFTR (1)
cAMP (1)
FLAP (1)
BMI-1 (1)
BCRP (1)
ATP Citrate Lyase (1)
Aromatase (1)
Arginase (1)
Apelin receptor (1)
Aminopeptidase (1)
Adenosine deaminase (1)
Acyltransferase (1)
ACK (1)
Endothelin Receptor (1)
FXR (1)
PKM (1)
Melanin-concentrating Hormone Receptor (MCHR) (1)
PAK (1)
PAI-1 (1)
OXPHOS (1)
OCT (1)
Nucleoside Antimetabolite/Analog (1)
NPC1L1 (1)
NMDAR (1)
Na+/Ca2+ Exchanger (1)
Myosin (1)
Monoamine Oxidase (1)
LTR (1)
Glucokinase (1)
Liver X Receptor (1)
LDL (1)
Kinesin (1)
Indoleamine 2,3-Dioxygenase (IDO) (1)
ABC (1)
Hydroxylase (1)
hCE (1)
Haspin Kinase (1)
GPX (1)
GluR (1)
YAP (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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