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TargetMol | Compound Library

抗前列腺癌化合物库现货

Anti-Prostate Cancer Compound Library

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产品编号 L2195

前列腺癌是指发生在前列腺的上皮性恶性肿瘤,是男性生殖系统中常见的恶性肿瘤,具有复杂的疾病发病机制。Androgen Receptor、Hedgehog、TGF-β、Wnt、PI3K-AKT-mTOR 等多个信号通路和靶点参与前列腺癌的进展。 TargetMol 抗前列腺癌化合物库收集了2256 种与前列腺癌相关的化合物,包括已经报道具有前列腺癌治疗作用的化合物,以及靶向前列腺癌相关靶点的化合物,是抗前列腺癌药物研发的良好工具。

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产品编号 L2195

抗前列腺癌化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 2256种与前列腺癌相关的化合物,可以用于高通量和高内涵筛选;
  • 部分化合物已上市或已进入临床期;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
NF-κB
PI3K
VEGFR
EGFR
Reactive Oxygen Species
COX
mTOR
ERK
Akt
PARP
CDK
Endogenous Metabolite
JAK
Wnt/beta-catenin
AMPK
p38 MAPK
GSK-3
STAT
FGFR
Androgen Receptor
PDGFR
Antibacterial
Raf
MEK
Src
c-Kit
Ras
FLT
JNK
MAPK
IκB/IKK
TNF
Histone Methyltransferase
DNA-PK
S6 Kinase
Caspase
Parasite
ATM/ATR
Hedgehog/Smoothened
Cytochromes P450
IL Receptor
Tyrosine Kinases
Potassium Channel
c-Met/HGFR
Antifungal
PDK
RIP kinase
Antibiotic
HER
Ferroptosis
PPAR
Aurora Kinase
Bcr-Abl
c-RET
Pim
NOD
HIV Protease
Antioxidant
Influenza Virus
PKC
Mitophagy
Gamma-secretase
Epigenetic Reader Domain
NO Synthase
Casein Kinase
Calcium Channel
IRAK
PKA
Bcl-2 Family
PD-1/PD-L1
IGF-1R
Estrogen/progestogen Receptor
MMP
Rho
ROS
PI4K
Lipoxygenase
DNA/RNA Synthesis
Microtubule Associated
Smo
p53
NOD-like Receptor (NLR)
Nrf2
c-Fms
HDAC
Mitochondrial Metabolism
Topoisomerase
Virus Protease
Dehydrogenase
NOS
Prostaglandin Receptor
GABA Receptor
HIF/HIF Prolyl-Hydroxylase
Tyrosinase
Syk
ROCK
Beta Amyloid
Estrogen Receptor/ERR
Trk receptor
Chk
TGF-beta/Smad
Interleukin
PDE
FAK
Sodium Channel
AChR
Phosphatase
Kras
Drug Metabolite
PLK
TLR
SIK
5-HT Receptor
PTEN
E1/E2/E3 Enzyme
GNRH Receptor
Antiviral
HSP
MELK
Proteasome
TAM Receptor
DYRK
Adrenergic Receptor
P-gp
CSF-1R
Antifection
HSV
Cholinesterase (ChE)
PGE Synthase
NADPH
Tie-2
HIF
SARS-CoV
Glucocorticoid Receptor
TRP/TRPV Channel
SGK
Carbonic Anhydrase
RAAS
ASK
HCV Protease
Integrin
Transferase
HBV
Ephrin Receptor
MNK
MLK
LDL
Cannabinoid Receptor
Porcupine
IAP
transporter
Free radical scavengers
Reductase
ALK
Histamine Receptor
Serine Protease
Glucosidase
Histone Acetyltransferase
TOPK
Anti-infection
Glutathione Peroxidase
Opioid Receptor
Progesterone Receptor
Aryl Hydrocarbon Receptor
ATPase
c-Myc
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Cholecystokinin Receptor
CXCR
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PSMA
IRE1
Mdm2
DNA Alkylation
GPCR
BACE
KLF
Retinoid Receptor
CaMK
Phospholipase
GTPase
Chloride channel
IFNAR
Fatty Acid Synthase
LRRK2
BTK
RAR/RXR
YAP
Endothelin Receptor
MRP
ROR
DUB
NADPH-oxidase
Adenosine Receptor
S1P Receptor
cAMP
CCR
NMDAR
Discoidin Domain Receptor (DDR)
GluR
Serine/threonin kinase
ADC Cytotoxin
STING
RANKL/RANK
Dopamine Receptor
FAAH
MAO
PERK
Beta-Secretase
Gap Junction Protein
Acyltransferase
Reverse Transcriptase
ABC Transporter
Monoamine Transporter
RSV
PKM
BCRP
DPP-4
Haspin Kinase
Wee1
DHFR
Platelet aggregation
cGAS
DAPK
BMI-1
Survivin
Cysteine Protease
DNA Methyltransferase
Adenosine Deaminase
Somatostatin
Nucleoside Antimetabolite/Analog
OCT
PAFR
PYK2
Glutathione reductase
Aromatase
Decarboxylase
Sirtuin
OXPHOS
Hydroxylase
VDA
PAI-1
UGT
gp120/CD4
Kinesin
Aminopeptidase
NPC1L1
Glucokinase
FLAP
SGLT
ATP Citrate Lyase
CRISPR/Cas9
Proton pump
Indoleamine 2,3-Dioxygenase (IDO)
CFTR
Methionine Adenosyltransferase (MAT)
iGluR
AhR
Monoamine Oxidase
CD73
hCE
LTR
GPX
Myosin
Melanin-concentrating Hormone Receptor (MCHR)
FXR
Liver X Receptor
DNA
GST
Sigma receptor
Apelin receptor
Arginase
Na+/Ca2+ Exchanger
MicroRNA
PAK
Hck

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