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TargetMol | Compound Library

抗前列腺癌化合物库现货

Anti-Prostate Cancer Compound Library
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货号 L2195

前列腺癌是指发生在前列腺的上皮性恶性肿瘤,是男性生殖系统中常见的恶性肿瘤,具有复杂的疾病发病机制。Androgen Receptor、Hedgehog、TGF-β、Wnt、PI3K-AKT-mTOR 等多个信号通路和靶点参与前列腺癌的进展。 TargetMol 抗前列腺癌化合物库收集了2256 种与前列腺癌相关的化合物,包括已经报道具有前列腺癌治疗作用的化合物,以及靶向前列腺癌相关靶点的化合物,是抗前列腺癌药物研发的良好工具。

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货号 L2195

抗前列腺癌化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 2256种与前列腺癌相关的化合物,可以用于高通量和高内涵筛选;
  • 部分化合物已上市或已进入临床期;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
NF-κB
PI3K
ROS
VEGFR
Reactive Oxygen Species
EGFR
COX
Ras
mTOR
Akt
ERK
Endogenous Metabolite
p38 MAPK
PARP
Wnt/beta-catenin
CDK
STAT
JAK
GSK-3
AMPK
Antibacterial
FGFR
Androgen Receptor
PDGFR
Raf
Caspase
MEK
JNK
Src
FLT
c-Kit
Parasite
MAPK
TNF
IκB/IKK
S6 Kinase
Histone Methyltransferase
DNA-PK
NO Synthase
Cytochromes P450
Bcl-2 Family
Hedgehog/Smoothened
ATM/ATR
PPAR
Interleukin
Antifungal
c-Met/HGFR
Potassium Channel
Bcr-Abl
Tyrosine Kinases
Antibiotic
IL Receptor
DNA/RNA Synthesis
RIP kinase
Influenza Virus
HIV Protease
PKC
Aurora Kinase
HER
PDK
Ferroptosis
NOD
Kras
Mitophagy
c-RET
Antioxidant
Pim
Gamma-secretase
Calcium Channel
Epigenetic Reader Domain
MMP
Casein Kinase
NOD-like Receptor (NLR)
IGF-1R
PD-1/PD-L1
PI4K
PKA
Dehydrogenase
Virus Protease
Smo
IRAK
HIF/HIF Prolyl-Hydroxylase
Estrogen/progestogen Receptor
Microtubule Associated
Nrf2
Estrogen Receptor/ERR
Rho
Lipoxygenase
c-Fms
Drug Metabolite
TGF-beta/Smad
Beta Amyloid
Mitochondrial Metabolism
Prostaglandin Receptor
p53
GABA Receptor
HDAC
NOS
Phosphatase
Topoisomerase
P-gp
TLR
Tyrosinase
FAK
AChR
ROCK
Chk
Trk receptor
PLK
Syk
HSP
PDE
PTEN
Sodium Channel
HSV
Tie-2
SARS-CoV
Antifection
E1/E2/E3 Enzyme
Cholinesterase (ChE)
Reductase
SIK
TRP/TRPV Channel
5-HT Receptor
Anti-infection
DYRK
Serine Protease
PGE Synthase
Survivin
ATPase
IAP
Proteasome
Integrin
CSF-1R
TAM Receptor
HCV Protease
Cannabinoid Receptor
MLK
NADPH
Adrenergic Receptor
CaMK
Antiviral
SGK
c-Myc
GNRH Receptor
Histone Acetyltransferase
MELK
Angiotensin-converting Enzyme (ACE)
MNK
ASK
Carbonic Anhydrase
PERK
HBV
RAAS
Glucosidase
OXPHOS
Transferase
Glucocorticoid Receptor
Ephrin Receptor
HIF
MDM-2/p53
Fatty Acid Synthase
Porcupine
Histamine Receptor
TOPK
Phospholipase
Glutathione Peroxidase
Aryl Hydrocarbon Receptor
Opioid Receptor
Free radical scavengers
Retinoid Receptor
IFNAR
RANKL/RANK
PSMA
transporter
GPCR
Adenosine Receptor
Progesterone Receptor
ALK
BTK
KLF
UGT
glycosidase
Hippo pathway
Cholecystokinin Receptor
DNA Alkylation
Beta-Secretase
Chloride channel
Serine/threonin kinase
Leukotriene Receptor
IRE1
LDL
STING
LRRK2
FKBP
BACE
DNA Methyltransferase
Mdm2
GTPase
PAK
Reverse Transcriptase
Gap Junction Protein
ROS Kinase
Apelin receptor
ROR
NMDAR
DUB
S1P Receptor
Dopamine Receptor
MRP
PYK2
Discoidin Domain Receptor (DDR)
Kinesin
PROTACs
ABC Transporter
FAAH
CCR
GluR
ATP Citrate Lyase
CFTR
Myosin
Endothelin Receptor
Acyltransferase
RAR/RXR
Cysteine Protease
FXR
Prolyl Endopeptidase (PREP)
CXCR
NADPH-oxidase
ADC Cytotoxin
YAP
Hck
Monoamine Oxidase
MAO
cAMP
MicroRNA
Glucokinase
Immunology/Inflammation related
PAFR
Haspin Kinase
DPP-4
Orphan Receptor
RSV
MIF
Somatostatin
Indoleamine 2,3-Dioxygenase (IDO)
Wee1
BCRP
Aminopeptidase
Methionine Adenosyltransferase (MAT)
Cuproptosis
DAPK
CD38
LTR
VDA
ATG
Nucleoside Antimetabolite/Analog
iGluR
Monoamine Transporter
DNA
Sirtuin
CD73
cGAS
Hydroxylase
Sigma receptor
Thyroid hormone receptor(THR)
Melanin-concentrating Hormone Receptor (MCHR)
NPC1L1
DHFR
FLAP
Glutathione reductase
Decarboxylase
Adenosine Deaminase
Proton pump
MyD88
DNA Alkylator/Crosslinker
Arrestin
Cadherin
Pyroptosis
GPX
PKM
Necroptosis
OCT
IDO
Na-K-Cl cotransporter
SGLT
Lipid
hCE
BMI-1
AhR
Y Box Binding Protein 1
Arginase
Na+/Ca2+ Exchanger
gp120/CD4
ASCT
Liver X Receptor
AIM2
PAI-1
GST
Aromatase
Platelet aggregation

Keywords