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TargetMol | Compound Library

抗前列腺癌化合物库现货

Anti-Prostate Cancer Compound Library

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产品编号 L2195

前列腺癌是指发生在前列腺的上皮性恶性肿瘤,是男性生殖系统中常见的恶性肿瘤,具有复杂的疾病发病机制。Androgen Receptor、Hedgehog、TGF-β、Wnt、PI3K-AKT-mTOR 等多个信号通路和靶点参与前列腺癌的进展。 TargetMol 抗前列腺癌化合物库收集了2256 种与前列腺癌相关的化合物,包括已经报道具有前列腺癌治疗作用的化合物,以及靶向前列腺癌相关靶点的化合物,是抗前列腺癌药物研发的良好工具。

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产品编号 L2195

抗前列腺癌化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 2256种与前列腺癌相关的化合物,可以用于高通量和高内涵筛选;
  • 部分化合物已上市或已进入临床期;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
NF-κB
PI3K
ROS
Reactive Oxygen Species
VEGFR
EGFR
COX
Ras
mTOR
ERK
Akt
Endogenous Metabolite
p38 MAPK
PARP
Wnt/beta-catenin
CDK
JAK
STAT
AMPK
GSK-3
Antibacterial
FGFR
Androgen Receptor
PDGFR
Raf
JNK
Caspase
MEK
Src
FLT
c-Kit
Parasite
MAPK
TNF
IκB/IKK
DNA-PK
S6 Kinase
Histone Methyltransferase
NO Synthase
Cytochromes P450
Bcl-2 Family
Hedgehog/Smoothened
ATM/ATR
PPAR
Interleukin
Antifungal
c-Met/HGFR
Tyrosine Kinases
IL Receptor
DNA/RNA Synthesis
Potassium Channel
Antibiotic
Bcr-Abl
HIV Protease
Ferroptosis
PKC
RIP kinase
Aurora Kinase
Influenza Virus
PDK
NOD
HER
Kras
Mitophagy
c-RET
Antioxidant
Pim
Calcium Channel
Epigenetic Reader Domain
Gamma-secretase
MMP
Casein Kinase
NOD-like Receptor (NLR)
IGF-1R
PD-1/PD-L1
Dehydrogenase
PKA
PI4K
Virus Protease
Smo
IRAK
Estrogen/progestogen Receptor
Nrf2
Microtubule Associated
HIF/HIF Prolyl-Hydroxylase
Estrogen Receptor/ERR
Rho
Lipoxygenase
Drug Metabolite
TGF-beta/Smad
Prostaglandin Receptor
Beta Amyloid
c-Fms
Mitochondrial Metabolism
GABA Receptor
p53
Phosphatase
Topoisomerase
P-gp
TLR
HDAC
Tyrosinase
NOS
ROCK
Trk receptor
AChR
FAK
PDE
PTEN
Chk
HSP
PLK
Syk
Sodium Channel
Tie-2
HSV
SARS-CoV
Reductase
DYRK
GNRH Receptor
TRP/TRPV Channel
SIK
E1/E2/E3 Enzyme
Antifection
Cholinesterase (ChE)
CaMK
5-HT Receptor
Anti-infection
Proteasome
ATPase
HCV Protease
Integrin
NADPH
c-Myc
Serine Protease
Adrenergic Receptor
CSF-1R
PGE Synthase
Antiviral
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MELK
SGK
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TAM Receptor
MLK
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Transferase
RAAS
PERK
HBV
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IAP
Glucosidase
Angiotensin-converting Enzyme (ACE)
OXPHOS
MNK
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Ephrin Receptor
transporter
ASK
HIF
MDM-2/p53
GPCR
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IFNAR
Histamine Receptor
Glutathione Peroxidase
TOPK
Progesterone Receptor
RANKL/RANK
Aryl Hydrocarbon Receptor
LDL
Opioid Receptor
Fatty Acid Synthase
PSMA
Porcupine
Free radical scavengers
ALK
Retinoid Receptor
Phospholipase
BTK
Mdm2
Chloride channel
BACE
GTPase
Cholecystokinin Receptor
Serine/threonin kinase
Leukotriene Receptor
IRE1
UGT
DNA Alkylation
PAK
glycosidase
Beta-Secretase
STING
LRRK2
FKBP
Reverse Transcriptase
KLF
Gap Junction Protein
DNA Methyltransferase
ROS Kinase
Apelin receptor
PROTACs
RAR/RXR
Dopamine Receptor
ROR
ADC Cytotoxin
YAP
MRP
Cysteine Protease
FXR
PYK2
MAO
Prolyl Endopeptidase (PREP)
Myosin
NMDAR
ABC Transporter
FAAH
CCR
CXCR
Endothelin Receptor
cAMP
GluR
DUB
ATP Citrate Lyase
Acyltransferase
Hippo pathway
Discoidin Domain Receptor (DDR)
NADPH-oxidase
CFTR
S1P Receptor
Monoamine Oxidase
Kinesin
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Proton pump
MicroRNA
NPC1L1
CD38
DHFR
MyD88
Y Box Binding Protein 1
Arginase
DNA Alkylator/Crosslinker
LTR
Arrestin
Na+/Ca2+ Exchanger
Necroptosis
gp120/CD4
MIF
VDA
OCT
ASCT
Hck
ATG
Nucleoside Antimetabolite/Analog
Liver X Receptor
Glucokinase
IDO
iGluR
Immunology/Inflammation related
FLAP
PAFR
Haspin Kinase
Na-K-Cl cotransporter
Monoamine Transporter
DPP-4
Somatostatin
Cadherin
Orphan Receptor
DNA
Indoleamine 2,3-Dioxygenase (IDO)
SGLT
Wee1
Lipid
BCRP
Glutathione reductase
Aminopeptidase
Sirtuin
CD73
AIM2
Decarboxylase
cGAS
hCE
PAI-1
Pyroptosis
RSV
Methionine Adenosyltransferase (MAT)
GST
GPX
Aromatase
CRISPR/Cas9
Hydroxylase
Adenosine Deaminase
Cuproptosis
DAPK
Platelet aggregation
BMI-1
Sigma receptor
AhR
PKM

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