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TargetMol | Compound Library

抗前列腺癌化合物库现货

Anti-Prostate Cancer Compound Library

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产品编号 L2195

前列腺癌是指发生在前列腺的上皮性恶性肿瘤,是男性生殖系统中常见的恶性肿瘤,具有复杂的疾病发病机制。Androgen Receptor、Hedgehog、TGF-β、Wnt、PI3K-AKT-mTOR 等多个信号通路和靶点参与前列腺癌的进展。 TargetMol 抗前列腺癌化合物库收集了2256 种与前列腺癌相关的化合物,包括已经报道具有前列腺癌治疗作用的化合物,以及靶向前列腺癌相关靶点的化合物,是抗前列腺癌药物研发的良好工具。

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产品编号 L2195

抗前列腺癌化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 2256种与前列腺癌相关的化合物,可以用于高通量和高内涵筛选;
  • 部分化合物已上市或已进入临床期;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
NF-κB
PI3K
Reactive Oxygen Species
VEGFR
EGFR
COX
Ras
mTOR
Endogenous Metabolite
Akt
ERK
PARP
p38 MAPK
Wnt/beta-catenin
CDK
JAK
AMPK
GSK-3
STAT
FGFR
Antibacterial
Androgen Receptor
PDGFR
Raf
MEK
JNK
FLT
Src
c-Kit
Parasite
Caspase
MAPK
IκB/IKK
TNF
S6 Kinase
DNA-PK
Histone Methyltransferase
Cytochromes P450
ATM/ATR
Hedgehog/Smoothened
Bcl-2 Family
PPAR
c-Met/HGFR
Tyrosine Kinases
Antifungal
IL Receptor
Potassium Channel
Bcr-Abl
Aurora Kinase
Influenza Virus
HIV Protease
Antibiotic
PKC
PDK
HER
RIP kinase
NO Synthase
Ferroptosis
NOD
Kras
Mitophagy
c-RET
Pim
Antioxidant
Calcium Channel
Epigenetic Reader Domain
DNA/RNA Synthesis
NOD-like Receptor (NLR)
Casein Kinase
Gamma-secretase
MMP
PKA
Interleukin
PI4K
IGF-1R
Smo
IRAK
PD-1/PD-L1
Dehydrogenase
Estrogen/progestogen Receptor
Microtubule Associated
ROS
HIF/HIF Prolyl-Hydroxylase
Virus Protease
Rho
Lipoxygenase
Nrf2
c-Fms
Drug Metabolite
Prostaglandin Receptor
p53
Mitochondrial Metabolism
GABA Receptor
HDAC
Phosphatase
Topoisomerase
Tyrosinase
Estrogen Receptor/ERR
TGF-beta/Smad
ROCK
Beta Amyloid
NOS
FAK
PTEN
P-gp
Chk
Trk receptor
Syk
Sodium Channel
PDE
Tie-2
HSP
AChR
TRP/TRPV Channel
5-HT Receptor
Anti-infection
E1/E2/E3 Enzyme
HSV
Cholinesterase (ChE)
Antifection
TLR
SIK
PLK
DYRK
GNRH Receptor
NADPH
Adrenergic Receptor
Antiviral
SGK
ATPase
PGE Synthase
HCV Protease
Cannabinoid Receptor
Proteasome
CSF-1R
SARS-CoV
TAM Receptor
Histone Acetyltransferase
MELK
Transferase
Glucocorticoid Receptor
transporter
Carbonic Anhydrase
HBV
IAP
ASK
OXPHOS
MLK
Integrin
Reductase
RAAS
Glucosidase
Angiotensin-converting Enzyme (ACE)
MNK
c-Myc
Ephrin Receptor
HIF
MDM-2/p53
CaMK
Porcupine
Survivin
Glutathione Peroxidase
Aryl Hydrocarbon Receptor
LDL
Opioid Receptor
Free radical scavengers
Retinoid Receptor
Histamine Receptor
TOPK
Phospholipase
Serine Protease
GPCR
Progesterone Receptor
ALK
BTK
BACE
IFNAR
RANKL/RANK
PSMA
DNA Methyltransferase
PERK
Hippo pathway
Chloride channel
Leukotriene Receptor
IRE1
LRRK2
FKBP
Cholecystokinin Receptor
DNA Alkylation
Beta-Secretase
KLF
Mdm2
GTPase
PAK
Reverse Transcriptase
ROS Kinase
ADC Cytotoxin
YAP
Monoamine Oxidase
ABC Transporter
FAAH
CCR
GluR
ATP Citrate Lyase
CFTR
Dopamine Receptor
MRP
PYK2
UGT
Fatty Acid Synthase
Discoidin Domain Receptor (DDR)
RAR/RXR
Serine/threonin kinase
Cysteine Protease
FXR
Prolyl Endopeptidase (PREP)
CXCR
STING
NADPH-oxidase
Myosin
Endothelin Receptor
Acyltransferase
Apelin receptor
ROR
NMDAR
DUB
S1P Receptor
Adenosine Receptor
MAO
cAMP
Gap Junction Protein
Necroptosis
OCT
Hck
IDO
Na-K-Cl cotransporter
SGLT
Lipid
hCE
BMI-1
AhR
CD38
LTR
VDA
ATG
Nucleoside Antimetabolite/Analog
iGluR
Monoamine Transporter
DNA
Sirtuin
CD73
cGAS
CRISPR/Cas9
Hydroxylase
Sigma receptor
MIF
Somatostatin
Indoleamine 2,3-Dioxygenase (IDO)
Wee1
BCRP
Aminopeptidase
Methionine Adenosyltransferase (MAT)
Cuproptosis
DAPK
Kinesin
Proton pump
DNA Alkylator/Crosslinker
Arrestin
Pyroptosis
GPX
PKM
Thyroid hormone receptor(THR)
Melanin-concentrating Hormone Receptor (MCHR)
NPC1L1
DHFR
FLAP
Glutathione reductase
Decarboxylase
Adenosine Deaminase
MicroRNA
Glucokinase
PAFR
Haspin Kinase
DPP-4
RSV
Y Box Binding Protein 1
Arginase
Na+/Ca2+ Exchanger
gp120/CD4
ASCT
Liver X Receptor
AIM2
PAI-1
GST
Aromatase
Platelet aggregation

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