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TargetMol | Compound Library

抗前列腺癌化合物库现货

Anti-Prostate Cancer Compound Library

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产品编号 L2195

前列腺癌是指发生在前列腺的上皮性恶性肿瘤,是男性生殖系统中常见的恶性肿瘤,具有复杂的疾病发病机制。Androgen Receptor、Hedgehog、TGF-β、Wnt、PI3K-AKT-mTOR 等多个信号通路和靶点参与前列腺癌的进展。 TargetMol 抗前列腺癌化合物库收集了2256 种与前列腺癌相关的化合物,包括已经报道具有前列腺癌治疗作用的化合物,以及靶向前列腺癌相关靶点的化合物,是抗前列腺癌药物研发的良好工具。

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产品编号 L2195

抗前列腺癌化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 2256种与前列腺癌相关的化合物,可以用于高通量和高内涵筛选;
  • 部分化合物已上市或已进入临床期;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
NF-κB
PI3K
Reactive Oxygen Species
VEGFR
EGFR
COX
Ras
mTOR
Endogenous Metabolite
Akt
ERK
PARP
p38 MAPK
CDK
Wnt/beta-catenin
JAK
AMPK
GSK-3
STAT
Antibacterial
FGFR
Androgen Receptor
PDGFR
Raf
MEK
JNK
Src
FLT
c-Kit
Caspase
Parasite
MAPK
IκB/IKK
TNF
DNA-PK
S6 Kinase
Histone Methyltransferase
Cytochromes P450
ATM/ATR
Hedgehog/Smoothened
Bcl-2 Family
c-Met/HGFR
PPAR
Tyrosine Kinases
Antifungal
IL Receptor
Potassium Channel
Antibiotic
Bcr-Abl
Aurora Kinase
Influenza Virus
Ferroptosis
NOD
RIP kinase
HIV Protease
HER
PKC
PDK
NO Synthase
Kras
c-RET
Mitophagy
Antioxidant
Pim
Calcium Channel
Epigenetic Reader Domain
Casein Kinase
DNA/RNA Synthesis
NOD-like Receptor (NLR)
Gamma-secretase
MMP
PKA
Interleukin
PI4K
IRAK
PD-1/PD-L1
Smo
IGF-1R
Estrogen/progestogen Receptor
Microtubule Associated
Virus Protease
Dehydrogenase
ROS
HIF/HIF Prolyl-Hydroxylase
Rho
Lipoxygenase
Nrf2
c-Fms
GABA Receptor
Drug Metabolite
Prostaglandin Receptor
p53
Mitochondrial Metabolism
Estrogen Receptor/ERR
TGF-beta/Smad
HDAC
Phosphatase
Tyrosinase
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NOS
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PTEN
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Syk
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PDE
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SIK
E1/E2/E3 Enzyme
HSV
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TRP/TRPV Channel
5-HT Receptor
Anti-infection
TLR
PLK
Histone Acetyltransferase
MELK
PGE Synthase
Proteasome
CSF-1R
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transporter
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GPCR
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Aryl Hydrocarbon Receptor
LDL
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Free radical scavengers
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Serine Protease
BTK
Mdm2
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PAK
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ROS Kinase
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Cholecystokinin Receptor
DNA Alkylation
Beta-Secretase
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IFNAR
RANKL/RANK
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FKBP
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PYK2
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YAP
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Thyroid hormone receptor(THR)
Melanin-concentrating Hormone Receptor (MCHR)
NPC1L1
DHFR
FLAP
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DNA
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DNA Alkylator/Crosslinker
Arrestin
Pyroptosis
GPX
PKM
MicroRNA
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PAFR
Haspin Kinase
DPP-4
RSV

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