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TargetMol | Compound Library

抗前列腺癌化合物库现货

Anti-Prostate Cancer Compound Library

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产品编号 L2195

前列腺癌是指发生在前列腺的上皮性恶性肿瘤,是男性生殖系统中常见的恶性肿瘤,具有复杂的疾病发病机制。Androgen Receptor、Hedgehog、TGF-β、Wnt、PI3K-AKT-mTOR 等多个信号通路和靶点参与前列腺癌的进展。 TargetMol 抗前列腺癌化合物库收集了2256 种与前列腺癌相关的化合物,包括已经报道具有前列腺癌治疗作用的化合物,以及靶向前列腺癌相关靶点的化合物,是抗前列腺癌药物研发的良好工具。

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产品编号 L2195

抗前列腺癌化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 2256种与前列腺癌相关的化合物,可以用于高通量和高内涵筛选;
  • 部分化合物已上市或已进入临床期;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
NF-κB
PI3K
Reactive Oxygen Species
VEGFR
EGFR
COX
Ras
mTOR
Endogenous Metabolite
Akt
ERK
PARP
p38 MAPK
Wnt/beta-catenin
CDK
JAK
AMPK
GSK-3
STAT
FGFR
Antibacterial
Androgen Receptor
PDGFR
Raf
MEK
Src
JNK
FLT
c-Kit
Parasite
Caspase
MAPK
IκB/IKK
TNF
DNA-PK
S6 Kinase
Histone Methyltransferase
Cytochromes P450
ATM/ATR
Hedgehog/Smoothened
Bcl-2 Family
c-Met/HGFR
PPAR
Antifungal
Tyrosine Kinases
IL Receptor
Potassium Channel
HIV Protease
Bcr-Abl
Aurora Kinase
Influenza Virus
Antibiotic
Ferroptosis
PKC
RIP kinase
PDK
NOD
HER
Kras
Mitophagy
c-RET
NO Synthase
Antioxidant
Pim
Calcium Channel
Epigenetic Reader Domain
Gamma-secretase
DNA/RNA Synthesis
Casein Kinase
NOD-like Receptor (NLR)
MMP
PKA
Interleukin
PI4K
Smo
IGF-1R
IRAK
PD-1/PD-L1
Estrogen/progestogen Receptor
Dehydrogenase
ROS
Microtubule Associated
HIF/HIF Prolyl-Hydroxylase
Virus Protease
Rho
Lipoxygenase
Nrf2
c-Fms
Drug Metabolite
Mitochondrial Metabolism
Prostaglandin Receptor
GABA Receptor
p53
Phosphatase
Estrogen Receptor/ERR
Topoisomerase
TGF-beta/Smad
HDAC
Tyrosinase
NOS
ROCK
Beta Amyloid
PTEN
Chk
P-gp
Trk receptor
Syk
Sodium Channel
FAK
Tie-2
PDE
HSP
AChR
DYRK
GNRH Receptor
TRP/TRPV Channel
SIK
E1/E2/E3 Enzyme
Antifection
HSV
Cholinesterase (ChE)
TLR
5-HT Receptor
PLK
Anti-infection
Proteasome
ATPase
HCV Protease
NADPH
Adrenergic Receptor
CSF-1R
PGE Synthase
Antiviral
SARS-CoV
Histone Acetyltransferase
MELK
SGK
Cannabinoid Receptor
TAM Receptor
Carbonic Anhydrase
Transferase
Integrin
Reductase
RAAS
c-Myc
HBV
Glucocorticoid Receptor
IAP
Glucosidase
Angiotensin-converting Enzyme (ACE)
OXPHOS
MNK
Ephrin Receptor
transporter
ASK
HIF
MDM-2/p53
MLK
GPCR
Histamine Receptor
Glutathione Peroxidase
TOPK
Progesterone Receptor
Serine Protease
Aryl Hydrocarbon Receptor
LDL
Opioid Receptor
CaMK
Survivin
Porcupine
Free radical scavengers
ALK
Retinoid Receptor
Phospholipase
BTK
Mdm2
Chloride channel
BACE
IFNAR
PERK
GTPase
Cholecystokinin Receptor
Leukotriene Receptor
RANKL/RANK
IRE1
DNA Alkylation
PAK
Beta-Secretase
PSMA
LRRK2
Hippo pathway
FKBP
Reverse Transcriptase
KLF
DNA Methyltransferase
ROS Kinase
Apelin receptor
RAR/RXR
Dopamine Receptor
ROR
ADC Cytotoxin
YAP
Adenosine Receptor
MRP
Serine/threonin kinase
Cysteine Protease
FXR
PYK2
MAO
Prolyl Endopeptidase (PREP)
Myosin
UGT
NMDAR
ABC Transporter
Fatty Acid Synthase
FAAH
CCR
CXCR
Endothelin Receptor
cAMP
GluR
DUB
ATP Citrate Lyase
Acyltransferase
STING
Discoidin Domain Receptor (DDR)
Gap Junction Protein
NADPH-oxidase
CFTR
S1P Receptor
Monoamine Oxidase
Thyroid hormone receptor(THR)
Melanin-concentrating Hormone Receptor (MCHR)
Proton pump
MicroRNA
NPC1L1
CD38
DHFR
Y Box Binding Protein 1
Arginase
DNA Alkylator/Crosslinker
LTR
Arrestin
Na+/Ca2+ Exchanger
Necroptosis
gp120/CD4
MIF
VDA
OCT
ASCT
Hck
ATG
Nucleoside Antimetabolite/Analog
Liver X Receptor
Glucokinase
IDO
iGluR
FLAP
PAFR
Haspin Kinase
Na-K-Cl cotransporter
Monoamine Transporter
DPP-4
Somatostatin
DNA
Indoleamine 2,3-Dioxygenase (IDO)
SGLT
Wee1
Lipid
BCRP
Glutathione reductase
Aminopeptidase
Sirtuin
CD73
AIM2
Decarboxylase
cGAS
hCE
PAI-1
Pyroptosis
RSV
Methionine Adenosyltransferase (MAT)
GST
GPX
Aromatase
CRISPR/Cas9
Hydroxylase
Adenosine Deaminase
Cuproptosis
DAPK
Platelet aggregation
BMI-1
Sigma receptor
AhR
Kinesin
PKM

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