248
85
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T24706 |
RBC10
RBC 10,RBC-10 |
GTPase | GPCR/G Protein |
RBC10 抑制 Ral 与其效应物 RALBP1 的结合,以及抑制 Ral 介导的鼠胚胎成纤维细胞的细胞扩散和人类癌细胞系的非贴壁依赖性生长。 | |||
T14358 |
Avoralstat
BCX4161 |
Others | Others |
Avoralstat (BCX4161) 是血浆激肽释放酶(PKK)抑制剂,具有口服活性,可用于遗传性血管性水肿的研究。 | |||
T28918 |
Talviraline
Bay 10-8979,HBY 097,Bay10-8979,Bay-108979,Bay108979,Bay 108979,Bay-10-8979 |
HIV Protease; DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Proteases/Proteasome |
Talviraline (Bay 10-8979) 是一种 RNA 引导的 DNA 聚合酶抑制剂。Talviraline 对多种人类细胞系以及新鲜人类外周血淋巴细胞和巨噬细胞中的 HIV-1 诱导的细胞杀伤和 HIV-1 复制具有很强的抑制作用。 | |||
T77632 |
Antiviral agent 34
|
Antiviral; DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Immunology/Inflammation |
Antiviral agent 34 是一种可口服且作用效果较强的抗病毒化合物,抑制甲型和乙型流感病毒。Antiviral agent 34 通过调节 RNA 聚合酶来抑制流感病毒的增殖。Antiviral agent 34 可用于研究病毒感染。 | |||
T36375 |
Ralaniten triacetate
EPI-506 |
Androgen Receptor | Endocrinology/Hormones |
Ralaniten triacetate (EPI-506) 是 Ralaniten 的前体,是一种具有口服活性的雄激素受体 N 端结构域 (AR-NTD) 抑制剂,具有抗癌活性,可用于研究前列腺癌和乳腺癌。 | |||
T77122 |
Praluzatamab
|
Others | Others |
Praluzatamab 是一种靶向活化白细胞粘附分子 (ALCAM/CD116) 的单克隆抗体。Praluzatamab 是 Praluzatamab ravtansine 的裸抗, 可用于合成抗体活性分子偶联物(Praluzatamab ravtansine)。Praluzatamab 可用于研究研究乳腺癌。 | |||
T13140 |
Umbralisib R-enantiomer
TGR-1202 R-enantiomer,RP5264 R-enantiomer |
PI3K | PI3K/Akt/mTOR signaling |
Umbralisib R-enantiomer (RP5264 R-enantiomer) 是 PI3K 的δ型抑制剂,是 TGR-1202 活性较低的对映体。Umbralisib R-enantiomer 对δ型 pi3激酶的 IC50,至少比抑制剂对其他 PI3K 亚型(A, β和γ)的 IC50低20倍。 | |||
T9449 |
Nitrofural
[(E)-(5-nitrofuran-2-yl)methylideneamino,(E)-2-((5-硝基呋喃-2-基)亚甲基)肼甲酰胺 |
Antibacterial | Microbiology/Virology |
Nitrofural 是 20 世纪已在临床应用中确立的硝基呋喃。 Nitrofural 在临床上对广泛的革兰氏阳性和革兰氏阴性细菌(包括许多常见的泌尿道病原体菌株)仍然有效。 | |||
T20549 |
Neutral red
|
Others | Others |
Neutral Red 是含氮 pH 指示剂(pKi=6.8),是类囊体内部酸化的指示剂。它能够将溶酶体染成红色。 | |||
T67904 |
Antiviral agent
|
HBV | Microbiology/Virology |
Antiviral agent是一种具有抗乙型肝炎活性的噻唑烷。 | |||
T0660 |
Beta-Tetralone
2-Tetralone,beta-四氢萘酮 |
P450 | Metabolism |
Beta-Tetralone (2-Tetralone) 是 tetralin 的酮衍生物。 | |||
T6482 |
Efaproxiral Sodium
乙丙昔罗钠,RSR13 sodium |
Reactive Oxygen Species | Immunology/Inflammation; Metabolism; NF-κB |
Efaproxiral Sodium (RSR13 sodium) 是血红蛋白 (Hb) 合成变构调节剂,能够减少血红蛋白氧 (O2) 的结合亲和力。 | |||
T9395 |
(1S,4R)-N-Desmethyl Sertraline Hydrochloride
|
Others | Others |
(1S,4R)-N-DesmethylSertralineHydrochloride 是一种Serotonin transporter 和 Norepinephrine transporter 抑制剂,IC5分别为19 nM 和35 nM. | |||
T7547 |
Ralfinamide mesylate
FCE-26742A (mesylate) |
Sodium Channel | Membrane transporter/Ion channel |
Ralfinamide mesylate (FCE-26742A (mesylate)) 是一种口服有效,来源于 α-aminoamide 的钠离子通道阻滞剂, 在缓解疼痛方面有研究价值。 | |||
T17111 |
Todralazine hydrochloride
Ecarazine hydrochloride,盐酸托屈嗪 |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Todralazine hydrochloride (Ecarazine hydrochloride) 是一种 β2AR 阻滞剂,具有抗氧化和自由基清除活性。 Todralazine hydrochloride 可用于抗高血压的研究。 | |||
T19748 |
Butralin
A-820,A820,A 820,丁烯酯甲酸,Tamex |
Others | Others |
Butralin (A-820) 是一种除草剂和植物生长控制剂。 | |||
T26939 |
Cadralazine
ISF 2469,卡屈嗪,ISF-2469,ISF2469 |
Others | Others |
Cadralazine (ISF 2469) 是一种外周小动脉血管扩张剂,可用于作为抗高血压药物的研究。 | |||
T28255 |
Opaviraline
GW420867X,GW-867,HBY-1293,GW867,GW-420867X |
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Opaviraline (GW-420867X) 是一种有效逆转录酶抑制剂,对Human immunodeficiency virus 1具有抑制作用,具有治疗HIV 感染的潜力。 | |||
T7349 |
Ralfinamide
(S)-2-[[4-[(2-氟苄基)氧基]苄基]氨基]丙酰胺,Priralfinamide,FCE-26742A |
Sodium Channel | Membrane transporter/Ion channel |
Ralfinamide (Priralfinamide) 是一种具有口服活性的,来源于 α-aminoamide 的钠离子通道阻滞剂, 在缓解疼痛方面有研究的价值。 | |||
T20508 |
Orfralure
|
||
Orfralure is a biochemical substance. | |||
T19999 |
1-Tetralol, (S)-
(S)-(+)-1,2,3,4-四氢-1-萘酚,(S)-Tetralin-1-ol,(S)-(+)-1,2,3,4-Tetrahydro-1-naphthol,(S)-1-Hydroxytetralin,J330.337C |
Others | Others |
1-Tetralol, (S)- ((S)-1-Hydroxytetralin) 可在细胞实验中用作 AKR1C1 的底物。 | |||
T5330 |
Fluralaner
AH252723,氟雷拉纳,A1443 |
GABA Receptor; Parasite | Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience |
Fluralaner (A1443) 是一种异恶唑啉杀外寄生虫剂。 它有效且选择性地抑制 GABA 受体通道阻滞剂 EBOB 与家蝇头膜的结合,IC50值为 455 pM。 | |||
T1613 |
Hydralazine hydrochloride
Hydralazine HCl,Apresoline,盐酸肼屈嗪 |
MAO; HIF/HIF Prolyl-Hydroxylase | Chromatin/Epigenetic; Metabolism; Neuroscience |
Hydralazine hydrochloride (Apresoline) 是一种直接作用的血管舒张剂,可抗高血压。 | |||
T2265 |
Bimiralisib
5-(4,6-dimorpholino-1,3,5-triazin-2-yl)-4-(trifluoromethyl)pyridin-2-amine,PQR309,PI3K-IN-2 |
Others; PI3K; S6 Kinase; mTOR | MAPK; Others; PI3K/Akt/mTOR signaling |
Bimiralisib (PI3K-IN-2) 是一种有效的,可渗透脑的 mTOR/PI3K 抑制剂,是一种 mTORC1和 mTORC2抑制剂。它能够抑制 PI3Kα,PI3Kδ,PI3Kβ,PI3Kγ和 mTOR,IC50分别为 33 nM,451 nM,661 nM,708 nM 和 89 nM。 | |||
T39350 |
Sebetralstat
KVD900 |
Others | Others |
Sebetralstat (KVD900) 是一种血浆激肽释放酶抑制剂,可用于代谢性疾病的研究。 | |||
T21355 |
6-Chloro-1-tetralone
6-Chloro-α-Tetralone,5-CHLORO-L-INDOMONE,6-chloro-3;5-CHLORO-1-INDOMONE,5-CHLORO-1-INDOMONE,6-chloro-3 |
Others | Others |
6-Chloro-1-tetralone (6-chloro-3;5-Chloro-1-Indomone) 是合成药物化合物的重要中间体。 | |||
T14527 |
Benfluralin
|
||
Benfluralin 是一种除草剂,是一种农用化学品,可用作芽前除草剂。 用于控制一系列粮食和非粮食作物中的草和其他杂草。 | |||
T63272 |
Edralbrutinib
TG-1701 |
BTK | Angiogenesis; Tyrosine Kinase/Adaptors |
Edralbrutinib (TG-1701) 是有效的BTK抑制剂,具有抗癌活性,可用于治疗肿瘤、免疫系统疾病、血液及淋巴系统疾病。Edralbrutinib可用于研究膜性肾小球肾炎和视神经脊髓炎。 | |||
T16569 |
Praliciguat
IW-1973 |
Others; Guanylate cyclase | GPCR/G Protein; Others |
Praliciguat (IW-1973) 是一种有效且具有口服活性的可溶性鸟苷酸环化酶 (sGC) 刺激剂,还增强 NO 信号传导,可作为血管扩张剂。在 HEK-293 细胞中,它能够刺激 sGC,EC50值为 197 nM。 | |||
T6120 |
Pralatrexate
Folotyn,10-炔丙基-10-去氮杂氨基蝶呤,10-Propargyl-10-deazaaminopterin,普拉曲沙 |
Apoptosis; DHFR; Antifolate; TAM Receptor | Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Tyrosine Kinase/Adaptors |
Pralatrexate (10-Propargyl-10-deazaaminopterin) 是一种抗叶酸剂,也是二氢叶酸还原酶抑制剂,Ki 值为 13.4 pM。它具有抗肿瘤活性,可研究复发/难治性 T 细胞淋巴瘤。它是叶酰聚谷氨酸合成酶的底物,具有改善的细胞摄取和保留能力。 | |||
T3526 |
Dasotraline hydrochloride
SEP-225289 hydrochloride,达索曲林盐酸盐 |
Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Norepinephrine | GPCR/G Protein; Neuroscience |
Dasotraline hydrochloride (SEP-225289 hydrochloride) 是具有阻断多巴胺 (IC50=4 nM),去甲肾上腺素 (IC50=6 nM) 和三羟色胺转运蛋白 (IC50=11 nM)的三重再摄取抑制剂。 | |||
T4635 |
Ralinepag
APD811 |
Others; Prostaglandin Receptor | GPCR/G Protein; Immunology/Inflammation; Others |
Ralinepag (APD811) 是一种可口服的非前列腺素前列环素 (IP) 受体激动剂,对人和大鼠 IP 受体以及人 DP1 受体的 EC50 分别为 8.5、530 和 850 nM。 | |||
T8900 |
Seralutinib
GB002 |
PDGFR | Angiogenesis; Tyrosine Kinase/Adaptors |
Seralutinib (GB002) 是可吸入的PDGFRα 和 PDGFRβ激酶抑制剂,可用于研究肺动脉高压。 | |||
T1111 |
Pralidoxime Chloride
2-PAM chloride,吡啶醛肟甲氯,2-Pyridinealdoxime methochloride,2-PAM (chloride) |
AChE | Neuroscience |
Pralidoxime Chloride (2-PAM chloride) 是一种肟类化合物,对中毒乙酰胆碱酯酶具有恢复作用,可用于有机磷中毒的研究。 | |||
T6632 |
Raltitrexed
ZD1694,雷替曲塞,D1694,ICI-D1694,Tomudex |
Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
Raltitrexed (D1694) 是一种抗代谢药物,通过抑制胸苷酸合成酶起作用,可用于化疗。 | |||
T22592 |
ATPγS tetralithium salt
ATP-gamma-S tetralithium salt |
PERK | Apoptosis |
ATPγS tetralithium salt 是真核生物翻译起始因子 eIF4A 的核苷酸水解和RNA解链活性的底物,与 p97 突变体和朊病毒相关。 | |||
T0059 |
Diphenylpyraline hydrochloride
盐酸双苯比拉林,4-Diphenylmethoxy-1-methylpiperidine hydrochloride |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Diphenylpyraline hydrochloride (4-Diphenylmethoxy-1-methylpiperidine hydrochloride) 是一种组胺 H1 受体的拮抗剂,抑制多巴胺的吸收。它是可口服的抗组胺试剂,具有抗胆碱和抗过敏作用,可用于缓解过敏性疾病,如鼻炎、花粉热和瘙痒性皮肤疾病等。 | |||
TP1929L1 |
Saralasin acetate(34273-10-4 free base)
|
RAAS | Endocrinology/Hormones |
Saralasin acetate(34273-10-4 free base) 是一种非选择性血管紧张素 II 拮抗剂。 | |||
T4976 |
Umbralisib
TGR-1202,RP5264,TGR 1202,TGR1202 |
PI3K | PI3K/Akt/mTOR signaling |
Umbralisib (TGR 1202) 是一种PI3Kδ抑制剂,IC50=22.2 nM,EC50=24.3 nM。它同时可抑制CK1ε,EC50=6.0 μM。 | |||
T60440 |
Antiviral agent 17
|
||
Antiviral agent 17 (Compound 4) 是一种抗感染剂,在人类复制子试验中显著保留其抗病毒作用,EC50值为0.015 μM。Antiviral agent 17 对小鼠诺如病毒(MNV)表现出良好的抗病毒活性。Antiviral agent 17 在研究传染性和恶性疾病方面具有潜力。 | |||
T1251 |
Dicloralurea
双(三氯乙醛基)脲,Dichlorolurea,双 (三氯乙醛基) 脲,DCU |
Others | Others |
Dicloralurea (DCU) 是一种兽用的食品添加剂,可用作生长刺激剂。 | |||
T6047 |
Ralimetinib dimesylate
LY2228820 dimesylate,Ralimetinib,LY2228820,Ralimetinib Mesylate |
Apoptosis; p38 MAPK; Autophagy | Apoptosis; Autophagy; MAPK |
Ralimetinib dimesylate (LY2228820 dimesylate) 是一种选择性,ATP 竞争性的 p38 MAPK α/β抑制剂,IC50分别为5.3 和 3.2 nM。 | |||
T10497 |
Benralizumab
BIW-8405,MEDI-563 |
Apoptosis; IL Receptor; Interleukin | Apoptosis; Immunology/Inflammation |
Benralizumab (MEDI-563) 是一种靶向白介素 5 受体 α (IL-5Rα) 单克隆抗体,通过增强抗体依赖性细胞介导的细胞毒性促使嗜酸性粒细胞快速进行反应。Benralizumab 可用于严重的嗜酸性哮喘,可用于预防慢性阻塞性肺病加重。 | |||
T3270 |
Dihydralazine sulfate
1,4-Dihydrazinophthalazine sulfate,硫酸双肼屈嗪,Hydralazine sulfate,Nepresol,Depressan,Dihydralazine sulphate |
Others | Others |
Dihydralazine sulfate (Nepresol) 是一种抗高血压的药物。 | |||
T2239L |
Raltegravir
雷特格韦,MK-0518 |
HIV Protease; Integrase | Microbiology/Virology; Proteases/Proteasome |
Raltegravir (MK-0518) 是一种HIV 整合酶抑制剂。 | |||
T28503 |
Ralitoline
GOE-4942,PD-117818,Ralitolina,CI-946,Ralitolinum |
||
Ralitoline (Ralitolinum) 是一种抗惊厥剂,具有抗癌活性和钠通道阻断活性。 | |||
T2365 |
Pilaralisib
SAR245408,XL-147 |
PI3K | PI3K/Akt/mTOR signaling |
Pilaralisib (XL-147) 是一种有效的、选择性的 I 类PI3Ks 抑制剂,能够抑制 PI3Kα (IC50:39 nM),PI3Kβ (IC50:383 nM),PI3Kγ (IC50:23 nM) 和 PI3Kδ (IC50:36 nM)。 | |||
T1338 |
Sucralfate
硫糖铝,Sucrose octasulfate–aluminum complex |
FGFR; Others; Antibacterial; Prostaglandin Receptor | Angiogenesis; GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Others; Tyrosine Kinase/Adaptors |
Sucralfate (Sucrose octasulfate–aluminum complex) 是一种口服活性胃保护剂。它抑制消化性活性,并与黏膜损伤时暴露的带负电荷的上皮下蛋白结合,形成一层粘性层,保护血管床和增殖区。它可用于预防和治疗胃肠道疾病。 | |||
T9183 |
Ralmitaront
RO6889450 |
Others | Others |
Ralmitaront (RO6889450) 是口服具有活力的口服微量胺相关受体 1 (TAAR1) 的部分激动剂。它是一种神经抑制剂,可用于研究神经相关疾病,如精神分裂症 (SCZ)、分裂情感性障碍。 | |||
T76975 |
Tomaralimab
OPN-305 |
TLR | Immunology/Inflammation |
Tomaralimab (OPN-305) 是一种人源化的靶向 TLR2 的 IgG4 单克隆抗体。Tomaralimab 可用于研究骨髓增生异常综合征 (MDS) 。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T5625 |
Zearalenone
玉米,Mycotoxin F2,玉米烯酮,RAL,F2 toxin,Toxin F2 |
Others | Others |
Zearalenone (F2 toxin) 是真菌毒素,主要由食物和饲料中的 Fusarium 产生。它会引起幼龄母猪乳房发育早熟或其它雌激素效应。它在猪、牛、羊体内具有雌激素活性,急性毒性低。 | |||
TN1008 |
Psoralenoside
|
CaMK; Calcium Channel; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience |
Psoralenoside 是源于补骨脂中的苯并呋喃苷,具有抗肿瘤、抗菌、促进成骨细胞增殖和雌激素样活性。它对组胺 H1、钙调素和电压门控 l 型钙通道具有较高的亲和力。 | |||
T5090 |
2-Methylbutyraldehyde
2-Ethylpropanal,RS)-2-Methylbutanal,2-甲基丁醛 |
Others | Others |
2-Methylbutyraldehyde (2-Ethylpropanal) 属于短链醛类化合物,白术饮片中的焦香味物质之一。 | |||
T13542 |
α-Zearalenol
|
Estrogen Receptor/ERR | Endocrinology/Hormones |
α-Zearalenol 是一种霉菌毒素,对雌激素受体具有高亲和力。它是 zearalenone (ZEN) 的一种衍生物,由于其异种雌激素效应可引起动物的生殖障碍。 | |||
T2943 |
5-Hydroxymethylfurfural
5-羟甲基糠醛,2-Hydroxymethyl-5-furfural,2-Formyl-5-hydroxymethylfuran,5-Hydroxymethyl-2-furaldehyde,5-(Hydroxymethyl)furan-2-carbaldehyde |
Others; Antifungal | Microbiology/Virology; Others |
5-Hydroxymethylfurfural (2-Formyl-5-hydroxymethylfuran) 是来自木质纤维素生物质,能抑制酵母的生长和发酵。 | |||
T8213 |
Isolinderalactone
|
NOS; STAT | Immunology/Inflammation; JAK/STAT signaling; Stem Cells |
Isolinderalactone 具有抗炎和抗癌能力,具有中等的 iNOS 抑制活性,IC50 值为 0.30 uM。 | |||
T1399 |
Sucralose
Trichlorosucrose,三氯蔗糖,E955 |
Others; Endogenous Metabolite | Metabolism; Others |
Sucralose (Trichlorosucrose) 是一种无营养的人工甜味剂 (sweetener) 和代糖,它能够激活保守神经的禁食响应,从而刺激啮齿动物产生食欲。 | |||
T7921 |
β-Cyclocitral
beta-Cyclocitral,β-环柠檬醛 |
Others | Others |
β-Cyclocitral 是 β-胡萝卜素的挥发性氧化衍生物,是微囊藻特有的掠食性动物防御信号。它是一种强大的驱虫剂。它是主要的挥发性萜类化合物之一,可以上调防御基因的表达,从而增强过量光照 (EL) 的适应性。 | |||
T3S0289 |
Araloside X
|
Calcium Channel | Membrane transporter/Ion channel; Metabolism |
Aralosides possess protective effect against experimental myocardial ischemia and infarction, the mechanism of myocardial protection may be attributed to the amelioration of FFA metabolic deterioration and membrane peroxidation induced by oxygen free radi | |||
T1549 |
Raloxifene hydrochloride
LY156758 hydrochloride,盐酸雷洛昔芬,Raloxifene HCl,LY139481 hydrochloride,Keoxifene hydrochloride,LY156758 (Keoxifene) HCl |
Estrogen Receptor/ERR; Others; MAO; Estrogen/progestogen Receptor; Autophagy | Autophagy; Endocrinology/Hormones; Metabolism; Neuroscience; Others |
Raloxifene hydrochloride (LY156758 hydrochloride) 是一种选择性且可口服的雌激素受体调节剂,用于预防绝经后妇女的骨质疏松症。它对骨骼和胆固醇代谢具有雌激素激动作用,但对乳腺和子宫组织具有完全的雌激素拮抗作用。 | |||
Fr12275 |
7-Methoxy-1-tetralone
|
Others | Others |
7-Methoxy-1-tetralone 可能具有杀虫活性。 | |||
T2942 |
Psoralen
Ficusin,Furocoumarin,补骨脂素,psoralene |
Apoptosis; Influenza Virus; HIV Protease; DNA/RNA Synthesis | Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Proteases/Proteasome |
Psoralen (Ficusin) 是从补骨脂种子中提取的一种香豆素。它具有如抗癌、抗氧化、抗抑郁、抗癌、抗菌、抗病毒等多种生物学特性。 | |||
T3399 |
Psoralidin
|
Others; Estrogen/progestogen Receptor; Reactive Oxygen Species; Lipoxygenase; Gamma-secretase; Akt; COX; Antibacterial | Cytoskeletal Signaling; Endocrinology/Hormones; Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience; NF-κB; Others; PI3K/Akt/mTOR signaling; Proteases/Proteasome; Stem Cells |
Psoralidin 是COX-2和5-LOX 的抑制剂,有抗癌,抗菌和抗炎作用。它显著下调NOTCH1信号传导,还极大地诱导活化氧产生。 | |||
T5657 |
Veratraldehyde
3,4-Dimethoxybenzaldehyde,藜芦醛 |
Antifungal | Microbiology/Virology |
Veratraldehyde (3,4-Dimethoxybenzaldehyde) 是一种能够使用于香料,农业化学和制药工业中的重要化学品。 | |||
T3418 |
Demethylzeylasteral
去甲泽拉木醛,Demethylzeylasteral (T-96) |
Apoptosis; UGT | Apoptosis; Metabolism |
Demethylzeylasteral (Demethylzeylasteral (T-96)) 分离自雷公藤,具有抗炎、免疫抑制和抗肿瘤活性。它通过阻断 TGF-β 信号通路,抑制三阴性乳腺癌的侵袭,它能显著减轻动脉粥样硬化。 | |||
TN1343 |
8-Geranyloxypsoralen
8-香叶草氧基补骨脂素 |
Anti-infection; P450; BACE | Metabolism; Microbiology/Virology; Neuroscience |
8-Geranyloxypsoralen 是一种呋喃香豆素,分离自葡萄柚,是 P450 3A4 的有效抑制剂(IC50:3.93 μM)。 | |||
T5S1897 |
Linderalactone
|
Apoptosis; Others; JAK | Angiogenesis; Apoptosis; Chromatin/Epigenetic; JAK/STAT signaling; Others; Stem Cells |
Linderalactone 是从乌药中分离出来的一种倍半萜烯内酯,通过调节凋亡相关蛋白的表达和抑制 JAK/STAT 信号通路来抑制癌细胞生长。它以 IC50值为 15 µM 来抑制肺癌 A-549 细胞的增殖。 | |||
T4S0290 |
Araloside A
Chikusetsusaponin IV,竹节参皂苷IV |
RAAS; Fas/FasL | Apoptosis; Endocrinology/Hormones |
Araloside A (Chikusetsusaponin IV) 是竹节参中的一种成分,对肾素renin 具有低抑制活性(IC50:77.4 μM)。 | |||
T4918 |
DL-Glyceraldehyde
Glyceric aldehyde,DL-甘油醛晶体 |
Reductase | Endocrinology/Hormones; Metabolism |
DL-Glyceraldehyde (Glyceric aldehyde) 是由酶甘油醛脱氢酶的作用产生的,该酶使用 NADP 作为辅因子将甘油转化为甘油醛。它是一种高活性化合物,可以修饰和交联蛋白质。 | |||
T2S1907 |
Coniferaldehyde
Ferulaldehyde,Ferulyl aldehyde,4-HYDROXY-3-METHOXYCINNAMALDEHYDE,松柏醛,Coniferyl aldehyde,松柏醛;4-羟基-3-甲氧基肉桂醛 |
Apoptosis; Antioxidant | Apoptosis; oxidation-reduction |
Coniferaldehyde (Ferulaldehyde) 是一种血红素加氧酶-1 的有效诱导剂,具有抗炎作用。在 RAW264.7 巨噬细胞中,它通过 PKCα/βII/Nrf-2/HO-1 依赖性途径来抑制 LPS 诱导的细胞凋亡。 | |||
T0896 |
Furaltadone hydrochloride
Furaltadone HCl,盐酸呋喃它酮 |
Antibacterial; Antibiotic; Parasite | Microbiology/Virology |
Furaltadone hydrochloride (Furaltadone HCl) 是硝基呋喃药,可研究肠沙门氏菌感染,治疗球虫病。Furaltadone 具有体外抑制葡萄球菌作用。 | |||
T3154 |
Citral
Geranialdehyde,alpha-Citral,柠檬醛,geranial |
Others | Others |
Citral (alpha-Citral) 是一种单萜,从柠檬草精油中获得,具有抗疼痛、抗炎作用。 | |||
TCP2934 |
5-Methylfurfural
5-Methyl furfural,5-Methyl-2-furaldehyde,5-甲基呋喃醛 |
Others | Others |
5-Methylfurfural (5-Methyl-2-furaldehyde) 是一种天然存在的调味剂,存在于香烟烟雾凝结物,烤土豆粉,甘草精油,储存的脱水橙粉,挥发性化合物的烤牛肉,香气浓缩的海绵蛋糕,咖啡,面包,茶和可可种。 | |||
TN3694 |
Coniferaldehyde
|
NOS; COX; Nrf2; PKC; Autophagy | Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling; Immunology/Inflammation; Neuroscience |
Coniferaldehyde 能显着抑制酒球菌菌株的生长活力。 Coniferaldehyde 通过诱导血红素加氧酶 1 (HO-1) 发挥抗炎特性。 | |||
TN1148 |
Isopsoralenoside
|
Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Antibacterial | Endocrinology/Hormones; Microbiology/Virology |
Isopsoralenoside 是补骨脂多糖中的一种苯并呋喃苷。它在消化道内容物中可迅速代谢为补骨脂素。它具有雌激素样活性、促进成骨细胞增殖活性、抗肿瘤活性和抗菌活性。 | |||
T5662 |
5-Hydroxy-1-tetralone
|
Others | Others |
5-hydroxy-1-tetralone 是一种荧光标记试剂,可用于生物样品中的鞘糖脂的测定。 | |||
T4930 |
ISOBUTYRALDEHYDE OXIME
|
Others | Others |
ISOBUTYRALDEHYDE OXIME 是衍生自 2-methylpropanal 的醛肟。它来源于异丁醛。 | |||
T2826 |
Asaraldehyde
Asarylaldehyde,2,4,5-trimethoxy-Benzaldehyde,Asaronaldehyde,细辛醛 |
COX | Immunology/Inflammation; Neuroscience |
Asaraldehyde (2,4,5-trimethoxy-Benzaldehyde) 是COX-2抑制剂,能够明显降低环加氧酶 II (COX-2) 的活性(IC50:100 μg/mL)。 | |||
TN4771 | Phyltetralin | ||
Phyltetralin has antihyperuricemic activity. | |||
TN2403 | Glabralide B | Others | Others |
Glabralide B is a natural product from plants | |||
T14548 |
Beta-Zearalanol
|
Others | Others |
Beta-Zearalenol, a derivative of zearalenone (ZEA) capable of conjugating with glucuronic acid[2], is a mycotoxin produced by Fusarium spp. It induces apoptosis and oxidative stress in mammalian reproductive cells[1]. | |||
TN4591 |
Murralongin
|
Others | Others |
Murralongin exhibits cytotoxicity against cholangiocarcinoma cell line, KKU-100. | |||
T67590 |
3-Furaldehyde
|
||
3-Furaldehyde 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 T67590,CAS号为 498-60-2。 | |||
TN3560 |
Cabralealactone
|
Antifection | Microbiology/Virology |
Cabralealactone displays antimycobacterial activity against Mycobacterium tuberculosis, it is weakly cytotoxic to a breast cancer (BC) cell line, it is moderately active against a small-cell lung cancer (NCI-H187) cell line. | |||
TN5229 |
Vibralactone B
|
Antifection | Microbiology/Virology |
Vibralactone B shows antibacterial activity, it can inhibit significantly the growth of E. coli and Pseudomonas aeruginosa, with MBC values of 50 and 100 ug/mL, respectively. | |||
T82282 |
Glycyuralin E
|
||
Glycyuralin E,一种从Glycyrrhiza uralensis中可分离的天然化合物。 | |||
TN3559 |
Cabraleahydroxylactone
|
HSV | Microbiology/Virology |
Cabraleahydroxylactone displays antimycobacterial activity against Mycobacterium tuberculosis, it is weakly cytotoxic to a breast cancer (BC) cell line.It shows antiviral activity against herpes simplex virus type-1 with an IC50 value of 3.20 ug/mL, in comparison with the standard acyclovir (IC50=1.90ug/mL). | |||
T79952 |
Kadsuralignan A
|
||
Kadsuralignan A(化合物1)为从五味子(Schisandra lancifolia)叶和茎中分离的一种二苯并环辛二烯木脂素,显示出抗HIV活性,其EC50值为2.23 μg/mL。 | |||
T38478 |
Mevalonic acid 5-pyrophosphate tetralithium
Mevalonicacid5-diphosphatetetralithium,Mevalonic acid 5-pyrophosphate tetralithium,5-Diphosphomevalonic acid tetralithium |
||
Mevalonic acid 5-pyrophosphate (also known as 5-Diphosphomevalonic acid) tetralithium is an endogenous metabolite involved in the mevalonate pathway. | |||
TN3557 |
Cabraleadiol
|
ATPase; Antifection | Membrane transporter/Ion channel; Microbiology/Virology |
Cabraleadiol displays antimycobacterial activity against Mycobacterium tuberculosis, it also is weakly cytotoxic to a breast cancer (BC) cell line. Cabraleadiol inhibits photosystem II (PS II) and induces the appearance of small G band which is related wi | |||
TN3556 |
Cabraleadiol 3-acetate
|
Others | Others |
Cabraleadiol 3-acetate是一种天然产物,属于楝科米仔兰属,其产品编号为 TN3556,CAS号为 35833-62-6。Cabraleadiol 3-acetate可用作对照参考。 | |||
TN3267 | 8-(7-Hydroxy-3,7-dimethyl-2,5-octadienyloxy)psoralen | Others | Others |
8-(7-Hydroxy-3,7-dimethyl-2,5-octadienyloxy)psoralen 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3267,CAS号为 144398-34-5。 | |||
TN4128 |
Geraldol
|
Others | Others |
Geraldol 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4128,CAS号为 21511-25-1。 | |||
TN4784 |
Picraline
|
SGLT | GPCR/G Protein |
A series of a hydroxy substituted derivatives 21-28 at C-17 of the Picraline-type alkaloids have been derived as having potent SGLT inhibitory activity. | |||
TN2926 |
3-Epicabraleahydroxylactone
|
Others | Others |
3-Epicabraleahydroxylactone has anti-tumor promoting effect, it has anti-carcinogenic activity by the inhibitory effect on the induction of Epstein-Barr virus early antigen(EBV-EA) by the tumor promoter. | |||
T13551 |
Araliadiol
|
Others | Others |
Araliadiol is a polyacetylenic compound isolated from the leaves of Aralia cordata Thunb. Araliadiol inhibits MCF-7 cell growth (IC50: 6.41 µg/mL). | |||
T13577 |
β-Zearalenol
|
Others | Others |
β-Zearalenol, a non-steroidal estrogenic mycotoxin synthesized by Fusarium species, potentially influences transcription and affects gene expression on the translational level. | |||
TN3266 |
8-(6-Hydroperoxy-3,7-dimethyl-2,7-octadienyloxy)psoralen
|
Others | Others |
8-(6-Hydroperoxy-3,7-dimethyl-2,7-octadienyloxy)psoralen 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3266,CAS号为 151121-39-0。 | |||
TN2925 |
3-Epicabraleadiol
|
Others | Others |
3-Epicabraleadiol是一种天然产物,属于山茶科山茶属,其产品编号为 TN2925,CAS号为 19942-04-2。3-Epicabraleadiol可用作对照参考。 | |||
TN5251 |
Walsuralactam A
|
Others | Others |
Walsuralactam A in the formula I, which is used as an active ingredient, and is used for treating and preventing the tumour. | |||
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