首页 工具
登录
购物车
口服活性化合物库

口服活性化合物库

现 货
产品编号 L9850 Orally Active Compound Library
  库化合物信息   Excel SDF

口服给药是临床给药尤其是长期用药的常用给药方式,也是安全、方便、经济的给药方法;口服生物利用度是药物经胃肠道黏膜吸收,经过肝脏进入体循环血液中的药量占口服剂量的百分比;口服生物利用度高的药物,较低剂量即可达到疗效,有效降低毒副作用;而口服生物利用度过低时,药理活性好的化合物也无法在靶部位充分的暴露,由此造成治疗的失败或者剂量过高产生较大的毒副作用,导致药物开发失败,限制了应用。 TargetMol 精心收集了 2484 种公开报道具有口服活性的化合物,可以用于药物再利用及口服活性药物的开发。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
获取报价
点击图片重新获取验证码

产品描述

  • 2484种口服活性化合物独特集合,可用于高通量筛选和高内涵筛选;
  • 部分药物已批准上市或处于临床试验中,生物活性和安全性得到验证;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • NMR和HPLC检测技术保证产品高纯度;
  • 所有化合物现货供应。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L9850)
点击图片重新获取验证码

客户使用化合物库发表的文献

收起

化合物库组成

Autophagy (297)
Apoptosis (271)
Antibacterial (206)
Antibiotic (190)
5-HT Receptor (133)
Endogenous Metabolite (110)
Adrenergic Receptor (102)
Dopamine Receptor (84)
Histamine Receptor (82)
COX (77)
Parasite (64)
HIV Protease (63)
AChR (61)
DNA/RNA Synthesis (57)
VEGFR (57)
Potassium Channel (54)
EGFR (44)
Sodium Channel (44)
PDGFR (43)
P450 (43)
Calcium Channel (42)
Glucocorticoid Receptor (41)
Estrogen/progestogen Receptor (41)
c-Kit (40)
FLT (39)
SARS-CoV (39)
PDE (37)
Ferroptosis (34)
CDK (33)
Antifungal (32)
PI3K (32)
Reactive Oxygen Species (31)
Dehydrogenase (31)
JAK (30)
FGFR (29)
RAAS (29)
Topoisomerase (29)
HCV Protease (28)
Src (27)
c-Met/HGFR (26)
NF-κB (26)
Mitophagy (26)
Reverse Transcriptase (26)
Influenza Virus (25)
PPAR (25)
Estrogen Receptor/ERR (23)
Serotonin Transporter (23)
GABA Receptor (23)
BTK (23)
Proteasome (23)
Bcr-Abl (22)
mTOR (22)
GPR (21)
HBV (21)
HDAC (21)
Androgen Receptor (20)
Microtubule Associated (20)
Prostaglandin Receptor (20)
TRP/TRPV Channel (19)
p38 MAPK (19)
PARP (18)
ribosome (18)
GluR (18)
ROS (18)
Adenosine Receptor (18)
Histone Methyltransferase (18)
Tyrosine Kinases (18)
Phosphatase (18)
Raf (18)
HSV (17)
Epigenetic Reader Domain (17)
Progesterone Receptor (17)
HIF/HIF Prolyl-Hydroxylase (17)
TNF (17)
Opioid Receptor (17)
Proton pump (17)
DPP-4 (16)
ALK (16)
MEK (16)
Nucleoside Antimetabolite/Analog (16)
AChE (16)
HER (15)
Norepinephrine (15)
Trk receptor (15)
iGluR (15)
Virus Protease (14)
S1P Receptor (14)
ERK (14)
SGLT (13)
MAPK (13)
P-gp (13)
TAM Receptor (13)
Beta Amyloid (13)
c-RET (13)
LPL Receptor (13)
Transferase (13)
Thrombin (12)
ROCK (12)
MRP (12)
STAT (12)
c-Fms (12)
MMP (11)
MAO (11)
DNA gyrase (11)
Retinoid Receptor (11)
Phospholipase (11)
AMPK (11)
Aurora Kinase (11)
Syk (10)
NADPH (10)
HSP (10)
Wnt/beta-catenin (10)
Integrin (10)
Interleukin (10)
Endothelin Receptor (10)
DNA Alkylator/Crosslinker (10)
ATPase (10)
Akt (10)
CSF-1R (9)
IL Receptor (9)
HMG-CoA Reductase (9)
E1/E2/E3 Enzyme (9)
PKC (9)
CCR (9)
Caspase (9)
Guanylate cyclase (9)
Lipoxygenase (9)
Antifection (9)
TLR (9)
Mitochondrial Metabolism (9)
Fatty Acid Synthase (9)
CXCR (9)
Ras (9)
Gamma-secretase (9)
Acyltransferase (9)
ROR (8)
BCL (8)
IGF-1R (8)
PLK (8)
Factor Xa (8)
GSK-3 (8)
Complement System (8)
Thyroid hormone receptor(THR) (8)
Monoamine Oxidase (8)
ATM/ATR (7)
ABC (7)
ROS Kinase (7)
CFTR (7)
Ligand for E3 Ligase (7)
Nrf2 (7)
NO Synthase (7)
LTR (7)
Antifolate (7)
DHFR (7)
NMDAR (7)
Neurokinin receptor (7)
Beta-Secretase (7)
Hydroxylase (7)
Carbonic Anhydrase (7)
Antiviral (7)
HIF (7)
GHSR (6)
Smo (6)
Antioxidant (6)
CaMK (6)
ASK (6)
OX Receptor (6)
Leukotriene Receptor (6)
Hedgehog/Smoothened (6)
DNA Alkylation (6)
FAK (6)
DNA Methyltransferase (6)
Reductase (6)
Glutathione Peroxidase (6)
Aminopeptidase (6)
TGF-beta/Smad (6)
RSV (6)
P2Y Receptor (6)
Stearoyl-CoA Desaturase (SCD) (5)
Serine/threonin kinase (5)
Melatonin Receptor (5)
Serine Protease (5)
IAP (5)
Lipase (5)
Sigma receptor (5)
PAK (5)
Ephrin Receptor (5)
FXR (5)
IκB/IKK (5)
Isocitrate Dehydrogenase (IDH) (5)
BACE (5)
Vasopressin Receptor (5)
Casein Kinase (5)
Indoleamine 2,3-Dioxygenase (IDO) (5)
Cannabinoid Receptor (5)
NADPH-oxidase (4)
Xanthine Oxidase (4)
P2X Receptor (4)
p53 (4)
PAI-1 (4)
PGE Synthase (4)
CaSR (4)
PKA (4)
Sirtuin (4)
Aromatase (4)
Pim (4)
Monoamine Transporter (4)
MT Receptor (4)
Cysteine Protease (4)
GNRH Receptor (4)
Histone Demethylase (4)
transporter (4)
DNA-PK (4)
IRAK (4)
DNA (4)
Mdm2 (4)
Aryl Hydrocarbon Receptor (4)
PERK (3)
Porcupine (3)
JNK (3)
AhR (3)
CRM1 (3)
Neprilysin (3)
Molecular Glues (3)
DUB (3)
IFNAR (3)
Histone Acetyltransferase (3)
TOPK (3)
FAAH (3)
FLAP (3)
UGT (3)
Free radical scavengers (3)
RIP kinase (3)
Glucosidase (3)
Glucokinase (3)
Glucagon Receptor (3)
PD-1/PD-L1 (3)
Drug Metabolite (3)
PAD (3)
Chk (3)
cholecystokinin (3)
Discoidin Domain Receptor (DDR) (3)
S6 Kinase (3)
Amino Acids and Derivatives (3)
Liver X Receptor (3)
Neuropeptide Y Receptor (3)
Annexin A (3)
NOD-like Receptor (NLR) (3)
Glutathione reductase (2)
Hck (2)
Protease-activated Receptor (2)
MNK (2)
SGK (2)
BMI-1 (2)
Hexokinase (2)
Tyrosinase (2)
Acetyl-CoA Carboxylase (2)
Rho (2)
GST (2)
Adenosine deaminase (2)
STING (2)
NOD (2)
Thrombopoietin Receptor (2)
Tie-2 (2)
Telomerase (2)
Integrase (2)
Imidazoline Receptor (2)
PDK (2)
CAT (2)
CETP (2)
LDL (2)
OXPHOS (2)
PI4K (2)
LRRK2 (2)
Lipid (2)
MALT (2)
IDO (2)
Platelet aggregation (2)
advanced glycation end products (2)
Ligands for Target Protein for PROTAC (2)
CGRP Receptor (2)
Somatostatin (1)
SIK (1)
ACK (1)
Angiotensin-converting Enzyme (ACE) (1)
Adiponectin receptor (1)
Taste receptor (1)
Anti-infection (1)
Survivin (1)
Gap Junction Protein (1)
ATP Citrate Lyase (1)
Hydrogenase (1)
MLK (1)
Decarboxylase (1)
Methionine Adenosyltransferase (MAT) (1)
LPA Receptor (1)
LHRH (1)
Kinesin (1)
IRE1 (1)
DYRK (1)
Myosin (1)
Epoxide Hydrolase (1)
Haspin Kinase (1)
GRK (1)
GPX (1)
GPCR19 (1)
GlyT (1)
Glutaminase (1)
GluCls (1)
Monocarboxylate transporter (1)
Na+/Ca2+ Exchanger (1)
BCRP (1)
PAFR (1)
Pyroptosis (1)
PYK2 (1)
Bradykinin Receptor (1)
PROTAC Linker (1)
Prolyl Endopeptidase (PREP) (1)
cAMP (1)
PKM (1)
Cell wall (1)
p97 (1)
Na-K-Cl cotransporter (1)
Chloride channel (1)
OAT (1)
c-Myc (1)
NPC1L1 (1)
CRISPR/Cas9 (1)
Neurotensin Receptor (1)
NEDD8 (1)
NAMPT (1)
NOS (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
陶术
生物
TargetMol®中国区唯一合作伙伴
点击进入陶术生物官网陶术生物
联系我们
400-820-0310

上海市静安区江场三路238号8楼