Cat. No. | Product Name | CAS No. | Purity | Chemical Structure |
---|---|---|---|---|
T0039 | Dapoxetine
达波西汀
|
119356-77-3 | 98% |
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Dapoxetine 是一种选择性5-羟色胺再摄取抑制剂,用于治疗早泄。 | ||||
T3086 | Mesoridazine Besylate
苯磺酸美索达嗪
|
32672-69-8 | 98% |
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Mesoridazine Besylate 是一种哌啶类精神安定药,属于称为吩噻嗪类的药物,用于治疗精神分裂症。它是硫利达嗪的代谢物。 | ||||
T62269 | F 14679
化合物F 14679
|
208109-38-0 | 98% |
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F 14679 是一种有效的5-HT1A 激动剂(pKi=10.23),具有 Ca2t 的最大反应与5-HT 相似。 | ||||
T28414 | Piclozotan
化合物Piclozotan
|
182415-09-4 | 98% |
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Piclozotan (anhydrous) 是一种 5-HT1A 受体激动剂,在短暂的大脑中动脉闭塞(t-MCAO)模型中表现出显着的神经保护活性,可以改善晚期帕金森病患者的运动并发症。 | ||||
T4348 | Syk Inhibitor II
化合物Syk Inhibitor II
|
726695-51-8 | 98% |
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Syk Inhibitor II 是一种可渗透细胞、具有 ATP 竞争性的嘧啶-甲酰胺化合物,可选择性且可逆地抑制 Syk,IC50为 41 nM。 | ||||
T8702 | SKF-83566
化合物SKF-83566
|
99295-33-7 | 98% |
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SKF-83566 是一种具有血脑渗透性和口服活性的 D1 样多巴胺受体拮抗剂和一种较弱的竞争性 5-HT2 受体拮抗剂,Ki 为 11 nM。它是竞争性多巴胺转运蛋白抑制剂,可用于研究帕金森氏症和对尼古丁渴望的缓解的相关研究。 | ||||
T1769 | Pardoprunox
帕多芦诺
|
269718-84-5 | 98% |
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Pardoprunox 是多巴胺受体D2、D3部分激动剂和5-HT1A 激动剂,pEC50分别为 8、9.2 和 6.3。 | ||||
TN1415 | Auraptenol
化合物Auraptenol
|
1221-43-8 | 98% |
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Auraptenol possesses robust antidepressant-like efficacy in mice. | ||||
T15100 | Desmethyl cariprazine
化合物 T15100
|
839712-15-1 | 98% |
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Desmethyl cariprazine is a Cariprazine active metabolite. Cariprazine, an antipsychotic drug candidate, shows a high affinity for the D3 (Ki: 0.085 nM) and D2 (K... | ||||
T17095 | TIK-301
化合物 T17095
|
118702-11-7 | 98% |
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TIK-301 is a chlorinated melatonin derivative and a potent, high-affinity, and orally active melatonin MT1 and MT2 receptors agonist (Kis: 0.081 nM and 0.042 nM,... | ||||
T11949 | Masupirdine mesylate
化合物 T11949
|
1791396-46-7 | 98% |
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Masupirdine mesylate (SUVN-502 mesylate) shows high selectivity over 5-HT2A receptor and other 100 target sites, and has potential for treatment of Alzheimer's d... | ||||
T19381 | Isobutyryl-L-carnitine
化合物 T19381
|
25518-49-4 | 98% |
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Isobutyryl-L-carnitine is a member of the class of compounds known as acylcarnitines. Isobutyryl-L-carnitine is a product of the acyl-CoA dehydrogenases. | ||||
T13339 | Wf-516
化合物 T13339
|
310392-94-0 | 98% |
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Wf-516 is a 5-HT reuptake inhibitor (Kis: 5 nM and 40 nM for 5-HT1A receptor and 5-HT2A receptor in humans, respectively), and with potent antidepressant activit... | ||||
TN4713 | Onitisin
化合物 TN4713
|
53823-03-3 | 98% |
|
Onitisin, onitinoside and onitin can inhibit the contraction of isolated guinea-pig ileum. | ||||
T10380 | AS19
化合物 T10380
|
1000578-26-6 | 98% |
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AS19 is a potent, selective 5-HT7 receptor agonist (IC50: 0.83 nM; Ki: 0.6 nM). AS19 is selective for 5-HT7 over 5-HT1A, 5-HT1B, 5-HT1D, and 5-HT5A receptors (Ki... | ||||
T15026 | Cyamemazine
化合物 T15026
|
3546-03-0 | 98% |
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Cyamemazine, contains the phenothiazine chromophore, is a neuroleptic agent used as an anxiolytic. Cyamemazine is a potent 5-HT3 (Ki: 12 nM), 5-HT2A (Ki: 1.5 nM)... | ||||
T13021 | Sulamserod
化合物 T13021
|
219757-90-1 | 98% |
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Sulamserod is an antagonist of 5-HT4 receptor, has antiarrhythmic activities. | ||||
T16433 | Pancopride
化合物 T16433
|
121650-80-4 | 98% |
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Pancopride is a new effective and selective antagonist of the 5-HT3 receptor. | ||||
T12262L | NPS ALX Compound 4a dihydrochloride
化合物 T12262L
|
1781934-44-8 | 98% |
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NPS ALX Compound 4a dihydrochloride is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM) | ||||
T10114 | 3-Hydroxy agomelatine
化合物 T10114
|
166526-99-4 | 98% |
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3-Hydroxy agomelatine is an Agomelatine metabolite and a 5-HT2C receptor antagonist (IC50: 3.2 μM; Ki: 1.8 μM). |