规格

价格

库存

数量

1 mg

¥ 541

现货

5 mg

¥ 1,250

现货

10 mg

¥ 1,830

现货

25 mg

¥ 2,890

现货

50 mg

¥ 3,980

现货

100 mg

¥ 5,370

现货

200 mg

¥ 6,900

现货

1 mL x 10 mM (in DMSO)

¥ 1,430

现货

生物活性

产品描述	CP 96021 is a group of 5-HT1 receptors and 5-HT2 receptors antagonists that have anti-inflammatory properties and are non-non-self anti-ulcer compounds for the treatment of gastrointestinal tract and respiratory asthma.
靶点活性	LTD4:0.46mg/kg（ED50）, PAF:0.16 mg/kg(ED50)
体内活性	CP-96021 inhibits iv LTD4- and iv PAF-induced bronchoconstriction in guinea pigs with ED50s of 0.46 and 0.16 mg/kg p.o. respectively. CP-96021 effectively blocks the combined airway obstructive effects of endogenously released PAF and LTD4 stimulated by aerosolized antigen challenge in guinea pigs with an ED50s of 1.8 mg/kg p.o[1]

化学信息

分子量	492.57
分子式	C₂₉H₂₁FN₄OS
CAS No.	139401-43-7
Smiles	CC=1N(C=2C(N1)=CN=CC2)C3=CC=C(OCC4=CC(/C=C/C5=NC=6C(S5)=CC=C(F)C6)=CC=C4)C=C3
密度	1.31 g/cm3 (Predicted)