首页 工具
登录
购物车
Adrenergic Receptor

Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.
1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16
Cat. No. Product Name CAS No. Purity Chemical Structure
TCS2185 Yohimbine
育亨宾
146-48-5
Yohimbine 是一种有效的、相对非选择性的α2 - 肾上腺素能受体拮抗剂,IC50=0.6μM。
T1769 Pardoprunox
帕多芦诺
269718-84-5
Pardoprunox (SLV-308) 是多巴胺受体D2、D3部分激动剂和5-HT1A 激动剂,pEC50分别为 8、9.2 和 6.3。
TN4882 Quinine HCl
化合物 TN4882
130-89-2 98%
Quinine HCl produces alpha-adrenergic blockade. Quinine modifies catecholamine- and calcium-induced myocardial contractile force responses.
T5450 DL-071-IT
化合物DL-071-IT
55104-39-7 98%
DL-071-IT (Afurolol Hydrochloride) 是一种有效的非选择性β-肾上腺素受体拮抗剂。 DL-071-IT 表现出内在的拟交感神经活性和弱的膜稳定活性。
T13470 (±)-Levomepromazine-d6
化合物 T13470
1189805-51-3 98%
(±)-Methotrimeprazine (D6) is the deuterium labeled Methotrimeprazine, which is an antagonist of D3 dopamine and Histamine H1 receptor.
T78567 Moprolol
化合物 Moprolol
5741-22-0 98%
Moprolol ((±)-Moprolol)为β-肾上腺素能受体阻滞剂,主要应用于原发性高血压研究。
T79641 (±)-N-Methylcoclaurine
化合物 (±)-N-Methylcoclaurine
1472-62-4 98%
(±)-N-Methylcoclaurine为选择性α2-肾上腺素受体拮抗剂。
T80175 Conopeptide rho-TIA
化合物 Conopeptide rho-TIA
381725-58-2 98%
Conopeptide rho-TIA为从掠食性海螺Conus tulipa毒液中提炼的多肽,对人类α1B-Adrenergic Receptor呈现非竞争性抑制作用,同时对α1A-Adrenergic Receptor和α1D-Adrenergic Receptor表现出竞争性抑制。Conopeptide rho-TI...
T80477 Muscarinic toxin 3
化合物 Muscarinic toxin 3
873336-87-9 98%
Muscarinic toxin 3 (MT3) 是高效的非竞争性mAChR及adrenoceptors拮抗剂,对M1、M4、α1A、α1B、α1D、α2A、α2B、α2C受体展示出不同程度的选择性,其pIC50值分别为6.71、8.79、8.86、7.57、8.13、8.49、6.5、7.29。该化合物具有显著的肾上腺...
TN1797 Isorhoifolin
异野漆树苷
552-57-8 98%
Isorhoifolin and vicenin II are main compounds of ethyl acetate fraction (EAcF) obtained from Erythrina velutina leaves, EAcF increases the cardiac contractile f...
T81798 Mibenratide TFA
化合物 Mibenratide TFA
98%
Mibenratide TFA,一种小环肽及肾上腺素能 β1 受体 (adrenergic β1 receptor) 拮抗剂,适用于心力衰竭研究。
T15042 D2343
化合物 T15042
72734-63-5 98%
D2343 is an agonist of β2-adrenoceptor. It also is an inhibitor of α1- adrenoceptor.
T6663 Scopine hydrochloride
盐酸东莨菪醇
85700-55-6 98%
Scopine hydrochloride (6,7-Epoxytropine hydrochloride) 是一种 Anisodine 的代谢物。
T16769 Ro 363
化合物 T16769
74513-77-2 98%
RO 363 is an effective inotropic stimulant and is a cardiovascular modulator that decreases diastolic blood pressure and pronounces increases in myocardial contr...
TN2267 Tetrahydroalstonine
四氢鸭脚木碱
6474-90-4 98%
Tetrahydroalstonine 是从 Rhazya stricta 的果实中提取出来的吲哚类生物碱,是一种具有选择性的 α2-肾上腺素受体拮抗剂。Tetrahydroalstonine 在Rauwolfia tetraphylla 中表现出抗精神病活性。
TN3368 Akuammigine
化合物 TN3368
642-17-1 98%
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
T11786 KUL-7211 racemate
化合物 T11786
911196-40-2 98%
KUL 7211 is a selective β-adrenoceptor agonist. KUL 7211 racemate is the racemate of KUL 7211.
T12815 (S)-Terazosin
(S)-特拉唑嗪
109351-33-9 98%
(S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor with...
T13285 Vatinoxan hydrochloride
化合物 T13285
130466-38-5 98%
Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.
T6562 Latrepirdine dihydrochloride
化合物Latrepirdine
97657-92-6 98%
Latrepirdine dihydrochloride (Dimebolin dihydrochloride) 是一种具有口服活性和神经活性的多种药物靶点的拮抗剂,可刺激淀粉样前体蛋白分解代谢和 β-淀粉样蛋白分泌。
Yohimbine
TCS2185
Yohimbine 是一种有效的、相对非选择性的α2 - 肾上腺素能受体拮抗剂,IC50=0.6μM。
Pardoprunox
T1769
Pardoprunox (SLV-308) 是多巴胺受体D2、D3部分激动剂和5-HT1A 激动剂,pEC50分别为 8、9.2 和 6.3。
Quinine HCl
TN4882
Quinine HCl produces alpha-adrenergic blockade. Quinine modifies catecholamine- and calcium-induced myocardial contractile force responses.
DL-071-IT
T5450
DL-071-IT (Afurolol Hydrochloride) 是一种有效的非选择性β-肾上腺素受体拮抗剂。 DL-071-IT 表现出内在的拟交感神经活性和弱的膜稳定活性。
(±)-Levomepromazine-d6
T13470
(±)-Methotrimeprazine (D6) is the deuterium labeled Methotrimeprazine, which is an antagonist of D3 dopamine and Histamine H1 receptor.
Moprolol
T78567
Moprolol ((±)-Moprolol)为β-肾上腺素能受体阻滞剂,主要应用于原发性高血压研究。
(±)-N-Methylcoclaurine
T79641
(±)-N-Methylcoclaurine为选择性α2-肾上腺素受体拮抗剂。
Conopeptide rho-TIA
T80175
Conopeptide rho-TIA为从掠食性海螺Conus tulipa毒液中提炼的多肽,对人类α1B-Adrenergic Receptor呈现非竞争性抑制作用,同时对α1A-Adrenergic Receptor和α1D-Adrenergic Receptor表现出竞争性抑制。Conopeptide rho-TI...
Muscarinic toxin 3
T80477
Muscarinic toxin 3 (MT3) 是高效的非竞争性mAChR及adrenoceptors拮抗剂,对M1、M4、α1A、α1B、α1D、α2A、α2B、α2C受体展示出不同程度的选择性,其pIC50值分别为6.71、8.79、8.86、7.57、8.13、8.49、6.5、7.29。该化合物具有显著的肾上腺...
Isorhoifolin
TN1797
Isorhoifolin and vicenin II are main compounds of ethyl acetate fraction (EAcF) obtained from Erythrina velutina leaves, EAcF increases the cardiac contractile f...
Mibenratide TFA
T81798
Mibenratide TFA,一种小环肽及肾上腺素能 β1 受体 (adrenergic β1 receptor) 拮抗剂,适用于心力衰竭研究。
D2343
T15042
D2343 is an agonist of β2-adrenoceptor. It also is an inhibitor of α1- adrenoceptor.
Scopine hydrochloride
T6663
Scopine hydrochloride (6,7-Epoxytropine hydrochloride) 是一种 Anisodine 的代谢物。
Ro 363
T16769
RO 363 is an effective inotropic stimulant and is a cardiovascular modulator that decreases diastolic blood pressure and pronounces increases in myocardial contr...
Tetrahydroalstonine
TN2267
Tetrahydroalstonine 是从 Rhazya stricta 的果实中提取出来的吲哚类生物碱,是一种具有选择性的 α2-肾上腺素受体拮抗剂。Tetrahydroalstonine 在Rauwolfia tetraphylla 中表现出抗精神病活性。
Akuammigine
TN3368
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
KUL-7211 racemate
T11786
KUL 7211 is a selective β-adrenoceptor agonist. KUL 7211 racemate is the racemate of KUL 7211.
(S)-Terazosin
T12815
(S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor with...
Vatinoxan hydrochloride
T13285
Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.
Latrepirdine dihydrochloride
T6562
Latrepirdine dihydrochloride (Dimebolin dihydrochloride) 是一种具有口服活性和神经活性的多种药物靶点的拮抗剂,可刺激淀粉样前体蛋白分解代谢和 β-淀粉样蛋白分泌。
1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16
联系我们
400-820-0310

上海市静安区江场三路238号8楼