Cat. No. | Product Name | CAS No. | Purity | Chemical Structure |
---|---|---|---|---|
TN2144 | Resveratroloside
白藜芦醇-4'-O-葡萄糖苷
|
38963-95-0 |
|
|
Resveratroloside 是α-glucosidase 的竞争性抑制剂,可以对血糖水平进行调节,对心脏具有保护作用。 | ||||
TN4800 | Pisatin
化合物 TN4800
|
20186-22-5 | 98% |
|
Pisatin is an isoflavonoid phytoalexin synthesized by pea (Pisum sativum L.). | ||||
TN3294 | 8alpha-(2-Methylacryloyloxy)hirsutinolide 13-O-acetate
化合物 TN3294
|
67667-71-4 | 98% |
|
8alpha-(2-Methylacryloyloxy)hirsutinolide 13-O-acetate shows inhibitory activity toward CYP2A6 and MAO-A and MAO-B enzymes. | ||||
TQ0109 | Cephaeline dihydrochloride
盐酸吐根酚碱
|
5853-29-2 | 98% |
|
(-)-Cephaeline (dihydrochloride) is an enantiomer of Cephaeline. Cephaeline is a selective CYP2D6 inhibitor (IC50: 121 μM). | ||||
T10535 | BI 653048
化合物 T10535
|
1198784-72-3 | 98% |
|
BI 653048 is a selective and orally active agonist of nonsteroidal glucocorticoid (IC50: 55 nM). BI 653048 is also an HCV NS3 protease inhibitor. | ||||
TN4424 | Lecanoric acid
化合物 TN4424
|
480-56-8 | 98% |
|
Lecanoric acid shows antioxidant activity with an IC50 value of 79-95 ug/ml, it at 100 ug/ml conc. shows high growth stimulating activity in terms of increased d... | ||||
TN4277 | Isocupressic acid
化合物 TN4277
|
1909-91-7 | 98% |
|
Isocupressic acid induces abortion in pregnant cows when ingested primarily during the last trimester, it decrease affects the angiogenesis of the female reprodu... | ||||
TMA2106 | (-)-Sparteine
化合物 TMA2106
|
24915-04-6 | 98% |
|
Sparteine is a class 1a antiarrhythmic agent, a sodium channel blocker. The deficient debrisoquine hydroxylation of Sparteine is due to the absence of P-450IID1 ... | ||||
TN5278 | Zederone
化合物 TN5278
|
7727-79-9 | 98% |
|
Zederone has anti-bacterial activity,it inhibits gram-positive bacteria activity. Zederone induces hepatotoxicity implicated the induction of Cyps, which leads t... | ||||
TN3300 | 8alpha-Tigloyloxyhirsutinolide 13-O-acetate
化合物 TN3300
|
83182-58-5 | 98% |
|
8alpha-Tigloyloxyhirsutinolide 13-O-acetate shows inhibitory activity toward CYP2A6 and MAO-A and MAO-B enzymes. 8alpha-Tigloyloxyhirsutinolide 13-O-acetate has ... | ||||
TMA0164 | 15-Hydroxydehydroabietic acid
化合物 TMA0164
|
54113-95-0 | 98% |
|
15-Hydroxydehydroabietic acid exhibits a promising alpha-glucosidase inhibitory activity, it also shows significant antibacterial activities. | ||||
TN2147 | Retrorsine
倒千里光碱
|
480-54-6 | 98% |
|
Retrorsine 特异性地抑制肝细胞增殖,并在肝损伤后唤起小肝细胞样祖细胞。逆转录酶可用于肝细胞损伤的研究。 | ||||
T10891 | CRTH2-IN-1
化合物 T10891
|
926661-54-3 | 98% |
|
CRTH2-IN-1 is a selective prostaglandin D2 receptor DP2 (CRTH2) antagonist, a Ramatroban analog, with an IC50 of 6 nM in the human DP2 binding assay. | ||||
TN1378 | α-Viniferin
α-葡萄素
|
62218-13-7 | 98% |
|
α-Viniferin 属于一类有机化合物,也称为2-芳基苯并呋喃类黄酮,是前列腺素H2合成酶抑制剂。具有抗阿尔茨海默病、抗结核、抗肿瘤、抗炎、抗糖尿病等多种药理活性 | ||||
TN3080 | 5,6,7-Trimethoxycoumarin
化合物 TN3080
|
55085-47-7 | 98% |
|
5,6,7-Trimethoxycoumarin shows moderate inhibitory activity against Micrococcus luteus, it also displays an intermediate cytotoxic effects against brine shrimp l... | ||||
T6051 | Orteronel
化合物(S)-Orteronel
|
566939-85-3 | 98% |
|
(S)-Orteronel ((S)-Orteronel) 是人17,20-裂解酶 (17,20-lyase, CYP17) 选择性抑制剂(IC50:38 nM),CYP17对(S)-Orteronel 选择性比对 11-hydroxylase 及 CYP3A4 高 1000 多倍。 | ||||
T11964 | MCH-1 antagonist 1
化合物 T11964
|
1039825-68-7 | 98% |
|
MCH-1 antagonist 1 also inhibits CYP3A4 (IC50: 10μM).MCH-1 antagonist 1 is a potent melanin concentrating hormone (MCH-1) antagonist (Ki: 2.6 nM). | ||||
TQ0296 | N-Nornuciferine
N-去甲荷叶碱
|
4846-19-9 | 98% |
|
N-Nornuciferine, an aporphine alkaloid in lotus leaf, significantly inhibits CYP2D6 (IC50: 3.76 μM, Ki: 2.34 μM). | ||||
TN4928 | Rutacridone
化合物 TN4928
|
17948-33-3 | 98% |
|
Rutacridone has mutagenicity. | ||||
TN2687 | 2,3',4,6-Tetrahydroxybenzophenone
化合物 TN2687
|
26271-33-0 | 98% |
|
2,3',4,6-Tetrahydroxybenzophenone possesses significant antioxidant activity. |