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Factor VIIa

Factor VIIa(FVIIa)是一种在血液凝固过程中起关键作用的丝氨酸蛋白酶。它是由肝脏合成的Factor VII的活化形式,通过维生素K依赖的γ-羧化作用成熟。FVIIa在凝血级联反应中扮演着启动者的角色,主要通过与组织因子(TF)结合形成复合物,激活Factor X和Factor IX,进而启动外源性凝血途径。这一过程对于止血和血栓形成至关重要。FVIIa的活性受多种因素调节,包括抗凝蛋白如组织因子途径抑制物(TFPI)和抗凝血酶III。FVIIa在维持血液凝固平衡中起着精细的调节作用,和出血性疾病有关。

EMD-503982
T27257768370-75-8In house
EMD-503982 是潜在的因子Xa和因子VIIa抑制剂,具有潜在的抗癌抗肿瘤活性,可用于研究血栓栓塞性疾病和神经系统疾病。
  • ¥ 1980 TargetMol
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TargetMol | Inhibitor Hot
Cytochalasin D
T322922144-77-0
Cytochalasin D is an actin inhibitor, the removal of actin stress fibers is crucial for the chondrogenic differentiation. It may be an inhibitor of some fertilization processes such as sperm penetration or sperm head decondensation. Cytochalasin D inhibit
  • ¥ 2430
In stock
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PCI-27483
T3469871266-63-6In house
PCI-27483 是一种FVIIa/tissue factor 抑制剂,具有抗肿瘤的作用。
  • ¥ 823
In stock
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BMS-593214
T716411004551-40-9In house
BMS-593214 是一种选择性活性位点定向因子 VIIa 抑制剂,也是 VIIa 激活底物 FX 的非竞争性抑制剂,具有抗血栓形成和抗出血活性。BMS-593214 可用于研究电诱导颈动脉血栓形成 (AT)和线诱导腔静脉血栓形成 (VT)。
  • ¥ 2170
In stock
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ARC19499
T751521350667-54-7
ARC19499 是一种核酸适配体, 与组织因子通路抑制剂(TFPI)特异性结合,阻断 TFPI 对factor Xa 和 TF factor VIIa 复合物的抑制作用。ARC19499 纠正血友病A 和B 血浆中的凝血酶生成,并恢复凝血。
  • 待询
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