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PGK1

PGK1(Phosphoglycerate kinase 1)是糖酵解过程中产生ATP的第一个关键代谢酶,参与肿瘤的糖酵解途径,能够影响肿瘤生长、迁移、侵袭、基因表达、能量代谢、分子调控,因此与多种疾病相关,如癌症、神经退行性疾病和心血管疾病。

CBR-470-1
T400632416095-06-0
CBR-470-1 是一种有效的糖酵解磷酸甘油酸激酶1 (PGK1) 抑制剂,通过增加甲基乙二醛的水平来激活 NRF2。 CBR-470-1 是一种非共价的 Nrf2 激活剂,具有神经保护活性,通过激活 Keap1-Nrf2 级联反应来保护 SH-SY5Y 神经元细胞免受 MPP+ 诱导的细胞毒性。
  • ¥ 239
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Acriflavine Hydrochloride
T198328063-24-9
Acriflavine Hydrochloride (Acriflavine HCl) 是一种 HIF-1α 抑制剂。它通过靶向 HIF-1α 介导的途径并在体外和体内降低 PGK1、VEGF 和 HIF-1α 的水平发挥作用。
  • ¥ 289
In stock
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Z57346765
T876591016340-64-9
Z57346765是一种特异性的PGK1(Phosphoglycerate kinase 1)抑制剂,通过降低糖酵解过程中PGK1的代谢酶活性,抑制PGK1依赖的细胞增殖。临床期中,Z57346765对局部晚期肾透明细胞癌(KIRC)具有剂量依赖的抑制作用,通过诱导与细胞代谢、DNA复制以及细胞周期相关的基因表达发生变化。
  • ¥ 447
In stock
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