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Sulfotransferase

Sulfotransferase(SULT)是一类催化硫酸基(SO₃)从磷酸腺苷磷硫酸(PAPS)转移到小分子羟基或氨基上的酶,广泛参与激素、胆酸、神经递质、药物和外源化合物的代谢与解毒。人类 SULT 家族包含多个亚型(如 SULT1、SULT2 等),在肝、肠、脑等组织呈差异表达;SULT 的底物特异性、多态性与表达调控直接影响药物代谢、激素稳态及某些疾病易感性。

Chst15-IN-1
Chst15-IN-1
T396312158198-77-5
Chst15-IN-1 是一种选择性、可逆且共价的 Chst15 酶抑制剂,能够抑制硫酸软骨素E(CS-E)及相关硫转移酶的硫酸化过程,从而减弱硫酸软骨素蛋白聚糖(CSPGs)的抑制效应,被认为具有促进神经修复的潜力。
  • ¥ 329
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