isomer

(Z)-JIB-04 (NSC 693627) 是 JIB-04 的 Z 型异构体。其中 JIB-04 有 E 型和 Z 型异构体两种形式。而(Z)-JIB-04 (NSC 693627) 在表观遗传分析中无活性。

W-9 hydrochloride 是一种钙调蛋白拮抗剂。

Azulene (Bicyclo[5.3.0]Decapentaene) 是萘的异构体，具有高抗HIV 活性。它是从洋甘菊精油中分离出来的一种化学支架。

5-O-Cinnamoylquinic acid 是一种天然产物。

Allocholic acid 是一种胆汁酸，在脊椎动物中发现，在肝脏再生和致癌过程中会重新出现，也是成熟嗅觉系统的特定性刺激物。

INCB3344 is a potent CCR2 antagonist. INCB3344 R-isomer is the R-isomer of INCB3344.

Eltanexor Z-isomer exhibits different inhibitory effects on Z138, MM15, 3T3 cell lines, with IC50s of 100 nM-50 μM, < 100 nM, > 30 μM, respectively.Eltanexor Z-isomer is the less active isomer of KPT-8602. KPT-8602 is a potent CRM1 inhibitor.

LY-411575 isomer 1 is a potent γ-secretase inhibitor. LY-411575 isomer 1 is an isomer of LY411575.

LY-411575 isomer 2 是 LY411575 的异构体。其中 LY411575 是一种高效的 γ-secretase 抑制剂。

LY-411575 isomer 3 是 LY411575 的异构体。其中 LY411575 是一种高效的 γ-secretase 抑制剂。

Longilactone, delta-4(18)-Isomer, 2alpha-alcoho 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T125797，CAS号为 149155-28-2。

Talabostat isomer mesylate, an isomer of talabostat mesylate, is a potent, nonselective, and orally available inhibitor of dipeptidyl peptidase IV (DPP-IV) with a Ki of 0.18 nM. Talabostat (PT100, Val-boroPro) is notable for its efficacy in inhibiting DPP-IV.

TTA-Q6(isomer) is an isomer of TTA-Q6. TTA-Q6 is a selective antagonist of the T-type Ca2+ channel.

NVP-BHG712 isomer 是一种 NVP-BHG712 的位置异构体，能够与EPHA2和EPHB4显示保守非键结合。

T3-ATA S-isomer, the S-isomer of T3-ATA, represents the active form of the thyroid hormone.

T4-ATA S-isomer, the active form of the thyroid hormone, represents the S-isomer of T4-ATA.

AB-FUBINACA 3-fluorobenzyl isomer 为一种具备高亲和力的吲唑类合成大麻素，主要影响中枢神经系统内的CB1受体（Ki= 0.9 nM)，并展现出抗惊厥活性。

Edoxaban Isomer is an impurity of Edoxaban, which is a novel inhibitor of factor Xa.

BAY-598 R-异构体是BAY589的R-异构体，它可用作参考化合物。它是是赖氨酸N-甲基转移酶（SMYD2）的抑制剂，对SMYD2比蛋白酶激活的受体1（PAR1）具有选择性。

Trichostatin A S-isomer is the s-isomer of Trichostatin A. Trichostatin A is a histone deacetylase inhibitors (HDIs or HDACIs) that have a broad spectrum of epigenetic activities. Trichostatin A inhibits HDACs 1, 3, 4, 6 and 10 with IC50 values around 20

TSR011-isomer, a TrKA ALK inhibitor, is used potentially for the treatment of solid tumours and lymphoma.

AZD6482 (S-isomer) is a potent, selective, ATP-competitive PI3Kβ inhibitor (IC(50) 0.01 μm), which can inhibit insulin-induced in vitro glucose uptake by human adipocytes (IC(50) is 4.4 μm).

Midodrine is a vasopressor antihypertensive agent for the treatment of symptomatic postural hypotension.

Endoxifen E-isomer hydrochloride (E-Endoxifen hydrochloride) 是 Endoxifen 的 E-异构体，是 Endoxifen Z-isomer 原料中主要的杂质，具有抗雌激素作用。