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AChR

AChR

An acetylcholine receptor (abbreviated AChR) is an integral membrane protein that responds to the binding of acetylcholine, a neurotransmitter.
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Cat. No. Product Name CAS No. Purity Chemical Structure
TN2217 Sophoflavescenol
槐苦参醇
216450-65-6 99.65%
Sophoflavescenol 是异戊烯基黄酮类化合物,能够抑制PDE5的活性,IC50=0.013 μM。它也抑制 RLAR,HRAR,BACE1,AChE 和 BChE,IC50值分别为 0.30 µM,0.17 µM,10.98 µM,8.37 µM 和 8.21 µM。
TN1798 Isorosmanol
异迷迭香酚
93780-80-4 98.85%
Isorosmanol 具有抗氧化、神经保护和神经营养作用,可能用于老年性疾病,如认知功能下降和色素沉着。
T0346 Camylofine
卡米罗芬
54-30-8 98%
Camylofine (Avacan) 是抗胆碱剂,也是一种平滑肌松弛剂。
TN1519 (S)-Coclaurine
化合物Coclaurine
486-39-5 97.72%
(S)-Coclaurine (Coclaurine) 是一种从 Sarcopetalum harveyanum 中分离出来的,是一种 nAChR 拮抗剂。
T8702 SKF-83566
化合物SKF-83566
99295-33-7 95.00%
SKF-83566 是一种具有血脑渗透性和口服活性的 D1 样多巴胺受体拮抗剂和一种较弱的竞争性 5-HT2 受体拮抗剂,Ki 为 11 nM。它是竞争性多巴胺转运蛋白抑制剂,可用于研究帕金森氏症和对尼古丁渴望的缓解的相关研究。
T68019 Ursulcholic acid
熊硫胆酸
88426-32-8 100%
Ursulcholic acid (Ursulcholic) 是一种可溶于水的抗胆碱能化合物。
T1236 Pentolinium Tartrate
酒石酸喷托铵
52-62-0
Pentolinium Tartrate (Pendine) 是烟碱拮抗剂,已被用作高血压的神经节阻滞剂。
T0218 Biperiden
比哌立登
514-65-8
Biperiden (Bipariden) 是中枢 M1胆碱受体阻断剂,有抗帕金森症活性。
T13129 Terodiline hydrochloride
盐酸特罗地林
7082-21-5 98%
Terodiline hydrochloride is an antagonist of M1-selective muscarinic receptor (mAChR)(Kbs of 15, 160, 280, and 198 nM in rabbit vas deferens (M1), atria (M2), bl...
T6721 Vinblastine
长春质碱
865-21-4 98%
Vinblastine 抑制微管形成并抑制 nAChR 活性,IC50 为 8.9 μM,用于治疗某些类型的癌症。
TN4837 Pseudotaraxasterol
化合物 TN4837
464-98-2 98%
Pseudotaraxasterol shows cytotoxic activity against MOLT-4 cells.
TN3696 Conodurine
化合物 TN3696
2665-57-8 98%
Conodurine shows leishmanicidal and antibacterial activities, it shows inhibition activity for acetyl (AChE) and butyrylcholinesterase (BuChE).
TN1559 Dehydrodicentrine
去氢荷包牡丹碱
19843-03-9 98%
Dehydrodicentrine showed strong acetylcholinesterase (AChE) inhibitory effects with the IC50 value of 2.98 μM.
T12020 Metixene hydrochloride
盐酸麦塞散
1553-34-0 98%
Metixene hydrochloride is an anticholinergic antiparkinsonian agent.
TN1645 Flavokawain C
2',4-二羟基-4',6'-二甲氧基查耳酮
56798-34-6 98%
Flavokawain C is a melanogenesis inhibitor, it inhibited melanogenesis with IC50 values of 6.9 μM. Flavokawain C has anti-tumor activity, it inhibited cell cycle...
TN1653 Fustin
黄颜木素
20725-03-5 98%
Fustin 是植物漆树 (Rhus verniciflua Stokes) 的植物性黄烷醇成分。 Fustin 对 6-羟基多巴胺诱导的神经元细胞死亡具有保护作用。
TN3380 Alloisoimperatorin
化合物 TN3380
35214-83-6 98%
Alloisoimperatorin is a candidate of AChE inhibitors, it displays potent antioxidant effects against the DPPH radical and against renal epithelial cell injury by...
T13713 GP531
化合物 T13713
142344-87-4 98%
GP531 is a second-generation adenosine regulating agent. It is pharmacologically silent under basal conditions but increases localized endogenous adenosine durin...
TN2505 1,5-Diphenylpentan-1-one
化合物 TN2505
39686-51-6 98%
1,5-Diphenylpentan-1-one shows poor insecticidal and acetylcholinesterase inhibitory activities.
TN4652 Niazimicin
化合物 TN4652
147821-49-6 98%
Niazimicin are NF-B and PI3K inhibitors, which shows antimicrobial, hypotensive and spasmolytic activities. Niazimicin has potent antitumor promoting activity in...
Sophoflavescenol
TN2217
Sophoflavescenol 是异戊烯基黄酮类化合物,能够抑制PDE5的活性,IC50=0.013 μM。它也抑制 RLAR,HRAR,BACE1,AChE 和 BChE,IC50值分别为 0.30 µM,0.17 µM,10.98 µM,8.37 µM 和 8.21 µM。
Isorosmanol
TN1798
Isorosmanol 具有抗氧化、神经保护和神经营养作用,可能用于老年性疾病,如认知功能下降和色素沉着。
Camylofine
T0346
Camylofine (Avacan) 是抗胆碱剂,也是一种平滑肌松弛剂。
(S)-Coclaurine
TN1519
(S)-Coclaurine (Coclaurine) 是一种从 Sarcopetalum harveyanum 中分离出来的,是一种 nAChR 拮抗剂。
SKF-83566
T8702
SKF-83566 是一种具有血脑渗透性和口服活性的 D1 样多巴胺受体拮抗剂和一种较弱的竞争性 5-HT2 受体拮抗剂,Ki 为 11 nM。它是竞争性多巴胺转运蛋白抑制剂,可用于研究帕金森氏症和对尼古丁渴望的缓解的相关研究。
Ursulcholic acid
T68019
Ursulcholic acid (Ursulcholic) 是一种可溶于水的抗胆碱能化合物。
Pentolinium Tartrate
T1236
Pentolinium Tartrate (Pendine) 是烟碱拮抗剂,已被用作高血压的神经节阻滞剂。
Biperiden
T0218
Biperiden (Bipariden) 是中枢 M1胆碱受体阻断剂,有抗帕金森症活性。
Terodiline hydrochloride
T13129
Terodiline hydrochloride is an antagonist of M1-selective muscarinic receptor (mAChR)(Kbs of 15, 160, 280, and 198 nM in rabbit vas deferens (M1), atria (M2), bl...
Vinblastine
T6721
Vinblastine 抑制微管形成并抑制 nAChR 活性,IC50 为 8.9 μM,用于治疗某些类型的癌症。
Pseudotaraxasterol
TN4837
Pseudotaraxasterol shows cytotoxic activity against MOLT-4 cells.
Conodurine
TN3696
Conodurine shows leishmanicidal and antibacterial activities, it shows inhibition activity for acetyl (AChE) and butyrylcholinesterase (BuChE).
Dehydrodicentrine
TN1559
Dehydrodicentrine showed strong acetylcholinesterase (AChE) inhibitory effects with the IC50 value of 2.98 μM.
Metixene hydrochloride
T12020
Metixene hydrochloride is an anticholinergic antiparkinsonian agent.
Flavokawain C
TN1645
Flavokawain C is a melanogenesis inhibitor, it inhibited melanogenesis with IC50 values of 6.9 μM. Flavokawain C has anti-tumor activity, it inhibited cell cycle...
Fustin
TN1653
Fustin 是植物漆树 (Rhus verniciflua Stokes) 的植物性黄烷醇成分。 Fustin 对 6-羟基多巴胺诱导的神经元细胞死亡具有保护作用。
Alloisoimperatorin
TN3380
Alloisoimperatorin is a candidate of AChE inhibitors, it displays potent antioxidant effects against the DPPH radical and against renal epithelial cell injury by...
GP531
T13713
GP531 is a second-generation adenosine regulating agent. It is pharmacologically silent under basal conditions but increases localized endogenous adenosine durin...
1,5-Diphenylpentan-1-one
TN2505
1,5-Diphenylpentan-1-one shows poor insecticidal and acetylcholinesterase inhibitory activities.
Niazimicin
TN4652
Niazimicin are NF-B and PI3K inhibitors, which shows antimicrobial, hypotensive and spasmolytic activities. Niazimicin has potent antitumor promoting activity in...
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