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335

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T12829 Salmeterol

沙美特罗,GR33343X

Adrenergic Receptor GPCR/G Protein; Neuroscience
Salmeterol (GR33343X) 是一种选择性的人β2肾上腺素受体激动剂。它能够有效刺激 cAMP 积累,作用于 CHO 细胞,对人β2,β1和β3肾上腺素受体的 pEC50分别为 9.6、6.1 和 5.9。
T9098 DMG-PEG 2000

DMG-PEG2000

Others Others
DMG-PEG 2000 (DMG-PEG2000) 可用于脂质纳米颗粒制备,用于口服质粒 DNA 的体内传递途径,提高纳米颗粒的黏液渗透性和传递效率。它也可用于 siRNA 转染的脂质体的制备,能够提高转染效率。
T26889 Borofalan(10B)

L-4-Boronophenylalanine,4-10硼酸-L-苯丙氨酸

Others Others
Borofalan(10B) (L-4-Boronophenylalanine) 具有抗肿瘤作用,可用于研究复发性或局部晚期头颈癌。
T8799 (E/Z)-IT-603

IT603

Others; NF-κB NF-κB; Others
(E/Z)-IT-603 是一种c-Rel 抑制剂,其IC50=3 μM。它是 E-IT-603 和 Z-IT-603的混合物。它具有抗癌作用。它有望作为调节剂调节移植物抗宿主病和恶性病中的 T 细胞反应。
T19692 Deferitrin

GT 56252,GT 56 252,地夫立群,GT-56252,GT-56-252

Others Others
Deferitrin (GT-56-252) 是一种具有口服活性的三叉戟铁螯合剂,是去铁硫素 (DFT) 类似物。它有用于严重的 β 地中海贫血的潜力。它用于输血引起的慢性铁超负荷。
T6653 Salmeterol Xinafoate

Salmetedur,昔美酸沙美特罗,沙美特罗昔萘酸酯,GR 33343X xinafoate,Arial

HIV Protease; Adrenergic Receptor GPCR/G Protein; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Salmeterol Xinafoate (GR 33343X xinafoate) 是选择性人β2肾上腺素受体激动剂。Salmeterol 有效刺激 cAMP 积累,能够作用于 CHO 细胞,对人β2,β1和β3肾上腺素受体的 pEC50分别为 9.6、6.1 和 5.9。
T7532 Piperaquine

Parasite Microbiology/Virology
Piperaquine 是一种双喹啉化合物,可抑制来自疟疾​​感染患者的恶性疟原虫分离株的离体生长,IC50 范围为 11.8-217.3 nM。
T5002 Methyl Aminolevulinate Hydrochloride

5-Aminolevulinic acid methyl ester,Methyl δ-aminolevulinate hydrochloride,5-氨基酮戊酸甲酯盐酸盐,Methyl 5-aminolevulinate Hydrochloride,Aminolevulinic acid methyl ester Hydrochloride

Others Others
Methyl Aminolevulinate Hydrochloride (5-Aminolevulinic acid methyl ester) 是增敏剂,可用于光动力疗法。Methyl aminolevulinate 是一种前药,可代谢为原卟啉 IX。
T1840 Isoindigotin

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Isoindigotin 用于治疗 Y.
T0383 Fenspiride hydrochloride

Fenspiride HCl,Pneumorel,Fluiden,Decaspiride,盐酸芬司必利

Adrenergic Receptor; PDE; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
Fenspiride hydrochloride (Decaspiride) 是一种口服活性的非甾体抗炎剂,是 H1-组胺受体的拮抗剂,可用于呼吸系统疾病的研究。
T3285L Eslicarbazepine

艾司利卡西平,Pazzul,EC 810-248-9,BIA 2-194,Stedesa,Erelib

Beta-Secretase; Sodium Channel Membrane transporter/Ion channel; Neuroscience
Eslicarbazepine (Stedesa) 是口服有效抗惊厥试剂,在局部癫痫的辅助研究中具有价值。
T3285 Eslicarbazepine Acetate

Zebinix,Aptiom,BIA 2-093,Exalief,艾司利卡西平醋酸酯,Stedesa

Beta-Secretase; Sodium Channel Membrane transporter/Ion channel; Neuroscience
Eslicarbazepine Acetate (Zebinix) 是一种抗癫痫药物。Eslicarbazepine acetate 也是 β-内分泌酶(β-Secretase)和电压门控钠离子通道的双抑制剂。
T21838 1-Naphthyl 3,5-dinitrobenzoate

JMC-4

Lipoxygenase Metabolism
1-Naphthyl 3,5-dinitrobenzoate (JMC-4) 是 5-LOX 的抑制剂,可用于炎症治疗的研究。
T1655 Ambrisentan

BSF-208075,BSF 208075,安倍生坦,LU 208075

Endothelin Receptor GPCR/G Protein
Ambrisentan (BSF 208075) 是 ET A 型受体选择性拮抗剂。
T20600 Kaolin

Clay 347,Hydrated aluminum silicate,Bolus alba,HSDB 630,Altowhite,China clay,高岭土

Others Others
Kaolin (Bolus alba) 是一种以高岭石族矿物为主的粘土。 Kaolin 提高了这种监测血友病治疗方法的敏感性。
T0718 Brivudine

Bromovinyldeoxyuridine,BVDU,溴夫定

Others; HSV Microbiology/Virology; Others
Brivudine (BVDU) 是胸苷类似物,有抗病毒活性,用于早期急性带状疱疹的研究。
T26126 Roxindole

Roxindole is an effective autoreceptor-selective dopamine agonist with additional properties as a serotonin reuptake inhibitor and 5-HT1A agonist. It was originally developed for the therapy of schizophrenic syndromes.
T73590 8-Phenyl-2,6-dibromo-1,3,5,7-tetramethyl BODIPY

8-Phenyl-2,6-dibromo-1,3,5,7-tetramethyl BODIPY 可用于光动力疗法。
T0454L Florfenicol

SCH-25298,氟苯尼考,(-)-Florfenicol

Antibacterial; Antibiotic Microbiology/Virology
Florfenicol (SCH-25298) 是一种常见得兽用抗生素,能用于研究牛呼吸疾病,在水产养殖业中可以用来控制鲶鱼肠道败血病,也可诱导鸡蛋早期胚胎死亡,LC50 值为 1.07 μg/g。
T0085L Entecavir

BMS200475,SQ34676,恩替卡韦

HBV Microbiology/Virology
Entecavir (SQ34676) 是一种选择性 HBV 抑制剂,在 HepG2细胞中的 EC50值为3.75 nM。
T6708 Tolcapone

Tasmar,Ro 40-7592,托卡朋

Apoptosis; Beta Amyloid; Transferase Apoptosis; Metabolism; Neuroscience
Tolcapone (Ro 40-7592) 是一种选择性,具有口服活性的外周和中枢COMT 抑制剂,在肝脏中对 COMT 的IC50为 773 nM。它还是一种 α-syn 和 Aβ42 寡聚和原纤维形成的有效抑制剂,可诱导氧化应激导致神经母细胞瘤细胞凋亡和抑制肿瘤生长。
T0078L Lapatinib ditosylate monohydrate

Lapatinib ditosylate monohydrate,Lapatinib ditoluenesulfonate monohydrate,Lapatinib tosilate hydrate,Lapatinib tosilate,Tykerb,二甲苯磺酸拉帕替尼单水合物,Tyverb

EGFR; Ferroptosis; Autophagy Angiogenesis; Apoptosis; Autophagy; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Lapatinib ditosylate (Lapatinib tosilate) monohydrate 是一种有效的 EGFR 和 ErbB2 抑制剂,对 EGFR 和 ErbB2的 IC50值分别为 10.8 和 9.2 nM。它用于治疗晚期乳腺癌和其他实体瘤。
T4296 MTX-211

MTX 211

EGFR; PI3K Angiogenesis; JAK/STAT signaling; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors
MTX-211 是EGFR 和PI3K 的双重抑制剂,可用于癌症和其他疾病研究。
T15501 HPPH

光克洛,Photochlor

Others Others
HPPH (Photochlor) 是第二代的光敏剂,可用于光动力疗法 (PDT)。
T9252 LY2880070

Chk Cell Cycle/Checkpoint
LY2880070 是一种用于癌症治疗的新型检查点激酶 1 (CHK1) 抑制剂。
T6875 Lesinurad

RDEA594,雷西那德,来司诺雷

OAT Membrane transporter/Ion channel
Lesinurad (RDEA594) 是URAT1和OAT 抑制剂。Lesinurad 用作肾转运蛋白OAT1 和OAT3 的底物,Km 分别为 0.85 和 2 μM。
T4472 NMS-P118

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
NMS-P118是可口服的高选择性PARP-1抑制剂,用于癌症治疗,在HeLa 细胞中的IC50值为0.04 μM。
T0317 Buflomedil hydrochloride

Buflomedil HCl,Fonzylane,Loftyl,盐酸丁咯地尔,丁咯地尔盐酸盐

Adrenergic Receptor GPCR/G Protein; Neuroscience
Buflomedil hydrochloride (Fonzylane) 是一种血管扩张剂,可用于外周动脉疾病引发的一系列症状。
T1461 Candesartan

CV 11974,坎地沙坦

RAAS Endocrinology/Hormones
Candesartan (CV 11974) 是一种血管紧张素II 受体拮抗剂(IC50:0.26 nM)。
T4344 ALW-II-41-27

Eph receptor tyrosine kinase inhibitor

Ephrin Receptor Tyrosine Kinase/Adaptors
ALW-II-41-27 (Eph receptor tyrosine kinase inhibitor) 是一种 Eph 受体酪氨酸激酶抑制剂,可用于治疗癌症。
T34616 Seridopidine

ACR-343,ACR 343,ACR343

Dopamine Receptor GPCR/G Protein; Neuroscience
Seridopidine (ACR343) 是一种多巴胺能活性调节剂,可作为精神分裂症、帕金森病和抽动秽语综合征的口服疗法。
T1103 Aminoglutethimide

DL-Aminoglutethimide,氨鲁米特,BA-16038,NSC-330915

Aromatase Endocrinology/Hormones
Aminoglutethimide (BA-16038) 是一种芳香酶抑制剂,IC50=10 μM,用于治疗晚期 BREAST Y。
T17035 Temoporfin

替莫卟吩,替莫泊芬

Others Others
Temoporfin 能够用于头颈部鳞状细胞癌的光动力学研究。
T2334 Avanafil

阿伐那非,TA1790

PDE Metabolism
Avanafil (TA1790) 是一种高活性PDE-5抑制剂,IC50=5.2 nM,对PDE1,PDE6和PDE11活性较低。
T0083 Eplerenone

Epoxymexrenone,CGP 30083,依普利酮,SC-66110

Glucocorticoid Receptor Endocrinology/Hormones
Eplerenone (CGP 30083) 是一种竞争性的、选择性的、具有口服活性的醛固酮 (aldosterone) 拮抗剂,IC50=138 nM。它对孕酮,雄激素,雌激素和糖皮质激素受体的亲和力低,可用于研究高血压和心肌梗死后的心力衰竭。
T0055 Glafenine

Glafenin,格拉非宁

COX Immunology/Inflammation; Neuroscience
Glafenine (Glafenin) 是一种可用于缓解疼痛研究的非甾体抗炎药。
T0045 Heptaminol hydrochloride

盐酸庚胺醇,RP-2831 hydrochloride

Others Others
Heptaminol hydrochloride (RP-2831 hydrochloride) 是一种血管收缩剂,有用于低血压(特别是体位性低血压)的研究潜力。
T6561 Laquinimod

LAQ,ABR-215062,拉喹莫德

Apoptosis; Others; NF-κB Apoptosis; NF-κB; Others
Laquinimod (LAQ) 是一种免疫调节剂,可预防中枢神经系统的神经变性和炎症。
T0703 Flavoxate hydrochloride

Flavoxate HCl,盐酸黄酮哌酯,NSC-114649,DW61,Rec-7-0040

AChR Neuroscience
Flavoxate hydrochloride (DW61) 是一种毒蕈碱受体 AChR 拮抗剂, IC50为 12.2 μM。
T5135 Flupentixol dihydrochloride

盐酸氟哌噻吨,Fupentixol Dihydrochloride,Flupenthixol dihydrochloride,(E/Z)-Flupentixol Dihydrochloride

Dopamine Receptor GPCR/G Protein; Neuroscience
Flupentixol dihydrochloride 是噻克西酮类试剂,能够用于研究精神分裂症以及抗焦虑和抑郁障碍。
T2317 Almotriptan Malate

LAS 31416,PNU180638,马来酸阿莫曲坦

5-HT Receptor GPCR/G Protein; Neuroscience
Almotriptan Malate (PNU180638) 是一种选择性 5-HT1B/1D 受体激动剂,用于治疗成人偏头痛发作。
T1476 Pramipexole

SND 919,普拉克索

Dopamine Receptor GPCR/G Protein; Neuroscience
Pramipexole (SND 919) 是能够透过血脑屏障的 D2 型多巴胺受体的选择性激动剂,对 D2 型受体、D2、D3、D4亚型受体的Ki 分别为 2.2 nM、3.9 nM、0.5 nM、1.3 nM。它可用于研究帕金森综合症和腿多动综合征。
T0189L Pemetrexed disodium

培美曲塞二钠盐,LY-231514,LY231514 disodium,培美曲塞二钠,Pemetrexed

Apoptosis; DHFR; DNA/RNA Synthesis; Antifolate; Autophagy Apoptosis; Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
Pemetrexed disodium (LY-231514) 是一种叶酸拮抗剂,用于治疗非小细胞肺癌和恶性间皮瘤。它抑制胸苷酸合成酶,二氢叶酸还原酶和甘氨酰胺核苷酸甲酰转移酶的Ki 分别为 1.3 nM,7.2 nM 和 65 nM。
T2561 Macitentan

马西替坦,ACT-064992

Apoptosis; Endothelin Receptor Apoptosis; GPCR/G Protein
Macitentan (ACT-064992) 是一种内皮素受体拮抗剂,用于治疗肺动脉高压。
T1159 Leflunomide

SU101,RS-34821,HWA486,来氟米特

Others; Dehydrogenase; AhR Immunology/Inflammation; Metabolism; Others
Leflunomide (HWA486) 是嘧啶合成抑制剂,能够抑制二氢乳清酸脱氢酶,具有抗风湿的活性。
T7105 Zinc phthalocyanine

酞菁锌,ZnPc

Others Others
Zinc phthalocyanine (ZnPc) 可用于环己烷的光氧化,广泛应用于工业 (催化剂、光导体)和生物医学(光动力疗法、PDT)。
T0026 Sulfalene

磺胺林,Sulfalene(SMPZ),Sulfalen,SMP2,Butadiene sulfone,AS-18908,Sulfametopyrazine,3-Sulfolene

Antibacterial; Antibiotic; Parasite; Autophagy Autophagy; Microbiology/Virology
Sulfalene (SMP2) 是一种长效磺胺类抗生素,用于治疗慢性支气管炎、尿路感染和疟疾。
T64695 IR-808

MHI-148

IR-808 (MHI-148) 是一种近红外菁染料,可用于无创癌症成像、诊断和成像引导光热治疗。
T0407 Edaravone

依达拉奉右莰醇,依达拉奉,MCI-186

Apoptosis; MMP; Free radical scavengers Apoptosis; oxidation-reduction; Proteases/Proteasome
Edaravone (MCI-186) 是一种新型自由基清除剂,能够抑制大鼠与 MMP-9有关的脑出血。
T6307 Lubiprostone

芦比前列酮,SPI-0211,RU-0211,鲁比前列酮

Chloride channel Membrane transporter/Ion channel
Lubiprostone (RU-0211) 是一种 ClC-2 氯化物通道的激活剂,用于治疗特发性慢性便秘。

化合物

Salmeterol
Cat.No: T12829
Synonym: 沙美特罗,GR33343X
Target: Adrenergic Receptor
DMG-PEG 2000
Cat.No: T9098
Synonym: DMG-PEG2000
Target: Others
Borofalan(10B)
Cat.No: T26889
Synonym: L-4-Boronophenylalanine,4-10硼酸-L-苯丙氨酸
Target: Others
(E/Z)-IT-603
Cat.No: T8799
Synonym: IT603
Target: Others, NF-κB
Deferitrin
Cat.No: T19692
Synonym: GT 56252,GT 56 252,地夫立群,GT-56252,GT-56-252
Target: Others
Salmeterol Xinafoate
Cat.No: T6653
Synonym: Salmetedur,昔美酸沙美特罗,沙美特罗昔萘酸酯,GR 33343X xinafoate,Arial
Target: HIV Protease, Adrenergic Receptor
Piperaquine
Cat.No: T7532
Synonym:
Target: Parasite
Methyl Aminolevulinate Hydrochloride
Cat.No: T5002
Synonym: 5-Aminolevulinic acid methyl ester,Methyl δ-aminolevulinate hydrochloride,5-氨基酮戊酸甲酯盐酸盐,Methyl 5-aminolevulinate Hydrochloride,Aminolevulinic acid methyl ester Hydrochloride
Target: Others
Isoindigotin
Cat.No: T1840
Synonym:
Target: DNA/RNA Synthesis
Fenspiride hydrochloride
Cat.No: T0383
Synonym: Fenspiride HCl,Pneumorel,Fluiden,Decaspiride,盐酸芬司必利
Target: Adrenergic Receptor, PDE, Histamine Receptor
Eslicarbazepine
Cat.No: T3285L
Synonym: 艾司利卡西平,Pazzul,EC 810-248-9,BIA 2-194,Stedesa,Erelib
Target: Beta-Secretase, Sodium Channel
Eslicarbazepine Acetate
Cat.No: T3285
Synonym: Zebinix,Aptiom,BIA 2-093,Exalief,艾司利卡西平醋酸酯,Stedesa
Target: Beta-Secretase, Sodium Channel
1-Naphthyl 3,5-dinitrobenzoate
Cat.No: T21838
Synonym: JMC-4
Target: Lipoxygenase
Ambrisentan
Cat.No: T1655
Synonym: BSF-208075,BSF 208075,安倍生坦,LU 208075
Target: Endothelin Receptor
Kaolin
Cat.No: T20600
Synonym: Clay 347,Hydrated aluminum silicate,Bolus alba,HSDB 630,Altowhite,China clay,高岭土
Target: Others
Brivudine
Cat.No: T0718
Synonym: Bromovinyldeoxyuridine,BVDU,溴夫定
Target: Others, HSV
Roxindole
Cat.No: T26126
Synonym:
Target:
8-Phenyl-2,6-dibromo-1,3,5,7-tetramethyl BODIPY
Cat.No: T73590
Synonym:
Target:
Florfenicol
Cat.No: T0454L
Synonym: SCH-25298,氟苯尼考,(-)-Florfenicol
Target: Antibacterial, Antibiotic
Entecavir
Cat.No: T0085L
Synonym: BMS200475,SQ34676,恩替卡韦
Target: HBV
Tolcapone
Cat.No: T6708
Synonym: Tasmar,Ro 40-7592,托卡朋
Target: Apoptosis, Beta Amyloid, Transferase
Lapatinib ditosylate monohydrate
Cat.No: T0078L
Synonym: Lapatinib ditosylate monohydrate,Lapatinib ditoluenesulfonate monohydrate,Lapatinib tosilate hydrate,Lapatinib tosilate,Tykerb,二甲苯磺酸拉帕替尼单水合物,Tyverb
Target: EGFR, Ferroptosis, Autophagy
MTX-211
Cat.No: T4296
Synonym: MTX 211
Target: EGFR, PI3K
HPPH
Cat.No: T15501
Synonym: 光克洛,Photochlor
Target: Others
LY2880070
Cat.No: T9252
Synonym:
Target: Chk
Lesinurad
Cat.No: T6875
Synonym: RDEA594,雷西那德,来司诺雷
Target: OAT
NMS-P118
Cat.No: T4472
Synonym:
Target: PARP
Buflomedil hydrochloride
Cat.No: T0317
Synonym: Buflomedil HCl,Fonzylane,Loftyl,盐酸丁咯地尔,丁咯地尔盐酸盐
Target: Adrenergic Receptor
Candesartan
Cat.No: T1461
Synonym: CV 11974,坎地沙坦
Target: RAAS
ALW-II-41-27
Cat.No: T4344
Synonym: Eph receptor tyrosine kinase inhibitor
Target: Ephrin Receptor
Seridopidine
Cat.No: T34616
Synonym: ACR-343,ACR 343,ACR343
Target: Dopamine Receptor
Aminoglutethimide
Cat.No: T1103
Synonym: DL-Aminoglutethimide,氨鲁米特,BA-16038,NSC-330915
Target: Aromatase
Temoporfin
Cat.No: T17035
Synonym: 替莫卟吩,替莫泊芬
Target: Others
Avanafil
Cat.No: T2334
Synonym: 阿伐那非,TA1790
Target: PDE
Eplerenone
Cat.No: T0083
Synonym: Epoxymexrenone,CGP 30083,依普利酮,SC-66110
Target: Glucocorticoid Receptor
Glafenine
Cat.No: T0055
Synonym: Glafenin,格拉非宁
Target: COX
Heptaminol hydrochloride
Cat.No: T0045
Synonym: 盐酸庚胺醇,RP-2831 hydrochloride
Target: Others
Laquinimod
Cat.No: T6561
Synonym: LAQ,ABR-215062,拉喹莫德
Target: Apoptosis, Others, NF-κB
Flavoxate hydrochloride
Cat.No: T0703
Synonym: Flavoxate HCl,盐酸黄酮哌酯,NSC-114649,DW61,Rec-7-0040
Target: AChR
Flupentixol dihydrochloride
Cat.No: T5135
Synonym: 盐酸氟哌噻吨,Fupentixol Dihydrochloride,Flupenthixol dihydrochloride,(E/Z)-Flupentixol Dihydrochloride
Target: Dopamine Receptor
Almotriptan Malate
Cat.No: T2317
Synonym: LAS 31416,PNU180638,马来酸阿莫曲坦
Target: 5-HT Receptor
Pramipexole
Cat.No: T1476
Synonym: SND 919,普拉克索
Target: Dopamine Receptor
Pemetrexed disodium
Cat.No: T0189L
Synonym: 培美曲塞二钠盐,LY-231514,LY231514 disodium,培美曲塞二钠,Pemetrexed
Target: Apoptosis, DHFR, DNA/RNA Synthesis, Antifolate, Autophagy
Macitentan
Cat.No: T2561
Synonym: 马西替坦,ACT-064992
Target: Apoptosis, Endothelin Receptor
Leflunomide
Cat.No: T1159
Synonym: SU101,RS-34821,HWA486,来氟米特
Target: Others, Dehydrogenase, AhR
Zinc phthalocyanine
Cat.No: T7105
Synonym: 酞菁锌,ZnPc
Target: Others
Sulfalene
Cat.No: T0026
Synonym: 磺胺林,Sulfalene(SMPZ),Sulfalen,SMP2,Butadiene sulfone,AS-18908,Sulfametopyrazine,3-Sulfolene
Target: Antibacterial, Antibiotic, Parasite, Autophagy
IR-808
Cat.No: T64695
Synonym: MHI-148
Target:
Edaravone
Cat.No: T0407
Synonym: 依达拉奉右莰醇,依达拉奉,MCI-186
Target: Apoptosis, MMP, Free radical scavengers
Lubiprostone
Cat.No: T6307
Synonym: 芦比前列酮,SPI-0211,RU-0211,鲁比前列酮
Target: Chloride channel
Cat. No. Product Name Target Signaling Pathways
T15242 Ercalcidiol

25-hydroxy Vitamin D2

Endogenous Metabolite Metabolism
Ercalcidiol 是维生素 D2 的代谢物,可用于监测维生素 D 治疗。
T0729 Benzyl benzoate

Ascabiol,Novoscabin,Scabitox,苯甲酸苄酯,Benzoic acid benzyl ester

Parasite Microbiology/Virology
Benzyl benzoate (Benzoic acid benzyl ester) 是化妆品中的香料成分,可研究疥疮和蠕形螨相关的炎症性皮肤病。
T2136 Geniposidic Acid

京尼平甙酸,京尼平苷酸

Apoptosis; Others; Endogenous Metabolite Apoptosis; Metabolism; Others
Geniposidic acid 是一种环烯醚萜苷,用于治疗黄疸、炎症和肝脏疾病,具有辐射保护和抗癌活性。
T0690 Quinine

奎宁树

Potassium Channel; Platelet aggregation; Parasite Membrane transporter/Ion channel; Microbiology/Virology; Others
Quinine 是一种从金鸡纳树皮中提取的生物碱,用于预防和治疗疟疾。它也用于特发性肌肉痉挛,可抑制电压脉冲引起的 MT mSlo3 (KCa5.1) 通道 +100 mV 电流, 其IC50值为 169 μM,是一种钾离子通道抑制剂。
T7106 Menaquinone-4

四烯甲萘醌,Vitamin K2,Menaquinone K4

Others; Endogenous Metabolite Metabolism; Others
Menaquinone-4 (Vitamin K2) 是维生素 K 的一种,用作止血剂,有潜力用于骨质疏松的研究。
T3130 Testosterone phenylpropionate

Testosterone hydrocinnamate,苯丙酸睾酮,Retandrol,Testosterone 17-phenylpropionate

Others Others
Testosterone phenylpropionate (Testosterone 17-phenylpropionate) 是一种长效雄激素。d3-Testosterone phenylpropionate 可用作内标物。
T0186 Docetaxel trihydrate

RP-56976 (Trihydrate),RP56976 (NSC 628503) Trihydrate,多西他赛三水合物

Apoptosis; BCL; Microtubule Associated Apoptosis; Cytoskeletal Signaling
Docetaxel trihydrate (RP-56976 Trihydrate) 是一种抗肿瘤试剂,抑制微管解聚的IC50值为 0.2 μM。它是紫杉醇的半合成类似物,能减弱 bcl-2 和 bcl-xL 基因表达的影响。它阻滞G2/M 细胞周期,导致细胞凋亡。
T6662 Scopine

东莨菪醇,6,7-Epoxytropine

Adrenergic Receptor GPCR/G Protein; Neuroscience
Scopine (6,7-Epoxytropine) 是一种山莨菪碱的代谢物,是一种 α1-肾上腺素受体激动剂,用于治疗急性循环性休克。
T2543 Cabazitaxel

XRP6258,卡巴他塞,RPR-116258A,TXD 258,taxoid XRP6258

Microtubule Associated; Autophagy Autophagy; Cytoskeletal Signaling
Cabazitaxel (taxoid XRP6258) 是一种紫杉烷类的抗肿瘤剂,可用于治疗多西他赛失败后的去势抵抗性转移性前列腺癌。
T3033 Deoxycorticosterone acetate

醋酸去氧皮质酮,DOC acetate,Cortexone acetate,11-Deoxycorticosterone acetate,醋酸脱氧皮质酮

Glucocorticoid Receptor; Endogenous Metabolite; Adrenergic Receptor Endocrinology/Hormones; GPCR/G Protein; Metabolism; Neuroscience
Deoxycorticosterone acetate (Cortexone acetate) 是肾上腺产生的类固醇激素,具有盐皮质激素活性,并作为醛固酮的前体。
TN3967 Epieriocalyxin A

ERK; BCL; ROS; Caspase; DNA/RNA Synthesis; JNK Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Immunology/Inflammation; MAPK; Proteases/Proteasome
Epieriocalyxin A 可以抑制 Caco-2 结肠癌细胞的生长。它可能是未来结肠癌治疗的潜在药物。
T2764 (S)-10-Hydroxycamptothecin

10-羟喜树碱,10-羟基喜树碱,10-Hydroxycamptothecin,10-HCPT

Apoptosis; Topoisomerase Apoptosis; DNA Damage/DNA Repair
(S)-10-Hydroxycamptothecin (10-HCPT) 是一种从喜树中分离的 DNA 拓扑异构酶 I 抑制剂。它显著诱导细胞凋亡,可研究肝癌、胃癌、结肠癌和白血病。
T4A2456 Gamabufotalin

Gamabufagin,日本蟾蜍毒苷元

COX Immunology/Inflammation; Neuroscience
Gamabufotalin (Gamabufagin) 是一种蟾蜍甾烯,存在于蟾酥中。它稳定性高,毒性低,被广泛用于癌症的研究。
T21651 Lansoprazole sodium

兰索拉唑钠,Lansoprazole (sodium), AG-1749 sodium

Proton pump; Phospholipase; Antibacterial Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
Lansoprazole sodium (Lansoprazole (sodium)) 是一种质子泵抑制剂,是中性鞘磷脂酶的外泌体抑制剂,能抑制胃酸生成。
T19237 Cholesteryl oleate

胆固醇油酸酯,Oleoylcholesterol,Cholesterol Oleate,Cholesteryl cis-9-octadecenoate

Endogenous Metabolite Metabolism
Cholesteryl oleate (Cholesteryl cis-9-octadecenoate) 是胆固醇的酯化形式,可用于合成固体脂质纳米颗粒。
T6395 Astragaloside A

Astragalin A,黄芪甲苷,Astramembrannin I

Calcium Channel Membrane transporter/Ion channel; Metabolism
Astragaloside A (Astramembrannin I) 是从黄芪中分离得到的初级纯皂苷,已广泛用于心血管疾病的治疗。
T6S1373 Casticin

Quercetagetin 3,6,7,4'-Tetramethyl Ether,Vitexicarpin,蔓荆子黄素

STAT JAK/STAT signaling; Stem Cells
Casticin (Vitexicarpin) 是从蔓荆子中得到的一种甲氧基黄酮,可抑制STAT3的活化,具有抗有丝分裂和抗炎活性。
TN6791 Palvanil

Hexadecanamide

TRP/TRPV Channel Membrane transporter/Ion channel
Palvanil (Hexadecanamide) 是一种快速脱敏的 TRPV1 激动剂。它可能是治疗 IBS 的有前途的药物,因为它可以调节肠道蠕动并减轻内脏疼痛。
T0392 Artemisinin

Qinghaosu,Artemisinine,Qinghaosu,NSC 369397,青蒿素,Artemisinine

HCV Protease; Ferroptosis; Akt; Parasite Apoptosis; Cytoskeletal Signaling; Microbiology/Virology; PI3K/Akt/mTOR signaling; Proteases/Proteasome
Artemisinin (Qinghaosu) 是一种倍半萜烯内酯,是从青蒿植物的地上部分分离的一种抗疟疾药物。它有神经保护和抗癌作用。
TN1877 Lonicerin

忍冬苦苷,金银花

Apoptosis; Antibacterial Apoptosis; Microbiology/Virology
Lonicerin 是一种抗藻酸盐分泌蛋白的黄酮类化合物,对铜绿假单胞菌有抑制作用。它可预防脂多糖诱导的急性肺损伤的炎症和细胞凋亡。
T2941 Glucosamine hydrochloride

Chitosamine hydrochloride,盐酸氨基葡萄糖,2-Amino-2-deoxy-glucose HCl,Chitosamine HCl,D-(+)-Glucosamine hydrochloride

Reactive Oxygen Species; HIF/HIF Prolyl-Hydroxylase; Endogenous Metabolite; Autophagy Autophagy; Chromatin/Epigenetic; Immunology/Inflammation; Metabolism; NF-κB
Glucosamine hydrochloride (Chitosamine hydrochloride) 是软骨基质和滑液中糖胺聚糖的天然成分,常用作骨关节炎的治疗方法。它也是一种氨基糖,是糖基化蛋白和脂质生化合成的突出前体,用作膳食补充剂。
T2S1720 Huperzine B

AChE Neuroscience
Huperzine B 是一种从 Huperzia serrata 中分离出的石蒜生物碱,也是一种高度选择性的乙酰胆碱酯酶抑制剂,可以用于改善阿尔茨海默氏病。
T3787 Didymin

Isosakuranetin-7-O-rutinoside,Neoponcirin,香风草甙

Apoptosis; Others Apoptosis; Others
Didymin (Neoponcirin) 从柑橘类水果中提取的一种膳食类黄酮苷,具有抗氧化特性。它通过抑制 N-Myc 和上调 RKIP 诱导凋亡。
TN1341 8-Deoxygartanin

8-脱氧藤黄苷

Beta Amyloid; NF-κB; Parasite Microbiology/Virology; Neuroscience; NF-κB
8-Deoxygartanin 是山竹果中的异戊烯化呫吨酮。它是丁基胆碱酯酶选择性抑制剂,对阿尔茨海默病 (AD) 具有多功能活性,可能是有希望治疗 AD 的化合物。
T3S0057 Dihydrochelerythrine

12,13-Dihydrochelerythrine,二氢白屈菜红碱

Antifungal Microbiology/Virology
Dihydrochelerythrine (12,13-Dihydrochelerythrine) 是一种从榕树叶片分离出的天然化合物,具有抗真菌活性,有潜力治疗多丝蚴引起的严重感染。
TN1996 Nothofagin

ERK; IL Receptor; TNF Apoptosis; Immunology/Inflammation; MAPK
Nothofagin 具有抗氧化和抗血栓活性,它通过抑制高渗透性、CAMs 的表达以及白细胞的粘附和迁移具有抗炎活性,从而支持其作为血管炎症性疾病的治疗作用。
T6194 Fidaxomicin

非达米星,Tiacumicin B,OPT-80,Clostomicin B1,PAR-101

Apoptosis; DNA/RNA Synthesis; Antibacterial; Antibiotic Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Fidaxomicin (Tiacumicin B) 是一种大环RNA 聚合酶抑制剂,具有窄谱活性。它选择性地根除致病性艰难梭菌,对构成正常健康肠道菌群的多种细菌影响很小。
T0256 Citric acid trilithium salt tetrahydrate

Lithium citrate tribasic tetrahydrate,柠檬酸三锂盐四水合物,Trilithium citrate tetrahydrate

Dehydrogenase; GSK-3; HIF/HIF Prolyl-Hydroxylase; Antibacterial; GluR Chromatin/Epigenetic; Metabolism; Microbiology/Virology; Neuroscience; PI3K/Akt/mTOR signaling; Stem Cells
Citric acid trilithium salt tetrahydrate (Lithium citrate tribasic tetrahydrate) 是一种用于治疗精神疾病的药物。它也是一种医药和建筑材料, 可用于氨基酸定量分析时的梯度洗脱。
TN1040 Skullcapflavone II

COX; Antibacterial; TGF-beta/Smad Immunology/Inflammation; Microbiology/Virology; Neuroscience; Stem Cells
Skullcapflavone II 是从黄芩中提取的黄酮,具有抗炎作用。它对 M. aurum 和 M. bovisBCG 具有较强的抗菌活性。它还调节破骨细胞的分化、存活和功能。
T5S1285 (+)-(3R,8S)-Falcarindiol

Falcarindiol,镰叶芹二醇

Others Others
(+)-(3R,8S)-Falcarindiol 是一种从胡萝卜中得到的聚乙炔,有抗炎、抗肿瘤和抗脂质过氧化活性。它具有抗分歧杆菌作用,对Mycobacterium tuberculosisH37Ra 的 MIC 和 IC50值分别为 24 μM 和 6 μM。
T1284 Megestrol acetate

SC10363,醋酸甲地孕酮,BDH1298

Glucocorticoid Receptor; Estrogen/progestogen Receptor; Progesterone Receptor; HIV Protease; Autophagy Autophagy; Endocrinology/Hormones; Microbiology/Virology; Others; Proteases/Proteasome
Megestrol acetate (BDH1298) 是具有口服活性的合成孕激素。它还具有抗雄激素特性,可用于治疗厌食症和恶病质。
T2967 Stigmasterol

Stigmasterin,beta-Stigmasterol,豆甾醇

MMP; Endogenous Metabolite Metabolism; Proteases/Proteasome
Stigmasterol (Stigmasterin) 是一种植物性甾醇,具有抑制胆固醇的特性,此外在风湿性疾病的研究中被评价为抗硬化因子。
T3752 4-Hydroxybenzyl alcohol

4-Methylolphenol,P-Methylolphenol,对羟基苯甲醇

Apoptosis; Endogenous Metabolite Apoptosis; Metabolism
4-Hydroxybenzyl alcohol (P-Methylolphenol) 是广泛分布于各种植物中的一种酚类天然产物,具有抗炎、抗氧化和抗伤害感受活性。它抑制肿瘤血管生成和生长,有神经保护作用。
TN6774 Emodin 6-O-β-D-glucoside

大黄素-6-O-β-D-葡萄糖苷,Glucoemodin

Others Others
Emodin 6-O-β-D-glucoside (Glucoemodin) 是一种从 Reynoutria japonica 中提取的活性化合物。它具有显著的抗炎和屏障保护活性,可用于研究动脉粥样硬化及糖尿病并发症。
T2787 Picroside I

6'-Cinnamoylcatalpol,胡黄连苦苷I

MMP; STAT JAK/STAT signaling; Proteases/Proteasome; Stem Cells
Picroside I (6'-Cinnamoylcatalpol) 是胡黄连的一种天然产物,是有肝脏保护作用的代谢成分,可用于哮喘研究,有减轻炎症作用,还下调 pSTAT6 和 GATA3 表达。
T2966 Beta-Sitosterol

Cupreol,谷甾醇,Beta-Sitosterol,β-Sitosterol,Azuprostat,SKF 14463,beta-谷甾醇,22,23-Dihydrostigmasterol,Betaprost

Apoptosis; Lipase; Endogenous Metabolite Apoptosis; Metabolism
Beta-Sitosterol (SKF 14463) 是一种植物甾醇,干扰细胞周期、细胞凋亡、增殖、存活、侵袭、血管生成和炎症等多种细胞信号通路。
T4S1422 Praeruptorin E

白花前胡素 E,白花前胡素E

Others; Calcium Channel Membrane transporter/Ion channel; Metabolism; Others
Praeruptorin E 是白花前胡中的一种主要成分,是钙拮抗剂,pD2′值为 5.2。
T6S0721 Orientin

荭草苷,Lutexin,Luteolin-8-glucoside

Others Others
Orientin (Luteolin-8-glucoside) 是天然存在的生物活性类黄酮,是一种有前景的神经保护剂,具有多种生物特性,如抗炎、抗肿瘤、抗氧化、保护心脏等。它有用于神经性疼痛研究潜力。
T4S2126 Ginkgetin

银杏双黄酮,银杏素

Apoptosis; Wnt/beta-catenin; COX; STAT; Autophagy Apoptosis; Autophagy; Cytoskeletal Signaling; Immunology/Inflammation; JAK/STAT signaling; Neuroscience; Stem Cells
Ginkgetin 是从银杏叶中分离得到的一种双黄酮,具有抗肿瘤、抗炎、神经保护、抗真菌的作用。它也是 Wnt 信号抑制剂,IC50值为 5.92 μM。
T2S1865 Octyl gallate

Gallic acid octyl ester,n-Octylgallate,Octyl 3,4,5-trihydroxybenzoate,Progallin O,Stabilizer GA-8,没食子酸辛酯

Antioxidant; Influenza Virus; Reactive Oxygen Species; Antibacterial; Antifungal; HSV Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; oxidation-reduction
Octyl gallate (Octyl 3,4,5-trihydroxybenzoate) 具有抗菌、抗氧化作用,有选择性和敏感性的荧光特性,广泛用作食品添加剂。它对 HSV-1,水泡性口炎病毒和脊髓灰质炎病毒有显著的抗病毒作用。
T2S2215 Crebanine

Apoptosis; Others; Akt Apoptosis; Cytoskeletal Signaling; Others; PI3K/Akt/mTOR signaling
Crebanine 是来自于韦诺萨千金藤的一种生物碱,通过抑制 MAPKs 和 Akt 信号通路表现出抗炎活性,还具有抗心律失常的作用。它可诱导人类癌细胞的 G1阻滞和凋亡。
T8053 N-Acetyl-L-arginine

N-Α-乙酰-L-精氨酸,Ac-Arg-OH

Endogenous Metabolite Metabolism
N-Acetyl-L-arginine (Ac-Arg-OH) 是一种胍基诺化合物,被发现存在于血液渗析性肾不足儿童患者血清中的。
T4S1551 Cinnamaldehyde

Cinnamic Aldehyde,肉桂醛

HIF Angiogenesis; Chromatin/Epigenetic
Cinnamaldehyde (Cinnamic Aldehyde) 具有解热作用。 它是镇静剂。它抑制MDA-MB-435S 细胞的侵袭能力与下调miR-27a 的表达有关。它诱导活性氧的产生,发挥血管扩张和抗癌作用。 它似乎是一种有希望的候选药物,可作为与 5-氟尿嘧啶 (5-FU) 和奥沙利铂 (OXA) 这两种用于 CRC 治疗的化疗药物联合治疗的辅助剂。其作用的可能机制可能涉及药物代谢基因的调节。 它在抑制黑色素瘤的发生和发展方面具有一定的作用,其作用机制可能表现为抑制VEGF 和HIF-α的表达,从而使血管模拟和黑色素瘤细胞新生血管的形成,促进肿瘤的生长。
T4S1057 Tripdiolide

IL Receptor; TNF Apoptosis; Immunology/Inflammation
Tripdiolide has cytotoxic, and anti-rheumatic activities, it suppresses pro-inflammatory gene expression, may be effective therapy for lupus nephritis.
TN5327 11(13)-Dehydroivaxillin

11(13)-Dehydroivaxillin possesses a promising antiplasmodial activity, which can be exploited in malaria therapy.
TN6646 Fargesol

(-)-Fargesol is a nartural product from the flowers buds of Magnolia fargesii,the dried flower buds of M. fargesii, has been used as therapy for nasal empyema and headache.
TN3327 9-O-Methyl-4-hydroxyboeravinone B

Others Others
9-O-Methyl-4-hydroxyboeravinone B is a promising candidate for cancer therapy.
T11895 Luteolin-7-rutinoside

Others Others
Luteolin-7-rutinoside has both antifungal activities and anti-arthritic, can result in a combination therapy for the treatment of fungal arthritis due to C. albicans infection.
T1033L Monensin

Elancoban,Rumensin,莫能菌素

Monensin is an antiprotozoal agent produced by Streptomyces cinnamonensis. It has an inhibitory effect on the Wnt/β-catenin signaling cascade. Monensin is a prospective anticancer drug for the therapy of neoplasia with deregulated Wnt signaling.
T73925 α-D-Glucose-1-phosphate disodium hydrate

α-D-Glucose-1-phosphate disodium hydrate 为合成葡萄糖醛酸的初始原料之一,同时,在心脏病研究领域,亦被广泛应用作为细胞抑制剂、抗生素、免疫抑制剂与循环系统研究的关键材料。
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天然产物

Ercalcidiol
Cat.No: T15242
Synonym: 25-hydroxy Vitamin D2
Target: Endogenous Metabolite
Benzyl benzoate
Cat.No: T0729
Synonym: Ascabiol,Novoscabin,Scabitox,苯甲酸苄酯,Benzoic acid benzyl ester
Target: Parasite
Geniposidic Acid
Cat.No: T2136
Synonym: 京尼平甙酸,京尼平苷酸
Target: Apoptosis, Others, Endogenous Metabolite
Quinine
Cat.No: T0690
Synonym: 奎宁树
Target: Potassium Channel, Platelet aggregation, Parasite
Menaquinone-4
Cat.No: T7106
Synonym: 四烯甲萘醌,Vitamin K2,Menaquinone K4
Target: Others, Endogenous Metabolite
Testosterone phenylpropionate
Cat.No: T3130
Synonym: Testosterone hydrocinnamate,苯丙酸睾酮,Retandrol,Testosterone 17-phenylpropionate
Target: Others
Docetaxel trihydrate
Cat.No: T0186
Synonym: RP-56976 (Trihydrate),RP56976 (NSC 628503) Trihydrate,多西他赛三水合物
Target: Apoptosis, BCL, Microtubule Associated
Scopine
Cat.No: T6662
Synonym: 东莨菪醇,6,7-Epoxytropine
Target: Adrenergic Receptor
Cabazitaxel
Cat.No: T2543
Synonym: XRP6258,卡巴他塞,RPR-116258A,TXD 258,taxoid XRP6258
Target: Microtubule Associated, Autophagy
Deoxycorticosterone acetate
Cat.No: T3033
Synonym: 醋酸去氧皮质酮,DOC acetate,Cortexone acetate,11-Deoxycorticosterone acetate,醋酸脱氧皮质酮
Target: Glucocorticoid Receptor, Endogenous Metabolite, Adrenergic Receptor
Epieriocalyxin A
Cat.No: TN3967
Synonym:
Target: ERK, BCL, ROS, Caspase, DNA/RNA Synthesis, JNK
(S)-10-Hydroxycamptothecin
Cat.No: T2764
Synonym: 10-羟喜树碱,10-羟基喜树碱,10-Hydroxycamptothecin,10-HCPT
Target: Apoptosis, Topoisomerase
Gamabufotalin
Cat.No: T4A2456
Synonym: Gamabufagin,日本蟾蜍毒苷元
Target: COX
Lansoprazole sodium
Cat.No: T21651
Synonym: 兰索拉唑钠,Lansoprazole (sodium), AG-1749 sodium
Target: Proton pump, Phospholipase, Antibacterial
Cholesteryl oleate
Cat.No: T19237
Synonym: 胆固醇油酸酯,Oleoylcholesterol,Cholesterol Oleate,Cholesteryl cis-9-octadecenoate
Target: Endogenous Metabolite
Astragaloside A
Cat.No: T6395
Synonym: Astragalin A,黄芪甲苷,Astramembrannin I
Target: Calcium Channel
Casticin
Cat.No: T6S1373
Synonym: Quercetagetin 3,6,7,4'-Tetramethyl Ether,Vitexicarpin,蔓荆子黄素
Target: STAT
Palvanil
Cat.No: TN6791
Synonym: Hexadecanamide
Target: TRP/TRPV Channel
Artemisinin
Cat.No: T0392
Synonym: Qinghaosu,Artemisinine,Qinghaosu,NSC 369397,青蒿素,Artemisinine
Target: HCV Protease, Ferroptosis, Akt, Parasite
Lonicerin
Cat.No: TN1877
Synonym: 忍冬苦苷,金银花
Target: Apoptosis, Antibacterial
Glucosamine hydrochloride
Cat.No: T2941
Synonym: Chitosamine hydrochloride,盐酸氨基葡萄糖,2-Amino-2-deoxy-glucose HCl,Chitosamine HCl,D-(+)-Glucosamine hydrochloride
Target: Reactive Oxygen Species, HIF/HIF Prolyl-Hydroxylase, Endogenous Metabolite, Autophagy
Huperzine B
Cat.No: T2S1720
Synonym:
Target: AChE
Didymin
Cat.No: T3787
Synonym: Isosakuranetin-7-O-rutinoside,Neoponcirin,香风草甙
Target: Apoptosis, Others
8-Deoxygartanin
Cat.No: TN1341
Synonym: 8-脱氧藤黄苷
Target: Beta Amyloid, NF-κB, Parasite
Dihydrochelerythrine
Cat.No: T3S0057
Synonym: 12,13-Dihydrochelerythrine,二氢白屈菜红碱
Target: Antifungal
Nothofagin
Cat.No: TN1996
Synonym:
Target: ERK, IL Receptor, TNF
Fidaxomicin
Cat.No: T6194
Synonym: 非达米星,Tiacumicin B,OPT-80,Clostomicin B1,PAR-101
Target: Apoptosis, DNA/RNA Synthesis, Antibacterial, Antibiotic
Citric acid trilithium salt tetrahydrate
Cat.No: T0256
Synonym: Lithium citrate tribasic tetrahydrate,柠檬酸三锂盐四水合物,Trilithium citrate tetrahydrate
Target: Dehydrogenase, GSK-3, HIF/HIF Prolyl-Hydroxylase, Antibacterial, GluR
Skullcapflavone II
Cat.No: TN1040
Synonym:
Target: COX, Antibacterial, TGF-beta/Smad
(+)-(3R,8S)-Falcarindiol
Cat.No: T5S1285
Synonym: Falcarindiol,镰叶芹二醇
Target: Others
Megestrol acetate
Cat.No: T1284
Synonym: SC10363,醋酸甲地孕酮,BDH1298
Target: Glucocorticoid Receptor, Estrogen/progestogen Receptor, Progesterone Receptor, HIV Protease, Autophagy
Stigmasterol
Cat.No: T2967
Synonym: Stigmasterin,beta-Stigmasterol,豆甾醇
Target: MMP, Endogenous Metabolite
4-Hydroxybenzyl alcohol
Cat.No: T3752
Synonym: 4-Methylolphenol,P-Methylolphenol,对羟基苯甲醇
Target: Apoptosis, Endogenous Metabolite
Emodin 6-O-β-D-glucoside
Cat.No: TN6774
Synonym: 大黄素-6-O-β-D-葡萄糖苷,Glucoemodin
Target: Others
Picroside I
Cat.No: T2787
Synonym: 6'-Cinnamoylcatalpol,胡黄连苦苷I
Target: MMP, STAT
Beta-Sitosterol
Cat.No: T2966
Synonym: Cupreol,谷甾醇,Beta-Sitosterol,β-Sitosterol,Azuprostat,SKF 14463,beta-谷甾醇,22,23-Dihydrostigmasterol,Betaprost
Target: Apoptosis, Lipase, Endogenous Metabolite
Praeruptorin E
Cat.No: T4S1422
Synonym: 白花前胡素 E,白花前胡素E
Target: Others, Calcium Channel
Orientin
Cat.No: T6S0721
Synonym: 荭草苷,Lutexin,Luteolin-8-glucoside
Target: Others
Ginkgetin
Cat.No: T4S2126
Synonym: 银杏双黄酮,银杏素
Target: Apoptosis, Wnt/beta-catenin, COX, STAT, Autophagy
Octyl gallate
Cat.No: T2S1865
Synonym: Gallic acid octyl ester,n-Octylgallate,Octyl 3,4,5-trihydroxybenzoate,Progallin O,Stabilizer GA-8,没食子酸辛酯
Target: Antioxidant, Influenza Virus, Reactive Oxygen Species, Antibacterial, Antifungal, HSV
Crebanine
Cat.No: T2S2215
Synonym:
Target: Apoptosis, Others, Akt
N-Acetyl-L-arginine
Cat.No: T8053
Synonym: N-Α-乙酰-L-精氨酸,Ac-Arg-OH
Target: Endogenous Metabolite
Cinnamaldehyde
Cat.No: T4S1551
Synonym: Cinnamic Aldehyde,肉桂醛
Target: HIF
Tripdiolide
Cat.No: T4S1057
Synonym:
Target: IL Receptor, TNF
11(13)-Dehydroivaxillin
Cat.No: TN5327
Synonym:
Target:
Fargesol
Cat.No: TN6646
Synonym:
Target:
9-O-Methyl-4-hydroxyboeravinone B
Cat.No: TN3327
Synonym:
Target: Others
Luteolin-7-rutinoside
Cat.No: T11895
Synonym:
Target: Others
Monensin
Cat.No: T1033L
Synonym: Elancoban,Rumensin,莫能菌素
Target:
α-D-Glucose-1-phosphate disodium hydrate
Cat.No: T73925
Synonym:
Target:
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