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Histamine Receptor

Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.
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Cat. No. Product Name CAS No. Purity Chemical Structure
T25875 Noberastine
诺柏斯汀
110588-56-2 98%
Noberastine 是一种新型组胺 H1拮抗剂,具有强效和特异性的外周抗组胺活性。
T70489 Enerisant HCl
盐酸Enerisant
1152749-07-9 98%
Enerisant HCl是一种新型强效选择性组胺H3受体拮抗剂,是P-gp的底物,由细胞色素P450(CYP)和转运蛋白介导。
T25737 Linetastine
利奈他斯汀
159776-68-8 98%
Linetastine 是一种 5-脂氧合酶抑制剂(5-LOX),能抑制白三烯的产生,并能拮抗组胺的作用。Linetastine可用于研究哮喘、动脉粥样硬化和消化性溃疡。
T68921 Impromidine hydrochloride
英普咪定盐酸盐
65573-02-6 98%
Impromidine hydrochloride 是一种非常有效和特异性的组胺H2受体激动剂,可用于进行心血管研究。
T68150 Talastine
他拉斯汀
16188-61-7 98%
Talastine 是一种抗组胺化合物,可诱发过敏性皮疹。
T68056 Donetidine
多奈替丁
99248-32-5 98%
Donetidine 是一种组胺 H2 受体拮抗剂,可用于治疗消化系统疾病。
T19839 Oxatomide
奥沙米特
60607-34-3 98%
Oxatomide 是一种有效且具有口服活性的双重 H1 组胺受体 和 P2X7 受体双重拮抗剂,具有抗组胺和抗过敏活性。Oxatomide 可用于阻断人 P2X7 受体中 ATP 诱导的电流 ,IC50 为 0.95 μM。Oxatomide 对 ATP 诱导的 Ca2+ 内流具有抑制作用,IC50 值为 0.43 μ...
T31195 Dalcotidine
化合物Dalcotidine
120958-90-9 98%
Dalcotidine 是一种新型组胺H2受体拮抗剂,具有组胺H9受体拮抗活性和抗分泌作用,与豚鼠大脑皮层结合的Ki 值为0.040 对分离性豚鼠右心房组胺诱导的正变时反应的拮抗作用的KB 值为0.041。Dalcotidine 提高了溃疡愈合的质量,可能有助于降低溃疡的复发率和复发率。
T34709 ST-1006
化合物ST-1006
1196994-11-2 98%
ST-1006是一种强效组胺 H4受体激动剂(pKi:7.94)。ST-1006具有抗炎作用。ST-1006是一种有效的嗜碱性粒细胞迁移诱导剂,可诱导嗜碱性粒细胞迁移。 ST-1006 具有抗炎作用和止痒作用。
T68146 Sufotidine
舒福替丁
80343-63-1 98%
Sufotidine 是一种具有高度选择性的竞争性 H2 受体拮抗剂。
T16476 PF-03654746
化合物PF-03654746
935840-31-6 98%
PF-03654746 是组胺 H3 受体的选择性拮抗剂。 PF-03654746 提高了阿尔茨海默病的认知功效和疾病改善作用。 PF-03654746 可用于治疗过敏性鼻炎的研究。
T3037 Cyclizine dihydrochloride
赛克利嗪二盐酸
5897-18-7 98%
Cyclizine dihydrochloride 是一种哌嗪衍生物,是选择性组胺H1受体拮抗剂,可用于恶心、呕吐和头晕的研究。
TN3699 Corchoionoside C
化合物 TN3699
185414-25-9 98%
Corchoionoside C has antioxidant activity, shows strong scavenging activities on DPPH radical, it also shows weak antifungal activity. Corchoionosides A, B, and ...
T10770 Cetirizine D8
化合物 T10770
774596-22-4 98%
Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
T11729 JTE-952
化合物 T11729
1255303-54-8 98%
JTE-952 is a oral, potent active and selective Type II inhibitor of colony stimulating factor-1 receptor (CSF-1R or cFMS, type III receptor tyrosine kinase), wit...
T15590 Iodophenpropit dihydrobromide
化合物 T15590
145196-87-8 98%
Iodophenpropit dihydrobromide is an effective and selective antagonist of the histamine H3 receptor. The binding of [125I]Iodophenpropit is readily reversible, s...
TN3483 Bakkenolide D
化合物 TN3483
18456-03-6 98%
Bakkenolide D has anti-allergic effect, it and bakkenolide D demonstrates inhibitory effect on the trachea contraction induced by histamine in vitro, they have o...
T12630 (R)-(-)-α-Methylhistamine dihydrobromide
(R)(−)-α-甲基组胺 二盐酸盐
868698-49-1 98%
(R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 nM).
TN2155 Rhodiocyanoside A
化合物Rhodiocyanoside A
168433-86-1 98%
Rhodiocyanoside A has antiallergic activity, it exhibits inhibitory activity on the histamine release from rat peritoneal exudate cells sensitized with anti-DNP ...
T11088 Doxepin D3 Hydrochloride
化合物 T11088
347840-07-7 98%
Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin...
Noberastine
T25875
Noberastine 是一种新型组胺 H1拮抗剂,具有强效和特异性的外周抗组胺活性。
Enerisant HCl
T70489
Enerisant HCl是一种新型强效选择性组胺H3受体拮抗剂,是P-gp的底物,由细胞色素P450(CYP)和转运蛋白介导。
Linetastine
T25737
Linetastine 是一种 5-脂氧合酶抑制剂(5-LOX),能抑制白三烯的产生,并能拮抗组胺的作用。Linetastine可用于研究哮喘、动脉粥样硬化和消化性溃疡。
Impromidine hydrochloride
T68921
Impromidine hydrochloride 是一种非常有效和特异性的组胺H2受体激动剂,可用于进行心血管研究。
Talastine
T68150
Talastine 是一种抗组胺化合物,可诱发过敏性皮疹。
Donetidine
T68056
Donetidine 是一种组胺 H2 受体拮抗剂,可用于治疗消化系统疾病。
Oxatomide
T19839
Oxatomide 是一种有效且具有口服活性的双重 H1 组胺受体 和 P2X7 受体双重拮抗剂,具有抗组胺和抗过敏活性。Oxatomide 可用于阻断人 P2X7 受体中 ATP 诱导的电流 ,IC50 为 0.95 μM。Oxatomide 对 ATP 诱导的 Ca2+ 内流具有抑制作用,IC50 值为 0.43 μ...
Dalcotidine
T31195
Dalcotidine 是一种新型组胺H2受体拮抗剂,具有组胺H9受体拮抗活性和抗分泌作用,与豚鼠大脑皮层结合的Ki 值为0.040 对分离性豚鼠右心房组胺诱导的正变时反应的拮抗作用的KB 值为0.041。Dalcotidine 提高了溃疡愈合的质量,可能有助于降低溃疡的复发率和复发率。
ST-1006
T34709
ST-1006是一种强效组胺 H4受体激动剂(pKi:7.94)。ST-1006具有抗炎作用。ST-1006是一种有效的嗜碱性粒细胞迁移诱导剂,可诱导嗜碱性粒细胞迁移。 ST-1006 具有抗炎作用和止痒作用。
Sufotidine
T68146
Sufotidine 是一种具有高度选择性的竞争性 H2 受体拮抗剂。
PF-03654746
T16476
PF-03654746 是组胺 H3 受体的选择性拮抗剂。 PF-03654746 提高了阿尔茨海默病的认知功效和疾病改善作用。 PF-03654746 可用于治疗过敏性鼻炎的研究。
Cyclizine dihydrochloride
T3037
Cyclizine dihydrochloride 是一种哌嗪衍生物,是选择性组胺H1受体拮抗剂,可用于恶心、呕吐和头晕的研究。
Corchoionoside C
TN3699
Corchoionoside C has antioxidant activity, shows strong scavenging activities on DPPH radical, it also shows weak antifungal activity. Corchoionosides A, B, and ...
Cetirizine D8
T10770
Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
JTE-952
T11729
JTE-952 is a oral, potent active and selective Type II inhibitor of colony stimulating factor-1 receptor (CSF-1R or cFMS, type III receptor tyrosine kinase), wit...
Iodophenpropit dihydrobromide
T15590
Iodophenpropit dihydrobromide is an effective and selective antagonist of the histamine H3 receptor. The binding of [125I]Iodophenpropit is readily reversible, s...
Bakkenolide D
TN3483
Bakkenolide D has anti-allergic effect, it and bakkenolide D demonstrates inhibitory effect on the trachea contraction induced by histamine in vitro, they have o...
(R)-(-)-α-Methylhistamine dihydrobromide
T12630
(R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 nM).
Rhodiocyanoside A
TN2155
Rhodiocyanoside A has antiallergic activity, it exhibits inhibitory activity on the histamine release from rat peritoneal exudate cells sensitized with anti-DNP ...
Doxepin D3 Hydrochloride
T11088
Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin...
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