Cat. No. | Product Name | CAS No. | Purity | Chemical Structure |
---|---|---|---|---|
T25875 | Noberastine
诺柏斯汀
|
110588-56-2 | 98% |
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Noberastine 是一种新型组胺 H1拮抗剂,具有强效和特异性的外周抗组胺活性。 | ||||
T70489 | Enerisant HCl
盐酸Enerisant
|
1152749-07-9 | 98% |
|
Enerisant HCl是一种新型强效选择性组胺H3受体拮抗剂,是P-gp的底物,由细胞色素P450(CYP)和转运蛋白介导。 | ||||
T25737 | Linetastine
利奈他斯汀
|
159776-68-8 | 98% |
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Linetastine 是一种 5-脂氧合酶抑制剂(5-LOX),能抑制白三烯的产生,并能拮抗组胺的作用。Linetastine可用于研究哮喘、动脉粥样硬化和消化性溃疡。 | ||||
T68921 | Impromidine hydrochloride
英普咪定盐酸盐
|
65573-02-6 | 98% |
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Impromidine hydrochloride 是一种非常有效和特异性的组胺H2受体激动剂,可用于进行心血管研究。 | ||||
T68150 | Talastine
他拉斯汀
|
16188-61-7 | 98% |
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Talastine 是一种抗组胺化合物,可诱发过敏性皮疹。 | ||||
T68056 | Donetidine
多奈替丁
|
99248-32-5 | 98% |
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Donetidine 是一种组胺 H2 受体拮抗剂,可用于治疗消化系统疾病。 | ||||
T19839 | Oxatomide
奥沙米特
|
60607-34-3 | 98% |
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Oxatomide 是一种有效且具有口服活性的双重 H1 组胺受体 和 P2X7 受体双重拮抗剂,具有抗组胺和抗过敏活性。Oxatomide 可用于阻断人 P2X7 受体中 ATP 诱导的电流 ,IC50 为 0.95 μM。Oxatomide 对 ATP 诱导的 Ca2+ 内流具有抑制作用,IC50 值为 0.43 μ... | ||||
T31195 | Dalcotidine
化合物Dalcotidine
|
120958-90-9 | 98% |
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Dalcotidine 是一种新型组胺H2受体拮抗剂,具有组胺H9受体拮抗活性和抗分泌作用,与豚鼠大脑皮层结合的Ki 值为0.040 对分离性豚鼠右心房组胺诱导的正变时反应的拮抗作用的KB 值为0.041。Dalcotidine 提高了溃疡愈合的质量,可能有助于降低溃疡的复发率和复发率。 | ||||
T34709 | ST-1006
化合物ST-1006
|
1196994-11-2 | 98% |
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ST-1006是一种强效组胺 H4受体激动剂(pKi:7.94)。ST-1006具有抗炎作用。ST-1006是一种有效的嗜碱性粒细胞迁移诱导剂,可诱导嗜碱性粒细胞迁移。 ST-1006 具有抗炎作用和止痒作用。 | ||||
T68146 | Sufotidine
舒福替丁
|
80343-63-1 | 98% |
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Sufotidine 是一种具有高度选择性的竞争性 H2 受体拮抗剂。 | ||||
T16476 | PF-03654746
化合物PF-03654746
|
935840-31-6 | 98% |
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PF-03654746 是组胺 H3 受体的选择性拮抗剂。 PF-03654746 提高了阿尔茨海默病的认知功效和疾病改善作用。 PF-03654746 可用于治疗过敏性鼻炎的研究。 | ||||
T3037 | Cyclizine dihydrochloride
赛克利嗪二盐酸
|
5897-18-7 | 98% |
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Cyclizine dihydrochloride 是一种哌嗪衍生物,是选择性组胺H1受体拮抗剂,可用于恶心、呕吐和头晕的研究。 | ||||
TN3699 | Corchoionoside C
化合物 TN3699
|
185414-25-9 | 98% |
|
Corchoionoside C has antioxidant activity, shows strong scavenging activities on DPPH radical, it also shows weak antifungal activity. Corchoionosides A, B, and ... | ||||
T10770 | Cetirizine D8
化合物 T10770
|
774596-22-4 | 98% |
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Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist. | ||||
T11729 | JTE-952
化合物 T11729
|
1255303-54-8 | 98% |
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JTE-952 is a oral, potent active and selective Type II inhibitor of colony stimulating factor-1 receptor (CSF-1R or cFMS, type III receptor tyrosine kinase), wit... | ||||
T15590 | Iodophenpropit dihydrobromide
化合物 T15590
|
145196-87-8 | 98% |
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Iodophenpropit dihydrobromide is an effective and selective antagonist of the histamine H3 receptor. The binding of [125I]Iodophenpropit is readily reversible, s... | ||||
TN3483 | Bakkenolide D
化合物 TN3483
|
18456-03-6 | 98% |
|
Bakkenolide D has anti-allergic effect, it and bakkenolide D demonstrates inhibitory effect on the trachea contraction induced by histamine in vitro, they have o... | ||||
T12630 | (R)-(-)-α-Methylhistamine dihydrobromide
(R)(−)-α-甲基组胺 二盐酸盐
|
868698-49-1 | 98% |
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(R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 nM). | ||||
TN2155 | Rhodiocyanoside A
化合物Rhodiocyanoside A
|
168433-86-1 | 98% |
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Rhodiocyanoside A has antiallergic activity, it exhibits inhibitory activity on the histamine release from rat peritoneal exudate cells sensitized with anti-DNP ... | ||||
T11088 | Doxepin D3 Hydrochloride
化合物 T11088
|
347840-07-7 | 98% |
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Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin... |