Cat. No. | Product Name | CAS No. | Purity | Chemical Structure |
---|---|---|---|---|
T72084 | (R)-BI-2852
化合物T72084
|
2375482-49-6 | 98% |
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(R)-5-hydroxy-3-(2-((((1-((1-methyl-1H-imidazol-4-yl)methyl)-1H-indol-6-yl)methyl)amino)methyl)-1H-indol-3-yl)isoindolin-1-one 可用作RAS 家族蛋白的抑制剂 ,是治疗和预防肿瘤的化合物。 (R)... | ||||
T30778 | CCG-257081
化合物CCG-257081
|
1922098-90-5 | 98% |
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CCG-257081 是心肌素相关转录因子和血清反应因子 (MRTF/SRF) 的抑制剂,通过抑制 Rho/MRTF/SRF 通路来发挥作用。CCG-257081已在多个小鼠模型中显示出预防博莱霉素诱导的纤维化的功效。CCG-257081 可用于预防癌症和纤维化的研究。 | ||||
T1931 | 6H05
化合物6H05
|
1469338-01-9 | 98% |
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6H05 是致癌突变体 K-Ras(G12C) 的选择性变构抑制剂。 | ||||
T62228 | KRAS G12D inhibitor 14
KRAS G12D抑制剂14
|
2765254-39-3 | 98% |
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KRAS G12D inhibitor 14 是一种 KRAS G12D 的有效抑制剂,能够结合 KRAS G12D 蛋白 (Kd: 33 nM)。KRAS G12D inhibitor 14 抑制 KRAS G12D (KRAS G12D-GTP) 的活性形式,但对 KRAS G13D 无抑制作用。 | ||||
T10374 | ARS-1323-alkyne
化合物ARS-1323-alkyne
|
2436544-27-1 | 98% |
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ARS-1323-alkyne 是switch-II pocket (S-IIP)抑制剂,能够特异性报告活体细胞中 KRASG12C 核苷酸的状态。 | ||||
T11770 | KRAS G12C inhibitor 16
化合物 T11770
|
2349392-79-4 | 98% |
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KRAS G12C inhibitor 16 is a potent KRAS G12C inhibitor. | ||||
T11776 | KRas G12C inhibitor 1
化合物 T11776
|
2158297-28-8 | 98% |
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KRas G12C inhibitor 1 is a compound that inhibits KRas G12C. | ||||
T11773 | KRAS inhibitor-6
化合物 T11773
|
2022986-61-2 | 98% |
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KRAS inhibitor-6 is a potent KRAS G12C inhibitor. | ||||
T16023 | MC 976
化合物 T16023
|
129831-99-8 | 98% |
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MC 976 is a derivative of Vitamin D3. | ||||
T11769 | KRAS G12C inhibitor 15
化合物 T11769
|
2349393-21-9 | 98% |
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KRAS G12C inhibitor 15 is a potent KRAS G12C inhibitor . | ||||
T11775 | KRAS inhibitor-8
化合物 T11775
|
2022986-70-3 | 98% |
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KRAS inhibitor-8 is a potent KRAS G12C inhibitor. | ||||
T12452 | Digeranyl bisphosphonate
化合物Digeranyl bisphosphonate
|
878143-03-4 | 98% |
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Digeranyl bisphosphonate 是一种有效的香叶基焦磷酸香叶酯 (GGPP) 合酶抑制剂,对 Rac1 的香叶基焦磷酸化有抑制作用。Digeranyl bisphosphonate 诱导细胞发生自噬却不诱导细胞凋亡。 | ||||
T11771 | KRAS G12C inhibitor 17
化合物 T11771
|
2349393-04-8 | 98% |
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KRAS G12C inhibitor 17 is a potent KRAS G12C inhibitor. | ||||
T11767 | KRAS G12C inhibitor 13
化合物 T11767
|
2241719-75-3 | 98% |
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KRAS G12C inhibitor 13 is a KRAS G12C inhibitor . | ||||
T11774 | KRAS inhibitor-7
化合物 T11774
|
2022986-68-9 | 98% |
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KRAS inhibitor-7 is a potent KRAS G12C inhibitor. | ||||
T11768 | KRAS G12C inhibitor 14
化合物 T11768
|
2349393-95-7 | 98% |
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KRAS G12C inhibitor 14 是一种有效的 KRAS G12C 抑制剂(IC50= 18 nM)。 | ||||
T11780 | KRAS G12C inhibitor 5
化合物 T11780
|
2158297-63-1 | 98% |
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KRAS G12C inhibitor 5 is a KRas G12C inhibitor. | ||||
T11744 | KB-5246
化合物 T11744
|
119474-55-4 | 98% |
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KB-5246, displays antibacterial activities.is a tetracyclic quinolone. | ||||
T11778 | KRas G12C inhibitor 3
化合物 T11778
|
2206735-75-1 | 98% |
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KRas G12C inhibitor 3 is a compound that inhibits KRas G12C. | ||||
T13844 | PROTAC K-Ras Degrader-1
化合物 T13844
|
2378258-52-5 | 98% |
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PROTAC K-Ras Degrader-1 is potent degrader of K-Ras based PROTAC. |