175
69
2
514
5
Cat. No. | Product Name | Form | Specificity Of Inhibition |
---|---|---|---|
C0051 |
Penicillin-Streptomycin Solution (100×), Sterile
青霉素-链霉素双抗溶液(100×),灭菌 |
Sol<em>uti</em>on in bottle | |
C0052 |
Penicillin-Streptomycin-Amphotericin B Solution (100×), Sterile
青霉素-链霉素-两性霉素B三抗溶液(100×),灭菌 |
Sol<em>uti</em>on in bottle |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T7777 |
M4284
M 4284 |
Antibacterial | Microbiology/Virology |
M4284 (M 4284) 是一种选择性和口服活性的联苯甘露糖苷 FimH 拮抗剂。它对不同宿主遗传背景和肠道微生物群落环境中的不同 UPEC(由尿路致病性大肠杆菌引起的尿路感染(UTI))菌株具有活性 | |||
T8139 |
Sulfamethoxazole sodium
新诺明钠,Ro 4-2130 sodium,磺胺甲恶唑钠 |
Others; Antibacterial; Antibiotic | Microbiology/Virology; Others |
Sulfamethoxazole sodium (Ro 4-2130 sodium) 是一种磺胺类抗菌素。它常用于各种尿道病原体的研究,与 Trimethoprim 联用,可用于尿路感染的研究。 | |||
T35337L |
Teduglutide acetate
|
Glucagon Receptor | GPCR/G Protein |
Teduglutide acetate 是一种 GLP-2 类似物,可使小肠黏膜肥大。它通过改变 claudin-10 的分布部分恢复小肠上皮功能,促进钠再循环以进行钠耦合葡萄糖转运和水吸收。 | |||
T19850 |
Semaglutide
索玛鲁肽,司美格鲁肽,索马鲁肽 |
Glucagon Receptor | GPCR/G Protein |
Semaglutide 是人胰高血糖素样肽-1受体激动剂,是一种人胰高血糖素样肽-1 的长效类似物。它有用于 2 型糖尿病研究的潜力。 | |||
T7618 |
Pyributicarb
TSH-888,稗草畏 |
P450 | Metabolism |
Pyributicarb (TSH-888) 是氨基甲酸酯型除草剂,能够有效激活CYP3A4基因及人类孕烷 X 受体。 | |||
T76702 |
Sutimlimab
|
Complement System | Immunology/Inflammation |
Sutimlimab 是一种新型靶向补体蛋白 C1 的单克隆抗体。Sutimlimab 常当作 C1 抑制剂使用,用于治疗冷凝集素病相关溶血。 | |||
T8567 |
amflutizole
|
Xanthine Oxidase | Metabolism |
amflutizole 用于治疗痛风,是一种黄嘌呤氧化酶抑制剂。 | |||
T4387 |
evobrutinib
MSC2364447C,M2951 |
BTK | Angiogenesis; Tyrosine Kinase/Adaptors |
Evobrutinib(M2951) 也称为 M-2951 和 MSC-2364447C,是布鲁顿酪氨酸激酶(BTK) 的高选择性抑制剂,BTK 对包括 B 淋巴细胞和巨噬细胞在内的各种免疫细胞的发育和功能很重要。临床前研究表明它可能对某些自身免疫性疾病有治疗作用。 | |||
T0081 |
Lafutidine
拉呋替丁,FRG-8813 |
5-HT Receptor; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Lafutidine (FRG-8813) 是一种组胺受体 H2RA 拮抗剂,可抑制胃酸分泌,具有胃粘膜保护作用,可用于研究胃食管反流疾病。 | |||
T27413 |
Trimebutine CTB salt
GIC1001 |
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
Trimebutine CTB salt (GIC-1001) 是一种阿片受体激动剂,可用于研究疼痛。 | |||
T12152 |
N-piperidine Ibrutinib hydrochloride
|
BTK | Angiogenesis; Tyrosine Kinase/Adaptors |
N-piperidine Ibrutinib hydrochloride 是一种强效的 BTK 抑制剂,是BTK 配体,抑制 WT BTK 和 C481S BTK ,可用于合成一系列 PROTAC 分子。N-piperidine Ibrutinib hydrochloride具有潜在的抗癌活性,可抑制癌细胞的生长和增殖。 | |||
T61268 |
Vutiglabridin
HSG4112 |
Phosphatase | Metabolism |
Vutiglabridin (HSG4112) 是一种新型且安全的PON2调节剂,是一个外消旋化合物。Vutiglabridin 是Glabridin 的优化结构类似物,比Glabridin 在减重效果和化学稳定性方面更加优越。Vutiglabridin 通过靶向线粒体对氧磷酶-2改善mptp 诱导的帕金森病小鼠的神经变性。Vutiglabridin 是一种治疗肥胖的临床2期药物,在PD 模型中对对线粒体PON2具有治疗作用。Vutiglabridin 渗透到大脑,结合PON2,恢复1-甲基-4-苯基吡啶(MPP*)诱导的SH-SY5Y 神经母细胞瘤细胞线粒体功能障碍。Vutiglabridin 在小鼠实验中 显著减轻了1-甲基-4苯基-1,2,3,6-四氢吡啶(MPTP)诱导的PD 模型小鼠的运动障碍和多巴胺能神经元损伤。 | |||
TP1472 |
Tyroserleutide
|
Others | Others |
Tyroserleutide 是一种可从猪脾脏的降解产物中分离得到的小分子三肽,在体内外均对肿瘤生长具有抑制作用。 | |||
TP1796 |
Albiglutide TFA (782500-75-8 free base)
Albiglutide TFA |
Glucagon Receptor | GPCR/G Protein |
Albiglutide TFA (782500-75-8 free base) (Albiglutide TFA) 是一种长效 GLP-1 受体激动剂,用于治疗 2 型糖尿病 (T2DM)。 | |||
T8460 |
Olmutinib
HM61713,BI1482694 |
EGFR | Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors |
Olmutinib (BI1482694) 是一种新型表皮生长因子受体酪氨酸激酶抑制剂。 | |||
T21404 |
Fluticasone furoate
Veramyst,Allermist,Avamys,糠酸氟替卡松,Fluticasone furoate |
Glucocorticoid Receptor | Endocrinology/Hormones |
Fluticasone furoate (Avamys) 是一种合成的三氟化皮质类固醇,衍生自氟替卡松,Kd 为 0.3 nM。Fluticasone furoate 具有有效的抗炎、抗哮喘活性和低全身暴露。Fluticasone furoate 可用作过敏性鼻炎治疗研究的鼻喷雾剂。 | |||
T61913 |
Cavutilide
|
EGFR | Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors |
Cavutilide具有抗心律失常活性,抑制 hERG K(+)通道,可用于研究心力衰竭和持续性心房颤动。 | |||
T26926 |
Butibufen
FF 105,FF-106,FF 106,FF106 |
Lipoxygenase | Metabolism |
Butibufen (FF-106) 是一种具有口服活性的非甾体抗炎化合物,是潜在的环氧合酶抑制剂,具有止痛和解热活性,抑制尿素合成。Butibufen 可用于研究风湿性疾病。 | |||
T16730 |
Remibrutinib
|
BTK | Angiogenesis; Tyrosine Kinase/Adaptors |
Remibrutinib 是有效的、口服具有活力的 bruton tyrosine kinase 抑制剂 (IC50:1 nM),在血液中抑制 BTK 活性的 IC50的值为 0.23 μM。它具有研究慢性荨麻疹的潜力。 | |||
T1667 |
Tandutinib
MLN518,CT53518,NSC726292,坦度替尼 |
Apoptosis; FLT; CSF-1R; PDGFR; Src; c-Kit | Angiogenesis; Apoptosis; Tyrosine Kinase/Adaptors |
Tandutinib (CT53518) 是一种选择性 FLT3抑制剂,其 IC50为 0.22 μM。它还抑制c-Kit 和PDGFR,其IC50分别为 0.17 μM 和 0.20 μM。它可穿透血脑屏障,用于急性骨髓性白血病。 | |||
T7175 |
Alflutinib mesylate
甲磺酸伏美替尼,AST2818 mesylate |
EGFR | Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors |
Alflutinib mesylate (AST2818 mesylate) 是一种不可逆的酪氨酸激酶抑制剂,可选择性抑制 EGFR 突变。 | |||
T9125 |
Tolebrutinib
PRN2246,SAR442168 |
BTK | Angiogenesis; Tyrosine Kinase/Adaptors |
Tolebrutinib (PRN2246) 是一种选择性、有效的、具有口服活性、可透过血脑屏障的布鲁顿氏酪氨酸激酶抑制剂,能够作用于 Ramos B 细胞 (IC50:0.4 nM)、HMC 小胶质细胞 (IC50:0.7 nM)。它对中枢神经系统免疫具有功效。它可用于多发性硬化症的研究。 | |||
T6541 |
Ibutilide Fumarate
Corvert Fumarate,U70226E,富马酸伊布利特 |
Calcium Channel; Sodium Channel | Membrane transporter/Ion channel; Metabolism |
Ibutilide Fumarate (U70226E) 是一种 III 类抗心律失常药物,可作用于急性心梗阻塞。 | |||
T9408 |
N-piperidine Ibrutinib
|
BTK | Angiogenesis; Tyrosine Kinase/Adaptors |
N-piperidine Ibrutinib 是一种有效的 BTK 抑制剂,对 WT BTK 和 C481S BTK 的 IC50 分别为 51.0 和 30.7 nM。它可作为BTK 配体用于一系列PROTAC 的合成,如SJF620。 SJF620 是一种有效的 PROTAC BTK 降解剂,DC50 为 7.9 nM。 | |||
TP1103 |
Cotadutide acetate
MEDI0382 acetate,Cotadutide acetate (1686108-82-6 Free base) |
Glucagon Receptor | GPCR/G Protein |
Cotadutide acetate (MEDI0382 acetate) 是一种有效的胰高血糖素样肽-1 (GLP-1) 和胰高血糖素受体肽双重激动剂,EC50 分别为 6.9 pM 和 10.2 pM。 | |||
T33479 |
Monoxerutin
Z 12007,MonoHER,7-Monohydroxyethylrutosid |
Antioxidant | oxidation-reduction |
Monoxerutin (MonoHER) 是一种血管扩张剂,具有抗氧化活性,可防止阿霉素诱导的小鼠心脏毒性,可用于研究急性呼吸系统综合征。 | |||
T12542 |
Rilzabrutinib
PRN1008 |
EGFR; Others; HER; BTK | Angiogenesis; JAK/STAT signaling; Others; Tyrosine Kinase/Adaptors |
Rilzabrutinib (PRN1008) 是一种可逆的、选择性的、有口服活性的布鲁顿氏酪氨酸激酶(BTK)共价抑制剂,其 IC50=1.3 nM。 | |||
T1501 |
Rifabutin
LM-427,Ansamycin,利福布汀,利福布丁 |
HSP; DNA/RNA Synthesis; Antibacterial; Antibiotic | Cell Cycle/Checkpoint; Cytoskeletal Signaling; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology |
Rifabutin (LM-427) 是半合成的安莎霉素抗生素,抑制 DNA 依赖性 RNA 聚合酶,有抗分枝杆菌作用。 | |||
T0918 |
Trimebutine
曲美布汀,Mebutin |
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
Trimebutine (Mebutin) 是阿片受体激动剂,有抗毒蕈碱活性。它是解痉剂,可调节肠道和结肠运动,并通过抗毒蕈碱和弱μ-阿片受体激动剂作用缓解腹痛。 | |||
T22254 |
Alflutinib
AST2818,ASK120067 |
EGFR; P450 | Angiogenesis; JAK/STAT signaling; Metabolism; Tyrosine Kinase/Adaptors |
Alflutinib (ASK120067) 是 EGFR 抑制剂。 它对 T790M 的性耐药突变以及 EGFR 活性突变具有抑制作用。它对于癌症疾病,特别是非小细胞肺癌(NSC-LC)方面具有研究潜力。 | |||
TQ0242 |
Fenebrutinib
GDC-0853 |
BTK | Angiogenesis; Tyrosine Kinase/Adaptors |
Fenebrutinib (GDC-0853) 是一种选择性的、有效的、具有口服活性的、非共价的布鲁顿酪氨酸激酶抑制剂,对野生型 Btk,及突变型 C481S,C481R,T474I,T474M 的 Ki 分别为 0.91 nM,1.6,1.3,12.6 和 3.4 nM。有用于类风湿关节炎和系统性红斑狼疮研究的潜力。 | |||
T36287 |
Pirtobrutinib
|
BTK | Angiogenesis; Tyrosine Kinase/Adaptors |
Pirtobrutinib (LOXO-305) is an advanced BTK inhibitor that displays high selectivity and operates through a non-covalent mechanism. This compound effectively inhibits various BTK C481 substitution mutations, leading to tumor regression in BTK-dependent lymphoma tumors in mouse xenograft models. Furthermore, Pirtobrutinib exhibits remarkable selectivity for BTK, with more than a 300-fold difference compared to 370 other kinases tested. Notably, at a concentration of 1 μM, Pirtobrutinib demonstrat... | |||
T5044 |
Futibatinib
TAS120,FGFR-IN-1 |
FGFR | Angiogenesis; Tyrosine Kinase/Adaptors |
Futibatinib (FGFR-IN-1) 是口服具有活力的、选择性强的、高生物利用度的、不可逆的 FGFR 抑制剂。它抑制突变型和野生型 FGFR2,且 IC50相似(wild-type FGFR2=0.9 nM; V5651=1-3 nM; N550H=3.6 nM; E566G=2.4 nM)。 | |||
T14337 |
Buloxibutid
AT2 receptor agonist C21 |
RAAS | Endocrinology/Hormones |
Buloxibutid (AT2 receptor agonist C21) 是一种新型且具有选择性小分子 angiotensin II AT2 receptor (血管紧张素 II AT2 受体)激动剂,对 AT2 受体和 AT1 受体的 Ki 值分别为 0.4 nM 和 10 μM。 | |||
T3626 |
Acalabrutinib
ACP-196,阿可替尼 |
BTK | Angiogenesis; Tyrosine Kinase/Adaptors |
Acalabrutinib (ACP-196) 是一种不可逆的、高效的、具有口服活性、选择性的第二代BTK 抑制剂。它与 BTK 的 ATP 结合口袋中的 Cys481 共价结合。它在慢性淋巴细胞性白血病 (CLL) 小鼠模型中显示出强大的靶向作用和功效。 | |||
T13447 |
(R)-Zanubrutinib
(R)-BGB-3111 |
BTK | Angiogenesis; Tyrosine Kinase/Adaptors |
(R)-Zanubrutinib ((R)-BGB-3111) 是布鲁顿酪氨酸激酶(BTK)的选择性抑制剂。 | |||
T7584 |
zanubrutinib
赞鲁替尼,BGB-3111,泽布替尼 |
BTK | Angiogenesis; Tyrosine Kinase/Adaptors |
Zanubrutinib (BGB-3111) 是 Bruton tyrosine kinase(Btk) 的选择性抑制剂。 | |||
T67881 |
Acalabrutinib enantiomer
R-Acalabrutinib |
BTK | Angiogenesis; Tyrosine Kinase/Adaptors |
Acalabrutinib enantiomer (R-Acalabrutinib) 是一类属于布鲁顿酪氨酸激酶(BTK)抑制剂的化合物。Acalabrutinib enantiomer 可用于癌症、自身免疫性疾病和慢性炎症等领域的研究。 | |||
T6918 |
Olmutinib
HM61713, BI 1482694,奥莫替尼,BI 1482694,HM61713 |
EGFR; BTK | Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors |
Olmutinib (HM61713, BI 1482694) 是可口服的不可逆 EGFR 酪氨酸激酶抑制剂,其与激酶结构域附近的半胱氨酸残基结合,可用于非小细胞肺癌的研究。 | |||
T6876 |
Liraglutide
利拉鲁肽,Liraglutidum,利拉糖肽,Victoza,Liraglutida,NN2211 |
Glucagon Receptor | GPCR/G Protein |
Liraglutide (Liraglutida) 是胰高血糖素样肽-1 受体激动剂,用于 2 型糖尿病的研究。 | |||
TQ0236 |
Tirabrutinib
ONO-4059,GS-4059,Velexbru |
BTK | Angiogenesis; Tyrosine Kinase/Adaptors |
Tirabrutinib (GS-4059) (ONO-4059) 是一种口服有效的高选择性 Bruton’s Tyrosine Kinase (BTK) 抑制剂 (能透过血脑屏障),其 IC50 值为 6.8 nM。Tirabrutinib 不可逆共价结合 BTK 并抑制异常 B 细胞受体信号传导。Tirabrutinib 可用于自身免疫性疾病和血液学恶性肿瘤的研究。 | |||
T8636 |
Ibrutinib deacryloylpiperidine
IBT4A,5-(4-phenoxyphenyl)-7H-pyrrolo[2,3-d]pyriMidin-4-ylaMine,伊布替尼中间体N-2 |
BTK | Angiogenesis; Tyrosine Kinase/Adaptors |
Ibrutinib deacryloylpiperidine (IBT4A) 是 Ibrutinib 的杂质之一。它是一种不可逆的、选择性的 Btk 抑制剂 (IC50:0.5 nM)。 | |||
T16679 |
Belzutifan
PT2977,MK-6482 |
HIF | Angiogenesis; Chromatin/Epigenetic |
Belzutifan (MK-6482) 是具有口服活性的 HIF-2α选择性抑制剂,IC50为 9 nM。Belzutifan 具有提高的效力和改善的药代动力学特征。Belzutifan (MK-6482) 可以抑制透明细胞肾细胞癌。 | |||
T5913 |
Sulbutiamine
舒布硫胺,Bisibuthiamine |
Antioxidant | oxidation-reduction |
Sulbutiamine (Bisibuthiamine) 是合成的维生素 B1 类似物,可用于研究无力症。 | |||
T0188 |
Fluticasone (propionate)
丙酸氟替卡松,CCI-187881,氟替卡松丙酸酯,Fluticasone propionate |
Glucocorticoid Receptor; Virus Protease; Estrogen/progestogen Receptor; Phospholipase; Endogenous Metabolite | Endocrinology/Hormones; Metabolism; Microbiology/Virology |
Fluticasone propionate (CCI-187881) 是一种选择性糖皮质激素受体激动剂,是一种局部抗炎激素,亲和力KD 为 0.5 nM。具有抗病毒活性。 | |||
T78097L |
Mazdutide acetate(2259884-03-0 free base)
Mazdutide acetate(2259884-03-0 free base),OXM-3 acetate,LY-3305677 acetate,IBI-362 acetate |
Glucagon Receptor | GPCR/G Protein |
Mazdutide acetate 是一种高效的胰高血糖素样肽 (GLP-1R) 与胰高血糖素受体 (GCGR) 的共激动剂,是一种胃泌酸调节素类似物。Mazdutide acetate可刺激小鼠胰岛的胰岛素分泌 ,可用于研究肥胖和 2 型糖尿病 (T2D) 。 | |||
T17220 |
Vecabrutinib
SNS-062 |
Tyrosine Kinases; BTK | Angiogenesis; Tyrosine Kinase/Adaptors |
Vecabrutinib (SNS-062) (SNS-062) 是一种有效的,非共价的 BTK 和 ITK 抑制剂,Kd 值分别为 0.3 nM 和 2.2 nM。Vecabrutinib 对 ITK 的 IC50 值为 24 nM。 | |||
T5407 |
Branebrutinib
BMS986195 |
BTK | Angiogenesis; Tyrosine Kinase/Adaptors |
Branebrutinib (BMS986195) 是一个高效的、不可逆的、共价的、选择抑的布鲁顿氏酪氨酸激酶(BTK)的制剂 (IC50:0.1 nM)。 | |||
TQ0039 |
(±)-Zanubrutinib
(±)-BGB-3111 |
BTK | Angiogenesis; Tyrosine Kinase/Adaptors |
(±)-Zanubrutinib ((±)-BGB-3111) 是一种有效的口服Bruton’s 酪氨酸激酶(Btk)抑制剂,具有优越的口服生物利用度,可实现更高的暴露量和更完整的靶点抑制。 | |||
T1937 |
Spautin-1
Spautin 1 |
Apoptosis; DUB; Autophagy | Apoptosis; Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Ubiquitination |
Spautin-1是一种特异性自噬抑制剂,可抑制泛素特异性肽酶 USP10和 USP13,IC50s 约为0.6到0.7 μM。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1313 |
Nitrofurantoin
Furadantine,呋喃妥因,Macrodantin,Furadonine |
Antibacterial; Antibiotic | Microbiology/Virology |
Nitrofurantoin (Furadantine) 是一种具有口服活性的广谱内酰胺酶抗菌剂。它是一种抗生素,可研究尿路感染。 | |||
T0473 |
Arbutin
Uva,p-Arbutin,p-Arbutin,熊果苷,β-Arbutin |
Tyrosinase | Proteases/Proteasome |
Arbutin (p-Arbutin) 是一种从熊果植物 Arctostaphylos uvaursi 中分离出的天然多酚,具有抗氧化,抗炎和抗肿瘤特性。它是一种脱色剂,也是一种黑色素细胞中酪氨酸酶的竞争性抑制剂,对单酚酶的 Kiapp 值为 1.42 mM;对二酚酶Kiapp 的值为 0.9 mM。 | |||
T22417 |
Rutin hydrate
芦丁,Rutoside,Sophorin,Quercetin-3-O-rutinoside |
Beta Amyloid; Others; Autophagy | Autophagy; Neuroscience; Others |
Rutin hydrate (Sophorin) 是一种广泛存在于多种植物中的黄酮类天然产物,具有降糖、抗炎、抗氧化、神经保护、肾脏保护、肝脏保护和降低 Aβ 低聚物活性等多种生物活性。它能穿过血脑屏障,通过抑制细胞凋亡、线粒体功能紊乱和氧化应激抑制万古霉素诱导的肾小管细胞凋亡。 | |||
T67708 |
Thiolutin
Acetopyrrothin |
Antibacterial; Antibiotic | Microbiology/Virology |
Thiolutin (Acetopyrrothin) 是一种内皮细胞粘附抑制剂,由链霉菌产生。 Thiolutin 具有抗生素和抗血管生成特性。 Thiolutin 可快速诱导 Hsp27 的磷酸化。 | |||
T16552 |
Pleuromutilin
Mutilin 14-glycolate,Drosophilin B,截短侧耳素 |
Antibacterial; Antibiotic | Microbiology/Virology |
Pleuromutilin (Drosophilin B) 通过与细菌的 50S 核糖体亚基结合来抑制细菌蛋白质的合成。 | |||
TN1065 |
Hirsutine
|
Apoptosis | Apoptosis |
Hirsutine 是一种来自钩藤的吲哚生物碱,可诱导细胞凋亡,是一种登革热病毒抑制剂,且毒性低。它具有抗癌、心脏保护、抗高血压、抗心律失常和血管舒张活性。 | |||
TN1461 |
(-)-Butin
Butin,漆黄素 ( 紫铆素) |
Akt; PI3K; Nrf2 | Cytoskeletal Signaling; Immunology/Inflammation; PI3K/Akt/mTOR signaling |
(-)-Butin (Butin) 是 Butin 的 S 对映体。其中 Butin 是一种分离自黄檀的心材中的生物活性黄酮类化合物,具有显著的抗血小板、抗氧化、抗炎作用。 | |||
T4911 |
α-Arbutin
4-hydroxyphenyl-D-lucopyranoside,alpha-Arbutoside,α-熊果苷,alpha-Arbutin |
Tyrosinase | Proteases/Proteasome |
α-Arbutin (4-hydroxyphenyl-D-lucopyranoside) 是一种流行的、有效的皮肤增白剂,也是一种酪氨酸酶 (tyrosinase) 抑制剂。 | |||
T19898 |
Methylarbutin
ß-PMP-Glc;4-Methoxyphenyl β-D-Glucopyranoside,ß-PMP-Glc,4-Methoxyphenyl β-D-Glucopyranoside |
Others | Others |
Methylarbutin (ß-PMP-Glc;4-Methoxyphenyl β-D-Glucopyranoside) 是一种冰重结晶抑制剂 (IRI)。 | |||
T0795 |
Rutin
Quercetin 3-O-rutinoside,芦丁,Rutoside |
Beta Amyloid; Prostaglandin Receptor; Autophagy | Autophagy; GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Rutin (Quercetin 3-O-rutinoside) 属于黄酮类天然产物,具有血脑屏障渗透性。Rutin 具有广泛的生物活性,包括抗氧化、抗炎、抗肿瘤、降血糖、神经保护、抗菌、抗衰老等等。 | |||
T3816 |
Velutin
|
NF-κB; HIF/HIF Prolyl-Hydroxylase | Chromatin/Epigenetic; Metabolism; NF-κB |
Velutin 是一种苷元,提取自槲寄生中,能够抑制黑色素生物合成。它利用 NF-κB 途径减少破骨细胞分化和下调 HIF-1α。 | |||
T13818 |
Phytohemagglutinin
PHA-M,植物血球凝集素,PHA,植物血凝素 |
Apoptosis | Apoptosis |
Phytohemagglutinin (PHA-M) 是一种普通豆菜豆的主要种子凝集素,聚集在子叶的薄壁细胞中。它是一种 T 细胞激活剂,能够刺激人单核白细胞,可诱导 ChAT mRNA 表达,增强 ACh 合成。 | |||
T6463 |
Deoxyarbutin
|
Tyrosinase | Proteases/Proteasome |
Deoxyarbutin 能够抑制酪氨酸酶活性和黑色素合成,具有显著而持久的美白效果,表现出强烈的抗氧化作用。 | |||
T60104 |
Mycophenolic acid-β-D-glucuronide solution
|
Others | Others |
Mycophenolic acid glucuronide 是人血浆中mycophenolic acid 的葡糖甙代谢产物。 | |||
T3817 |
Darutigenol
|
Others | Others |
Darutigenol 是一种戊二萜,从Siegesbecikia orientalis L.中分离得到。 | |||
T0772 |
Troxerutin
曲克芦丁,Trihydroxyethylrutin,维脑路通 |
NOD-like Receptor (NLR) | Immunology/Inflammation |
Troxerutin (Trihydroxyethylrutin) 是一种天然生物类黄酮芦丁的三羟乙基化衍生物,也被称为维生素 P4,可抑制活性氧的产生并抑制 ER 应激介导的NOD 活化。 | |||
T4S2164 |
Narirutin
Naringenin-7-O-rutinoside,Isonaringin,芸香柚皮苷,柚皮芸香苷 |
Others; Antibacterial | Microbiology/Virology; Others |
Narirutin (Naringenin-7-O-rutinoside) 是从Citrus unshiu 中分离的活性成分之一,具有抗氧化和抗炎活性。它是一种具有抗结核效力的shikimate 激酶抑制剂。 | |||
TN1738 | Homoarbutin | Others | Others |
Homoarbutin is a natural product | |||
TN5646 |
Antiarol rutinoside
3,4,5-Trimethoxyphenyl rutinoside |
||
Antiarol rutinoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5646,CAS号为 261351-23-9。 | |||
TN3298 |
8alpha-Hydroxyhirsutinolide
|
TNF; NF-κB | Apoptosis; NF-κB |
8alpha-Hydroxyhirsutinolide shows anti-inflammatory activity, it inhibits TNF-α-induced NF-κB activity with the IC(50) value of 1.9 uM. | |||
T81072 |
Suffruticosol A
|
||
Suffruticosol A是一种从P. lactiflora种子中分离得到的神经保护剂,能够逆转由Scopolamine诱导的细胞神经退行性损伤。该化合物还能改善海马体胆碱能缺陷并部分增强BDNF信号传导,从而在Scopolamine诱导模型中显示出改善神经功能的作用,可恢复小鼠记忆与认知行为。 | |||
T81731 |
Myricetin-3-O-rutinoside
|
||
Myricetin-3-O-rutinoside(Compound 3)是从Picea abies中分离出的天然化合物。 | |||
T81507 |
Petunidin 3-rutinoside
|
||
Petunidin 3-rutinoside,一种可从Sambucus canadensis分离的天然产物。 | |||
TN6915 |
Quercetin-7-O-rutinoside
|
||
Quercetin-7-O-rutinoside is a natural product. | |||
TN2129 |
Quercetin-3-o-rutinose
|
Others | Others |
Quercetin-3-o-rutinose has antioxidative activity, it exerts strong DPPH radical-scavenging activity. | |||
TN5572 |
9β-Hydroxydarutigenol
|
||
9β-Hydroxydarutigenol 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5572,CAS号为 1188282-00-9。 | |||
T70355 |
Flutimide
|
Others | Others |
Flutimide是一种针对流感病毒核酸内切酶的选择性抑制剂,具有3 μM的IC50值,表现出细胞培养中的抗病毒活性,适用于流感等急性传染性呼吸道疾病的研究。 | |||
TN3293 | 8alpha-(2-Methylacryloyloxy)-1-O-methylhirsutinolide 13-O-acetate | Others | Others |
8alpha-(2-Methylacryloyloxy)-1-O-methylhirsutinolide 13-O-acetate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3293,CAS号为 883872-71-7。 | |||
TN1313 |
6-Hydroxykaempferol 3-Rutinoside -6-glucoside
|
Others | Others |
6-Hydroxykaempferol 3-Rutinoside -6-glucoside是一种天然产物,属于菊科金线菊属,其产品编号为 TN1313,CAS号为 145134-63-0。6-Hydroxykaempferol 3-Rutinoside -6-glucoside可用作对照参考。 | |||
TN5085 |
Syringetin-3-O-rutinoside
|
Others | Others |
Syringetin-3-O-rutinoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5085,CAS号为 53430-50-5。 | |||
TN6285 |
Beiwutine
|
||
Beiwutine 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6285,CAS号为 76918-93-9。 | |||
TN3236 |
7-Hydroxydarutigenol
|
Others | Others |
7-Hydroxydarutigenol 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3236,CAS号为 1188281-99-3。 | |||
T38016 |
Hirsutide
|
Others | Others |
Hirsutide is a cyclotetrapeptide fungal metabolite produced by the entomopathogenic fungus Hirsutella. It has antibacterial activity against C. pyogenes, S. aureus, P. aeruginosa, and K. pneumonia (MICs = 25, 13, 6, and 21 μg/cm3, respectively). Hirsutide also has antifungal activity against C. albicans, M. audouinii, A. niger, and Ganoderma (MICs = 13, 6, 25, and 6 μg/cm3, respectively). | |||
TN3295 |
8alpha-(2-Methylacryloyloxy)hirsutinolide
|
Others | Others |
8alpha-(2-Methylacryloyloxy)hirsutinolide 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3295,CAS号为 188293-70-1。 | |||
TN6255 |
3,7,8-Tri-O-methylellagic acid 2-O-rutinoside
3,3',4'-Tri-O-methylellagic acid 4-O-rutinoside |
||
3,7,8-Tri-O-methylellagic acid 2-O-rutinoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6255,CAS号为 56470-18-9。 | |||
TN4781 |
Physcion 8-O-rutinoside
|
Others | Others |
Physcion 8-O-rutinoside is a natural product from Rhamnus libanoticus. | |||
TN1320 |
6-O-Caffeoylarbutin
|
Others | Others |
6'-O-caffeoylarbutin may serve as a skin-whitening ingredient with the merits of potent melanin inhibition,less toxicity and reversible melanin synthesis after stopping use. | |||
TN6620 |
Peonidin-3-O-rutinoside chloride
|
||
Peonidin-3-O-rutinoside chloride 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6620,CAS号为 27539-32-8。 | |||
TN1311 |
5,6,7,4'-Tetrahydroxyflavonol 3-O-rutinoside
6-Hydroxykaempferol 3-beta-rutinoside,6-羟基山柰酚-3-O-芸香糖苷 |
Others | Others |
6-Hydroxykaempferol 3-beta-rutinoside is a natural product | |||
T41035 |
Methoxyeugenol 4-O-rutinoside
|
Others | Others |
Methoxyeugenol 4-O-rutinoside (compound 9) is a phenyl glucoside present in Daphniphyllum angustifolium bark. | |||
TN7477 |
Isorhamnetin-3-O-rutinoside-7-O-glucoside
|
Others | Others |
T77201 |
Rutin trihydrate
|
Others | Others |
Rutin (Rutoside) trihydrate 是多功能天然黄酮苷,展现出抗氧化、抗炎、抗糖尿病及抗癌效果。此外,该化合物还具有心脏保护和神经保护活性。 | |||
TN4033 |
Eugenol rutinoside
|
Others | Others |
Eugenol rutinoside 是一种存在于dendropanax dentiger 中的天然产物。 | |||
TN6344 |
Velutinam
|
||
Velutinam 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6344,CAS号为 146428-62-8。 | |||
TN5807 |
Ethyl rutinoside
|
||
Ethyl rutinoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5807,CAS号为 187539-57-7。 | |||
TN4539 |
Methyl chanofruticosinate
|
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Methyl chanofruticosinate has weak anti-HIV-1 activity. | |||
TN3111 |
5-Glutinen-3-ol
|
Others | Others |
5-Glutinen-3-ol is a natural product from Clausena excavata. | |||
TN3294 |
8alpha-(2-Methylacryloyloxy)hirsutinolide 13-O-acetate
|
NADPH-oxidase; P450; MAO | Immunology/Inflammation; Metabolism; Neuroscience |
8alpha-(2-Methylacryloyloxy)hirsutinolide 13-O-acetate shows inhibitory activity toward CYP2A6 and MAO-A and MAO-B enzymes. | |||
T81933 |
Limocitrin-3-rutinoside
|
||
Limocitrin-3-rutinoside,一种类黄酮成员及糖苷,可从桃(Prunus persica)果实中提取。 | |||
TN5571 |
16-O-Acetyldarutigenol
|
||
16-O-Acetyldarutigenol是一种天然产物,属于菊科豨莶属,其产品编号为 TN5571,CAS号为 1188282-01-0。16-O-Acetyldarutigenol可用作对照参考。 | |||
------------------------ 更多 ------------------------ |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-03044 |
Bikunin/AMBP Protein, Human, Recombinant (aa 1-203, His)
α-1-microglobulin/bikunin precursor,ITI,EDC1,alpha-1-microgl... |
Human | HEK293 Cells |
Bikunin/AMBP Protein, Human, Recombinant (aa 1-203, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 22.3 kDa and the accession number is P02760. | |||
TMPY-00326 |
Bikunin/AMBP Protein, Human, Recombinant (mFc)
ITI,HCP,HI30,IATIL,A1M,ITIL,UTI,ITILC,EDC1,alpha-1-... |
Human | HEK293 Cells |
Bikunin/AMBP Protein, Human, Recombinant (mFc) is expressed in HEK293 mammalian cells with mFc tag. The predicted molecular weight is 47.2 kDa and the accession number is P02760. | |||
TMPY-00363 |
Bikunin/AMBP Protein, Human, Recombinant (aa 206-348, His)
EDC1,ITILC,UTI,α-1-microglobulin/bikunin precursor,... |
Human | P. pastoris (Yeast) |
Bikunin/AMBP Protein, Human, Recombinant (aa 206-348, His) is expressed in yeast with His tag. The predicted molecular weight is 17.4 kDa and the accession number is CAA38587.1. | |||
TMPY-05823 |
Influenza B (B/Colorado/06/2017) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
Influenza B | HEK293 Cells |
Influenza B (B/Colorado/06/2017) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 58.86 kDa and the accession number is A0A2Z5E1Y3. | |||
TMPY-00152 |
Influenza A H3N2 (A/Texas/50/2012) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H3N2 | Baculovirus Insect Cells |
Influenza A H3N2 (A/Texas/50/2012) Hemagglutinin/HA Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 59.3 kDa. | |||
TMPY-01193 |
Influenza A H1N1 (A/Brevig Mission/1/1918) Hemagglutinin Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H1N1 | HEK293 Cells |
Influenza A H1N1 (A/Brevig Mission/1/1918) Hemagglutinin Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 37.5 kDa and the accession number is Q9WFX3. | |||
TMPY-01501 |
Influenza A H1N1 (A/Puerto Rico/8/1934) Hemagglutinin/HA Protein (HEK293, His)
Harvey rat sarcoma viral oncogene homolog |
H1N1 | HEK293 Cells |
Influenza A H1N1 (A/Puerto Rico/8/1934) Hemagglutinin/HA Protein (HEK293, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 59 kDa and the accession number is P03452. | |||
TMPY-00416 |
Influenza A H10N8 (A/Jiangxi-Donghu/346/2013) Hemagglutinin/HA0 Protein
Harvey rat sarcoma viral oncogene homolog |
H10N8 | Baculovirus Insect Cells |
Influenza A H10N8 (A/Jiangxi-Donghu/346/2013) Hemagglutinin/HA0 Protein is expressed in Baculovirus insect cells. The predicted molecular weight is 60.6 kDa. | |||
TMPY-05533 |
Influenza A H1N1 (A/Michigan/45/2015) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H1N1 | HEK293 Cells |
Influenza A H1N1 (A/Michigan/45/2015) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 59.2 kDa. | |||
TMPY-05908 |
Influenza A H1N1 (A/swine/England/267/2007) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H1N1 | HEK293 Cells |
Influenza A H1N1 (A/swine/England/267/2007) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 58.3 kDa and the accession number is A0A0K0NE88. | |||
TMPY-01129 |
Influenza A H5N1 (A/Vietnam/1194/2004) Hemagglutinin/HA Protein (RERRRKKR to TETR, HA1+HA2, uncleaved, His)
Harvey rat sarcoma viral oncogene homolog |
H5N1 | HEK293 Cells |
Influenza A H5N1 (A/Vietnam/1194/2004) Hemagglutinin/HA Protein (RERRRKKR to TETR, HA1+HA2, uncleaved, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 59 kDa and the accession number is Q6DQ34. | |||
TMPY-00113 |
Influenza A H3N2 (A/Wisconsin/67/2005) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H3N2 | Baculovirus Insect Cells |
Influenza A H3N2 (A/Wisconsin/67/2005) Hemagglutinin/HA Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 59.3 kDa and the accession number is B4URC5. | |||
TMPY-01525 |
Influenza A H3N2 (A/Aichi/2/1968) Hemagglutinin/HA1 Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H3N2 | HEK293 Cells |
Influenza A H3N2 (A/Aichi/2/1968) Hemagglutinin/HA1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 37.6 kDa and the accession number is P03437. | |||
TMPY-05021 |
Influenza B (B/Brisbane/60/2008) Hemagglutinin/HA Protein
Harvey rat sarcoma viral oncogene homolog |
Influenza B | Baculovirus Insect Cells |
Influenza B (B/Brisbane/60/2008) Hemagglutinin/HA Protein is expressed in Baculovirus insect cells. The predicted molecular weight is 61.7kDa and the accession number is C0LT35. | |||
TMPY-04293 |
Influenza A H3N2 (A/Perth/16/2009) Hemagglutinin/HA0 Protein
Harvey rat sarcoma viral oncogene homolog |
H3N2 | Baculovirus Insect Cells |
Influenza A H3N2 (A/Perth/16/2009) Hemagglutinin/HA0 Protein is expressed in Baculovirus insect cells. The predicted molecular weight is 61.9 kDa and the accession number is C6KNH7. | |||
TMPY-00012 |
Influenza A H3N2 (A/Texas/50/2012) Hemagglutinin/HA1 Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H3N2 | HEK293 Cells |
Influenza A H3N2 (A/Texas/50/2012) Hemagglutinin/HA1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 38.1 kDa and the accession number is R4L4F3. | |||
TMPY-05918 |
Influenza A H1N1 (A/Guangdong-Maonan/SWL1536/2019)/(A/Hawaii/70/2019) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H1N1 | HEK293 Cells |
Influenza A H1N1 (A/Guangdong-Maonan/SWL1536/2019)/(A/Hawaii/70/2019) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 59.2 kDa and the accession number is A0A5Q2EZ09. | |||
TMPY-02343 |
Influenza B (B/Brisbane/60/2008) Hemagglutinin/HA1 Protein (His)
Harvey rat sarcoma viral oncogene homolog |
Influenza B | HEK293 Cells |
Influenza B (B/Brisbane/60/2008) Hemagglutinin/HA1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 39.1 kDa and the accession number is C0LT38. | |||
TMPY-04524 |
Influenza B (B/PHUKET/3073/2013) Hemagglutinin/HA1 Protein (His)
Harvey rat sarcoma viral oncogene homolog |
Influenza B | HEK293 Cells |
Influenza B (B/PHUKET/3073/2013) Hemagglutinin/HA1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 39.1 kDa. | |||
TMPY-01134 |
Influenza A H1N1 (A/Brisbane/59/2007) Hemagglutinin Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H1N1 | HEK293 Cells |
Influenza A H1N1 (A/Brisbane/59/2007) Hemagglutinin Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 37.7 kDa and the accession number is B0VX44. | |||
TMPY-01528 |
Influenza A H5N1 (A/Hong Kong/483/1997) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H5N1 | HEK293 Cells |
Influenza A H5N1 (A/Hong Kong/483/1997) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 59.7 kDa and the accession number is O92930. | |||
TMPY-00109 |
Influenza A H1N1 (A/WSN/1933) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H1N1 | Baculovirus Insect Cells |
Influenza A H1N1 (A/WSN/1933) Hemagglutinin/HA Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 59.1 kDa and the accession number is B4URE7. | |||
TMPY-01522 |
Influenza A H1N1 (A/Solomon Islands/3/2006) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H1N1 | HEK293 Cells |
Influenza A H1N1 (A/Solomon Islands/3/2006) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 59 kDa and the accession number is A7Y8I1. | |||
TMPY-01519 |
Influenza A H1N1 (A/New Caledonia/20/1999) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H1N1 | HEK293 Cells |
Influenza A H1N1 (A/New Caledonia/20/1999) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 59 kDa and the accession number is Q6WG00. | |||
TMPY-00642 |
Influenza A H1N1 (A/California/07/2009) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H1N1 | Baculovirus Insect Cells |
Influenza A H1N1 (A/California/07/2009) Hemagglutinin/HA Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 59 kDa and the accession number is C3W5X2. | |||
TMPY-00744 |
Influenza A H5N1 (A/VietNam/1203/2004) Hemagglutinin/HA Protein (His & Fc)
Harvey rat sarcoma viral oncogene homolog |
H5N1 | HEK293 Cells |
Influenza A H5N1 (A/VietNam/1203/2004) Hemagglutinin/HA Protein (His & Fc) is expressed in HEK293 mammalian cells with His and Fc tag. The predicted molecular weight is 85.7 kDa and the accession number is Q5EP31. | |||
TMPY-04701 |
Influenza B (B/PHUKET/3073/2013) Hemagglutinin/HA0 Protein
Harvey rat sarcoma viral oncogene homolog |
Influenza B | Baculovirus Insect Cells |
Influenza B (B/PHUKET/3073/2013) Hemagglutinin/HA0 Protein is expressed in Baculovirus insect cells. The predicted molecular weight is 61.7 kDa. | |||
TMPY-00951 |
Influenza A H5N1 (A/Anhui/1/2005) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H5N1 | HEK293 Cells |
Influenza A H5N1 (A/Anhui/1/2005) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 59 kDa and the accession number is Q1WDM0. | |||
TMPY-05922 |
Influenza B (B/Washington/02/2019) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
Influenza B | HEK293 Cells |
Influenza B (B/Washington/02/2019) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 58.6 kDa. | |||
TMPY-00954 |
Influenza A H1N1 (A/Brisbane/59/2007) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H1N1 | HEK293 Cells |
Influenza A H1N1 (A/Brisbane/59/2007) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 59 kDa and the accession number is B0VX44. | |||
TMPY-03937 |
Influenza A H3N2 (A/Hong Kong/1/1968) Hemagglutinin/HA Protein (aa 1-530, His)
Harvey rat sarcoma viral oncogene homolog |
H3N2 | Baculovirus Insect Cells |
Influenza A H3N2 (A/Hong Kong/1/1968) Hemagglutinin/HA Protein (aa 1-530, His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 59 kDa and the accession number is Q91MA7.1. | |||
TMPY-02524 |
Influenza B (B/Brisbane/60/2008) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
Influenza B | HEK293 Cells |
Influenza B (B/Brisbane/60/2008) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 60 kDa and the accession number is C0LT35. | |||
TMPY-05010 |
Influenza A H9N2 (A/Hong Kong/3239/2008) Hemagglutinin/HA1 Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H9N2 | HEK293 Cells |
Influenza A H9N2 (A/Hong Kong/3239/2008) Hemagglutinin/HA1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 37.2 kDa and the accession number is D3G601. | |||
TMPY-01491 |
Influenza A H1N1 (A/Puerto Rico/8/1934) Hemagglutinin Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H1N1 | HEK293 Cells |
Influenza A H1N1 (A/Puerto Rico/8/1934) Hemagglutinin Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 38 kDa and the accession number is P03452. | |||
TMPY-05566 |
Siglec-2/CD22 Protein, Human, Recombinant (His, Solution)
CD22 molecule,SIGLEC-2,SIGLEC2 |
Human | HEK293 Cells |
Siglec-2/CD22 Protein, Human, Recombinant (His, Solution) is expressed in HEK293 mammalian cells with His tag. The accession number is P20273-1. | |||
TMPY-01131 |
Influenza A H1N1 (A/California/04/2009) Hemagglutinin/HA1 Protein(His)
Harvey rat sarcoma viral oncogene homolog |
H1N1 | HEK293 Cells |
Influenza A H1N1 (A/California/04/2009) Hemagglutinin/HA1 Protein(His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 38 kDa and the accession number is C3W5S1. | |||
TMPY-00955 |
Influenza B (B/Florida/4/2006) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
Influenza B | HEK293 Cells |
Influenza B (B/Florida/4/2006) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 60 kDa and the accession number is B1AG46. | |||
TMPY-02662 |
Influenza A H10N8 (A/Jiangxi-Donghu/346/2013) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H10N8 | Baculovirus Insect Cells |
Influenza A H10N8 (A/Jiangxi-Donghu/346/2013) Hemagglutinin/HA Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 57.9 kDa. | |||
TMPY-04658 |
Influenza A H3N2 (A/Switzerland/9715293/2013) Hemagglutinin/HA0 Protein
Harvey rat sarcoma viral oncogene homolog |
H3N2 | Baculovirus Insect Cells |
Influenza A H3N2 (A/Switzerland/9715293/2013) Hemagglutinin/HA0 Protein is expressed in Baculovirus insect cells. The predicted molecular weight is 61.8 kDa. | |||
TMPY-04783 |
Influenza A H3N2 (A/Wuhan/359/1995) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H3N2 | Baculovirus Insect Cells |
Influenza A H3N2 (A/Wuhan/359/1995) Hemagglutinin/HA Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 59.2 kDa and the accession number is J9R649. | |||
TMPY-01301 |
Influenza A H9N2 (A/Hong Kong/1073/99) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H9N2 | HEK293 Cells |
Influenza A H9N2 (A/Hong Kong/1073/99) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 58 kDa and the accession number is Q9ICY5. | |||
TMPY-00278 |
Influenza A H3N2 (A/Victoria/361/2011) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H3N2 | Baculovirus Insect Cells |
Influenza A H3N2 (A/Victoria/361/2011) Hemagglutinin/HA Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 59.4 kDa and the accession number is L0HR89. | |||
TMPY-02612 |
Influenza A H3N2 (A/Perth/16/2009) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H3N2 | HEK293 Cells |
Influenza A H3N2 (A/Perth/16/2009) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 59 kDa and the accession number is C6KNH7. | |||
TMPY-04682 |
Influenza B (B/PHUKET/3073/2013) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
Influenza B | Baculovirus Insect Cells |
Influenza B (B/PHUKET/3073/2013) Hemagglutinin/HA Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 59.1 kDa. | |||
TMPY-00314 |
Influenza B (B/Yamagata/16/1988) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
Influenza B | Baculovirus Insect Cells |
Influenza B (B/Yamagata/16/1988) Hemagglutinin/HA Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 59 kDa. | |||
TMPY-03836 |
Influenza A H7N9 (A/Anhui/1/2013) Hemagglutinin/HA1 Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H7N9 | HEK293 Cells |
Influenza A H7N9 (A/Anhui/1/2013) Hemagglutinin/HA1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 36.2 kDa and the accession number is M9TFV7. | |||
TMPY-05920 |
Influenza A H3N2 (A/Kansas/14/2017) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H3N2 | HEK293 Cells |
Influenza A H3N2 (A/Kansas/14/2017) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 59 kDa and the accession number is A0A346MM15. | |||
TMPY-00956 |
Influenza A H1N1 (A/California/04/2009) Hemagglutinin/HA Protein ( (Native, HA1+HA2, uncleaved),His)
Harvey rat sarcoma viral oncogene homolog |
H1N1 | HEK293 Cells |
Influenza A H1N1 (A/California/04/2009) Hemagglutinin/HA Protein ( (Native, HA1+HA2, uncleaved),His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 59 kDa and the accession number is C3W5S1. | |||
TMPY-04090 |
Influenza A H7N9 (A/Shanghai/2/2013) Hemagglutinin/HA Protein (HEK293, His)
Harvey rat sarcoma viral oncogene homolog |
H7N9 | HEK293 Cells |
Influenza A H7N9 (A/Shanghai/2/2013) Hemagglutinin/HA Protein (HEK293, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 57.6 kDa. | |||
TMPY-00957 |
Influenza A H3N2 (A/Brisbane/10/2007) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H3N2 | HEK293 Cells |
Influenza A H3N2 (A/Brisbane/10/2007) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 59 kDa and the accession number is A8W8K8. | |||
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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TMIH-0067 |
Acalabrutinib Metabolite 27-d4
|
||
Acalabrutinib Metabolite 27-d4 是 Acalabrutinib Metabolite 27 的氘代化合物。 | |||
TMIH-0065 |
Acalabrutinib-d4
|
||
Acalabrutinib-d4 是 Acalabrutinib 的氘代化合物。Acalabrutinib 的 CAS 号为 1420477-60-6。Acalabrutinib 是一种不可逆的、高效的、具有口服活性、选择性的第二代BTK抑制剂。它与 BTK 的 ATP 结合口袋中的 Cys481 共价结合。它在慢性淋巴细胞性白血病 (CLL) 小鼠模型中显示出强大的靶向作用和功效。 | |||
TMIH-0610 |
Zanubrutinib-d5
|
||
Zanubrutinib-d5 是 Zanubrutinib 的氘代化合物。Zanubrutinib 的 CAS 号为 1691249-45-2。Zanubrutinib 是 Bruton tyrosine kinase(Btk) 的选择性抑制剂。 | |||
T11601 |
Ibrutinib-d5
PCI-32765 D5,Ibrutinib D5 |
Others | Others |
Ibrutinib D5 is a deuterium-labeled Ibrutinib. Ibrutinib is an irreversible Btk inhibitor. | |||
TMIH-0066 |
Acalabrutinib intermediate-d4
|
||
Acalabrutinib intermediate-d4 是 Acalabrutinib intermediate 的氘代化合物。Acalabrutinib intermediate 的 CAS 号为 1420478-90-5。 |