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Sodium Channel

Sodium Channel

Sodium channels are integral membrane proteins that form ion channels, conducting sodium ions (Na+) through a cell's plasma membrane.
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Cat. No. Product Name CAS No. Purity Chemical Structure
T3021 Bulleyaconitine A
草乌甲素
107668-79-1 98%
Bulleyaconi cine A 是一种分离自乌头属植物的抗炎活性化合物,也可用于缓解疼痛的研究。
T0037 Halazone
哈拉宗
80-13-7 98%
Halazone 是一种非典型的磺酰胺衍生物,有抗菌活性。它也是碳酸酐酶 II 抑制剂,Kd 值为 1.45 µM。它广泛用于饮用水消毒,可保护钠通道免于灭活。
TN3910 Ecdysone
蜕皮激素
3604-87-3 98%
Ecdysone 是存在于昆虫和草药中的主要类固醇激素,可以激活盐皮质激素受体并诱导细胞凋亡。Ecdysone 的活性代谢物 20-羟基蜕皮激素在协调发育过渡和体内稳态睡眠调节中起重要作用。
T6782 Benzocaine hydrochloride
化合物Benzocaine hydrochloride
23239-88-5 98%
Benzocaine hydrochloride 是一种表面麻醉剂,通过阻止脉冲沿神经纤维和神经末梢传递而起作用。
T3029 Sparteine sulfate
硫酸司巴丁
299-39-8 98%
Sparteine sulfate 是一种 1a 类抗心律失常药和钠通道阻滞剂。它可以螯合二价钙和镁。
TN3042 4-Hydroxycinnamamide
化合物 TN3042
194940-15-3 98%
4-Hydroxycinnamamide has antioxidant activity. 4-Hydroxycinnamamide derivatives are specific inhibitors of tyrosine-specific protein kinases.
T2173 Veratridine
藜芦定
71-62-5 98%
Veratridine 是一种生物碱,来自百合科植物。Veratridine 是一种钠通道激动剂, 对 Nav1.7 的峰值电流具有抑制作用,IC50为 18.39 µM。
TP1852 Myomodulin
肌调蛋白
110570-93-9 98%
Myomodulin 是一种存在于软体动物、昆虫和腹足类动物中的神经肽。它存在于两个已确定的海兔神经元中,它们包含肌调节蛋白 A、ARC 运动神经元 B16 和腹部神经元 L10。
TN4697 Odoroside H
化合物 TN4697
18810-25-8 98%
Odoroside H has anticancer activities, the cytotoxic effects are induced by the inhibition of the plasma membrane bound Na(+)/K(+)-ATPase.
TN5141 Thevetin B
黄夹甙 B
27127-79-3 98%
Thevetin B 是一种强心苷,是Na+-, K+-依赖性腺苷三磷酸酶 (Na+,K+-ATPase) 的抑制剂,来自 Thevetia peruviana。
TCA2511 11Beta-hydroxyprogesterone
11β-羟孕酮
600-57-7 98%
The progesterone derivatives 11 alpha- and 11 beta-hydroxyprogesterone are potent inhibitors of 11 beta-hydroxysteroid dehydrogenase (isoforms 1 and 2) in vitro ...
TN4276 Isocudraniaxanthone B
化合物 TN4276
199851-52-0 98%
Isocudraniaxanthone B may have antimalarial activity.
T12951 Sodium Channel inhibitor 2
化合物 T12951
653573-60-5 98%
Sodium Channel inhibitor 2 is a blocker of sodium channel.
TN5234 Vindorosine
化合物 TN5234
5231-60-7 98%
Vindorosine has blood vessel relaxation effect, possible underlying mechanisms involving the inhibition of Ca(2+) entry via L-type Ca(2+) channels in vascular sm...
T16887 Sipatrigine
化合物 T16887
130800-90-7 98%
Sipatrigine is a glutamate release inhibitor and voltage-dependent sodium channel.
TN2306 Wilfordine
雷公藤定碱
37239-51-3 98%
Wilfordine is an insecticidally active alkaloid, Na+-K+-ATPase may be an acting target of wilfordine against some larvae of insect.
TN5060 Stauntosaponin A
化合物 TN5060
1417887-91-2 98%
Stauntosaponin A and stauntosaponin B show moderate inhibitory activities against Na+/K+-ATPase with IC50 values of 21 and 29 uM, respectively.
TN4183 Hardwickiic acid
左旋哈氏豆属酸
1782-65-6 98%
Hardwickiic acid 是一种从Pulicaria gnaphalodes 中提取的天然化合物,是一种抗伤害性感受作用化合物。Hardwickiic acid 能阻断河豚毒素敏感的电压依赖性钠通道 (sodium channels)。Hardwickiic acid 具有抗炎和杀虫活性。
T16707 QX-314 bromide
化合物 T16707
24003-58-5 98%
QX-314 bromide is a blocker of the membrane-impermeable permanently charged sodium channel.
T13830 Propoxycaine hydrochloride
盐酸丙氧卡因
550-83-4 98%
Propoxycaine hydrochloride is an inhibit of voltage-gated sodium channels.
Bulleyaconitine A
T3021
Bulleyaconi cine A 是一种分离自乌头属植物的抗炎活性化合物,也可用于缓解疼痛的研究。
Halazone
T0037
Halazone 是一种非典型的磺酰胺衍生物,有抗菌活性。它也是碳酸酐酶 II 抑制剂,Kd 值为 1.45 µM。它广泛用于饮用水消毒,可保护钠通道免于灭活。
Ecdysone
TN3910
Ecdysone 是存在于昆虫和草药中的主要类固醇激素,可以激活盐皮质激素受体并诱导细胞凋亡。Ecdysone 的活性代谢物 20-羟基蜕皮激素在协调发育过渡和体内稳态睡眠调节中起重要作用。
Benzocaine hydrochloride
T6782
Benzocaine hydrochloride 是一种表面麻醉剂,通过阻止脉冲沿神经纤维和神经末梢传递而起作用。
Sparteine sulfate
T3029
Sparteine sulfate 是一种 1a 类抗心律失常药和钠通道阻滞剂。它可以螯合二价钙和镁。
4-Hydroxycinnamamide
TN3042
4-Hydroxycinnamamide has antioxidant activity. 4-Hydroxycinnamamide derivatives are specific inhibitors of tyrosine-specific protein kinases.
Veratridine
T2173
Veratridine 是一种生物碱,来自百合科植物。Veratridine 是一种钠通道激动剂, 对 Nav1.7 的峰值电流具有抑制作用,IC50为 18.39 µM。
Myomodulin
TP1852
Myomodulin 是一种存在于软体动物、昆虫和腹足类动物中的神经肽。它存在于两个已确定的海兔神经元中,它们包含肌调节蛋白 A、ARC 运动神经元 B16 和腹部神经元 L10。
Odoroside H
TN4697
Odoroside H has anticancer activities, the cytotoxic effects are induced by the inhibition of the plasma membrane bound Na(+)/K(+)-ATPase.
Thevetin B
TN5141
Thevetin B 是一种强心苷,是Na+-, K+-依赖性腺苷三磷酸酶 (Na+,K+-ATPase) 的抑制剂,来自 Thevetia peruviana。
11Beta-hydroxyprogesterone
TCA2511
The progesterone derivatives 11 alpha- and 11 beta-hydroxyprogesterone are potent inhibitors of 11 beta-hydroxysteroid dehydrogenase (isoforms 1 and 2) in vitro ...
Isocudraniaxanthone B
TN4276
Isocudraniaxanthone B may have antimalarial activity.
Sodium Channel inhibitor 2
T12951
Sodium Channel inhibitor 2 is a blocker of sodium channel.
Vindorosine
TN5234
Vindorosine has blood vessel relaxation effect, possible underlying mechanisms involving the inhibition of Ca(2+) entry via L-type Ca(2+) channels in vascular sm...
Sipatrigine
T16887
Sipatrigine is a glutamate release inhibitor and voltage-dependent sodium channel.
Wilfordine
TN2306
Wilfordine is an insecticidally active alkaloid, Na+-K+-ATPase may be an acting target of wilfordine against some larvae of insect.
Stauntosaponin A
TN5060
Stauntosaponin A and stauntosaponin B show moderate inhibitory activities against Na+/K+-ATPase with IC50 values of 21 and 29 uM, respectively.
Hardwickiic acid
TN4183
Hardwickiic acid 是一种从Pulicaria gnaphalodes 中提取的天然化合物,是一种抗伤害性感受作用化合物。Hardwickiic acid 能阻断河豚毒素敏感的电压依赖性钠通道 (sodium channels)。Hardwickiic acid 具有抗炎和杀虫活性。
QX-314 bromide
T16707
QX-314 bromide is a blocker of the membrane-impermeable permanently charged sodium channel.
Propoxycaine hydrochloride
T13830
Propoxycaine hydrochloride is an inhibit of voltage-gated sodium channels.
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