t82

T 82 is an antagonist of 5-HT3 and inhibitor of acetylcholinesterase (AChE) and used for the treatment of Alzheimer's Disease.

T-82 is an acetylcholinesterase inhibitor that may ameliorate the impairment of memory induced by acetylcholinergic dysfunction.

FT827 是选择性泛素特异性蛋白酶 7（USP7）共价抑制剂（Ki=4.2 µM，Kd=7.8 μM），靶向 USP7 的自抑制载脂蛋白形式的催化中心,可用于研究癌症。

OT-82 是一种具有口服活性、选择性和高效性的 NAMPT 抑制剂，具有抗癌活性和细胞毒性，可在携带 EWS 异种移植物的小鼠中损害了肿瘤生长并延长了存活时间。OT-82 可用于研究白血病。

15a-Hydroxy-3,11,23-trioxo-lanost-8,20-dien-26-oic acid is a Lanostane triterpenoid compound with the ability to inhibit NO production in LPS-induced microglia.

(3β,7β,12β,20Z)-3,7,12-Trihydroxy-11,15,23-trioxo-lanost-8,20-dien-26-oic acid, a lanostane triterpenoid, demonstrates significant inhibitory effects on nitric oxide (NO) production in BV-2 microglia cells induced by n LPS, with an IC50 value of 9.55 uM. Moreover, this compound possesses anti-inflammatory properties.

Antibacterial agent 82 (compound 7p) 是一种抗菌剂。

Anticancer agent 82 是 FiVe1 衍生物，是一种口服有效的选择性抗癌剂。FiVe1 能够结合 III 型中间丝蛋白vimentin(VIM)，诱导 Ser56 过度磷酸化，导致有丝分裂的选择性中断和转化表达 VIM 的间充质癌细胞的多核化。Anticancer agent 82 比 FiVe1 表现出更好的口服利用度和药代动力学特征。

Metofenazate difumarate is a selective calmodulin inhibitor.

Antitumor agent-82是一种有效的抗肿瘤剂。Antitumor agent-82 显示出抗增殖活性。Antitumor agent-82 通过 ATG5 ATG7信号通路诱导细胞自噬 (Autophagy)。

Antifungalagent 82 (compound G34)是一种高效的抗真菌剂，对Valsa mali具有显著的体外活性，其EC50值仅为0.57 μg mL。该化合物在40 mg L的浓度下，还能够有效地在体内保护植物免受V. mali的侵害。