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GluR

GluR

Glutamate receptors are synaptic and non synaptic receptors located primarily on the membranes of neuronal and glial cells.Glutamate receptors are responsible for the glutamate-mediated postsynaptic excitation of neural cells, and are important for neural communication, memory formation, learning, and regulation.
TargetMol
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Cat. No. Product Name CAS No. Purity Chemical Structure
T4009 NS 1209
化合物NS 1209
205645-02-9
TargetMol Chemical Structure NS 1209
NS 1209 (SPD 502) 是一种 AMPA 受体拮抗剂。
T15369 Gamma-DGG
化合物 T15369
6729-55-1 98%
TargetMol Chemical Structure gamma-DGG
gamma-DGG is a competitive blocker of AMPA receptor.
T11906 LY 541850
化合物 T11906
852679-76-6 98%
TargetMol Chemical Structure LY 541850
LY541850 is a selective orthosteric mGlu2 agonist and mGlu3 antagonist with IC50 values of 0.161 μM and 0.038 μM, respectively.LY 541850 is claimed from human io...
T15692 L-AP4
化合物 T15692
23052-81-5 98%
TargetMol Chemical Structure L-AP4
L-APB is an effective and specific agonist for the group III mGluRs (EC50s: 0.13, 0.29, 1.0, 249 μM for mGlu4, mGlu8, mGlu6, and mGlu7 receptors, respectively).
T11907 Pomaglumetad methionil anhydrous
化合物 T11907
635318-55-7 98%
TargetMol Chemical Structure Pomaglumetad methionil anhydrous
LY2140023 has the potential for schizophrenia.LY2140023 is an orally active prodrug of LY404039. LY404039 is a selective metabotropic glutamate 2/3 receptor agon...
T12520 Pomaglumetad methionil
化合物 T12520
956385-05-0 98%
TargetMol Chemical Structure Pomaglumetad methionil
Pomaglumetad methionil is an oral methionine prodrug of the potent specific agonist of mGlu2/3 receptor LY404039.
T12025 MFZ 10-7 hydrochloride
化合物 T12025
1779796-36-9 98%
TargetMol Chemical Structure MFZ 10-7 hydrochloride
MFZ 10-7 hydrochloride is a highly potent and selective negative allosteric modulator of mGluR5 NAM
T11911 LY3020371 hydrochloride
化合物 T11911
1377615-44-5 98%
TargetMol Chemical Structure LY3020371 hydrochloride
LY3020371 hydrochloride exerts an antidepressant-like signature in vivo. LY3020371 hydrochloride is a potent, selective metabotropic glutamate 2/3 receptor (mGlu...
T21935 AMN082
化合物AMN 082 dihydrochloride
97075-46-2 98%
TargetMol Chemical Structure AMN082
AMN082 (AMN 082 dihydrochloride) 是可口服,可透过血脑屏障的选择性mGluR7激动剂,通过跨膜区的变构位点直接激活受体信号,具有抗抑郁作用。
T13319 VU0652835
化合物 T13319
1848252-81-2 98%
TargetMol Chemical Structure VU0652835
VU0652835 is a negative allosteric modulator of metabotropic glutamate receptor subtype 5 (mGlu5) (IC50: 81 nM).
T15618 JNJ-46281222
化合物 T15618
1254980-38-5 98%
TargetMol Chemical Structure JNJ-46281222
JNJ-46281222 is an metabotropic glutamate (mGlu) 2-selective, highly potent PAM (positive allosteric modulator). It has nanomolar affinity (Kd = 1.7 nM) and a hi...
T11311L Foliglurax
化合物 T11311L
1883329-51-8 98%
TargetMol Chemical Structure Foliglurax
Foliglurax is a highly selective brain-penetrant metabotropic glutamate receptor 4 positive allosteric modulator (mGluR4 PAM) (EC50: 79 nM).
T15823 LYPLAL1-IN-1
化合物 T15823
1966129-74-7 98%
TargetMol Chemical Structure LYPLAL1-IN-1
LYPLAL1-IN-1 is a selective covalent small-molecule inhibitor of Lysophospholipase-like 1 (IC50: 0.006 μM). LYPLAL1-IN-1 also enhances glucose production.
T12118 MSOP
化合物 T12118
66515-29-5 98%
TargetMol Chemical Structure MSOP
MSOP is a selective antagonist of group III metabotropic glutamate receptor (KD of 51 μM for the L-AP4-sensitive presynaptic mGluR).
T17248 VU6001376
化合物 T17248
1968546-34-0 98%
TargetMol Chemical Structure VU6001376
VU6001376 is an effective and selective positive allosteric modulator of the metabotropic glutamate receptor 4 (EC50: 50.1 nM).
T38789 BMS-984923
化合物 BMS-984923
1375752-78-5 98%
TargetMol Chemical Structure BMS-984923
BMS-984923 是可口服且具有血脑屏障透过性的 mGluR5 沉默异构调节剂,抑制β-淀粉样蛋白寡聚体诱导的异常突触信号传导,可用于研究阿尔茨海默症。
TQ0114 CMPDA
化合物CMPDA
380607-77-2 98%
TargetMol Chemical Structure CMPDA
CMPDA is a positive allosteric modulator of AMPA receptors (EC50s: 45.4 nM/63.4 nM for GluA2i/GluA2o receptor).
T14615 Biphenylindanone A
化合物 T14615
866823-73-6 98%
TargetMol Chemical Structure Biphenylindanone A
Biphenylindanone A is a selective potentiator of human mGluR2 (hmGluR2),and for the treatment of neurological disorders.
T23288 (S)-3,4-DCPG
化合物(S)-3,4-DCPG
201730-11-2 98%
TargetMol Chemical Structure (S)-3,4-DCPG
(S)-3,4-DCPG ((S)-3,4-Dicarboxyphenylglycine) 是人代谢型谷氨酸受体 8a (mGluR8a) 的选择性激动剂。
T6725 VU 0357121
化合物VU 0357121
433967-28-3 99.99%
TargetMol Chemical Structure VU 0357121
VU 0357121 是一种高选择性的mGlu5R 正变构调节剂 ,EC50为 33 nM。
NS 1209
T4009
NS 1209 (SPD 502) 是一种 AMPA 受体拮抗剂。
gamma-DGG
T15369
gamma-DGG is a competitive blocker of AMPA receptor.
LY 541850
T11906
LY541850 is a selective orthosteric mGlu2 agonist and mGlu3 antagonist with IC50 values of 0.161 μM and 0.038 μM, respectively.LY 541850 is claimed from human io...
L-AP4
T15692
L-APB is an effective and specific agonist for the group III mGluRs (EC50s: 0.13, 0.29, 1.0, 249 μM for mGlu4, mGlu8, mGlu6, and mGlu7 receptors, respectively).
Pomaglumetad methionil anhydrous
T11907
LY2140023 has the potential for schizophrenia.LY2140023 is an orally active prodrug of LY404039. LY404039 is a selective metabotropic glutamate 2/3 receptor agon...
Pomaglumetad methionil
T12520
Pomaglumetad methionil is an oral methionine prodrug of the potent specific agonist of mGlu2/3 receptor LY404039.
MFZ 10-7 hydrochloride
T12025
MFZ 10-7 hydrochloride is a highly potent and selective negative allosteric modulator of mGluR5 NAM
LY3020371 hydrochloride
T11911
LY3020371 hydrochloride exerts an antidepressant-like signature in vivo. LY3020371 hydrochloride is a potent, selective metabotropic glutamate 2/3 receptor (mGlu...
AMN082
T21935
AMN082 (AMN 082 dihydrochloride) 是可口服,可透过血脑屏障的选择性mGluR7激动剂,通过跨膜区的变构位点直接激活受体信号,具有抗抑郁作用。
VU0652835
T13319
VU0652835 is a negative allosteric modulator of metabotropic glutamate receptor subtype 5 (mGlu5) (IC50: 81 nM).
JNJ-46281222
T15618
JNJ-46281222 is an metabotropic glutamate (mGlu) 2-selective, highly potent PAM (positive allosteric modulator). It has nanomolar affinity (Kd = 1.7 nM) and a hi...
Foliglurax
T11311L
Foliglurax is a highly selective brain-penetrant metabotropic glutamate receptor 4 positive allosteric modulator (mGluR4 PAM) (EC50: 79 nM).
LYPLAL1-IN-1
T15823
LYPLAL1-IN-1 is a selective covalent small-molecule inhibitor of Lysophospholipase-like 1 (IC50: 0.006 μM). LYPLAL1-IN-1 also enhances glucose production.
MSOP
T12118
MSOP is a selective antagonist of group III metabotropic glutamate receptor (KD of 51 μM for the L-AP4-sensitive presynaptic mGluR).
VU6001376
T17248
VU6001376 is an effective and selective positive allosteric modulator of the metabotropic glutamate receptor 4 (EC50: 50.1 nM).
BMS-984923
T38789
BMS-984923 是可口服且具有血脑屏障透过性的 mGluR5 沉默异构调节剂,抑制β-淀粉样蛋白寡聚体诱导的异常突触信号传导,可用于研究阿尔茨海默症。
CMPDA
TQ0114
CMPDA is a positive allosteric modulator of AMPA receptors (EC50s: 45.4 nM/63.4 nM for GluA2i/GluA2o receptor).
Biphenylindanone A
T14615
Biphenylindanone A is a selective potentiator of human mGluR2 (hmGluR2),and for the treatment of neurological disorders.
(S)-3,4-DCPG
T23288
(S)-3,4-DCPG ((S)-3,4-Dicarboxyphenylglycine) 是人代谢型谷氨酸受体 8a (mGluR8a) 的选择性激动剂。
VU 0357121
T6725
VU 0357121 是一种高选择性的mGlu5R 正变构调节剂 ,EC50为 33 nM。
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