Cat. No. | Product Name | CAS No. | Purity | Chemical Structure |
---|---|---|---|---|
T14123 | ACT 178882
化合物 T14123
|
1007392-69-9 | 98% |
|
ACT 178882 is a new Renin inhibitor (IC50: 1.4 nM). | ||||
T16544 | Pivalopril
化合物 T16544
|
81045-50-3 | 98% |
|
Pivalopril is a new orally active inhibitor of angiotensin-converting enzyme. | ||||
T11809 | L162441
化合物 T11809
|
154512-46-6 | 98% |
|
L162441 is an antagonist of Angiotensin type 1 receptor. | ||||
T10323 | Angiotensin II (3-8), human TFA
化合物 T10323
|
T10323 | 98% |
|
Angiotensin II (3-8), human (TFA) is an angiotensin AT1 receptor agonist with less activity. | ||||
T16573 | Pratosartan
化合物 T16573
|
153804-05-8 | 98% |
|
Pratosartan is a selective antagonist of angiotensin II receptor. | ||||
T19187 | Aliskiren D6 hemifumarate
化合物 T19187
|
T19187 | 98% |
|
Aliskiren (CGP 60536) D6 hemifumarate is a deuterium-labeled Aliskiren hemifumarate. Aliskiren hemifumarate is a direct and orally active renin inhibitor (IC50: ... | ||||
T16385 | Omapatrilat
化合物 T16385
|
167305-00-2 | 98% |
|
Omapatrilat is a metalloprotease ACE and NEP dual inhibitor (Ki: 0.64 and 0.45 nM, respectively). | ||||
T6444 | Cilazapril Monohydrate
西拉普利水合物
|
92077-78-6 | 98% |
|
Cilazapril Monohydrate (Justor) 是一种血管紧张素转化酶抑制剂,能够作用于高血压和充血性心力衰竭的研究。 | ||||
T11808 | L162389
化合物 T11808
|
169281-53-2 | 98% |
|
L162389 is a potent angiotensin AT1 receptor antagonist with Ki of 28 nM. | ||||
T7616 | A 779
化合物A 779(3TFA)
|
159432-28-7 | 98% |
|
A 779 是一种 G 蛋白偶联受体 Mas 的有效拮抗剂,Mas 受体是Ang1-7 receptor,与传统的AngII 不同。 | ||||
T12704 | Rentiapril
化合物 T12704
|
80830-42-8 | 98% |
|
Rentiapril is an orally active inhibitor of angiotensin converting enzyme (ACE), with antihypertensive activity. | ||||
TN4431 | Leucosceptoside A
米团花苷A
|
83529-62-8 | 98% |
|
Leucosceptoside A shows inhibitory activity against PKCalpha with the IC50 value of 19.0 microM; it also exhibits strong inhibitory capacity against α-glucosidas... | ||||
TN1464 | Camellianin A
山茶黄酮苷 A
|
109232-77-1 | 98% |
|
Camellianin A has anticancer activity, it can inhibit the proliferation of the human hepatocellular liver carcinoma Hep G2 and human breast adenocarcinoma MCF-7 ... | ||||
T5824 | Angiotensin II (3-8), human
化合物Angiotensin IV
|
12676-15-2 | 98% |
|
Angiotensin II (3-8), human 是活性稍弱的血管紧张素AT1受体激动剂。 | ||||
T6627 | Phosphoramidon Disodium
磷酰胺二钠
|
164204-38-0 | 98% |
|
Phosphoramidon Disodium (Phosphoramidon Disodium Salt) Salt 是一种金属蛋白酶 (metalloprotease) 抑制剂 。Phosphoramidon Disodium Salt 抑制内皮素转化酶 (ECE) ,中性肽内切酶 (NEP) 和血管紧张素转换酶 (... | ||||
T11642 | Imidaprilate
化合物 T11642
|
89371-44-8 | 98% |
|
Imidaprilate is an active metabolite of TA-6366, acts as a potent angiotensin-converting enzyme (ACE) inhibitor (IC50: 2.6 nM). It is used in the research of the... | ||||
T7575 | [Sar1, Ile8]-Angiotensin II
化合物[Sar1, Ile8]-Angiotensin II(3TFA)
|
37827-06-8 | 98% |
|
[Sar1, Ile8]-Angiotensin II 是一种在血管平滑肌细胞中有多种作用(如正常动脉的收缩,培养的细胞或病变血管的肥大或增生等)的多肽,。 | ||||
T2318 | Sacubitril/Valsartan
沙库必曲/缬沙坦
|
936623-90-4 | 99.94% |
|
Sacubitril/Valsartan (LCZ696) 是由 Valsartan (an ARB) 和 Sacubitril (AHU377) 组成,摩尔比为 1:1,是一种首创的,口服有效的血管紧张素受体-脑啡肽酶 (ARN) 双抑制剂,用于研究高血压和心力衰竭。它可通过抑制炎症、氧化应激和细胞凋亡来改善糖尿性心肌... | ||||
T6542 | Imidapril hydrochloride
盐酸咪达普利
|
89396-94-1 | 99.94% |
|
Imidapril hydrochloride (Tanapril) 是一种血管紧张素转换酶 (ACE) 抑制剂,具有抗高血压活性。 | ||||
T3753 | Sinapinic Acid
芥子酸
|
530-59-6 | 99.92% |
|
Sinapinic Acid (Synapoic acid) 是从 Hydnophytum formicarumJack. 根中分离到的酚类,是HDAC 抑制剂,对ACE-I 的活性也有抑制作用。它有抗肿瘤活性,诱导肿瘤细胞凋亡,具有抗氧化、抗糖尿病的作用。 |