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Targets Recommended: FLT

218

抑制剂 & 化合物

3

天然产物

1

TargetMol 试剂盒

14

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Cat. No. Product Name Form Specificity Of Inhibition
CL0094 FLT3 inhibitor kit

FLT3 inhibitor kit

TargetMol 试剂盒

FLT3 inhibitor kit
Cat.No: CL0094
Cat. No. Product Name Target Signaling Pathways
T11299 FLT3-IN-4

FLT3 inhibitor 9u

FLT Angiogenesis; Tyrosine Kinase/Adaptors
FLT3-IN-4 (FLT3 inhibitor 9u) 是一种口服有效的 Fms 样酪氨酸受体激酶 3 (FLT3; IC50= 7 nM) 抑制剂,可用于急性髓性白血病的研究。
T27011 CHMFL-FLT3-122

CHMFLFLT3122,CHMFL FLT3 122

FLT Angiogenesis; Tyrosine Kinase/Adaptors
CHMFL-FLT3-122 是一种强效口服 FLT3 激酶抑制剂,用于治疗 FLT3-ITD 阳性急性髓性白血病。CHMFL-FLT3-122能显著抑制 MV4-11细胞异种移植模型(50 mg/kg)的肿瘤生长,且在体内无明显毒性。
T1938 FLT3-IN-2

FLT Angiogenesis; Tyrosine Kinase/Adaptors
FLT3-IN-2 是 FLT3 抑制剂(IC50<1 μM)。
T9843 FLT3-IN-16

FLT3-IN-16 是一种有效的FLT3酪氨酸激酶抑制剂,其IC50值为 1.1 μM。FLT3-IN-16 可用于研究急性髓系白血病。
T11298 FLT3-IN-3

FLT Angiogenesis; Tyrosine Kinase/Adaptors
FLT3-IN-3FLT3抑制剂,能够抑制 FLT3 WT (IC50:13 nM) 和 FLT3 D835Y (IC50:8 nM) 。
T9856 FLT3-IN-10

2-Oxazolamine, 5-(4-fluorophenyl)-N-phenyl-

FLT Angiogenesis; Tyrosine Kinase/Adaptors
FLT3-IN-10 (2-Oxazolamine, 5-(4-fluorophenyl)-N-phenyl-) (compound 7c) 是有效的 FMS 样酪氨酸激酶 3 (FLT3) 抑制剂。FLT3-IN-10 具有治疗 FLT3 突变的急性髓性白血病 (AML) 的潜力。
T2051 SKLB4771

FLT3-​IN-​1,FLT3-IN-1

FLT Angiogenesis; Tyrosine Kinase/Adaptors
SKLB4771 (FLT3-IN-1) 是一种新型的、高效的 Flt3 抑制剂 (IC50:10nM)。
T6138 TCS 359

FLT3 Inhibitor

FLT Angiogenesis; Tyrosine Kinase/Adaptors
TCS 359 (FLT3 Inhibitor) 是 2-酰基氨基噻吩-3-甲酰胺,是选择性FLT3抑制剂(IC50:42 nM),能够抑制 MV4-11 细胞增殖(IC50:340 nM)。
T24067 Flt3 Inhibitor IV

Flt3 Inhibitor-IV,Flt3-IN-IV

Flt3 Inhibitor IV is a potent ATP-competitive Flt3 inhibitor.
T11300 FLT3-IN-6

Others Others
FLT3-IN-6 is a potent and selective inhibitor of FLT3-ITD (FLT3 mutation) with an IC50 of 1.336 nM.
T11707 JAK2/FLT3-IN-1

JNK MAPK
JAK2/FLT3-IN-1 has anti-cancer activity. JAK2/FLT3-IN-1 is a potent and orally effective dual JAK2/FLT3 (Janus kinase 2/ FMS-like tyrosine kinase 3) inhibitor with IC50 values of 0.7 nM, 4 nM, 26 nM and 39 nM for JAK2, FLT3, JAK1 and JAK3, respectively.
T24438 MDK5466

MDK-5466,MDK 5466,E21,Flt3-IN-III,Flt3 Inhibitor III

MDK5466 is an Flt3 inhibitor that acts by preventing glutamate-induced cell death.
T62824 FLT3/ITD-IN-3

FLT3/ITD-IN-3 (Compound 19) 是一种 FLT3-ITD 的有效抑制剂,能够作用于 FLT3D835Y (IC50: 0.3 nM)、FLT3 (IC50: 0.4 nM) 和 FLT3-ITD (IC50: 0.9 nM)。 FLT3/ITD-IN-3FLT3 的磷酸化显示出有效抑制作用,能够有效抗急性髓系白血病细胞的增殖。
T61415 FLT3/ITD-IN-1

FLT3/ITD-IN-1 (Compound 1) is a highly potent inhibitor of FLT3 internal tandem duplications (FLT3-ITD). It exhibits remarkable inhibitory effects against FLT3 and FLT3-ITD, with impressive IC50 values of 38.2 nM and 144.1 nM, respectively. Moreover, FLT3/ITD-IN-1 shows exceptional antiproliferative activities against several acute myeloid leukemia cell lines [1].
T82392 FLT3-IN-23

FLT3-IN-23作为JFMS样脂氨酸激酶3(FLT3)的抑制剂,表现出7.42 nM的IC50值。该化合物针对带有多种FLT3-TKD与FLT3-ITD-TKD突变的BaF3细胞显示出显著的抗增殖效果。
T82393 FLT3/CHK1-IN-1

FLT3/CHK-IN-1(Compound 18)为FLT3/CHK1双重抑制剂,其对c-KIT的选择性超1700倍,同时显著降低对hERG的亲和力,IC50为58.4 μM。在MV-4-11细胞接种小鼠异种移植模型中有效抑制肿瘤生长。
T63058 FLT3-IN-14

FLT3-IN-14 是一种 FLT3 的有效抑制剂,能够作用于 FLT3-WT (IC50: 5.6 nM) 和 FLT3-ITD (IC50: 1.4 nM)。FLT3-IN-14 能够抑制 FLT3 (Y591) 磷酸化,将细胞周期停滞在 G1 期并诱导细胞凋亡。
T62607 FLT3-IN-15

FLT3-IN-15 是一种口服具有活力的、有效的 FLT3 抑制剂,能够作用于 FLT3 (IC50: 0.87 nM) 和 FLT3/D835Y (IC50: 0.32 nM)。FLT3-IN-15 能够用于急性髓系白血病的研究。
T63174 FLT3-IN-17

FLT3-IN-17 是一种 FAK 抑制剂 (IC50: 12 nM)。FLT3-IN-17 能够抑制 CYPs 和 FLT3 突变体的活性,对 D835Y 的 IC50<0.5 nM。FLT3-IN-17 能够用于癌症的研究。
T62801 FLT3/TrKA-IN-1

FLT3/TrKA-IN-1 是一种有效的 FLT3/TrKA 双激酶抑制剂,能够作用于 FLT3 (IC50: 43.8 nM)、FLT3-ITD (IC50: 97.2 nM)、FLT3-TKD (IC50: 92.5 nM) 和 TrKA (IC50: 23.6 nM)。FLT3/TrKA-IN-1 能够将细胞周期阻滞在 G0/G1 期,并诱导细胞凋亡 (apoptosis),具有抗增殖作用。FLT3/TrKA-IN-1 具有潜力进行急性髓性白血病 (AML) 的研究。
T62863 FLT3/ITD-IN-4

FLT3/ITD-IN-4 (Compound 16) 是一种选择性的 FLT3 内部串联重复突变 (FLT3-ITD) 抑制剂 (IC50: 2.3 nM)。FLT3/ITD-IN-4 能够用于研究急性骨髓性白血病。
T63274 FLT3/ITD-IN-2

FLT3/ITD-IN-2 是 FLT3-ITD 的有效抑制剂,能够作用于 FLT3D835Y (IC50: 0.3 nM)、FLT3(IC50: 0.4 nM)和 FLT3-ITD(IC50: 1.0 nM)。FLT3/ITD-IN-2 能够有效的抑制 FLT3 的磷酸化,能够有效的抑制急性髓系白血病细胞的增殖。
T61977 FLT3/D835Y-IN-1

FLT3/D835Y-IN-1 (化合物13a) 是一种选择性的、口服活性的FLT3FLT3/D835Y 抑制剂,IC50分别为 0.26 nM 和 0.18 nM。FLT3/D835Y-IN-1 具有抗癌作用,可以用于急性髓系白血病的研究。
T63135 FLT3/CDK4-IN-1

FLT3/CDK4-IN-1 是一种高度选择性的、有效的、口服具有活力的 FLT3/CDK4 双重抑制剂,作用于 FLT3 (IC50: 7 nM) 与 CDK4 (IC50: 11 nM)。FLT3/CDK4-IN-1 在体内具有良好的抗肿瘤效果,对某些癌细胞表现出抗增殖作用。
T62260 FLT3-IN-11

FLT3-IN-11 (compound 30) 是一种口服具活力的、有效的、具有选择性的 FLT3 激酶抑制剂,能够作用于野生型 FLT3 (IC50: 7.22 nM) 和 FLT3-D835Y (IC50: 4.95 nM)。FLT3-IN-11 对 FLT3 的选择性比 c-KIT 高>1000 倍。FLT3-IN-11 表现出显著的抗急性髓性白血病 (AML) 作用,对 MV4-11 细胞的 IC50 值为 3.2 nM。
T61101 FLT3-IN-13

FLT3-IN-13 (compound 20) is a highly effective inhibitor targeting both topoisomerase II and FLT3 proteins in leukemic cells. It exhibits potent activity against these targets, with IC50 values of 2.26 μM for both. Moreover, FLT3-IN-13 induces cell cycle arrest at the G2/M phase and promotes apoptosis. Notably, it displays considerable anticytotoxic activity, specifically against leukemia [1].
T79596 FLT3-IN-20

FLT3-IN-20(compound 34f)作为一种高效FLT3抑制剂,对FLT3-D835Y和FLT3-ITD具有强效性,IC50值分别仅为1 nM和4 nM。该化合物在携带FLT3-ITD突变的AML细胞系MV4-11和MOLM-13中展现出显著的抗增殖效果,其中IC50值分别为7 nM和9 nM;对于带有FLT3-ITD-D835Y突变的MOLM-13变体,其IC50值为4 nM。FLT3-IN-20主要用于肿瘤治疗研究领域。
T79391 FLT3-IN-21

FLT3-IN-21(复合物LC-3)是一种高效的FLT3抑制剂,具有促进细胞凋亡的能力,其对FLT3酶的半抑制浓度(IC50)为8.4 nM。该化合物能够使细胞周期在G1期停滞,并对FLT3-ITD阳性的AML细胞系MV-4-11显示出显著的抑制作用(IC50:5.3 nM)。在小鼠体内,FLT3-IN-21以每日10 mg/kg的剂量可以有效抑制MV-4-11细胞异种移植瘤的生长,肿瘤生长抑制率(TGI)达到92.16%。
T62412 FLT3-IN-12

FLT3-IN-12 是一种选择性的、有效的、口服具有活力的 FLT3 激酶抑制剂,能够作用于 FLT3-WT (IC50: 1.48 nM) 和 FLT3-D835Y (IC50: 2.87 nM)。FLT3-IN-12 选择性比 c-KIT 高 (>1000 倍)。FLT3-IN-12 表现出显著的抗急性髓性白血病效果,对 MV4-11 细胞 的 IC50 值为 0.75 nM。
T79420 FLT3-IN-22

FLT3-IN-22(化合物22f)是一款高效的FLT3抑制剂,具有针对FLT3FLT3/D835Y极低的IC50值,分别为0.941 nM和0.199 nM。在MV4-11细胞和携带FLT3变异的Ba/F3细胞系中(涵盖FLT3-D835Y及FLT3-F691L),此抑制剂显示出显著的抗增殖能力。
T78176 FLT3-IN-19

FLT3-IN-19(Comp 50),作为一种选择性FLT3抑制剂,展现出0.213 nM的IC50。适用于AML研究。
T73142 FLT3-IN-18

FLT3-IN-18是一种高效且选择性的FLT3抑制剂,具有0.003 μM的IC50值。该化合物能够诱导(apoptosis)并使细胞周期在G1期停滞,同时抑制FLT3和STAT5的磷酸化,显示出对急性髓系白血病(AML)研究的潜力。
T38562 AKN-028

FLT Angiogenesis; Tyrosine Kinase/Adaptors
AKN-028 是酪氨酸激酶 FLT3的抑制剂,可剂量依赖性的诱导 FLT3的自磷酸化。
T74707 PROTAC FLT3/CDK9 degrader-1

PROTACFLT3/CDK9 degrader-1 是一种有效的FLT3和CDK9双PROTAC 降解剂。PROTACFLT3/CDK9 degrader-1 诱导细胞凋亡 (Apoptosis) 并有效降解靶蛋白FLT3和 CDK9。PROTACFLT3/CDK9 degrader-1具有研究 FLT3-ITD 突变型 AML 的潜力。
T64104 JAK2/FLT3-IN-1 TFA

JAK2/FLT3-IN-1 (TFA) 是一种口服具有活力的 JAK2/FLT3 双重抑制剂,表现出抗癌效果,能够作用于 JAK2 (IC50: 0.7 nM),FLT3 (IC50: 4 nM),JAK1 (IC50: 26 nM) 和 JAK3 (IC50: 39 nM)。
T63629 PDGFRα/FLT3-ITD-IN-2

PDGFRα/FLT3-ITD-IN-2 是 PDGFRα (IC50>20 μM) 和 FLT3 (IC50: 0.004 μM) 的有效抑制剂。PDGFRα/FLT3-ITD-IN-2 对急性髓系白血病或慢性嗜酸性粒细胞白血病表现出研究潜力。
T63454 PDGFRα/FLT3-ITD-IN-1

PDGFRα/FLT3-ITD-IN-1 是 PDGFRα/FLT3 的有效抑制剂,他们的 IC50 值分别大于 0.036 和 0.003 μM。 PDGFRα/FLT3-ITD-IN-1 对急性髓系白血病或慢性嗜酸性粒细胞白血病表现出研究潜力。
T2340 AC1NS4RE

Tyrosinase Proteases/Proteasome
是一种化学合成中的砌块
T63127 PDGFRα/FLT3-ITD-IN-3

PDGFRα/FLT3-ITD-IN-3 (Compound 18d) 是一种有效的 PDGFRα (IC50: 0.153 μM)、FLT3 (IC50: 0.004 μM) 抑制剂。PDGFRα/FLT3-ITD-IN-3 具有潜力进行急性髓系白血病或慢性嗜酸性粒细胞白血病的研究。
T2066 Quizartinib

AC220,奎扎替尼

Apoptosis; FLT; Autophagy; Ligands for Target Protein for PROTAC Angiogenesis; Apoptosis; Autophagy; PROTAC; Tyrosine Kinase/Adaptors
Quizartinib (AC220) 是一种具有口服活性的高选择性Ⅱ 型 FLT3酪氨酸激酶抑制剂,可诱导细胞凋亡。它抑制 Wt FLT3 和 突变型 FLT3-ITD 自磷酸化,IC50分别为 4.1 nM 和 1.1 nM。它可通过优化的 linker 与 VHL 配体连接,从而形成 PROTAC Flt3 降解剂。
T15335 FN-1501

FLT; CDK Angiogenesis; Cell Cycle/Checkpoint; Tyrosine Kinase/Adaptors
FN-1501 是一种有效的 FLT3 和 CDK 抑制剂,具有抗肿瘤的活性,对 CDK2/cyclin A、CDK4/cyclin D1、CDK6/cyclin D1 和 FLT3 的 IC50值分别为 2.47、0.85、1.96 和 0.28 nM。
T4428 CCT241736

FLT; Aurora Kinase Angiogenesis; Cell Cycle/Checkpoint; Chromatin/Epigenetic; Tyrosine Kinase/Adaptors
CCT241736 是一种口服生物可利用的双重 FLT3/Aurora 激酶抑制剂,还抑制临床相关的 FLT3 耐药突变体,包括 FLT3-ITD 和 FLT3。它是 CCT137690 的高级类似物,是治疗人类恶性肿瘤的临床前开发候选物。
T2272 BPR1J-097

BPR1J097

FLT Angiogenesis; Tyrosine Kinase/Adaptors
BPR1-J097 是新型的、强效的FLT3抑制剂 (IC50:11 nM)。
T6756 AMG 925

FLT; CDK Angiogenesis; Cell Cycle/Checkpoint; Tyrosine Kinase/Adaptors
AMG 925 是一种选择性FLT3/CDK4双重抑制剂,IC50分别为 1 nM 和 3 nM。
T9473 4SC-203

FLT Angiogenesis; Tyrosine Kinase/Adaptors
4SC-203 是一种具有潜在的抗肿瘤活性的多激酶抑制剂。它对 FLT3/STK1、 FLT3 的突变形式以及 VEGFRs 具有选择性抑制作用。
T1667 Tandutinib

MLN518,CT53518,NSC726292,坦度替尼

Apoptosis; FLT; CSF-1R; PDGFR; Src; c-Kit Angiogenesis; Apoptosis; Tyrosine Kinase/Adaptors
Tandutinib (CT53518) 是一种选择性 FLT3抑制剂,其 IC50为 0.22 μM。它还抑制c-Kit 和PDGFR,其IC50分别为 0.17 μM 和 0.20 μM。它可穿透血脑屏障,用于急性骨髓性白血病。
T6020 Pacritinib

SB1518

FLT; Tyrosine Kinases; JAK Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells; Tyrosine Kinase/Adaptors
Pacritinib (SB1518) 是一种野生型 JAK2和 JAK2V617F 突变型抑制剂,IC50分别为 23 和 19 nM。它也抑制 FLT3及其突变型 FLT3D835Y,IC50分别为 22 和 6 nM。
T3065 TG101209

Apoptosis; FLT; c-RET; JAK; Autophagy Angiogenesis; Apoptosis; Autophagy; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells; Tyrosine Kinase/Adaptors
TG101209 是一种选择性有效的 JAK2抑制剂,IC50值为 6 nM。它能抑制 Flt3和RET 的活性,IC50值分别为 25 nM 和 17 nM。
T7673 ATH686

ATH 686

Apoptosis; FLT Angiogenesis; Apoptosis; Tyrosine Kinase/Adaptors
ATH686 是一种选择性的,ATP 竞争性的FLT3抑制剂,具有抗白血病作用。它靶向突变 FLT3 蛋白激酶活性,并通过诱导凋亡和抑制细胞周期来抑制具有 FLT3 突变的细胞的增殖。
T8317 5'-Fluoroindirubinoxime

5'-FIO

FLT Angiogenesis; Tyrosine Kinase/Adaptors
5'-Fluoroindirubinoxime (5'-FIO) 是一种 Indirubin 的衍生物,是一种 FLT3 的抑制剂(IC50:15 nM)。

化合物

FLT3-IN-4
Cat.No: T11299
Synonym: FLT3 inhibitor 9u
Target: FLT
CHMFL-FLT3-122
Cat.No: T27011
Synonym: CHMFLFLT3122,CHMFL FLT3 122
Target: FLT
FLT3-IN-2
Cat.No: T1938
Synonym:
Target: FLT
FLT3-IN-16
Cat.No: T9843
Synonym:
Target:
FLT3-IN-3
Cat.No: T11298
Synonym:
Target: FLT
FLT3-IN-10
Cat.No: T9856
Synonym: 2-Oxazolamine, 5-(4-fluorophenyl)-N-phenyl-
Target: FLT
SKLB4771
Cat.No: T2051
Synonym: FLT3-​IN-​1,FLT3-IN-1
Target: FLT
TCS 359
Cat.No: T6138
Synonym: FLT3 Inhibitor
Target: FLT
Flt3 Inhibitor IV
Cat.No: T24067
Synonym: Flt3 Inhibitor-IV,Flt3-IN-IV
Target:
FLT3-IN-6
Cat.No: T11300
Synonym:
Target: Others
JAK2/FLT3-IN-1
Cat.No: T11707
Synonym:
Target: JNK
MDK5466
Cat.No: T24438
Synonym: MDK-5466,MDK 5466,E21,Flt3-IN-III,Flt3 Inhibitor III
Target:
FLT3/ITD-IN-3
Cat.No: T62824
Synonym:
Target:
FLT3/ITD-IN-1
Cat.No: T61415
Synonym:
Target:
FLT3-IN-23
Cat.No: T82392
Synonym:
Target:
FLT3/CHK1-IN-1
Cat.No: T82393
Synonym:
Target:
FLT3-IN-14
Cat.No: T63058
Synonym:
Target:
FLT3-IN-15
Cat.No: T62607
Synonym:
Target:
FLT3-IN-17
Cat.No: T63174
Synonym:
Target:
FLT3/TrKA-IN-1
Cat.No: T62801
Synonym:
Target:
FLT3/ITD-IN-4
Cat.No: T62863
Synonym:
Target:
FLT3/ITD-IN-2
Cat.No: T63274
Synonym:
Target:
FLT3/D835Y-IN-1
Cat.No: T61977
Synonym:
Target:
FLT3/CDK4-IN-1
Cat.No: T63135
Synonym:
Target:
FLT3-IN-11
Cat.No: T62260
Synonym:
Target:
FLT3-IN-13
Cat.No: T61101
Synonym:
Target:
FLT3-IN-20
Cat.No: T79596
Synonym:
Target:
FLT3-IN-21
Cat.No: T79391
Synonym:
Target:
FLT3-IN-12
Cat.No: T62412
Synonym:
Target:
FLT3-IN-22
Cat.No: T79420
Synonym:
Target:
FLT3-IN-19
Cat.No: T78176
Synonym:
Target:
FLT3-IN-18
Cat.No: T73142
Synonym:
Target:
AKN-028
Cat.No: T38562
Synonym:
Target: FLT
PROTAC FLT3/CDK9 degrader-1
Cat.No: T74707
Synonym:
Target:
JAK2/FLT3-IN-1 TFA
Cat.No: T64104
Synonym:
Target:
PDGFRα/FLT3-ITD-IN-2
Cat.No: T63629
Synonym:
Target:
PDGFRα/FLT3-ITD-IN-1
Cat.No: T63454
Synonym:
Target:
AC1NS4RE
Cat.No: T2340
Synonym:
Target: Tyrosinase
PDGFRα/FLT3-ITD-IN-3
Cat.No: T63127
Synonym:
Target:
Quizartinib
Cat.No: T2066
Synonym: AC220,奎扎替尼
Target: Apoptosis, FLT, Autophagy, Ligands for Target Protein for PROTAC
FN-1501
Cat.No: T15335
Synonym:
Target: FLT, CDK
CCT241736
Cat.No: T4428
Synonym:
Target: FLT, Aurora Kinase
BPR1J-097
Cat.No: T2272
Synonym: BPR1J097
Target: FLT
AMG 925
Cat.No: T6756
Synonym:
Target: FLT, CDK
4SC-203
Cat.No: T9473
Synonym:
Target: FLT
Tandutinib
Cat.No: T1667
Synonym: MLN518,CT53518,NSC726292,坦度替尼
Target: Apoptosis, FLT, CSF-1R, PDGFR, Src, c-Kit
Pacritinib
Cat.No: T6020
Synonym: SB1518
Target: FLT, Tyrosine Kinases, JAK
TG101209
Cat.No: T3065
Synonym:
Target: Apoptosis, FLT, c-RET, JAK, Autophagy
ATH686
Cat.No: T7673
Synonym: ATH 686
Target: Apoptosis, FLT
5'-Fluoroindirubinoxime
Cat.No: T8317
Synonym: 5'-FIO
Target: FLT
Cat. No. Product Name Target Signaling Pathways
T6S0033 Crotonoside

巴豆苷;异鸟苷,巴豆苷,Isoguanosine,2-HYDROXYADENOSINE

Others; FLT; HDAC Angiogenesis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Others; Tyrosine Kinase/Adaptors
Crotonoside (Isoguanosine) 是从中草药巴豆中分离出来的一种天然产物。 它抑制 FLT3 和 HDAC3/6,有治疗急性髓性白血病 (AML)的研究潜力。
T14055 5Z-7-Oxozeaenol

FR148083,L783279,LL-Z 1640-2

VEGFR; FLT; MEK; MAPK; PDGFR; Antibiotic; Src Angiogenesis; MAPK; Microbiology/Virology; Tyrosine Kinase/Adaptors
5Z-7-Oxozeaenol (FR148083) 是一种天然抗原生动物抑制剂,不可逆的选择性抑制 TAK1和 VEGF-R2,IC50值分别为 8 nM 和 52 nM。
T15542 Hypothemycin

Others Others
Hypothemycin is a fungal polyketide and is a multikinase inhibitor (Kis: 10/70 nM, 17/38 nM, 90 nM, 900 nM/1.5 μM, and 8.4/2.4 μM for VEGFR2/VEGFR1, MEK1/MEK2, FLT-3, PDGFRβ/PDGFRα, and ERK1/ERK2, respectively).

天然产物

Crotonoside
Cat.No: T6S0033
Synonym: 巴豆苷;异鸟苷,巴豆苷,Isoguanosine,2-HYDROXYADENOSINE
Target: Others, FLT, HDAC
5Z-7-Oxozeaenol
Cat.No: T14055
Synonym: FR148083,L783279,LL-Z 1640-2
Target: VEGFR, FLT, MEK, MAPK, PDGFR, Antibiotic, Src
Hypothemycin
Cat.No: T15542
Synonym:
Target: Others
Cat. No. Product Name Species Expression System
TMPK-00125 FLT3 Ligand Protein, Human, Recombinant (hFc)

FLT3LG,FL,Flt3 ligand,SL...

Human HEK293 Cells
Flt3 Ligand, also known as FL, is an alpha -helical cytokine that promotes the differentiation of multiple hematopoietic cell lineages.Stimulates the proliferation of early hematopoietic cells by activating FLT3. Synergizes well with a number of other colony stimulating factors and interleukins. FLT3 Ligand Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with C-hFc tag. The predicted molecular weight is 44.8 kDa and the accession number is P49771-1.
TMPK-00929 FLT3 Protein, Mouse, Recombinant (hFc)

FL,FLT3LG,Flt3L,SL cytok...

Mouse HEK293 Cells
Flt3 Ligand, also known as FL, is an alpha -helical cytokine that promotes the differentiation of multiple hematopoietic cell lineages.Stimulates the proliferation of early hematopoietic cells by activating FLT3. Synergizes well with a number of other colony stimulating factors and interleukins. FLT3 Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with C-hFc tag. The predicted molecular weight is 84.78 kDa and the accession number is Q00342.
TMPY-06873 FLT3 Ligand Protein, Human, Recombinant

FLT3LG,fms related tyrosine kinase 3

Human E. coli
FLT3 Ligand Protein, Human, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 17.75 kDa and the accession number is P49771-1.
TMPY-03066 FLT3 Ligand Protein, Mouse, Recombinant (hFc)

Ly72L,Flt3lg,fms related tyrosine kinase <...

Mouse HEK293 Cells
FLT3 Ligand Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 45.4 kDa and the accession number is P49772-1.
TMPY-03215 FLT3 Ligand Protein, Human, Recombinant (His)

fms related tyrosine kinase 3 ligand,FLT

Human Baculovirus Insect Cells
FLT3 Ligand Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 20.2 kDa and the accession number is P49771-1.
TMPY-01247 FLT3 Protein, Human, Recombinant (T227M, His)

FLK2,FLK-2,CD135,STK1,fms-related tyrosine kinase <...

Human HEK293 Cells
FLT3 Protein, Human, Recombinant (T227M, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 59.7 kDa and the accession number is P36888-1.
TMPK-00523 FLT3 Protein, Cynomolgus, Recombinant (hFc)

FLT-3,FLK2,STK-1,CD135

Cynomolgus HEK293 Cells
FLT3 Protein, Cynomolgus, Recombinant (hFc) is expressed in HEK293 mammalian cells with C-hFc tag. The predicted molecular weight is 84.58 kDa and the accession number is A0A2K5VQ48.
TMPK-00416 FLT3 Protein, Human, Recombinant (His & Avi), Biotinylated

STK-1,FLK2,CD135,FLT-3

Human CHO Cells
FLT3 Protein, Human, Recombinant (His & Avi), Biotinylated is expressed in CHO mammalian cells with C-His-Avi tag. The predicted molecular weight is 61.20 kDa and the accession number is P36888-1.
TMPY-05738 FLT3 Protein, Human, Recombinant (hFc)

FLK2,CD135,fms-related tyrosine kinase 3,F...

Human HEK293 Cells
FLT3 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 85.06 kDa and the accession number is P36888-1.
TMPJ-00123 FLT3LG Protein, Mouse, Recombinant (His)

Fms-related tyrosine kinase 3 ligand (Flt<...

Mouse HEK293 Cells
Fms-related tyrosine kinase 3 ligand(Flt3L) is a single-pass type I membrane protein and consists of 232 amino acids. Flt3L is a hematopoietic four helical bundle cytokine, structurally homologous to stem cell factor and colony stimulating factor. Flt3L synergizes well with a number of other colony stimulating factors and interleukins. Flt3L stimulates the proliferation and differentiation of various blood cell progentiors by activating FLT3.
TMPY-03704 FLT3 Protein, Mouse, Recombinant (His)

wmfl,Flk-2,Flk2,Flt-3,CD135,B2

Mouse HEK293 Cells
FLT3 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 69.4 kDa and the accession number is EDL05832.1.
TMPY-05332 FLT3 Ligand Protein, Rat, Recombinant (His)

fms related tyrosine kinase 3 ligand

Rat Baculovirus Insect Cells
FLT3 Ligand Protein, Rat, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 19.7 kDa and the accession number is NP_001292868.1.
TMPY-06938 FLT3 Protein, Human, Recombinant (hFc & Avi), Biotinylated

fms-related tyrosine kinase 3,CD135,STK1,F...

Human HEK293 Cells
FLT3 Protein, Human, Recombinant (hFc & Avi), Biotinylated is expressed in HEK293 mammalian cells with hFc and Avi tag. The predicted molecular weight is 86.87 kDa and the accession number is NP_004110.2.
TMPY-02842 UBE2L6 Protein, Human, Recombinant (His)

UBCH8,ubiquitin-conjugating enzyme E2L 6,RIG-B

Human E. coli
UBCH8, also known as UBE2L6, belongs to the ubiquitin-conjugating enzyme family. The family of ubiquitin-conjugating (E2) enzymes is characterized by the presence of a highly conserved ubiquitin-conjugating (UBC) domain. These domains accommodate the ATP-activated ubiquitin (Ub) or ubiquitin-like (UBL) protein via a covalently linked thioester onto its active-site residue. E2 enzymes act via selective protein-protein interactions with the E1 and E3 enzymes and connect activation to covalent modi...

重组蛋白

FLT3 Ligand Protein, Human, Recombinant (hFc)
Cat.No: TMPK-00125
Species: Human
Expression System: HEK293 Cells
FLT3 Protein, Mouse, Recombinant (hFc)
Cat.No: TMPK-00929
Species: Mouse
Expression System: HEK293 Cells
FLT3 Ligand Protein, Human, Recombinant
Cat.No: TMPY-06873
Species: Human
Expression System: E. coli
FLT3 Ligand Protein, Mouse, Recombinant (hFc)
Cat.No: TMPY-03066
Species: Mouse
Expression System: HEK293 Cells
FLT3 Ligand Protein, Human, Recombinant (His)
Cat.No: TMPY-03215
Species: Human
Expression System: Baculovirus Insect Cells
FLT3 Protein, Human, Recombinant (T227M, His)
Cat.No: TMPY-01247
Species: Human
Expression System: HEK293 Cells
FLT3 Protein, Cynomolgus, Recombinant (hFc)
Cat.No: TMPK-00523
Species: Cynomolgus
Expression System: HEK293 Cells
FLT3 Protein, Human, Recombinant (His & Avi), Biotinylated
Cat.No: TMPK-00416
Species: Human
Expression System: CHO Cells
FLT3 Protein, Human, Recombinant (hFc)
Cat.No: TMPY-05738
Species: Human
Expression System: HEK293 Cells
FLT3LG Protein, Mouse, Recombinant (His)
Cat.No: TMPJ-00123
Species: Mouse
Expression System: HEK293 Cells
FLT3 Protein, Mouse, Recombinant (His)
Cat.No: TMPY-03704
Species: Mouse
Expression System: HEK293 Cells
FLT3 Ligand Protein, Rat, Recombinant (His)
Cat.No: TMPY-05332
Species: Rat
Expression System: Baculovirus Insect Cells
FLT3 Protein, Human, Recombinant (hFc & Avi), Biotinylated
Cat.No: TMPY-06938
Species: Human
Expression System: HEK293 Cells
UBE2L6 Protein, Human, Recombinant (His)
Cat.No: TMPY-02842
Species: Human
Expression System: E. coli
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