Cat. No. | Product Name | CAS No. | Purity | Chemical Structure |
---|---|---|---|---|
TQ0141 | Taltobulin
他托布林
|
228266-40-8 | 99.54% |
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Taltobulin (HTI-286) 是一种三肽半胱氨酸的合成类似物,是一种微管蛋白抑制剂,在体外抑制肝肿瘤细胞增殖和体内肿瘤生长。Taltobulin 具有细胞毒性,诱导有丝分裂停滞以及凋亡 (apoptosis),可用于研究乳腺癌和与微管组织相关的疾病。 | ||||
T13807 | OSIP-486823
化合物OSIP-486823
|
200803-37-8 | 98.59% |
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OSIP-486823(CP248) 是一种新型有效的微管干扰剂,对蛋白激酶 G (PKG) 和微管均具有亲和力。 | ||||
T36848 | Combretastatin A-1
康普瑞汀A-1
|
109971-63-3 | 97.49% |
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Combretastatin A-1 是一种有效的微管抑制剂,具有抗肿瘤和抗血管活性,通过微管蛋白解聚介导的 AKT 失活抑制 Wnt/β-catenin 通路发挥作用,可用于研究肝癌。 | ||||
T16997 | Tasidotin hydrochloride
化合物 T16997
|
623174-20-9 | 98% |
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Tasidotin hydrochloride is a peptide analog of the antimitotic depsipeptide dolastatin 15. Tasidotin hydrochloride is an inhibitor of microtubule assembly and mi... | ||||
T17229 | Verubulin
化合物 T17229
|
827031-83-4 | 98% |
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Verubulin is a microtubule-disrupting agent with potent and broad-spectrum in vitro and in vivo cytotoxic activities. | ||||
T6721 | Vinblastine
长春质碱
|
865-21-4 | 98% |
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Vinblastine 抑制微管形成并抑制 nAChR 活性,IC50 为 8.9 μM,用于治疗某些类型的癌症。 | ||||
TQ0112 | Tubulysin A
化合物Tubulysin A
|
205304-86-5 | 98% |
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Tubulysin A is a natural product from myxobacterial. It has many function in vitro assays, including anti-microtubule, anti-mitotic, an apoptosis inducer, antica... | ||||
T13227 | Tubulin inhibitor 1
化合物 T13227
|
2237054-53-2 | 98% |
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Tubulin inhibitor 1 is an inhibitor of tubulin, inhibits tubulin polymerization, with potent anti-tumor activity, induces cellular apoptosis causes and cellular ... | ||||
T10428 | AZ82
化合物 AZ82
|
1449578-65-7 | 98% |
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AZ82 是一种具有选择性和高效性的驱动蛋白样蛋白 KIFC1 抑制剂,抑制 PCa 细胞胞质和细胞核中 KIFC1 的表达,诱导前列腺癌细胞多极有丝分裂和细胞凋亡。 | ||||
T11712 | Jasplakinolide
肌动蛋白多聚化肽
|
102396-24-7 | 98% |
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Jasplakinolide(Jaspamide) 是一种来自海洋海绵 (marine sponge) 的天然环状肽,是一种有效的肌动蛋白聚合反应 (actin polymerization) 诱导剂。Jasplakinolide 具有抗真菌和抗肿瘤活性,可以稳定先前存在的肌动蛋白丝。Jasplakinolide 与鬼笔... | ||||
T12805 | S-methyl DM1
化合物 T12805
|
912569-84-7 | 98% |
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S-methyl DM1 is a thiomethyl derivative of Maytansine. S-methyl DM1 binds to tubulin(Kd of 0.93 μM) and inhibts microtubule polymerization. | ||||
T12052 | Mivobulin
化合物 T12052
|
122332-18-7 | 98% |
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Mivobulin is an inhibitor of tubulin . | ||||
T13901 | SS28
化合物 T13901
|
141172-08-9 | 98% |
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SS28 inhibits tubulin polymerization to cause cell cycle arrest at G2/M phase. | ||||
T16543 | Pironetin
化合物 T16543
|
151519-02-7 | 98% |
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Pironetin binds to α-tubulin and is an effective inhibitor of microtubule polymerization. It also has cell cycle arrest and antitumor activity. Pironetin is an α... | ||||
T6722 | Vinflunine Tartrate
长春氟宁酒石酸盐
|
1201898-17-0 | 98% |
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Vinflunine Tartrate 是一种独特的新型长春花生物碱,具有抑制有丝分裂和微管蛋白相互作用活性的特性。 | ||||
T16387 | Ombrabulin
化合物 T16387
|
181816-48-8 | 98% |
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Ombrabulin is a derivative of CA-4 phosphate. It is known to show antivascular effects through selective disruption of the tubulin cytoskeleton of endothelial ce... | ||||
T12823 | S516
化合物 T12823
|
1016543-77-3 | 98% |
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S516 is an active CKD-516 metabolite and is a potent inhibitor of tubulin polymerization(IC50 of 4.29 μM), has marked antitumor activity. | ||||
TQ0202 | Epothilone D
埃博霉素
|
189453-10-9 | 98% |
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Epothilone D (KOS 862) is an effective microtubule stabilizer. | ||||
T16386 | Ombrabulin hydrochloride
化合物 T16386
|
253426-24-3 | 98% |
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Ombrabulin hydrochloride 是一种合成的、具有选择性的 CA-4 磷酸酯或 Ombrabulin 的衍生物,能破坏内皮细胞的微管蛋白细胞骨架,具有抗血管作用。Ombrabulin 是是一种微管蛋白聚合抑制剂,是 combretastatin a -4化合物类的一员,是一种水溶性的微管蛋白解聚肿瘤血管... | ||||
T13225 | Tubulin inhibitor 7
化合物 T13225
|
1309925-41-4 | 98% |
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Tubulin inhibitor 7 is an inhibitor of tubulin and a potent inhibitor of multiple cancer cell lines (tubulin polymerization (IC50: 0.52 μM), K562 cell growth (IC... |