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细胞凋亡化合物库

细胞凋亡化合物库

产品编号 L9000 Apoptosis Compound Library
  库化合物信息   Excel SDF

细胞凋亡是一种发生在多细胞生物中的程序性细胞死亡。相对于细胞坏死,细胞凋亡是受基因调控的主动过程,细胞凋亡时会发生特征性的形态学变化,产生称为凋亡小体的细胞碎片被吞噬细胞吞噬。细胞凋亡受到促凋亡因子(Fas 受体和 caspases)和抑凋亡因子(Bcl-2蛋白和 IAP)的调控,异常凋亡过程牵涉到多种疾病中,细胞凋亡的抑制可导致癌症、自身免疫性疾病、炎性疾病和病毒感染。另一方面,过度的细胞凋亡可能导致神经退行性疾病、血液疾病和组织损伤。目前在细胞凋亡与癌症发生和自身免疫性疾病之间的关系有着很多研究,人们希望激发癌细胞的细胞凋亡,以达到治疗癌症的目的。“细胞凋亡在神经退化性疾病中所扮演的角色(如阿兹海默氏症、亨丁顿舞蹈症、帕金森病、肌肉萎缩性侧索硬化症),是目前热门的研究领域。” TargetMol 细胞凋亡化合物库精选 1796 种与凋亡相关的生物活性小分子化合物,适用于癌症和神经退行性疾病相关研究。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
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产品描述

  • 1796种与凋亡相关的生物活性小分子化合物的特有集合,多用于研究肿瘤发生发展机制和抗癌药物筛选等。可用于高通量筛选和高内涵筛选;
  • 靶点含Bcl-2、Caspase、p53、TNF-α和survivin等;
  • 通过前期临床研究和临床实验,生物活性和安全性已经得到验证;
  • 其中一些活性化合物已得到FDA批准上市;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR和HPLC检测技术保证产品高纯度和高质量;
  • 所有化合物现货供应。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L9000)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

Apoptosis (1016)
Autophagy (369)
Endogenous Metabolite (114)
Ferroptosis (100)
NF-κB (93)
Antibacterial (89)
TNF (85)
EGFR (75)
Caspase (66)
BCL (59)
Reactive Oxygen Species (55)
JAK (54)
COX (50)
STAT (50)
DNA/RNA Synthesis (49)
p38 MAPK (48)
CDK (48)
ERK (48)
VEGFR (47)
Raf (46)
PI3K (44)
Antibiotic (42)
FLT (38)
Mitophagy (37)
HDAC (37)
HIV Protease (36)
Src (36)
PDGFR (34)
Antifungal (34)
Akt (34)
Parasite (34)
MEK (33)
p53 (32)
c-Kit (31)
c-RET (30)
Microtubule Associated (30)
mTOR (29)
Influenza Virus (28)
IL Receptor (28)
JNK (28)
FGFR (27)
Epigenetic Reader Domain (26)
Antioxidant (26)
E1/E2/E3 Enzyme (26)
Dehydrogenase (25)
Bcr-Abl (23)
HSP (22)
AMPK (22)
Aurora Kinase (22)
PARP (21)
Ras (21)
PKC (21)
PPAR (20)
Topoisomerase (20)
Nucleoside Antimetabolite/Analog (19)
Proteasome (19)
Interleukin (19)
RIP kinase (18)
Tyrosine Kinases (18)
Mdm2 (18)
HER (17)
AChR (16)
Virus Protease (16)
Mitochondrial Metabolism (16)
Histone Methyltransferase (16)
Phosphatase (16)
PERK (16)
MAPK (15)
Serine/threonin kinase (15)
Sirtuin (15)
c-Met/HGFR (14)
P450 (14)
IκB/IKK (14)
ROS (14)
NO Synthase (13)
GSK-3 (13)
DNA Alkylator/Crosslinker (13)
MMP (13)
Potassium Channel (12)
RAAS (12)
IAP (12)
HSV (12)
Lipoxygenase (12)
Calcium Channel (12)
Estrogen Receptor/ERR (11)
Estrogen/progestogen Receptor (11)
c-Myc (11)
ATPase (11)
Tyrosinase (11)
Wnt/beta-catenin (11)
PKA (11)
TRP/TRPV Channel (11)
IGF-1R (10)
PD-1/PD-L1 (10)
PDE (10)
DNA-PK (10)
Dopamine Receptor (10)
FAK (10)
Gamma-secretase (9)
Beta Amyloid (9)
Pim (9)
Chk (9)
DUB (9)
Histamine Receptor (9)
Sodium Channel (9)
Syk (9)
TAM Receptor (9)
Retinoid Receptor (9)
Phospholipase (8)
Nrf2 (8)
SARS-CoV (8)
AChE (8)
TGF-beta/Smad (8)
PLK (8)
Trk receptor (8)
TLR (8)
5-HT Receptor (8)
Drug Metabolite (8)
c-Fms (8)
Fatty Acid Synthase (8)
DNA Alkylation (7)
NADPH (7)
Reverse Transcriptase (7)
Casein Kinase (7)
Adrenergic Receptor (7)
HIF/HIF Prolyl-Hydroxylase (7)
HBV (7)
GPR (7)
PDK (7)
HMG-CoA Reductase (7)
HIF (7)
HCV Protease (7)
P-gp (7)
Histone Acetyltransferase (6)
S6 Kinase (6)
Antifolate (6)
BTK (6)
Kinesin (6)
CaMK (6)
Cysteine Protease (6)
ALK (6)
Prostaglandin Receptor (6)
NOS (5)
GluR (5)
Glutathione Peroxidase (5)
MAO (5)
UGT (5)
Monoamine Oxidase (5)
ROCK (5)
S1P Receptor (5)
Anti-infection (5)
Rho (5)
Opioid Receptor (5)
Integrin (5)
DHFR (4)
Serine Protease (4)
ASK (4)
Aryl Hydrocarbon Receptor (4)
PTEN (4)
ROR (4)
ATM/ATR (4)
DPP-4 (4)
DNA Methyltransferase (4)
OXPHOS (4)
PAK (4)
MRP (4)
CSF-1R (4)
iGluR (4)
Antiviral (4)
Histone Demethylase (4)
MLK (4)
Telomerase (4)
GABA Receptor (4)
Transferase (4)
Proton pump (3)
IRE1 (3)
TOPK (3)
PAI-1 (3)
CRISPR/Cas9 (3)
Adenosine Receptor (3)
Pyroptosis (3)
IFNAR (3)
DNA (3)
Acyltransferase (3)
PGE Synthase (3)
Hexokinase (3)
GPX (3)
MNK (3)
Leukotriene Receptor (3)
STING (3)
FXR (3)
NADPH-oxidase (3)
NAMPT (3)
Glucocorticoid Receptor (3)
Glucokinase (3)
NOD-like Receptor (NLR) (3)
LTR (3)
Survivin (3)
Lipid (3)
Reductase (3)
Progesterone Receptor (2)
Antifection (2)
BACE (2)
BMI-1 (2)
Aromatase (2)
VDA (2)
VDAC (2)
cAMP (2)
Aminopeptidase (2)
Xanthine Oxidase (2)
Smo (2)
SGK (2)
Androgen Receptor (2)
YAP (2)
CRM1 (2)
Immunology/Inflammation related (2)
LRRK2 (2)
LPL Receptor (2)
Myosin (2)
Liver X Receptor (2)
FLAP (2)
NOD (2)
IRAK (2)
P2 Receptor (2)
P2X Receptor (2)
Free radical scavengers (2)
PAFR (2)
Hck (2)
Hedgehog/Smoothened (2)
PAD (2)
KSP (1)
Arginase (1)
lysosomal autophagy (1)
Stearoyl-CoA Desaturase (SCD) (1)
ACK (1)
Wee1 (1)
Hydrogenase (1)
Glutathione reductase (1)
Lipase (1)
Adenosine deaminase (1)
Guanylate cyclase (1)
Thrombin (1)
Indoleamine 2,3-Dioxygenase (IDO) (1)
Tie-2 (1)
KLF (1)
GNRH Receptor (1)
Amino Acids and Derivatives (1)
Somatostatin (1)
transporter (1)
GTPase (1)
IDO (1)
AhR (1)
GST (1)
Sigma receptor (1)
Melatonin Receptor (1)
OCT (1)
cholecystokinin (1)
PKM (1)
Chloride channel (1)
CFTR (1)
CXCR (1)
p97 (1)
Dynamin (1)
Endothelin Receptor (1)
PYK2 (1)
Ephrin Receptor (1)
Carbonic Anhydrase (1)
RAR/RXR  (1)
Epoxide Hydrolase (1)
FAAH (1)
MTH1 (1)
Fas/FasL (1)
NPC1L1 (1)
Beta-Secretase (1)
Norepinephrine (1)
NMDAR (1)
RSV (1)
Neurokinin receptor (1)
Neprilysin (1)
Na+/Ca2+ Exchanger (1)
FOXO1 (1)
SGLT (1)
PI4K (1)
SIK (1)
Hippo pathway (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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