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TargetMol | Compound Library

细胞凋亡化合物库现货

Apoptosis Compound Library

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产品编号 L9000

细胞凋亡是一种发生在多细胞生物中的程序性细胞死亡。相对于细胞坏死,细胞凋亡是受基因调控的主动过程,细胞凋亡时会发生特征性的形态学变化,产生称为凋亡小体的细胞碎片被吞噬细胞吞噬。细胞凋亡受到促凋亡因子(Fas 受体和 caspases)和抑凋亡因子(Bcl-2蛋白和 IAP)的调控,异常凋亡过程牵涉到多种疾病中,细胞凋亡的抑制可导致癌症、自身免疫性疾病、炎性疾病和病毒感染。另一方面,过度的细胞凋亡可能导致神经退行性疾病、血液疾病和组织损伤。目前在细胞凋亡与癌症发生和自身免疫性疾病之间的关系有着很多研究,人们希望激发癌细胞的细胞凋亡,以达到治疗癌症的目的。“细胞凋亡在神经退化性疾病中所扮演的角色(如阿兹海默氏症、亨丁顿舞蹈症、帕金森病、肌肉萎缩性侧索硬化症),是目前热门的研究领域。” TargetMol 细胞凋亡化合物库精选 2394 种与凋亡相关的生物活性小分子化合物,适用于癌症和神经退行性疾病相关研究。

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产品编号 L9000

细胞凋亡化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 2394种与凋亡相关的生物活性小分子化合物的特有集合,多用于研究肿瘤发生发展机制和抗癌药物筛选等。可用于高通量筛选和高内涵筛选;
  • 靶点含Bcl-2、Caspase、p53、TNF-α和survivin等;
  • 通过前期临床研究和临床实验,生物活性和安全性已经得到验证;
  • 其中一些活性化合物已得到FDA批准上市;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR和HPLC检测技术保证产品高纯度和高质量;
  • 所有化合物现货供应。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Apoptosis
Autophagy
Endogenous Metabolite
EGFR
TNF
NF-κB
Antibacterial
Caspase
Ferroptosis
Bcl-2 Family
Reactive Oxygen Species
JAK
Akt
STAT
MDM-2/p53
CDK
p38 MAPK
PI3K
COX
ERK
DNA/RNA Synthesis
Ras
VEGFR
Parasite
p53
Antibiotic
Raf
Antioxidant
IL Receptor
Microtubule Associated
Antifungal
Interleukin
HDAC
FLT
Src
JNK
RIP kinase
mTOR
PARP
AMPK
c-RET
MEK
HIV Protease
PERK
Mitophagy
PDGFR
MAPK
FGFR
E1/E2/E3 Enzyme
c-Kit
Dehydrogenase
Nucleoside Antimetabolite/Analog
Tyrosine Kinases
Aurora Kinase
Epigenetic Reader Domain
HSP
Nrf2
Influenza Virus
Mdm2
PPAR
Topoisomerase
Bcr-Abl
ROS
Cytochromes P450
NO Synthase
c-Met/HGFR
Virus Protease
PKC
Mitochondrial Metabolism
Phosphatase
GSK-3
Wnt/beta-catenin
Potassium Channel
PD-1/PD-L1
Proteasome
Pim
IAP
MMP
Histone Methyltransferase
Sirtuin
HER
Calcium Channel
IκB/IKK
HSV
Lipoxygenase
IGF-1R
FAK
HIF/HIF Prolyl-Hydroxylase
PDE
SARS-CoV
Anti-infection
Estrogen Receptor/ERR
Molecular Glues
TGF-beta/Smad
ATPase
DNA-PK
Estrogen/progestogen Receptor
DNA Alkylator/Crosslinker
RAAS
PKA
Chk
DUB
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Beta Amyloid
Kras
AChR
Syk
S6 Kinase
PROTACs
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Necroptosis
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TLR
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Bcl-6
TRP/TRPV Channel
Adrenergic Receptor
Gamma-secretase
Drug Metabolite
Antiviral
Prostaglandin Receptor
ALK
Casein Kinase
PDK
Phospholipase
5-HT Receptor
HMG-CoA Reductase
Dopamine Receptor
Histamine Receptor
OXPHOS
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Pyroptosis
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c-Fms
HIF
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ASK
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HBV
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PTEN
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MAO
Immunology/Inflammation related
iGluR
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DAPK
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Opioid Receptor
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Angiotensin-converting Enzyme (ACE)
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ADC Cytotoxin
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IFNAR
DYRK
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FXR
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CSF-1R
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PAK
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transporter
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Liver X Receptor
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PYK2
NR4A
Aryl Hydrocarbon Receptor
IDO
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P2X Receptor
BTK
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OCT
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NAMPT
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NMDAR
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PAD
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STING
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PKM
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