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NF-κB 通路分子库

NF-κB 通路分子库

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产品编号 L3800 NF-κB Signaling Compound Library
  库化合物信息   Excel SDF

NF-κB 为一个转录因子蛋白家族,包括5个亚单位,两个亚单位形成的同源或异源二聚体与靶基因上特定的序列结合调节基因转录,不同的 NF-κB 二聚体在选择结合序列时可能略有差异,这是 NF-κB 通过不同的二聚体形式对不同基因的表达进行精细调节的一种方式。在静息的细胞中,NF-κB 和 IκB 形成复合体,以无活性形式存在于胞浆中。当细胞受细胞外信号刺激后,IκB 激酶(IκB kinase, IKK)将 IκB 磷酸化,使NF-κB 暴露核定位位点。游离的NF-κB 迅速移位到细胞核,与特异性序列结合,诱导相关基因转录。参与免疫反应的早期和炎症反应各阶段的许多分子都受NF-κB 的调控,包括:TNF-α、IL-1β、IL-2、IL-6、IL-8、IL-12、趋化因子、粘附分子、集落刺激因子等。此外,与细胞凋亡有关的分子如:肿瘤坏死因子受体相关因子-1(TRAF-1),抗细胞凋亡的蛋白-1和-2(IAP1/ IAP2),TNF 受体相关因子(TRAF)也都受NF-κB 的调控。

TargetMol NF-κB 信号通路分子库是由740 个NF-κB 信号通路相关的小分子化合物组成的独特集合,用于NF-κB 信号通路相关的研究及药物的筛选,可用于高通量、高内涵筛选。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
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产品描述

  • 740 个NF-κB信号通路相关的小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 是NF-κB信号通路研究及相关药物筛选的有效工具;??
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L3800)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

NF-κB (232)
Reactive Oxygen Species (163)
Apoptosis (142)
HDAC (109)
Autophagy (91)
TNF (83)
Endogenous Metabolite (64)
ROS (52)
Antibacterial (46)
Nrf2 (46)
COX (42)
IκB/IKK (40)
IL Receptor (34)
RIP kinase (27)
p38 MAPK (24)
ERK (24)
NOD (23)
Ferroptosis (21)
Antioxidant (20)
NO Synthase (20)
HIV Protease (19)
IRAK (18)
JNK (16)
Antifungal (15)
Influenza Virus (15)
STAT (14)
NOD-like Receptor (NLR) (13)
Akt (13)
ROS Kinase (11)
Antibiotic (11)
Mitophagy (10)
PPAR (10)
NOS (10)
P450 (10)
Calcium Channel (9)
Caspase (9)
Interleukin (9)
Parasite (9)
Mitochondrial Metabolism (9)
Lipoxygenase (8)
EGFR (8)
Virus Protease (8)
PDE (8)
MMP (8)
HIF/HIF Prolyl-Hydroxylase (7)
p53 (7)
TLR (7)
ALK (7)
PI3K (7)
Tyrosinase (7)
DNA/RNA Synthesis (7)
CDK (7)
GABA Receptor (6)
Beta Amyloid (6)
MAPK (6)
Topoisomerase (6)
Sodium Channel (6)
JAK (6)
Estrogen/progestogen Receptor (6)
Potassium Channel (5)
AChE (5)
Xanthine Oxidase (5)
AMPK (5)
Dehydrogenase (5)
AChR (5)
Wnt/beta-catenin (4)
MALT (4)
BCL (4)
c-Met/HGFR (4)
E1/E2/E3 Enzyme (4)
Proteasome (4)
HSP (3)
S6 Kinase (3)
Antifection (3)
IGF-1R (3)
5-HT Receptor (3)
Prostaglandin Receptor (3)
PKC (3)
SARS-CoV (3)
Ligand for E3 Ligase (3)
MAO (3)
Opioid Receptor (3)
MEK (3)
PGE Synthase (3)
Anti-infection (3)
Sirtuin (3)
Adenosine Receptor (3)
FGFR (3)
FLT (3)
Free radical scavengers (3)
Gamma-secretase (3)
VEGFR (3)
TRP/TRPV Channel (3)
Trk receptor (3)
Src (3)
transporter (3)
NADPH (3)
HER (3)
HIF (3)
TGF-beta/Smad (2)
Bcr-Abl (2)
Casein Kinase (2)
Cannabinoid Receptor (2)
Estrogen Receptor/ERR (2)
CaMK (2)
STING (2)
mTOR (2)
Syk (2)
RAAS (2)
PDK (2)
Tyrosine Kinases (2)
Antiviral (2)
Reverse Transcriptase (2)
P-gp (2)
Retinoid Receptor (2)
PKA (2)
RANKL/RANK (2)
Transferase (2)
ATPase (2)
FAK (2)
Molecular Glues (2)
Chloride channel (2)
Leukotriene Receptor (2)
Histamine Receptor (2)
LTR (2)
HSV (2)
IFNAR (2)
Microtubule Associated (2)
GST (2)
GSK-3 (2)
Glutathione Peroxidase (2)
GluR (2)
Drug Metabolite (2)
Immunology/Inflammation related (2)
ROR (1)
SGLT (1)
iGluR (1)
IAP (1)
RSV (1)
S1P Receptor (1)
DUB (1)
Serine Protease (1)
Reductase (1)
Serine/threonin kinase (1)
DYRK (1)
Histone Acetyltransferase (1)
Amylase (1)
Somatostatin (1)
RAR/RXR  (1)
Hedgehog/Smoothened (1)
HCV Protease (1)
HBV (1)
Aminopeptidase (1)
Adrenergic Receptor (1)
Haspin Kinase (1)
Glutathione reductase (1)
Adenosine deaminase (1)
Glucosidase (1)
Glucocorticoid Receptor (1)
Epigenetic Reader Domain (1)
Aromatase (1)
PTEN (1)
Indoleamine 2,3-Dioxygenase (IDO) (1)
cAMP (1)
LRRK2 (1)
BTK (1)
OXPHOS (1)
c-Kit (1)
Mdm2 (1)
OCT (1)
Carbonic Anhydrase (1)
PAK (1)
Chk (1)
CCR (1)
CFTR (1)
Necroptosis (1)
NADPH-oxidase (1)
MLK (1)
cGAS (1)
PAD (1)
BACE (1)
DNA Methyltransferase (1)
PKM (1)
Monoamine Oxidase (1)
Integrin (1)
Discoidin Domain Receptor (DDR) (1)
Aryl Hydrocarbon Receptor (1)
ATM/ATR (1)
PLK (1)
Platelet aggregation (1)
Cysteine Protease (1)
PARP (1)
Complement System (1)
c-Myc (1)
Phospholipase (1)
LDL (1)
Liver X Receptor (1)
PDGFR (1)
Aurora Kinase (1)
NPC1L1 (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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